CO4940420A1 - Nuevo metodo de tratamiento - Google Patents

Nuevo metodo de tratamiento

Info

Publication number
CO4940420A1
CO4940420A1 CO98040747A CO98040747A CO4940420A1 CO 4940420 A1 CO4940420 A1 CO 4940420A1 CO 98040747 A CO98040747 A CO 98040747A CO 98040747 A CO98040747 A CO 98040747A CO 4940420 A1 CO4940420 A1 CO 4940420A1
Authority
CO
Colombia
Prior art keywords
dione
benzyl
benzopyran
thiazolidine
dihydro
Prior art date
Application number
CO98040747A
Other languages
English (en)
Spanish (es)
Inventor
Robin Edwin Buckingham
Stephen Alistair Smith
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of CO4940420A1 publication Critical patent/CO4940420A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/64Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CO98040747A 1997-07-18 1998-07-17 Nuevo metodo de tratamiento CO4940420A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9715295A GB9715295D0 (en) 1997-07-18 1997-07-18 Novel method of treatment

Publications (1)

Publication Number Publication Date
CO4940420A1 true CO4940420A1 (es) 2000-07-24

Family

ID=10816167

Family Applications (1)

Application Number Title Priority Date Filing Date
CO98040747A CO4940420A1 (es) 1997-07-18 1998-07-17 Nuevo metodo de tratamiento

Country Status (39)

Country Link
EP (1) EP1001783B1 (enExample)
JP (2) JP2001510159A (enExample)
KR (1) KR100671918B1 (enExample)
CN (1) CN1264303A (enExample)
AP (1) AP1352A (enExample)
AR (1) AR016349A1 (enExample)
AT (1) ATE305790T1 (enExample)
AU (1) AU8448898A (enExample)
BG (1) BG64785B1 (enExample)
BR (1) BR9810445A (enExample)
CA (1) CA2296653C (enExample)
CO (1) CO4940420A1 (enExample)
CY (1) CY1105254T1 (enExample)
DE (1) DE69831808T2 (enExample)
DK (1) DK1001783T3 (enExample)
DZ (1) DZ2562A1 (enExample)
EA (1) EA003021B1 (enExample)
ES (1) ES2251093T3 (enExample)
GB (1) GB9715295D0 (enExample)
HU (1) HUP0003629A3 (enExample)
ID (1) ID24211A (enExample)
IL (1) IL134046A0 (enExample)
IN (1) IN189275B (enExample)
MA (1) MA24607A1 (enExample)
MY (1) MY155219A (enExample)
NO (1) NO325727B1 (enExample)
NZ (2) NZ511608A (enExample)
OA (1) OA11279A (enExample)
PE (1) PE99599A1 (enExample)
PL (2) PL197844B1 (enExample)
SA (1) SA98190468B1 (enExample)
SI (1) SI1001783T1 (enExample)
SK (1) SK285484B6 (enExample)
TR (1) TR200000134T2 (enExample)
TW (1) TW505516B (enExample)
UA (1) UA70303C2 (enExample)
UY (1) UY25102A1 (enExample)
WO (1) WO1999003477A1 (enExample)
ZA (1) ZA986363B (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6011049A (en) * 1997-02-19 2000-01-04 Warner-Lambert Company Combinations for diabetes
US6099862A (en) * 1998-08-31 2000-08-08 Andrx Corporation Oral dosage form for the controlled release of a biguanide and sulfonylurea
EA007610B1 (ru) * 1998-11-12 2006-12-29 Смитклайн Бичам Плс Таблетка с энтеропокрытием, обеспечивающая отсроченное высвобождение
SE9902918D0 (sv) * 1999-08-13 1999-08-13 Pharmacia & Upjohn Ab Methods for identification of compounds stimulating insulin secretion
MY125516A (en) * 1999-11-16 2006-08-30 Smithkline Beecham Plc Novel composition based on thiazolidinedione and metformin and use
AU1403501A (en) * 1999-11-16 2001-05-30 Smithkline Beecham Plc Novel composition and use
FR2812547B1 (fr) * 2000-08-04 2002-10-31 Lipha Composition pharmaceutique comprenant une association metformine et derive de thiazolidinedione et son utilisation pour la preparation de medicaments destines a traiter le diabete
WO2002055009A1 (en) 2001-01-12 2002-07-18 Sun Pharmaceutical Industries Limited Spaced drug delivery system
ITFI20010126A1 (it) * 2001-07-09 2003-01-09 Molteni & C Composizioni farmaceutiche per uso orale,contenenti,in combinazione,metformina e gliclazide
JP2004536843A (ja) * 2001-07-10 2004-12-09 エアロファーム テクノロジー インコーポレイテッド ピオグリタゾンおよびビグアナイドを含むコア製剤
WO2003105809A1 (en) 2002-06-17 2003-12-24 Themis Laboratories Private Limited Multilayer tablets containing thiazolidinedione and biguanides and methods for producing them
AU2003272504A1 (en) * 2002-09-20 2004-04-08 Andrx Labs Llc Multistage formulation containing a biguanide and thiazolidindione derivatives
UA80991C2 (en) 2002-10-07 2007-11-26 Solid preparation containing an insulin resistance improving drug and an active ingredient useful as a remedy for diabetes
CN1874774B (zh) 2003-10-31 2011-04-13 武田药品工业株式会社 包含胰岛素致敏剂、胰岛素促分泌素和聚氧乙烯脱水山梨醇脂肪酸酯的固体制剂
MXPA05010977A (es) * 2005-10-12 2007-04-11 Abdala Leopoldo Espinosa Composiciones farmaceuticas que comprenden sustancias antidiabeticas combinadas para su uso en diabetes mellitus.
KR100812538B1 (ko) * 2006-10-23 2008-03-11 한올제약주식회사 약물 제어방출형 메트포르민-글리메피리드 복합제제
CN101417130B (zh) * 2007-10-22 2010-10-06 鲁南制药集团股份有限公司 一种治疗ⅱ型糖尿病及其并发症的药物组合物
US11607441B2 (en) 2017-10-20 2023-03-21 Novmetapharma Co., Ltd. Pharmaceutical composition for preventing or treating diabetes, containing zinc salt, cyclo-hispro and antidiabetic drug as active ingredients

