SI1689726T1 - Derivati 5-(benz-(z)-iliden)-tiazolidin-4-ona kot imunosupresivna sredstva - Google Patents

Derivati 5-(benz-(z)-iliden)-tiazolidin-4-ona kot imunosupresivna sredstva

Info

Publication number
SI1689726T1
SI1689726T1 SI200431556T SI200431556T SI1689726T1 SI 1689726 T1 SI1689726 T1 SI 1689726T1 SI 200431556 T SI200431556 T SI 200431556T SI 200431556 T SI200431556 T SI 200431556T SI 1689726 T1 SI1689726 T1 SI 1689726T1
Authority
SI
Slovenia
Prior art keywords
thiazolidin
benz
ylidene
derivatives
immunosuppressant agents
Prior art date
Application number
SI200431556T
Other languages
English (en)
Inventor
Martin Bolli
Michael Scherz
Claus Mueller
Boris Mathys
Christoph Binkert
Oliver Nayler
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34639216&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1689726(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of SI1689726T1 publication Critical patent/SI1689726T1/sl

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    • C—CHEMISTRY; METALLURGY
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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/54—Nitrogen and either oxygen or sulfur atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
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    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
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    • C07D277/38—Nitrogen atoms
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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Veterinary Medicine (AREA)
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
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  • Neurology (AREA)
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  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
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SI200431556T 2003-11-21 2004-11-16 Derivati 5-(benz-(z)-iliden)-tiazolidin-4-ona kot imunosupresivna sredstva SI1689726T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP0313072 2003-11-21
EP04819591A EP1689726B1 (en) 2003-11-21 2004-11-16 5-(benz- (z) -ylidene) -thiazolidin-4-one derivatives as immunosuppressant agents
PCT/EP2004/012953 WO2005054215A1 (en) 2003-11-21 2004-11-16 5-(benz- (z) -ylidene) -thiazolidin-4-one derivatives as immunosuppressant agents

Publications (1)

Publication Number Publication Date
SI1689726T1 true SI1689726T1 (sl) 2011-01-31

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Family Applications (1)

Application Number Title Priority Date Filing Date
SI200431556T SI1689726T1 (sl) 2003-11-21 2004-11-16 Derivati 5-(benz-(z)-iliden)-tiazolidin-4-ona kot imunosupresivna sredstva

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Country Link
US (8) US7435828B2 (sl)
EP (2) EP1689726B1 (sl)
JP (2) JP4061332B2 (sl)
KR (1) KR100783835B1 (sl)
CN (1) CN100567275C (sl)
AR (1) AR047128A1 (sl)
AT (1) ATE483698T1 (sl)
AU (1) AU2004295047B2 (sl)
BR (1) BRPI0416752B8 (sl)
CA (1) CA2545582C (sl)
CY (1) CY1111087T1 (sl)
DE (1) DE602004029493D1 (sl)
DK (1) DK1689726T3 (sl)
ES (1) ES2352555T3 (sl)
HR (1) HRP20100714T1 (sl)
IL (1) IL175758A (sl)
MY (1) MY145074A (sl)
NO (1) NO336734B1 (sl)
NZ (1) NZ547962A (sl)
PL (1) PL1689726T3 (sl)
PT (1) PT1689726E (sl)
RU (1) RU2379299C2 (sl)
SI (1) SI1689726T1 (sl)
TW (1) TWI323659B (sl)
WO (1) WO2005054215A1 (sl)
ZA (1) ZA200605077B (sl)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
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PL1689726T3 (pl) 2003-11-21 2011-05-31 Actelion Pharmaceuticals Ltd Pochodne 5-(benz-(z)-ylideno)tiazolidyn-4-onu jako środki immunosupresyjne
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