DK1315724T3 - Thiazolidindionderivat og dets anvendelse som antidiabetikum - Google Patents

Thiazolidindionderivat og dets anvendelse som antidiabetikum

Info

Publication number
DK1315724T3
DK1315724T3 DK01963256T DK01963256T DK1315724T3 DK 1315724 T3 DK1315724 T3 DK 1315724T3 DK 01963256 T DK01963256 T DK 01963256T DK 01963256 T DK01963256 T DK 01963256T DK 1315724 T3 DK1315724 T3 DK 1315724T3
Authority
DK
Denmark
Prior art keywords
compound
diabetic
thiazolidinedione derivative
thiazolidinedione
derivative
Prior art date
Application number
DK01963256T
Other languages
English (en)
Inventor
Andrew Simon Craig
Michael Millan
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Application granted granted Critical
Publication of DK1315724T3 publication Critical patent/DK1315724T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK01963256T 2000-09-05 2001-09-05 Thiazolidindionderivat og dets anvendelse som antidiabetikum DK1315724T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0021784.4A GB0021784D0 (en) 2000-09-05 2000-09-05 Novel pharmaceutical

Publications (1)

Publication Number Publication Date
DK1315724T3 true DK1315724T3 (da) 2006-02-20

Family

ID=9898884

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01963256T DK1315724T3 (da) 2000-09-05 2001-09-05 Thiazolidindionderivat og dets anvendelse som antidiabetikum

Country Status (14)

Country Link
US (1) US20040044043A1 (da)
EP (1) EP1315724B1 (da)
JP (1) JP2004508370A (da)
KR (1) KR100769008B1 (da)
CN (1) CN1239501C (da)
AT (1) ATE310000T1 (da)
AU (1) AU2001284285A1 (da)
CY (1) CY1105354T1 (da)
DE (1) DE60115062T2 (da)
DK (1) DK1315724T3 (da)
ES (1) ES2248385T3 (da)
GB (1) GB0021784D0 (da)
HK (1) HK1057751A1 (da)
WO (1) WO2002020520A1 (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE39384E1 (en) 1993-09-01 2006-11-07 Smithkline Beecham P.L.C. Substituted thiazolidinedione derivatives
DK1448559T3 (da) * 2001-11-21 2007-04-30 Smithkline Beecham Plc 5-(4-(2-(N-methyl-N-(2-pyridyl)amino)ethoxy)benzyl)thiazolodin-2,4-dionbenzensulfat; fremgangsmåde til dets fremstilling; polymorf i, II og III deraf; og dets anvendelse som farmaceutisk aktiv bestenddel
DE102005034406A1 (de) * 2005-07-22 2007-02-01 Ratiopharm Gmbh Neue Salze von Rosiglitazon
US7435741B2 (en) * 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
EP2043744A2 (en) * 2006-07-13 2009-04-08 SmithKline Beecham Corporation Chemical compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
US5741803A (en) * 1992-09-05 1998-04-21 Smithkline Beecham Plc Substituted thiazolidinedionle derivatives
GB9726566D0 (en) * 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical
GB9726568D0 (en) * 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical
GB9726563D0 (en) * 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical

Also Published As

Publication number Publication date
KR100769008B1 (ko) 2007-10-22
ES2248385T3 (es) 2006-03-16
JP2004508370A (ja) 2004-03-18
DE60115062T2 (de) 2006-06-29
AU2001284285A1 (en) 2002-03-22
DE60115062D1 (de) 2005-12-22
HK1057751A1 (en) 2004-04-16
GB0021784D0 (en) 2000-10-18
WO2002020520A1 (en) 2002-03-14
CN1471529A (zh) 2004-01-28
KR20030027112A (ko) 2003-04-03
CN1239501C (zh) 2006-02-01
CY1105354T1 (el) 2010-03-03
US20040044043A1 (en) 2004-03-04
EP1315724B1 (en) 2005-11-16
EP1315724A1 (en) 2003-06-04
ATE310000T1 (de) 2005-12-15

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