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5522636A (en) * 1978-08-04 1980-02-18 Takeda Chem Ind Ltd Thiazoliding derivative
JPS5697277A (en) * 1980-01-07 1981-08-05 Takeda Chem Ind Ltd Thiazolidine derivative
JPS6051189A (ja) * 1983-08-30 1985-03-22 Sankyo Co Ltd チアゾリジン誘導体およびその製造法
US4582839A (en) * 1984-03-21 1986-04-15 Takeda Chemical Industries, Ltd. 2,4-thiazolidinediones
CN1003445B (zh) * 1984-10-03 1989-03-01 武田药品工业株式会社 噻唑烷二酮衍生物,其制备方法和用途
JPH06779B2 (ja) * 1985-06-10 1994-01-05 武田薬品工業株式会社 チアゾリジオン誘導体およびそれを含んでなる医薬組成物
US4812570A (en) * 1986-07-24 1989-03-14 Takeda Chemical Industries, Ltd. Method for producing thiazolidinedione derivatives
US4791125A (en) * 1987-12-02 1988-12-13 Pfizer Inc. Thiazolidinediones as hypoglycemic and anti-atherosclerosis agents
WO1989008651A1 (en) * 1988-03-08 1989-09-21 Pfizer Inc. Hypoglycemic thiazolidinedione derivatives
US5061717A (en) * 1988-03-08 1991-10-29 Pfizer Inc. Thiazolidinedione hypoglycemic agents
WO1991007107A1 (en) * 1989-11-13 1991-05-30 Pfizer Inc. Oxazolidinedione hypoglycemic agents
JPH04210683A (ja) * 1990-12-06 1992-07-31 Terumo Corp チアゾリジン−2,4−ジオン誘導体およびこれを含有する糖尿病合併症治療薬
US5900435A (en) * 1991-08-26 1999-05-04 Pharmacia & Upjohn Company Composition, food product and uses of 3-guanidinopropionic acid
US5917052A (en) * 1994-09-28 1999-06-29 Shaman Pharmaceuticals, Inc. Hypoglycemic agent from cryptolepis
TWI238064B (en) * 1995-06-20 2005-08-21 Takeda Chemical Industries Ltd A pharmaceutical composition for prophylaxis and treatment of diabetes
CN1168451C (zh) * 1997-06-18 2004-09-29 史密丝克莱恩比彻姆有限公司 噻唑烷二酮和磺酰脲组合物在制备治疗糖尿病的药物中的用途

Also Published As

Publication number Publication date
TR200000134T2 (tr) 2000-09-21
CA2296653A1 (en) 1999-01-28
WO1999003477A1 (en) 1999-01-28
DZ2562A1 (fr) 2003-02-15
PL197844B1 (pl) 2008-05-30
SI1001783T1 (sl) 2006-02-28
AP2000001733A0 (en) 2000-03-31
KR100671918B1 (ko) 2007-01-22
IN189275B (enExample) 2003-01-25
HK1028550A1 (en) 2001-02-23
PE99599A1 (es) 1999-12-18
SK592000A3 (en) 2000-09-12
NO20000228L (no) 2000-01-17
EP1001783A1 (en) 2000-05-24
JP2005213273A (ja) 2005-08-11
AR016349A1 (es) 2001-07-04
SK285484B6 (sk) 2007-02-01
CN1264303A (zh) 2000-08-23
NZ511608A (en) 2002-12-20
MA24607A1 (fr) 1999-04-01
AU8448898A (en) 1999-02-10
BR9810445A (pt) 2000-09-05
ZA986363B (en) 2000-01-17
HUP0003629A3 (en) 2003-04-28
KR20010021947A (ko) 2001-03-15
ID24211A (id) 2000-07-13
UY25102A1 (es) 2000-12-29
ES2251093T3 (es) 2006-04-16
NO20000228D0 (no) 2000-01-17
ATE305790T1 (de) 2005-10-15
JP2001510159A (ja) 2001-07-31
OA11279A (en) 2003-07-31
DE69831808T2 (de) 2006-07-06
MY155219A (en) 2015-09-30
PL198017B1 (pl) 2008-05-30
TW505516B (en) 2002-10-11
AP1352A (en) 2004-12-24
HUP0003629A2 (hu) 2001-07-30
EA003021B1 (ru) 2002-12-26
IL134046A0 (en) 2001-04-30
CA2296653C (en) 2007-10-02
UA70303C2 (uk) 2004-10-15
DK1001783T3 (da) 2006-02-06
EA200000139A1 (ru) 2000-06-26
NZ501164A (en) 2001-06-29
NO325727B1 (no) 2008-07-07
BG104135A (en) 2000-10-31
GB9715295D0 (en) 1997-09-24
CY1105254T1 (el) 2010-03-03
BG64785B1 (bg) 2006-04-28
DE69831808D1 (de) 2006-02-16
EP1001783B1 (en) 2005-10-05
SA98190468B1 (ar) 2007-01-20
PL338126A1 (en) 2000-09-25

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