IL65977A - 1,4,9,10-tetrahydropyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-one derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

1,4,9,10-tetrahydropyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-one derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL65977A
IL65977A IL65977A IL6597782A IL65977A IL 65977 A IL65977 A IL 65977A IL 65977 A IL65977 A IL 65977A IL 6597782 A IL6597782 A IL 6597782A IL 65977 A IL65977 A IL 65977A
Authority
IL
Israel
Prior art keywords
tetrahydropyrazolo
diazepin
pyrido
derivatives
preparation
Prior art date
Application number
IL65977A
Other languages
English (en)
Other versions
IL65977A0 (en
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of IL65977A0 publication Critical patent/IL65977A0/xx
Publication of IL65977A publication Critical patent/IL65977A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL65977A 1981-06-06 1982-06-04 1,4,9,10-tetrahydropyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-one derivatives,their preparation and pharmaceutical compositions containing them IL65977A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813122670 DE3122670A1 (de) 1981-06-06 1981-06-06 "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen"

Publications (2)

Publication Number Publication Date
IL65977A0 IL65977A0 (en) 1982-09-30
IL65977A true IL65977A (en) 1984-12-31

Family

ID=6134176

Family Applications (1)

Application Number Title Priority Date Filing Date
IL65977A IL65977A (en) 1981-06-06 1982-06-04 1,4,9,10-tetrahydropyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-one derivatives,their preparation and pharmaceutical compositions containing them

Country Status (27)

Country Link
US (1) US4381303A (fr)
EP (1) EP0066774B1 (fr)
JP (1) JPS57212182A (fr)
KR (1) KR880001719B1 (fr)
AR (1) AR229124A1 (fr)
AT (1) ATE10744T1 (fr)
AU (1) AU552765B2 (fr)
CA (1) CA1167440A (fr)
CS (1) CS226743B2 (fr)
DD (1) DD202574A5 (fr)
DE (2) DE3122670A1 (fr)
DK (1) DK253382A (fr)
ES (1) ES512846A0 (fr)
FI (1) FI71560C (fr)
GB (1) GB2117755B (fr)
GR (1) GR76438B (fr)
HU (1) HU186067B (fr)
IE (1) IE53067B1 (fr)
IL (1) IL65977A (fr)
NO (1) NO158063C (fr)
NZ (1) NZ200859A (fr)
PH (1) PH17719A (fr)
PL (1) PL135845B1 (fr)
PT (1) PT75016B (fr)
SU (1) SU1103795A3 (fr)
YU (1) YU118282A (fr)
ZA (1) ZA823919B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3643666A1 (de) * 1986-12-20 1988-06-30 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US4749788A (en) * 1987-04-13 1988-06-07 A. H. Robins Company, Incorporated Process for the preparation of aryl-pyrido(1,4) benzodiazepines
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
ATE103918T1 (de) * 1989-06-28 1994-04-15 Boehringer Ingelheim Pharma 5,11-dihydro-6h-dipyrido(3,2-b:2',3'e>(1,4>diazepin-6-one und -thione und ihre verwendung bei der aids-vorbeugung oder behandlung.
CA2052946A1 (fr) * 1990-10-19 1992-04-20 Karl G. Grozinger Methode de preparation de 5,11-dihydro-6h-dipyrido¬3,2-b:2',3'-e|¬1,4|diazepines
ES2137113B1 (es) 1997-07-29 2000-09-16 Almirall Prodesfarma Sa Nuevos derivados de triazolo-piridazinas heterociclicos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3450694A (en) * 1966-02-23 1969-06-17 Abbott Lab Substituted benzoxazepines and benzothiazepines
DE2707269A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung
DK334580A (da) * 1979-08-03 1981-02-04 Byk Gulden Lomberg Chem Fab Fremgangsmaade til fremstilling af substituerede tetraazatricycler

Also Published As

Publication number Publication date
PT75016B (de) 1985-05-17
KR840000543A (ko) 1984-02-25
ZA823919B (en) 1984-02-29
PL135845B1 (en) 1985-12-31
YU118282A (en) 1986-04-30
ES8304571A1 (es) 1983-03-01
GB2117755A (en) 1983-10-19
NO158063C (no) 1988-07-06
AU552765B2 (en) 1986-06-19
DE3261530D1 (en) 1985-01-24
HU186067B (en) 1985-05-28
NZ200859A (en) 1985-08-16
IL65977A0 (en) 1982-09-30
PL236742A1 (en) 1984-03-26
NO158063B (no) 1988-03-28
GR76438B (fr) 1984-08-10
FI821992A0 (fi) 1982-06-04
IE53067B1 (en) 1988-05-25
FI71560B (fi) 1986-10-10
JPS57212182A (en) 1982-12-27
DE3122670A1 (de) 1982-12-23
IE821350L (en) 1982-12-06
DK253382A (da) 1982-12-07
DD202574A5 (de) 1983-09-21
EP0066774A1 (fr) 1982-12-15
ES512846A0 (es) 1983-03-01
ATE10744T1 (de) 1984-12-15
AR229124A1 (es) 1983-06-15
CS226743B2 (en) 1984-04-16
EP0066774B1 (fr) 1984-12-12
SU1103795A3 (ru) 1984-07-15
GB2117755B (en) 1985-01-30
NO821882L (no) 1982-12-07
PT75016A (de) 1982-07-01
US4381303A (en) 1983-04-26
CA1167440A (fr) 1984-05-15
KR880001719B1 (ko) 1988-09-08
PH17719A (en) 1984-11-21
FI71560C (fi) 1987-01-19
AU8460582A (en) 1982-12-16

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