CS264332B2 - Process for preparing aminoalcohols - Google Patents

Process for preparing aminoalcohols Download PDF

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Publication number
CS264332B2
CS264332B2 CS856904A CS690485A CS264332B2 CS 264332 B2 CS264332 B2 CS 264332B2 CS 856904 A CS856904 A CS 856904A CS 690485 A CS690485 A CS 690485A CS 264332 B2 CS264332 B2 CS 264332B2
Authority
CS
Czechoslovakia
Prior art keywords
compound
methyl
dihydrochloride
formula
ethanol
Prior art date
Application number
CS856904A
Other languages
Czech (cs)
English (en)
Other versions
CS690485A2 (en
Inventor
Mitsuo Masaki
Haruhiko Shinozaki
Masaru Satoh
Naoya Moritoh
Koichi Hashimoto
Toshiro Kamishiro
Original Assignee
Nippon Chemiphar Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Chemiphar Co filed Critical Nippon Chemiphar Co
Publication of CS690485A2 publication Critical patent/CS690485A2/cs
Publication of CS264332B2 publication Critical patent/CS264332B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CS856904A 1984-09-28 1985-09-26 Process for preparing aminoalcohols CS264332B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP59203623A JPS6183147A (ja) 1984-09-28 1984-09-28 新規なアミノアルコール誘導体およびその製造法並びにそれを有効成分とするグルタミン酸遮断剤

Publications (2)

Publication Number Publication Date
CS690485A2 CS690485A2 (en) 1988-11-15
CS264332B2 true CS264332B2 (en) 1989-07-12

Family

ID=16477107

Family Applications (1)

Application Number Title Priority Date Filing Date
CS856904A CS264332B2 (en) 1984-09-28 1985-09-26 Process for preparing aminoalcohols

Country Status (21)

Country Link
EP (1) EP0177245B1 (da)
JP (1) JPS6183147A (da)
KR (1) KR910002671B1 (da)
AR (1) AR242776A1 (da)
AT (1) ATE62480T1 (da)
AU (1) AU578737B2 (da)
BR (1) BR8504879A (da)
CA (1) CA1260467A (da)
CS (1) CS264332B2 (da)
DE (1) DE3582466D1 (da)
DK (1) DK167117B1 (da)
ES (1) ES8706610A1 (da)
HU (1) HU199774B (da)
IN (1) IN162767B (da)
MX (1) MX162733A (da)
MY (1) MY102921A (da)
NZ (1) NZ213628A (da)
PH (1) PH21169A (da)
RO (1) RO93388B (da)
SU (1) SU1433409A3 (da)
ZA (1) ZA857449B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5070196A (en) * 1986-02-01 1991-12-03 Nippon Chemiphar Co., Ltd. Alkylenediamine derivatives
CA1318913C (en) * 1986-02-01 1993-06-08 Toshiro Kamishiro Alkylenediamine derivatives
JPH0314562A (ja) * 1988-04-11 1991-01-23 Nippon Chemiphar Co Ltd 新規なアルキレンジアミン誘導体およびグルタミン酸遮断剤
AU2159692A (en) * 1991-06-06 1993-01-12 G.D. Searle & Co. N-(arylethyl)-n-alkyl-2-(1-pyrrolidinyl)ethylamine derivatives for cns disorders
IT1271623B (it) * 1994-03-21 1997-06-04 Lifegroup Spa N-acilderivati di aminoalcoli con acidi monocarbossilici e bicarbossilici con attivita' neuroprotettiva nelle patologie neurologiche correlate ad eccitotossicita'
CA2231013A1 (en) * 1997-04-30 1998-10-30 Eli Lilly And Company Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
DE10251170A1 (de) * 2002-10-31 2004-05-13 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Beta-Agonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
US20040127733A1 (en) 2002-10-31 2004-07-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg New beta-agonists, processes for preparing them and their use as pharmaceutical compositions
DE102004021779A1 (de) 2004-04-30 2005-11-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Beta-Agonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
DE102005052127A1 (de) 2005-10-28 2007-05-03 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue indol-haltige Beta-Agonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2600217A (en) * 1948-06-22 1952-06-10 American Cyanamid Co Diaryl-hydroxyalkyl-diamino compounds and preparation thereof
US3092636A (en) * 1959-10-21 1963-06-04 Upjohn Co Alpha-[2-(1-alkyleneimino) ethylamino]-alkanophenones and the corresponding alcohols
GB1200886A (en) * 1966-09-23 1970-08-05 Allen & Hanburys Ltd Phenylaminoethanol derivatives
US3517000A (en) * 1968-08-08 1970-06-23 American Home Prod Alpha-aminomethyl benzyl alcohols
FR2370472A2 (fr) * 1976-11-10 1978-06-09 Continental Pharma Amino-alcool heterocyclique, son sel et son procede de preparation
JPS6183170A (ja) * 1984-09-28 1986-04-26 Nippon Chemiphar Co Ltd 新規な１，３−オキサゾリジン−２−オン誘導体およびその製造法

Also Published As

Publication number Publication date
IN162767B (da) 1988-07-09
BR8504879A (pt) 1986-07-22
ES8706610A1 (es) 1987-07-01
EP0177245B1 (en) 1991-04-10
RO93388B (ro) 1988-01-03
DK439285D0 (da) 1985-09-27
SU1433409A3 (ru) 1988-10-23
PH21169A (en) 1987-08-07
ATE62480T1 (de) 1991-04-15
DK167117B1 (da) 1993-08-30
EP0177245A3 (en) 1987-07-01
KR910002671B1 (ko) 1991-05-03
MX162733A (es) 1991-06-24
HU199774B (en) 1990-03-28
NZ213628A (en) 1989-03-29
ZA857449B (en) 1986-06-25
JPH0517900B2 (da) 1993-03-10
AR242776A1 (es) 1993-05-31
HUT40613A (en) 1987-01-28
CA1260467A (en) 1989-09-26
EP0177245A2 (en) 1986-04-09
KR860002450A (ko) 1986-04-26
AU578737B2 (en) 1988-11-03
ES547283A0 (es) 1987-07-01
DE3582466D1 (de) 1991-05-16
MY102921A (en) 1993-03-31
CS690485A2 (en) 1988-11-15
RO93388A (ro) 1987-12-31
AU4768985A (en) 1986-04-10
JPS6183147A (ja) 1986-04-26
DK439285A (da) 1986-03-29

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