JP6066910B2 - 殺菌・殺カビ性ピラゾール - Google Patents

殺菌・殺カビ性ピラゾール Download PDF

Info

Publication number
JP6066910B2
JP6066910B2 JP2013527253A JP2013527253A JP6066910B2 JP 6066910 B2 JP6066910 B2 JP 6066910B2 JP 2013527253 A JP2013527253 A JP 2013527253A JP 2013527253 A JP2013527253 A JP 2013527253A JP 6066910 B2 JP6066910 B2 JP 6066910B2
Authority
JP
Japan
Prior art keywords
compound
alkyl
independently
methyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
JP2013527253A
Other languages
English (en)
Japanese (ja)
Other versions
JP2013536856A (ja
JP2013536856A5 (enExample
Inventor
ジェフリー・キース・ロング
メアリー・アン・ハナガン
エリック・アレン・マーシャル
パウラ・ルイーズ・シャープ
エイミー・エックス・ディング
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
EIDP Inc
Original Assignee
EI Du Pont de Nemours and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by EI Du Pont de Nemours and Co filed Critical EI Du Pont de Nemours and Co
Publication of JP2013536856A publication Critical patent/JP2013536856A/ja
Publication of JP2013536856A5 publication Critical patent/JP2013536856A5/ja
Application granted granted Critical
Publication of JP6066910B2 publication Critical patent/JP6066910B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2013527253A 2010-09-01 2011-08-31 殺菌・殺カビ性ピラゾール Expired - Fee Related JP6066910B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US37915910P 2010-09-01 2010-09-01
US61/379,159 2010-09-01
PCT/US2011/049908 WO2012030922A1 (en) 2010-09-01 2011-08-31 Fungicidal pyrazoles

Publications (3)

Publication Number Publication Date
JP2013536856A JP2013536856A (ja) 2013-09-26
JP2013536856A5 JP2013536856A5 (enExample) 2014-10-09
JP6066910B2 true JP6066910B2 (ja) 2017-01-25

Family

ID=44651972

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013527253A Expired - Fee Related JP6066910B2 (ja) 2010-09-01 2011-08-31 殺菌・殺カビ性ピラゾール

Country Status (14)

Country Link
US (2) US8754115B2 (enExample)
EP (1) EP2611297B1 (enExample)
JP (1) JP6066910B2 (enExample)
KR (1) KR20130139892A (enExample)
CN (2) CN103079406B (enExample)
AR (1) AR082869A1 (enExample)
AU (1) AU2011295998A1 (enExample)
BR (2) BR122017015898B1 (enExample)
ES (1) ES2546671T3 (enExample)
MX (1) MX2013002400A (enExample)
PL (1) PL2611297T3 (enExample)
TW (1) TW201245155A (enExample)
UY (1) UY33582A (enExample)
WO (1) WO2012030922A1 (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR075713A1 (es) 2009-03-03 2011-04-20 Du Pont Pirazoles fungicidas
TWI504350B (zh) 2010-09-01 2015-10-21 Du Pont 殺真菌吡唑及其混合物
TWI568721B (zh) 2012-02-01 2017-02-01 杜邦股份有限公司 殺真菌之吡唑混合物
US20140235689A1 (en) * 2013-02-20 2014-08-21 E I Du Pont De Nemours And Company Fungicidal pyrazoles
WO2014157569A1 (ja) 2013-03-28 2014-10-02 武田薬品工業株式会社 複素環化合物
TWI652012B (zh) * 2013-05-20 2019-03-01 杜邦股份有限公司 殺真菌吡唑的固態形式
WO2015026646A1 (en) 2013-08-20 2015-02-26 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
EA201690737A1 (ru) 2013-12-05 2016-10-31 Куреха Корпорейшн Сельскохозяйственное или садоводческое химическое средство, способ борьбы с болезнями растений и продукт для борьбы с болезнями растений
WO2015083437A1 (ja) * 2013-12-05 2015-06-11 株式会社クレハ 農園芸用薬剤、植物病害防除方法および植物病害防除用製品
WO2015089800A1 (en) 2013-12-19 2015-06-25 Eli Lilly And Company Fluorophenyl pyrazol compounds
CN106458925A (zh) * 2014-05-06 2017-02-22 杜邦公司 杀真菌吡唑类
JP2017522334A (ja) 2014-07-24 2017-08-10 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺真菌性ピラゾール誘導体
EP3271336A1 (en) 2015-03-19 2018-01-24 E. I. du Pont de Nemours and Company Fungicidal pyrazoles
WO2016201662A1 (en) * 2015-06-18 2016-12-22 Eli Lilly And Company Fluoropyridyl pyrazol compounds
EP3412658A1 (en) * 2017-06-09 2018-12-12 Solvay Sa Processes for the manufacture of sulfur-substitued pyrazole derivatives
BR112022007294A2 (pt) * 2019-10-18 2022-07-05 Fmc Corp Métodos para a preparação de ácido 5-bromo-2-(3-cloro-piridin-2-il)-2h-pirazol-3-carboxílico
IL291939B2 (en) * 2019-10-18 2023-04-01 Fmc Corp Method for preparing 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyralose-3-carboxylic acid
TW202241859A (zh) * 2021-01-29 2022-11-01 美商富曼西公司 用於製備５－溴－２－（３－氯－吡啶－２－基）－２ｈ－吡唑－３－甲酸之方法
WO2024150100A1 (en) * 2023-01-09 2024-07-18 Fluorinnovation L.L.C-Fz New process for manufacturing of 3-halomethyl-substituted 1-methyl-1h-pyrazole-4-carbonitriles and of derivatives thereof, and intermediates therefore
CN116606263B (zh) * 2023-05-26 2025-06-13 青岛科技大学 一种含氟苯联噻唑双酯类化合物及其用途
WO2025168620A1 (en) * 2024-02-07 2025-08-14 Bayer Aktiengesellschaft Heteroaryl-substituted 4,5-dihydro-1h-2,4,5-oxadiazines as novel fungicides

