AR012997A1 - Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene. - Google Patents

Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene.

Info

Publication number
AR012997A1
AR012997A1 ARP980102883A ARP980102883A AR012997A1 AR 012997 A1 AR012997 A1 AR 012997A1 AR P980102883 A ARP980102883 A AR P980102883A AR P980102883 A ARP980102883 A AR P980102883A AR 012997 A1 AR012997 A1 AR 012997A1
Authority
AR
Argentina
Prior art keywords
insulin
thiazolidin
amino
methyl
preparation
Prior art date
Application number
ARP980102883A
Other languages
English (en)
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of AR012997A1 publication Critical patent/AR012997A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/28Insulins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Hematology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)

Abstract

Uso de 5-[4-[2-(N-metil-N-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de un medicamento util para el tratamientode diabetes mellitus y procesos asociados a la diabetes mellitus en un mamífero , que comprendeuna cantidad eficaz, no toxica y farmacéuticamente eficaz dedicho compuesto e insulina, y composicion farmaéutica que los contiene.
ARP980102883A 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene. AR012997A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9712866.4A GB9712866D0 (en) 1997-06-18 1997-06-18 Novel method of treatment

Publications (1)

Publication Number Publication Date
AR012997A1 true AR012997A1 (es) 2000-11-22

Family

ID=10814527

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP980102886A AR015894A1 (es) 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4-diona e insulina para la preparacion de un medicamento y composicion farmaceuticaque contiene dichos compuestos
ARP980102883A AR012997A1 (es) 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP980102886A AR015894A1 (es) 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4-diona e insulina para la preparacion de un medicamento y composicion farmaceuticaque contiene dichos compuestos

Country Status (30)

Country Link
EP (1) EP0999837A1 (es)
JP (1) JP2002504138A (es)
KR (1) KR20010013843A (es)
CN (1) CN1133431C (es)
AP (1) AP1287A (es)
AR (2) AR015894A1 (es)
AU (1) AU8216398A (es)
BG (1) BG104059A (es)
BR (1) BR9810444A (es)
CA (1) CA2294141A1 (es)
CO (1) CO4940454A1 (es)
DZ (1) DZ2521A1 (es)
EA (1) EA004800B1 (es)
GB (1) GB9712866D0 (es)
HU (1) HUP0003260A3 (es)
ID (1) ID23951A (es)
IL (1) IL133143A0 (es)
IN (1) IN189723B (es)
MA (1) MA26511A1 (es)
NO (1) NO996265L (es)
OA (1) OA11517A (es)
PE (1) PE104499A1 (es)
PL (1) PL343123A1 (es)
SK (1) SK179399A3 (es)
TR (1) TR199903095T2 (es)
TW (1) TW587937B (es)
UA (1) UA70299C2 (es)
UY (1) UY25050A1 (es)
WO (1) WO1998057636A1 (es)
ZA (1) ZA985237B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6291495B1 (en) * 1997-02-24 2001-09-18 Robert B. Rieveley Method and composition for the treatment of diabetes
TWI249401B (en) 1999-04-14 2006-02-21 Takeda Chemical Industries Ltd Agent for improving ketosis
DZ3155A1 (fr) 1999-04-23 2000-11-02 Smithkline Beecham Plc Nouvelle composition pharmaceutique.
DK1133312T3 (da) * 1999-06-21 2008-01-02 Lilly Co Eli Synergistisk anvendelse af thiazolidindioner med glucagonlignende peptid-1 og agonister deraf til behandling af ikke-insulinafhængig diabetes
AU5760900A (en) 1999-06-25 2001-01-31 Minimed, Inc. Multiple agent diabetes therapy
US6468507B1 (en) * 2000-05-01 2002-10-22 Aeropharm Technology, Inc. Non-aqueous aerosol formulation comprising rosiglitazone maleate, a non-aqueous carrier, and an amino acid stabilizer
GB0023970D0 (en) * 2000-09-29 2000-11-15 Smithkline Beecham Plc Novel pharmaceutical
AU2002248464A1 (en) 2001-02-21 2002-09-12 Medtronic Minimed, Inc. Stabilized insulin formulations
US6531461B1 (en) 2001-06-04 2003-03-11 Louis Obyo Obyo Nelson Medicament for the treatment of diabetes
US20020198203A1 (en) * 2001-06-07 2002-12-26 Wyeth Combination of a PTPase inhibitor and a thiazolidinedione agent
US6737401B2 (en) 2001-06-28 2004-05-18 Metronic Minimed, Inc. Methods of evaluating protein formulation stability and surfactant-stabilized insulin formulations derived therefrom
BR0316091A (pt) * 2002-11-08 2005-09-27 Hoffmann La Roche Compostos, processo para a manufatura dos mesmos, composições farmacêuticas, método para o tratamento e/ou prevenção de enfermidades que são moduladas por agonistas ppar(a) e/ou ppar(y) e/ou utilização dos mesmos
US7264813B2 (en) 2003-09-24 2007-09-04 Nikken Sohonsha Corporation Therapeutic uses of Dunaliella powder
CN102389427A (zh) * 2011-10-10 2012-03-28 成都恒瑞制药有限公司 含有罗格列酮和盐酸西替利嗪的固体口服制剂

