ATE310000T1 - Ein thiazolidindionderivat und seine verwendung als antidiabetikum - Google Patents

Ein thiazolidindionderivat und seine verwendung als antidiabetikum

Info

Publication number
ATE310000T1
ATE310000T1 AT01963256T AT01963256T ATE310000T1 AT E310000 T1 ATE310000 T1 AT E310000T1 AT 01963256 T AT01963256 T AT 01963256T AT 01963256 T AT01963256 T AT 01963256T AT E310000 T1 ATE310000 T1 AT E310000T1
Authority
AT
Austria
Prior art keywords
compound
antidiabetic drug
thiazolidinedione derivative
thiazolidinedione
derivative
Prior art date
Application number
AT01963256T
Other languages
English (en)
Inventor
Andrew Simon Craig
Michael Millan
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Application granted granted Critical
Publication of ATE310000T1 publication Critical patent/ATE310000T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT01963256T 2000-09-05 2001-09-05 Ein thiazolidindionderivat und seine verwendung als antidiabetikum ATE310000T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0021784.4A GB0021784D0 (en) 2000-09-05 2000-09-05 Novel pharmaceutical
PCT/GB2001/003996 WO2002020520A1 (en) 2000-09-05 2001-09-05 A thiazolidinedione derivative and its use as antidiabetic

Publications (1)

Publication Number Publication Date
ATE310000T1 true ATE310000T1 (de) 2005-12-15

Family

ID=9898884

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01963256T ATE310000T1 (de) 2000-09-05 2001-09-05 Ein thiazolidindionderivat und seine verwendung als antidiabetikum

Country Status (14)

Country Link
US (1) US20040044043A1 (de)
EP (1) EP1315724B1 (de)
JP (1) JP2004508370A (de)
KR (1) KR100769008B1 (de)
CN (1) CN1239501C (de)
AT (1) ATE310000T1 (de)
AU (1) AU2001284285A1 (de)
CY (1) CY1105354T1 (de)
DE (1) DE60115062T2 (de)
DK (1) DK1315724T3 (de)
ES (1) ES2248385T3 (de)
GB (1) GB0021784D0 (de)
HK (1) HK1057751A1 (de)
WO (1) WO2002020520A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE39384E1 (en) 1993-09-01 2006-11-07 Smithkline Beecham P.L.C. Substituted thiazolidinedione derivatives
ES2278977T3 (es) * 2001-11-21 2007-08-16 Smithkline Beecham Plc Bencenosulfonato de 5-(4-(2-(n-metil-n-(2-piridil)amino)etoxi)bencil)tiazolidin-2,4-diona; procedimiento para su preparacion; polimorfos i, ii y iii de los mismos; y su uso como ingrediente activo farmaceutico.
DE102005034406A1 (de) * 2005-07-22 2007-02-01 Ratiopharm Gmbh Neue Salze von Rosiglitazon
US7435741B2 (en) 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
JP2009543805A (ja) * 2006-07-13 2009-12-10 スミスクライン ビーチャム コーポレーション インドリン誘導体及びgpr119作動物質

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
US5741803A (en) * 1992-09-05 1998-04-21 Smithkline Beecham Plc Substituted thiazolidinedionle derivatives
GB9726566D0 (en) * 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical
GB9726563D0 (en) * 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical
GB9726568D0 (en) * 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical

Also Published As

Publication number Publication date
CY1105354T1 (el) 2010-03-03
GB0021784D0 (en) 2000-10-18
EP1315724A1 (de) 2003-06-04
KR100769008B1 (ko) 2007-10-22
KR20030027112A (ko) 2003-04-03
CN1471529A (zh) 2004-01-28
DE60115062T2 (de) 2006-06-29
EP1315724B1 (de) 2005-11-16
ES2248385T3 (es) 2006-03-16
HK1057751A1 (en) 2004-04-16
WO2002020520A1 (en) 2002-03-14
AU2001284285A1 (en) 2002-03-22
CN1239501C (zh) 2006-02-01
DK1315724T3 (da) 2006-02-20
US20040044043A1 (en) 2004-03-04
DE60115062D1 (de) 2005-12-22
JP2004508370A (ja) 2004-03-18

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