Family Cites Families (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2891855A (en) 1954-08-16 1959-06-23 Geigy Ag J R Compositions and methods for influencing the growth of plants
US3235361A (en) 1962-10-29 1966-02-15 Du Pont Method for the control of undesirable vegetation
US3060084A (en) 1961-06-09 1962-10-23 Du Pont Improved homogeneous, readily dispersed, pesticidal concentrate
US3299566A (en) 1964-06-01 1967-01-24 Olin Mathieson Water soluble film containing agricultural chemicals
US3309192A (en) 1964-12-02 1967-03-14 Du Pont Method of controlling seedling weed grasses
US4144050A (en) 1969-02-05 1979-03-13 Hoechst Aktiengesellschaft Micro granules for pesticides and process for their manufacture
US3920442A (en) 1972-09-18 1975-11-18 Du Pont Water-dispersible pesticide aggregates
JPS5527916B2 (enExample) * 1973-02-05 1980-07-24
CA1060892A (en) * 1974-11-06 1979-08-21 Parke, Davis And Company Diazepine compounds and method for their production
US4172714A (en) 1976-12-20 1979-10-30 E. I. Du Pont De Nemours And Company Dry compactible, swellable herbicidal compositions and pellets produced therefrom
DE3246493A1 (de) 1982-12-16 1984-06-20 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von wasserdispergierbaren granulaten
AU559935B2 (en) * 1983-02-04 1987-03-26 Warner-Lambert Company Imidazolyl-pyrazolyl methanone derivatives
JPS6253970A (ja) * 1985-09-03 1987-03-09 Nippon Nohyaku Co Ltd ピラゾ−ル誘導体及びその製法
US5180587A (en) 1988-06-28 1993-01-19 E. I. Du Pont De Nemours And Company Tablet formulations of pesticides
DK0415688T3 (da) 1989-08-30 1999-08-23 Aeci Ltd Fremgangsmåde til fremstilling af et doseringssystem samt fremgangsmåde til behandling af en genstand eller et locus
JPH03141276A (ja) * 1989-10-24 1991-06-17 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
PL167613B1 (pl) 1990-03-12 1995-09-30 Du Pont Granulowana kompozycja rozpuszczalna lub dyspergowalna w wodzie PL
US5189040A (en) * 1990-05-28 1993-02-23 Sumitomo Chemical Company, Limited Pyrazole derivatives, method for producing the same and agricultural and/or horticultural fungicides containing the same as active ingredient
JPH04356480A (ja) * 1990-05-28 1992-12-10 Sumitomo Chem Co Ltd ピラゾール誘導体、その製造法およびそれを有効成分とする農園芸用殺菌剤
EP0480679B1 (en) 1990-10-11 1996-09-18 Sumitomo Chemical Company Limited Pesticidal composition
JPH0532662A (ja) * 1990-11-09 1993-02-09 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
JPH0551304A (ja) 1991-06-10 1993-03-02 Nippon Bayeragrochem Kk 除草剤組成物
JPH05279339A (ja) * 1992-01-22 1993-10-26 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
JPH0665237A (ja) * 1992-05-07 1994-03-08 Nissan Chem Ind Ltd 置換ピラゾール誘導体および農園芸用殺菌剤
US5939559A (en) * 1995-02-07 1999-08-17 Nissan Chemical Industries, Ltd. Pyrazole derivative and herbicidal composition
JP2865599B2 (ja) 1995-10-09 1999-03-08 株式会社横井製作所 埋設物の探査方法
DE10136065A1 (de) 2001-07-25 2003-02-13 Bayer Cropscience Ag Pyrazolylcarboxanilide
TW200724033A (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
CA2652859A1 (en) 2006-06-21 2007-12-27 E.I. Du Pont De Nemours And Company Pyrazinones as cellular proliferation inhibitors
GB0713479D0 (en) 2007-07-11 2007-08-22 Syngenta Participations Ag Substituted aromatic heterocyclic compounds as fungicides
PE20091953A1 (es) * 2008-05-08 2010-01-09 Du Pont Azoles sustituidos como fungicidas
AR075713A1 (es) 2009-03-03 2011-04-20 Du Pont Pirazoles fungicidas
WO2012023143A1 (en) 2010-08-19 2012-02-23 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
TWI504350B (zh) 2010-09-01 2015-10-21 Du Pont 殺真菌吡唑及其混合物

