CN103079406B - 杀真菌吡唑类 - Google Patents

杀真菌吡唑类 Download PDF

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Publication number
CN103079406B
CN103079406B CN201180042397.5A CN201180042397A CN103079406B CN 103079406 B CN103079406 B CN 103079406B CN 201180042397 A CN201180042397 A CN 201180042397A CN 103079406 B CN103079406 B CN 103079406B
Authority
CN
China
Prior art keywords
compound
formula
chloro
fluorophenyl
dimethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CN201180042397.5A
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English (en)
Chinese (zh)
Other versions
CN103079406A (zh
Inventor
J.K.龙
M.A.哈纳根
E.A.马歇尔
P.L.夏普
A.X.丁
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
FMC Corp
Original Assignee
EI Du Pont de Nemours and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by EI Du Pont de Nemours and Co filed Critical EI Du Pont de Nemours and Co
Priority to CN201510578968.7A priority Critical patent/CN105130900B/zh
Publication of CN103079406A publication Critical patent/CN103079406A/zh
Application granted granted Critical
Publication of CN103079406B publication Critical patent/CN103079406B/zh
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CN201180042397.5A 2010-09-01 2011-08-31 杀真菌吡唑类 Expired - Fee Related CN103079406B (zh)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN201510578968.7A CN105130900B (zh) 2010-09-01 2011-08-31 杀真菌吡唑类

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US37915910P 2010-09-01 2010-09-01
US61/379159 2010-09-01
PCT/US2011/049908 WO2012030922A1 (en) 2010-09-01 2011-08-31 Fungicidal pyrazoles

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CN201510578968.7A Division CN105130900B (zh) 2010-09-01 2011-08-31 杀真菌吡唑类

Publications (2)

Publication Number Publication Date
CN103079406A CN103079406A (zh) 2013-05-01
CN103079406B true CN103079406B (zh) 2016-03-30

Family

ID=44651972

Family Applications (2)

Application Number Title Priority Date Filing Date
CN201180042397.5A Expired - Fee Related CN103079406B (zh) 2010-09-01 2011-08-31 杀真菌吡唑类
CN201510578968.7A Expired - Fee Related CN105130900B (zh) 2010-09-01 2011-08-31 杀真菌吡唑类

Family Applications After (1)

Application Number Title Priority Date Filing Date
CN201510578968.7A Expired - Fee Related CN105130900B (zh) 2010-09-01 2011-08-31 杀真菌吡唑类

Country Status (14)

