CY1111087T1 - Παραγωγα 5-(βενζ-(ζ)-υλιδενο)-θειαζολιδιν-4-ονης ως ανοσοκατασταλτικοι παραγοντες - Google Patents
Παραγωγα 5-(βενζ-(ζ)-υλιδενο)-θειαζολιδιν-4-ονης ως ανοσοκατασταλτικοι παραγοντεςInfo
- Publication number
- CY1111087T1 CY1111087T1 CY20101101140T CY101101140T CY1111087T1 CY 1111087 T1 CY1111087 T1 CY 1111087T1 CY 20101101140 T CY20101101140 T CY 20101101140T CY 101101140 T CY101101140 T CY 101101140T CY 1111087 T1 CY1111087 T1 CY 1111087T1
- Authority
- CY
- Cyprus
- Prior art keywords
- thiazolidin
- benz
- derivatives
- ylideno
- immediately
- Prior art date
Links
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- C07—ORGANIC CHEMISTRY
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- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/54—Nitrogen and either oxygen or sulfur atoms
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
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Abstract
Η εφεύρεση αφορά σε φαρμακευτικές συνθέσεις οι οποίες περιέχουν τουλάχιστον ένα παράγωγο 5-βενζ-(Ζ)-υλιδενο)-θειαζολιδιν-4-όνης (I), για την πρόληψη ή θεραπευτική αντιμετώπιση διαταραχών που σχετίζονται με ένα ενεργοποιημένο ανοσοποιητικό σύστημα. Περαιτέρω, η εφεύρεση αφορά σε νέα παράγωγα θειαζολιδιν-4-όνης, συγκεκριμένα για χρήση ως φαρμακευτικά δραστικές ενώσεις. Οι εν λόγω ενώσεις επίσης δρουν ιδίως ως ανοσοκατασταλτικοί παράγοντες.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP0313072 | 2003-11-21 | ||
EP04819591A EP1689726B1 (en) | 2003-11-21 | 2004-11-16 | 5-(benz- (z) -ylidene) -thiazolidin-4-one derivatives as immunosuppressant agents |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1111087T1 true CY1111087T1 (el) | 2015-06-11 |
Family
ID=34639216
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20101101140T CY1111087T1 (el) | 2003-11-21 | 2010-12-10 | Παραγωγα 5-(βενζ-(ζ)-υλιδενο)-θειαζολιδιν-4-ονης ως ανοσοκατασταλτικοι παραγοντες |
Country Status (26)
Country | Link |
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US (8) | US7435828B2 (el) |
EP (2) | EP2295418A1 (el) |
JP (2) | JP4061332B2 (el) |
KR (1) | KR100783835B1 (el) |
CN (1) | CN100567275C (el) |
AR (1) | AR047128A1 (el) |
AT (1) | ATE483698T1 (el) |
AU (1) | AU2004295047B2 (el) |
BR (1) | BRPI0416752B8 (el) |
CA (1) | CA2545582C (el) |
CY (1) | CY1111087T1 (el) |
DE (1) | DE602004029493D1 (el) |
DK (1) | DK1689726T3 (el) |
ES (1) | ES2352555T3 (el) |
HR (1) | HRP20100714T1 (el) |
IL (1) | IL175758A (el) |
MY (1) | MY145074A (el) |
NO (1) | NO336734B1 (el) |
NZ (1) | NZ547962A (el) |
PL (1) | PL1689726T3 (el) |
PT (1) | PT1689726E (el) |
RU (1) | RU2379299C2 (el) |
SI (1) | SI1689726T1 (el) |
TW (1) | TWI323659B (el) |
WO (1) | WO2005054215A1 (el) |
ZA (1) | ZA200605077B (el) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SI1689726T1 (sl) | 2003-11-21 | 2011-01-31 | Actelion Pharmaceuticals Ltd | Derivati 5-(benz-(z)-iliden)-tiazolidin-4-ona kot imunosupresivna sredstva |
USRE43833E1 (en) | 2003-11-21 | 2012-11-27 | Actelion Pharmaceuticals Ltd. | Thiazolidin-4-one derivatives |
WO2005082901A1 (en) * | 2004-02-25 | 2005-09-09 | Smithkline Beecham Corporation | Novel chemical compounds |
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