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU228260B1 (en) * 1993-09-15 2013-02-28 Daiichi Sankyo Company Pharmaceutical compositions to treat impaired glucose tolerance
CN1192683A (zh) * 1995-08-10 1998-09-09 沃尼尔·朗伯公司 减少非胰岛素依赖型糖尿病患者外源性胰岛素给药量的方法
DK0859608T3 (da) * 1995-09-18 2004-06-14 Ligand Pharm Inc Behandling af NIDDM med RXR-agonister

Also Published As

Publication number Publication date
AP9901718A0 (en) 1999-12-31
PE104499A1 (es) 2000-01-13
CN1260715A (zh) 2000-07-19
IN189723B (es) 2003-04-19
AR015894A1 (es) 2001-05-30
CN1133431C (zh) 2004-01-07
KR20010013843A (ko) 2001-02-26
OA11517A (en) 2004-02-04
IL133143A0 (en) 2001-03-19
MA26511A1 (fr) 2004-12-20
UA70299C2 (en) 2004-10-15
EA200000042A1 (ru) 2000-08-28
SK179399A3 (en) 2000-11-07
HUP0003260A2 (hu) 2001-05-28
AU8216398A (en) 1999-01-04
ID23951A (id) 2000-06-08
EA004800B1 (ru) 2004-08-26
CO4940454A1 (es) 2000-07-24
EP0999837A1 (en) 2000-05-17
JP2002504138A (ja) 2002-02-05
BR9810444A (pt) 2000-09-05
DZ2521A1 (fr) 2003-02-08
GB9712866D0 (en) 1997-08-20
TW587937B (en) 2004-05-21
BG104059A (en) 2000-10-31
ZA985237B (en) 2000-02-17
CA2294141A1 (en) 1998-12-23
UY25050A1 (es) 2000-09-29
AP1287A (en) 2004-06-26
NO996265D0 (no) 1999-12-17
HUP0003260A3 (en) 2001-12-28
WO1998057636A1 (en) 1998-12-23
NO996265L (no) 1999-12-17
PL343123A1 (en) 2001-07-30
TR199903095T2 (xx) 2000-08-21

Similar Documents

Publication Publication Date Title
PE83199A1 (es) Composicion farmaceutica de tiazolidinadiona y biguanida para el tratamiento de la diabetes
AR012997A1 (es) Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene.
EA200601145A1 (ru) Таблетка замедленного высвобождения сенсибилизатора к инсулину и других антидиабетических агентов
AR057970A2 (es) Composiciones farmaceuticas para el tratamiento de la diabetes mellitus y condiciones asociadas con la diabetes mellitus y procedimientos para preprar dichas composiciones
PE99599A1 (es) Composicion farmaceutica para el tratamiento de la diabetes
MY135973A (en) Modified release compositions comprising 5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2, 4-dione, optionally in the form of pharmaceutically acceptable derivative
NZ513922A (en) Composition comprising 5-Ä4-Ä2-(N-methyl-N-2-pyridyl)-amino)ethoxy!benzyl!thiazolidine-2-4-dione
PE108199A1 (es) Composicion farmaceutica de tiazolidindiona y sulfonilurea
NZ515555A (en) Treatment of diabetes with thiazolidinedione and sulphonylurea
UY25051A1 (es) Composiciones para el tratamiento de diabetes mellitus
CY1105354T1 (el) Ένα παραγωγο θειαζολιδινοδιονης και η χρηση του σαν αντι-διαβητικο
EA200300345A1 (ru) Гидрохлоридная соль 5-[4-[2-(n-метил-n-(2-пиридил)амино)этокси]бензил]тиазолидин-2,4-диона
EA200300005A1 (ru) Соль тиазолидиндиона для лечения сахарного диабета
CY1107767T1 (el) Παραγωγο θειαζολιδινοδιονης και χρηση αυτου σαν αντιδιαβητικο
ECSP034467A (es) Farmaceutico novedoso
PE20001239A1 (es) Composicion de un sensibilizador de insulina
TH36758A (th) กรรมวิธีในการรักษาโรคเบาหวานด้วยไธอะโซลิดีนไดโอนและเมทฟอร์มิน
CO5150180A1 (es) Nueva composicion y uso liberacion modificada
ECSP003434A (es) Nuevos compuestos
ECSP003435A (es) Nuevos compuestos
TH21154B (th) กรรมวิธีในการรักษาโรคเบาหวานด้วยไธอะโซลิดีนไดโอนและเมทฟอร์มิน

Legal Events

Date Code Title Description
FA Abandonment or withdrawal