Country Link
US (2) US8754115B2 (enExample)
EP (1) EP2611297B1 (enExample)
JP (1) JP6066910B2 (enExample)
KR (1) KR20130139892A (enExample)
CN (2) CN103079406B (enExample)
AR (1) AR082869A1 (enExample)
AU (1) AU2011295998A1 (enExample)
BR (2) BR122017015898B1 (enExample)
ES (1) ES2546671T3 (enExample)
MX (1) MX2013002400A (enExample)
PL (1) PL2611297T3 (enExample)
TW (1) TW201245155A (enExample)
UY (1) UY33582A (enExample)
WO (1) WO2012030922A1 (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR075713A1 (es) 2009-03-03 2011-04-20 Du Pont Pirazoles fungicidas
TWI504350B (zh) 2010-09-01 2015-10-21 Du Pont 殺真菌吡唑及其混合物
TWI568721B (zh) 2012-02-01 2017-02-01 杜邦股份有限公司 殺真菌之吡唑混合物
US20140235689A1 (en) * 2013-02-20 2014-08-21 E I Du Pont De Nemours And Company Fungicidal pyrazoles
WO2014157569A1 (ja) 2013-03-28 2014-10-02 武田薬品工業株式会社 複素環化合物
TWI652012B (zh) * 2013-05-20 2019-03-01 杜邦股份有限公司 殺真菌吡唑的固態形式
WO2015026646A1 (en) 2013-08-20 2015-02-26 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
EA201690737A1 (ru) 2013-12-05 2016-10-31 Куреха Корпорейшн Сельскохозяйственное или садоводческое химическое средство, способ борьбы с болезнями растений и продукт для борьбы с болезнями растений
WO2015083437A1 (ja) * 2013-12-05 2015-06-11 株式会社クレハ 農園芸用薬剤、植物病害防除方法および植物病害防除用製品
WO2015089800A1 (en) 2013-12-19 2015-06-25 Eli Lilly And Company Fluorophenyl pyrazol compounds
CN106458925A (zh) * 2014-05-06 2017-02-22 杜邦公司 杀真菌吡唑类
JP2017522334A (ja) 2014-07-24 2017-08-10 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺真菌性ピラゾール誘導体
EP3271336A1 (en) 2015-03-19 2018-01-24 E. I. du Pont de Nemours and Company Fungicidal pyrazoles
WO2016201662A1 (en) * 2015-06-18 2016-12-22 Eli Lilly And Company Fluoropyridyl pyrazol compounds
EP3412658A1 (en) * 2017-06-09 2018-12-12 Solvay Sa Processes for the manufacture of sulfur-substitued pyrazole derivatives
BR112022007294A2 (pt) * 2019-10-18 2022-07-05 Fmc Corp Métodos para a preparação de ácido 5-bromo-2-(3-cloro-piridin-2-il)-2h-pirazol-3-carboxílico
IL291939B2 (en) * 2019-10-18 2023-04-01 Fmc Corp Method for preparing 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyralose-3-carboxylic acid
TW202241859A (zh) * 2021-01-29 2022-11-01 美商富曼西公司 用於製備５－溴－２－（３－氯－吡啶－２－基）－２ｈ－吡唑－３－甲酸之方法
WO2024150100A1 (en) * 2023-01-09 2024-07-18 Fluorinnovation L.L.C-Fz New process for manufacturing of 3-halomethyl-substituted 1-methyl-1h-pyrazole-4-carbonitriles and of derivatives thereof, and intermediates therefore
CN116606263B (zh) * 2023-05-26 2025-06-13 青岛科技大学 一种含氟苯联噻唑双酯类化合物及其用途
WO2025168620A1 (en) * 2024-02-07 2025-08-14 Bayer Aktiengesellschaft Heteroaryl-substituted 4,5-dihydro-1h-2,4,5-oxadiazines as novel fungicides

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101687845A (zh) * 2007-07-11 2010-03-31 先正达参股股份有限公司 用作杀真菌剂的异噻唑和吡唑衍生物

