CS226743B2 - Method of preparing new 1,4,9,10-tetrahydropyrazolo (4,3-e)pyrido (3,2-b) l,4)diazepin-10-ones - Google Patents
Method of preparing new 1,4,9,10-tetrahydropyrazolo (4,3-e)pyrido (3,2-b) l,4)diazepin-10-ones Download PDFInfo
- Publication number
- CS226743B2 CS226743B2 CS824137A CS413782A CS226743B2 CS 226743 B2 CS226743 B2 CS 226743B2 CS 824137 A CS824137 A CS 824137A CS 413782 A CS413782 A CS 413782A CS 226743 B2 CS226743 B2 CS 226743B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- alkyl group
- pyrido
- carbon atoms
- defined above
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19813122670 DE3122670A1 (de) | 1981-06-06 | 1981-06-06 | "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen" |
Publications (1)
Publication Number | Publication Date |
---|---|
CS226743B2 true CS226743B2 (en) | 1984-04-16 |
Family
ID=6134176
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS824137A CS226743B2 (en) | 1981-06-06 | 1982-06-03 | Method of preparing new 1,4,9,10-tetrahydropyrazolo (4,3-e)pyrido (3,2-b) l,4)diazepin-10-ones |
Country Status (27)
Country | Link |
---|---|
US (1) | US4381303A (fr) |
EP (1) | EP0066774B1 (fr) |
JP (1) | JPS57212182A (fr) |
KR (1) | KR880001719B1 (fr) |
AR (1) | AR229124A1 (fr) |
AT (1) | ATE10744T1 (fr) |
AU (1) | AU552765B2 (fr) |
CA (1) | CA1167440A (fr) |
CS (1) | CS226743B2 (fr) |
DD (1) | DD202574A5 (fr) |
DE (2) | DE3122670A1 (fr) |
DK (1) | DK253382A (fr) |
ES (1) | ES512846A0 (fr) |
FI (1) | FI71560C (fr) |
GB (1) | GB2117755B (fr) |
GR (1) | GR76438B (fr) |
HU (1) | HU186067B (fr) |
IE (1) | IE53067B1 (fr) |
IL (1) | IL65977A (fr) |
NO (1) | NO158063C (fr) |
NZ (1) | NZ200859A (fr) |
PH (1) | PH17719A (fr) |
PL (1) | PL135845B1 (fr) |
PT (1) | PT75016B (fr) |
SU (1) | SU1103795A3 (fr) |
YU (1) | YU118282A (fr) |
ZA (1) | ZA823919B (fr) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3643666A1 (de) * | 1986-12-20 | 1988-06-30 | Thomae Gmbh Dr K | Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
US4749788A (en) * | 1987-04-13 | 1988-06-07 | A. H. Robins Company, Incorporated | Process for the preparation of aryl-pyrido(1,4) benzodiazepines |
US5366972A (en) * | 1989-04-20 | 1994-11-22 | Boehringer Ingelheim Pharmaceuticals, Inc. | 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection |
DK0410148T3 (da) * | 1989-06-28 | 1994-08-08 | Boehringer Ingelheim Pharma | Hidtil ukendte 5,11-dihydro-6H-dipyrido(3,2-b:2,3-e)-(1,4)diazepin-6-oner og -thioner og deres anvendelse til forebyggelse eller behandling af AIDS |
CA2052946A1 (fr) * | 1990-10-19 | 1992-04-20 | Karl G. Grozinger | Methode de preparation de 5,11-dihydro-6h-dipyrido¬3,2-b:2',3'-e|¬1,4|diazepines |
ES2137113B1 (es) | 1997-07-29 | 2000-09-16 | Almirall Prodesfarma Sa | Nuevos derivados de triazolo-piridazinas heterociclicos. |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3450694A (en) * | 1966-02-23 | 1969-06-17 | Abbott Lab | Substituted benzoxazepines and benzothiazepines |
DE2707269A1 (de) * | 1977-02-19 | 1978-08-24 | Hoechst Ag | Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung |
DE3071581D1 (en) * | 1979-08-03 | 1986-06-05 | Byk Gulden Lomberg Chem Fab | Substituted tetraazatricyclic compounds, process for their preparation, their use and medicines containing them |
-
1981
- 1981-06-06 DE DE19813122670 patent/DE3122670A1/de not_active Withdrawn
-
1982
- 1982-05-13 US US06/377,911 patent/US4381303A/en not_active Expired - Fee Related
- 1982-05-25 DE DE8282104549T patent/DE3261530D1/de not_active Expired
- 1982-05-25 EP EP82104549A patent/EP0066774B1/fr not_active Expired
- 1982-05-25 AT AT82104549T patent/ATE10744T1/de not_active IP Right Cessation
- 1982-05-25 SU SU823441915A patent/SU1103795A3/ru active
- 1982-06-01 AR AR289564A patent/AR229124A1/es active
- 1982-06-02 GR GR68322A patent/GR76438B/el unknown
- 1982-06-03 DD DD82240437A patent/DD202574A5/de unknown
- 1982-06-03 YU YU01182/82A patent/YU118282A/xx unknown
- 1982-06-03 KR KR8202494A patent/KR880001719B1/ko active
- 1982-06-03 CS CS824137A patent/CS226743B2/cs unknown
- 1982-06-03 PL PL1982236742A patent/PL135845B1/pl unknown
- 1982-06-04 FI FI821992A patent/FI71560C/fi not_active IP Right Cessation
- 1982-06-04 PT PT75016A patent/PT75016B/pt unknown
- 1982-06-04 ZA ZA823919A patent/ZA823919B/xx unknown
- 1982-06-04 CA CA000404541A patent/CA1167440A/fr not_active Expired
- 1982-06-04 AU AU84605/82A patent/AU552765B2/en not_active Ceased
- 1982-06-04 IL IL65977A patent/IL65977A/xx unknown
- 1982-06-04 NZ NZ200859A patent/NZ200859A/en unknown
- 1982-06-04 IE IE1350/82A patent/IE53067B1/en unknown
- 1982-06-04 HU HU821823A patent/HU186067B/hu unknown
- 1982-06-04 PH PH27402A patent/PH17719A/en unknown
- 1982-06-04 DK DK253382A patent/DK253382A/da not_active Application Discontinuation
- 1982-06-04 JP JP57096080A patent/JPS57212182A/ja active Pending
- 1982-06-04 ES ES512846A patent/ES512846A0/es active Granted
- 1982-06-04 NO NO821882A patent/NO158063C/no unknown
- 1982-06-04 GB GB08216381A patent/GB2117755B/en not_active Expired
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