CN1990486A - N－氨基乙酰基－吡咯烷－2－腈和它们作为ddp－iv抑制剂的用途 - Google Patents

N－氨基乙酰基－吡咯烷－2－腈和它们作为ddp－iv抑制剂的用途 Download PDF

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CN1990486A
CN1990486A CNA2006101640208A CN200610164020A CN1990486A CN 1990486 A CN1990486 A CN 1990486A CN A2006101640208 A CNA2006101640208 A CN A2006101640208A CN 200610164020 A CN200610164020 A CN 200610164020A CN 1990486 A CN1990486 A CN 1990486A
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group
base
formula
different
general formula
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P·阿兰伊
L·巴拉兹
I·巴塔
S·巴托里
E·博龙凯
P·博维
K·卡奈
Z·卡普
E·苏珊
T·萨博
L·T·纳吉
K·鄂班－萨博
M·瓦伽
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Sanofi Aventis France
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CNA2006101640208A 2002-03-06 2003-03-04 N－氨基乙酰基－吡咯烷－2－腈和它们作为ddp－iv抑制剂的用途 Pending CN1990486A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU0200849A HUP0200849A2 (hu) 2002-03-06 2002-03-06 N-aminoacetil-2-ciano-pirrolidin-származékok, e vegyületeket tartalmazó gyógyszerkészítmények és eljárás előállításukra
HUP0200849 2002-03-06

Related Parent Applications (1)

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CNA038052636A Division CN1639159A (zh) 2002-03-06 2003-03-04 N－氨基乙酰基－吡咯烷－2－腈和它们作为ddp－iv抑制剂的用途

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CN1990486A true CN1990486A (zh) 2007-07-04

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ID=90001540

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CNA038052636A Pending CN1639159A (zh) 2002-03-06 2003-03-04 N－氨基乙酰基－吡咯烷－2－腈和它们作为ddp－iv抑制剂的用途
CNA2006101640208A Pending CN1990486A (zh) 2002-03-06 2003-03-04 N－氨基乙酰基－吡咯烷－2－腈和它们作为ddp－iv抑制剂的用途

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CNA038052636A Pending CN1639159A (zh) 2002-03-06 2003-03-04 N－氨基乙酰基－吡咯烷－2－腈和它们作为ddp－iv抑制剂的用途

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US (3) US7348327B2 (OSRAM)
EP (1) EP1487807B1 (OSRAM)
JP (1) JP4559737B2 (OSRAM)
KR (1) KR100977898B1 (OSRAM)
CN (2) CN1639159A (OSRAM)
AR (1) AR038868A1 (OSRAM)
AT (1) ATE443054T1 (OSRAM)
AU (1) AU2003209514B2 (OSRAM)
BR (1) BR0307960A (OSRAM)
CA (1) CA2475312C (OSRAM)
DE (1) DE60329282D1 (OSRAM)
EA (1) EA007410B1 (OSRAM)
EC (1) ECSP045274A (OSRAM)
HR (1) HRP20040910A2 (OSRAM)
HU (1) HUP0200849A2 (OSRAM)
IL (2) IL163286A (OSRAM)
IS (1) IS7434A (OSRAM)
MA (1) MA27105A1 (OSRAM)
MX (1) MXPA04008613A (OSRAM)
NO (1) NO20044221L (OSRAM)
NZ (1) NZ535662A (OSRAM)
PL (1) PL371099A1 (OSRAM)
RS (1) RS79004A (OSRAM)
TN (1) TNSN04141A1 (OSRAM)
TW (1) TWI250978B (OSRAM)
UA (1) UA78291C2 (OSRAM)
WO (1) WO2003074500A2 (OSRAM)
ZA (1) ZA200406467B (OSRAM)

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HUP0202001A2 (hu) * 2002-06-14 2005-08-29 Sanofi-Aventis DDP-IV gátló hatású azabiciklooktán- és nonánszármazékok
TW200401635A (en) * 2002-07-23 2004-02-01 Yamanouchi Pharma Co Ltd 2-Cyano-4-fluoropyrrolidine derivative or salt thereof
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7550590B2 (en) 2003-03-25 2009-06-23 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
ZA200508439B (en) 2003-05-05 2007-03-28 Probiodrug Ag Medical use of inhibitors of glutaminyl and glutamate cyclases
JP2007511467A (ja) 2003-05-14 2007-05-10 タケダ サン ディエゴ インコーポレイテッド ジペプチジルペプチダーゼインヒビター
WO2005016911A1 (en) 2003-08-13 2005-02-24 Takeda Pharmaceutical Company Limited 4-pyrimidone derivatives and their use as peptidyl peptidase inhibitors
HU227684B1 (en) 2003-08-29 2011-11-28 Sanofi Aventis Adamantane and azabicyclo-octane and nonane derivatives and their use as dpp-iv inhibitors
EP2338490A3 (en) 2003-11-03 2012-06-06 Probiodrug AG Combinations useful for the treatment of neuronal disorders
CN1905876B (zh) * 2003-11-17 2010-06-09 诺瓦提斯公司 二肽基肽酶iv抑制剂的用途
RU2385723C2 (ru) * 2003-11-17 2010-04-10 Новартис Аг Применение ингибиторов дипептидилпептидазы iv
NZ548351A (en) 2004-01-20 2009-08-28 Novartis Ag Direct compression formulation and process
EP1713780B1 (en) 2004-02-05 2012-01-18 Probiodrug AG Novel inhibitors of glutaminyl cyclase
CN101684089A (zh) * 2004-02-05 2010-03-31 杏林制药株式会社 双环酯类衍生物
FR2870538B1 (fr) 2004-05-19 2006-07-14 Servier Lab Nouveaux derives de pyrrolidines et de thiazolidines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
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EP1487807B1 (en) 2009-09-16
WO2003074500A3 (en) 2003-12-18
US20100210838A1 (en) 2010-08-19
NZ535662A (en) 2007-05-31
UA78291C2 (en) 2007-03-15
MA27105A1 (fr) 2004-12-20
HRP20040910A2 (en) 2006-02-28
KR20040091102A (ko) 2004-10-27
JP2005529078A (ja) 2005-09-29
RS79004A (sr) 2006-12-15
AR038868A1 (es) 2005-02-02
JP4559737B2 (ja) 2010-10-13
DE60329282D1 (de) 2009-10-29
TWI250978B (en) 2006-03-11
HUP0200849A2 (hu) 2004-08-30
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AU2003209514A1 (en) 2003-09-16
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CN1639159A (zh) 2005-07-13
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AU2003209514B2 (en) 2009-07-16
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US8063045B2 (en) 2011-11-22
BR0307960A (pt) 2005-02-15
IL177933A0 (en) 2006-12-31
EA200401157A1 (ru) 2005-06-30
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US7655663B2 (en) 2010-02-02
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