FI821992A0 - Nya 1,4,9,10-tetrahydro-pyratsolo/4,3-e/-pyrido/3,2-b//1,4/diazepin-10-oner, foerfarande foer deras framstaellning och dessa foereningar innehaollande laekemedel - Google Patents

Nya 1,4,9,10-tetrahydro-pyratsolo/4,3-e/-pyrido/3,2-b//1,4/diazepin-10-oner, foerfarande foer deras framstaellning och dessa foereningar innehaollande laekemedel

Info

Publication number
FI821992A0
FI821992A0 FI821992A FI821992A FI821992A0 FI 821992 A0 FI821992 A0 FI 821992A0 FI 821992 A FI821992 A FI 821992A FI 821992 A FI821992 A FI 821992A FI 821992 A0 FI821992 A0 FI 821992A0
Authority
FI
Finland
Prior art keywords
pyratsolo
oner
nya
diazepin
pyrido
Prior art date
Application number
FI821992A
Other languages
English (en)
Other versions
FI71560C (fi
FI71560B (fi
Inventor
Guenther Schmidt
Wolfhard Engel
Wolfgang Eberlein
Guenter Trummlitz
Guenther Engelhardt
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of FI821992A0 publication Critical patent/FI821992A0/fi
Application granted granted Critical
Publication of FI71560B publication Critical patent/FI71560B/fi
Publication of FI71560C publication Critical patent/FI71560C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI821992A 1981-06-06 1982-06-04 Foerfarande foer framstaellning av nya analgetiska, antiflogistiska och antipyretiska 1,4,9,10-tetrahydropyrazolo -/4,3-e/pyrido/3,2-b//1,4/diazepin-10-oner. FI71560C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3122670 1981-06-06
DE19813122670 DE3122670A1 (de) 1981-06-06 1981-06-06 "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen"

Publications (3)

Publication Number Publication Date
FI821992A0 true FI821992A0 (fi) 1982-06-04
FI71560B FI71560B (fi) 1986-10-10
FI71560C FI71560C (fi) 1987-01-19

Family

ID=6134176

Family Applications (1)

Application Number Title Priority Date Filing Date
FI821992A FI71560C (fi) 1981-06-06 1982-06-04 Foerfarande foer framstaellning av nya analgetiska, antiflogistiska och antipyretiska 1,4,9,10-tetrahydropyrazolo -/4,3-e/pyrido/3,2-b//1,4/diazepin-10-oner.

Country Status (27)

Country Link
US (1) US4381303A (fi)
EP (1) EP0066774B1 (fi)
JP (1) JPS57212182A (fi)
KR (1) KR880001719B1 (fi)
AR (1) AR229124A1 (fi)
AT (1) ATE10744T1 (fi)
AU (1) AU552765B2 (fi)
CA (1) CA1167440A (fi)
CS (1) CS226743B2 (fi)
DD (1) DD202574A5 (fi)
DE (2) DE3122670A1 (fi)
DK (1) DK253382A (fi)
ES (1) ES512846A0 (fi)
FI (1) FI71560C (fi)
GB (1) GB2117755B (fi)
GR (1) GR76438B (fi)
HU (1) HU186067B (fi)
IE (1) IE53067B1 (fi)
IL (1) IL65977A (fi)
NO (1) NO158063C (fi)
NZ (1) NZ200859A (fi)
PH (1) PH17719A (fi)
PL (1) PL135845B1 (fi)
PT (1) PT75016B (fi)
SU (1) SU1103795A3 (fi)
YU (1) YU118282A (fi)
ZA (1) ZA823919B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3643666A1 (de) * 1986-12-20 1988-06-30 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US4749788A (en) * 1987-04-13 1988-06-07 A. H. Robins Company, Incorporated Process for the preparation of aryl-pyrido(1,4) benzodiazepines
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
DK0410148T3 (da) * 1989-06-28 1994-08-08 Boehringer Ingelheim Pharma Hidtil ukendte 5,11-dihydro-6H-dipyrido(3,2-b:2,3-e)-(1,4)diazepin-6-oner og -thioner og deres anvendelse til forebyggelse eller behandling af AIDS
CA2052946A1 (en) * 1990-10-19 1992-04-20 Karl G. Grozinger Method for the preparation of 5,11-dihydro-6h-dipyrido ¬3,2-b:2', 3'-e| ¬1,4|diazepines
ES2137113B1 (es) 1997-07-29 2000-09-16 Almirall Prodesfarma Sa Nuevos derivados de triazolo-piridazinas heterociclicos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3450694A (en) * 1966-02-23 1969-06-17 Abbott Lab Substituted benzoxazepines and benzothiazepines
DE2707269A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung
CA1154762A (en) * 1979-08-03 1983-10-04 Georg Rainer Substituted tetraazatricyclic compounds, a process for their preparation, their use and medicaments containing them

Also Published As

Publication number Publication date
IL65977A0 (en) 1982-09-30
PL236742A1 (en) 1984-03-26
ES8304571A1 (es) 1983-03-01
DK253382A (da) 1982-12-07
DD202574A5 (de) 1983-09-21
SU1103795A3 (ru) 1984-07-15
IE53067B1 (en) 1988-05-25
AR229124A1 (es) 1983-06-15
PL135845B1 (en) 1985-12-31
NO821882L (no) 1982-12-07
FI71560C (fi) 1987-01-19
FI71560B (fi) 1986-10-10
NO158063B (no) 1988-03-28
HU186067B (en) 1985-05-28
JPS57212182A (en) 1982-12-27
US4381303A (en) 1983-04-26
YU118282A (en) 1986-04-30
IL65977A (en) 1984-12-31
DE3261530D1 (en) 1985-01-24
CS226743B2 (en) 1984-04-16
PH17719A (en) 1984-11-21
KR840000543A (ko) 1984-02-25
GB2117755A (en) 1983-10-19
ATE10744T1 (de) 1984-12-15
PT75016B (de) 1985-05-17
CA1167440A (en) 1984-05-15
NO158063C (no) 1988-07-06
NZ200859A (en) 1985-08-16
ES512846A0 (es) 1983-03-01
ZA823919B (en) 1984-02-29
AU552765B2 (en) 1986-06-19
IE821350L (en) 1982-12-06
GB2117755B (en) 1985-01-30
AU8460582A (en) 1982-12-16
PT75016A (de) 1982-07-01
KR880001719B1 (ko) 1988-09-08
EP0066774B1 (de) 1984-12-12
DE3122670A1 (de) 1982-12-23
GR76438B (fi) 1984-08-10
EP0066774A1 (de) 1982-12-15

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: DR. KARL THOMAE GESELLSCHAFT MIT