Also Published As

Publication number Publication date
BR112013004835A2 (pt) 2016-05-31
PL2611297T3 (pl) 2015-11-30
US20130143940A1 (en) 2013-06-06
BR112013004835B1 (pt) 2018-01-09
EP2611297A1 (en) 2013-07-10
KR20130139892A (ko) 2013-12-23
TW201245155A (en) 2012-11-16
UY33582A (es) 2012-03-30
CN105130900A (zh) 2015-12-09
CN103079406B (zh) 2016-03-30
US9131693B2 (en) 2015-09-15
AU2011295998A1 (en) 2013-02-21
US8754115B2 (en) 2014-06-17
JP2013536856A (ja) 2013-09-26
US20140221448A1 (en) 2014-08-07
WO2012030922A1 (en) 2012-03-08
MX2013002400A (es) 2013-06-05
BR122017015898B1 (pt) 2018-05-15
ES2546671T3 (es) 2015-09-25
AR082869A1 (es) 2013-01-16
EP2611297B1 (en) 2015-06-17
CN103079406A (zh) 2013-05-01
CN105130900B (zh) 2018-05-22

Similar Documents

Publication Publication Date Title
JP6066910B2 (ja) 殺菌・殺カビ性ピラゾール
JP6285090B2 (ja) 殺菌・殺カビ性ピラゾール
JP5580732B2 (ja) 置換ベンゼン殺菌・殺カビ剤
EP2867228B1 (en) Fungicidal heterocyclic carboxamides
US8815772B2 (en) Fungicidal heterocyclic carboxamides
JP2012503659A (ja) 殺菌・殺カビ性ピリダジン
WO2012023143A1 (en) Fungicidal pyrazoles
WO2013126283A1 (en) Fungicidal pyrazoles
JP2013501715A (ja) 殺菌・殺カビ性ジフェニル−置換ピリダジン
JP2011525922A (ja) 殺菌性ピリジン
JP2013541535A (ja) 殺菌・殺カビ性イミダゾール
JP2013509408A (ja) 複素二環置換されたアゾリルベンゼン殺菌・殺カビ剤
US20120329787A1 (en) Fungicidal pyranones and oxazinones
WO2018052838A1 (en) Fungicidal pyrazoles
JP2023513239A (ja) 殺真菌薬としての使用のための置換５，６－ジフェニル－３（２ｈ）－ピリダジノン
JP2018510155A (ja) 殺菌・殺カビ性ピラゾール
CN105683164A (zh) 杀真菌吡唑类
CA3229284A1 (en) Fungicidal substituted heterocycles

Legal Events

Date Code Title Description
A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20140820

A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20140820

A977 Report on retrieval

Free format text: JAPANESE INTERMEDIATE CODE: A971007

Effective date: 20150428

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20150526

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20150826

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20151125

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20160426

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20160726

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20160926

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20161026

TRDD Decision of grant or rejection written
A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

Effective date: 20161122

A61 First payment of annual fees (during grant procedure)

Free format text: JAPANESE INTERMEDIATE CODE: A61

Effective date: 20161220

R150 Certificate of patent or registration of utility model

Ref document number: 6066910

Country of ref document: JP

Free format text: JAPANESE INTERMEDIATE CODE: R150

S111 Request for change of ownership or part of ownership

Free format text: JAPANESE INTERMEDIATE CODE: R313113

S531 Written request for registration of change of domicile

Free format text: JAPANESE INTERMEDIATE CODE: R313531

R350 Written notification of registration of transfer

Free format text: JAPANESE INTERMEDIATE CODE: R350

LAPS Cancellation because of no payment of annual fees