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2891855A (en) 1954-08-16 1959-06-23 Geigy Ag J R Compositions and methods for influencing the growth of plants
US3235361A (en) 1962-10-29 1966-02-15 Du Pont Method for the control of undesirable vegetation
US3060084A (en) 1961-06-09 1962-10-23 Du Pont Improved homogeneous, readily dispersed, pesticidal concentrate
US3299566A (en) 1964-06-01 1967-01-24 Olin Mathieson Water soluble film containing agricultural chemicals
US3309192A (en) 1964-12-02 1967-03-14 Du Pont Method of controlling seedling weed grasses
US4144050A (en) 1969-02-05 1979-03-13 Hoechst Aktiengesellschaft Micro granules for pesticides and process for their manufacture
US3920442A (en) 1972-09-18 1975-11-18 Du Pont Water-dispersible pesticide aggregates
JPS5527916B2 (enExample) * 1973-02-05 1980-07-24
CA1060892A (en) * 1974-11-06 1979-08-21 Parke, Davis And Company Diazepine compounds and method for their production
US4172714A (en) 1976-12-20 1979-10-30 E. I. Du Pont De Nemours And Company Dry compactible, swellable herbicidal compositions and pellets produced therefrom
DE3246493A1 (de) 1982-12-16 1984-06-20 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von wasserdispergierbaren granulaten
AU559935B2 (en) * 1983-02-04 1987-03-26 Warner-Lambert Company Imidazolyl-pyrazolyl methanone derivatives
JPS6253970A (ja) * 1985-09-03 1987-03-09 Nippon Nohyaku Co Ltd ピラゾ−ル誘導体及びその製法
US5180587A (en) 1988-06-28 1993-01-19 E. I. Du Pont De Nemours And Company Tablet formulations of pesticides
DK0415688T3 (da) 1989-08-30 1999-08-23 Aeci Ltd Fremgangsmåde til fremstilling af et doseringssystem samt fremgangsmåde til behandling af en genstand eller et locus
JPH03141276A (ja) * 1989-10-24 1991-06-17 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
PL167613B1 (pl) 1990-03-12 1995-09-30 Du Pont Granulowana kompozycja rozpuszczalna lub dyspergowalna w wodzie PL
US5189040A (en) * 1990-05-28 1993-02-23 Sumitomo Chemical Company, Limited Pyrazole derivatives, method for producing the same and agricultural and/or horticultural fungicides containing the same as active ingredient
JPH04356480A (ja) * 1990-05-28 1992-12-10 Sumitomo Chem Co Ltd ピラゾール誘導体、その製造法およびそれを有効成分とする農園芸用殺菌剤
EP0480679B1 (en) 1990-10-11 1996-09-18 Sumitomo Chemical Company Limited Pesticidal composition
JPH0532662A (ja) * 1990-11-09 1993-02-09 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
JPH0551304A (ja) 1991-06-10 1993-03-02 Nippon Bayeragrochem Kk 除草剤組成物
JPH05279339A (ja) * 1992-01-22 1993-10-26 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
JPH0665237A (ja) * 1992-05-07 1994-03-08 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
US5939559A (en) * 1995-02-07 1999-08-17 Nissan Chemical Industries, Ltd. Pyrazole derivative and herbicidal composition
JP2865599B2 (ja) 1995-10-09 1999-03-08 株式会社横井製作所 埋設物の探査方法
DE10136065A1 (de) 2001-07-25 2003-02-13 Bayer Cropscience Ag Pyrazolylcarboxanilide
TW200724033A (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
CA2652859A1 (en) 2006-06-21 2007-12-27 E.I. Du Pont De Nemours And Company Pyrazinones as cellular proliferation inhibitors
PE20091953A1 (es) * 2008-05-08 2010-01-09 Du Pont Azoles sustituidos como fungicidas
AR075713A1 (es) 2009-03-03 2011-04-20 Du Pont Pirazoles fungicidas
WO2012023143A1 (en) 2010-08-19 2012-02-23 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
TWI504350B (zh) 2010-09-01 2015-10-21 Du Pont 殺真菌吡唑及其混合物

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101687845A (zh) * 2007-07-11 2010-03-31 先正达参股股份有限公司 用作杀真菌剂的异噻唑和吡唑衍生物

Also Published As

Publication number Publication date
BR112013004835A2 (pt) 2016-05-31
PL2611297T3 (pl) 2015-11-30
US20130143940A1 (en) 2013-06-06
BR112013004835B1 (pt) 2018-01-09
EP2611297A1 (en) 2013-07-10
KR20130139892A (ko) 2013-12-23
TW201245155A (en) 2012-11-16
UY33582A (es) 2012-03-30
CN105130900A (zh) 2015-12-09
US9131693B2 (en) 2015-09-15
AU2011295998A1 (en) 2013-02-21
US8754115B2 (en) 2014-06-17
JP2013536856A (ja) 2013-09-26
US20140221448A1 (en) 2014-08-07
JP6066910B2 (ja) 2017-01-25
WO2012030922A1 (en) 2012-03-08
MX2013002400A (es) 2013-06-05
BR122017015898B1 (pt) 2018-05-15
ES2546671T3 (es) 2015-09-25
AR082869A1 (es) 2013-01-16
EP2611297B1 (en) 2015-06-17
CN103079406A (zh) 2013-05-01
CN105130900B (zh) 2018-05-22

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C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
C14 Grant of patent or utility model
GR01 Patent grant
TR01 Transfer of patent right

Effective date of registration: 20180712

Address after: American Pennsylvania

Patentee after: FMC Corp.

Address before: Wilmington, Delaware, USA

Patentee before: E. I. du Pont de Nemours and Co.

TR01 Transfer of patent right
CF01 Termination of patent right due to non-payment of annual fee

Granted publication date: 20160330

Termination date: 20190831

CF01 Termination of patent right due to non-payment of annual fee