CY1111488T1 - Φαρμακοτεχνικη μορφη ενωσεων βορονικου οξεος - Google Patents

Φαρμακοτεχνικη μορφη ενωσεων βορονικου οξεος

Info

Publication number
CY1111488T1
CY1111488T1 CY20111100504T CY111100504T CY1111488T1 CY 1111488 T1 CY1111488 T1 CY 1111488T1 CY 20111100504 T CY20111100504 T CY 20111100504T CY 111100504 T CY111100504 T CY 111100504T CY 1111488 T1 CY1111488 T1 CY 1111488T1
Authority
CY
Cyprus
Prior art keywords
boronic acid
acid compounds
compounds
pharmaceutical form
sugar
Prior art date
Application number
CY20111100504T
Other languages
English (en)
Inventor
Shanker Gupta
Original Assignee
The United States Of America, Represented By The Secretary, Department Of Health And Human Services
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23004871&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1111488(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by The United States Of America, Represented By The Secretary, Department Of Health And Human Services filed Critical The United States Of America, Represented By The Secretary, Department Of Health And Human Services
Publication of CY1111488T1 publication Critical patent/CY1111488T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/04—Esters of boric acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02—Linear peptides containing at least one abnormal peptide link
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicinal Preparation (AREA)

Abstract

Η παρούσα εφεύρεση παρέχει σταθερές ενώσεις που παρασκευάζονται από βορονικό οξύ και λυοφιλοποιημένες ενώσεις αυτού του τύπου (1) στον οποίο τα Ζ1 και Ζ2 είναι ομάδες που παράγονται από σάκχαρο. Η εφεύρεση παρέχει επίσης μεθόδους για την παρασκευή τέτοιων ενώσεων. Η λυοφιλοποίηση ενός μίγματος που περιέχει μια ένωση βορονικού οξέος και μια ομάδα που προέρχεται από σάκχαρο παράγει μια σταθερή σύνθεση η οποία απελευθερώνει αμέσως την ένωση βορονικού οξέος κατόπιν ανασύστασης εντός υδατικών μέσων.
CY20111100504T 2001-01-25 2011-05-23 Φαρμακοτεχνικη μορφη ενωσεων βορονικου οξεος CY1111488T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26416001P 2001-01-25 2001-01-25
EP02709145A EP1355910B1 (en) 2001-01-25 2002-01-25 Formulation of boronic acid compounds

Publications (1)

Publication Number Publication Date
CY1111488T1 true CY1111488T1 (el) 2015-08-05

Family

ID=23004871

Family Applications (2)

Application Number Title Priority Date Filing Date
CY20111100504T CY1111488T1 (el) 2001-01-25 2011-05-23 Φαρμακοτεχνικη μορφη ενωσεων βορονικου οξεος
CY20181101322T CY1121142T1 (el) 2001-01-25 2018-12-11 Τυποποιηση ενωσεων βορονικου οξεος

Family Applications After (1)

Application Number Title Priority Date Filing Date
CY20181101322T CY1121142T1 (el) 2001-01-25 2018-12-11 Τυποποιηση ενωσεων βορονικου οξεος

Country Status (15)

Country Link
US (5) US6713446B2 (el)
EP (4) EP2251344B2 (el)
JP (2) JP4162491B2 (el)
AT (1) ATE501157T1 (el)
AU (1) AU2002243646B2 (el)
CA (2) CA2435146C (el)
CY (2) CY1111488T1 (el)
DE (1) DE60239384D1 (el)
DK (3) DK1355910T3 (el)
ES (2) ES2571219T3 (el)
FI (1) FI2251344T4 (el)
HK (1) HK1149936A1 (el)
PT (2) PT3078667T (el)
TR (1) TR201819416T4 (el)
WO (2) WO2002059131A1 (el)

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