CN1612852A - 脂氧素a4类似物 - Google Patents

脂氧素a4类似物 Download PDF

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Publication number
CN1612852A
CN1612852A CNA028268539A CN02826853A CN1612852A CN 1612852 A CN1612852 A CN 1612852A CN A028268539 A CNA028268539 A CN A028268539A CN 02826853 A CN02826853 A CN 02826853A CN 1612852 A CN1612852 A CN 1612852A
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Prior art keywords
alkyl
aryl
aralkyl
halogen
straight
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Chinese (zh)
Inventor
约翰·G.·鲍曼
威廉·J.·吉尔福德
约翰·F.·帕金森
维尔纳·斯库巴尔拉
巴布·苏布拉曼亚姆
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Bayer Pharma AG
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Schering AG
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23325714&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN1612852(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering AG filed Critical Schering AG
Publication of CN1612852A publication Critical patent/CN1612852A/zh
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    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/72Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 spiro-condensed with carbocyclic rings
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • A61K31/202Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having three or more double bonds, e.g. linolenic
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    • C07C229/12Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of acyclic carbon skeletons
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CNA028268539A 2001-11-06 2002-11-05 脂氧素a4类似物 Pending CN1612852A (zh)

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US33868401P 2001-11-06 2001-11-06
US60/338,684 2001-11-06

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CN101553456B (zh) * 2006-12-04 2013-08-28 拜耳知识产权有限责任公司 脂氧素a4类似物的晶体钾盐
CN102036714A (zh) * 2008-05-22 2011-04-27 拜耳先灵医药股份有限公司 晶体2-((2s,3r,4e,6e,10e,12s)-13-(4-氟苯氧基)-2,3,12-三羟基十三碳-4,6,10-三烯-8-炔)氧基)乙酸的无水形式和水合物形式

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