CH623813A5 - Process for the preparation of novel imidazole derivatives having an antifungal and antimicrobial action - Google Patents
Process for the preparation of novel imidazole derivatives having an antifungal and antimicrobial action Download PDFInfo
- Publication number
- CH623813A5 CH623813A5 CH1225575A CH1225575A CH623813A5 CH 623813 A5 CH623813 A5 CH 623813A5 CH 1225575 A CH1225575 A CH 1225575A CH 1225575 A CH1225575 A CH 1225575A CH 623813 A5 CH623813 A5 CH 623813A5
- Authority
- CH
- Switzerland
- Prior art keywords
- imidazole
- phenylethyl
- acid addition
- dichloro
- addition salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US50838474A | 1974-09-23 | 1974-09-23 | |
| US59362075A | 1975-07-07 | 1975-07-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH623813A5 true CH623813A5 (en) | 1981-06-30 |
Family
ID=27056177
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH1225575A CH623813A5 (en) | 1974-09-23 | 1975-09-22 | Process for the preparation of novel imidazole derivatives having an antifungal and antimicrobial action |
Country Status (19)
| Country | Link |
|---|---|
| JP (1) | JPS5910344B2 (fi) |
| AR (1) | AR224222A1 (fi) |
| AU (1) | AU496881B2 (fi) |
| CA (1) | CA1064040A (fi) |
| CH (1) | CH623813A5 (fi) |
| DE (1) | DE2541833A1 (fi) |
| DK (1) | DK155283C (fi) |
| FI (1) | FI64583C (fi) |
| FR (1) | FR2285126A1 (fi) |
| GB (1) | GB1485719A (fi) |
| HK (1) | HK8380A (fi) |
| IE (1) | IE43267B1 (fi) |
| IL (1) | IL47885A (fi) |
| MX (1) | MX4832E (fi) |
| MY (1) | MY8000270A (fi) |
| NL (1) | NL174462C (fi) |
| NO (1) | NO144345C (fi) |
| SE (1) | SE428471B (fi) |
| YU (3) | YU39746B (fi) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA755100B (en) * | 1974-09-23 | 1977-03-30 | Syntex Inc | 1-(b-(r-thio) phenethyl) imidazoles and derivatives thereof |
| EP0013786B1 (en) * | 1979-01-22 | 1982-10-06 | Syntex (U.S.A.) Inc. | Imidazole derivatives, pharmaceutical compositions containing them and their preparation |
| JPS63156228U (fi) * | 1987-04-01 | 1988-10-13 | ||
| DE3939525A1 (de) * | 1989-11-30 | 1991-06-06 | Hoechst Ag | Mit mehrfach ungesaettigten resten substituierte aryl-alkyl-azole, verfahren zu ihrer herstellung und ihre verwendung |
| IT1303672B1 (it) * | 1998-07-28 | 2001-02-23 | Nicox Sa | Sali nitrati di farmaci attivi nei disordini ossei |
| CN116063234B (zh) * | 2022-12-29 | 2023-11-24 | 山东京卫制药有限公司 | 一种硝酸硫康唑的制备方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU557755A3 (ru) * | 1968-08-19 | 1977-05-05 | Янссен Фармасьютика Н.В. (Фирма) | Способ получени производных имидазола |
| US3658813A (en) * | 1970-01-13 | 1972-04-25 | Janssen Pharmaceutica Nv | 1-(beta-aryl-beta-(r-oxy)-ethyl)-imidazoles |
| DE2041771C3 (de) * | 1970-08-22 | 1979-07-26 | Bayer Ag, 5090 Leverkusen | derivate |
| SE364275B (fi) * | 1971-06-17 | 1974-02-18 | Janssen Pharmaceutica Nv | |
| DE2242454A1 (de) * | 1972-08-29 | 1974-03-07 | Bayer Ag | 1-aethyl-imidazole, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
-
1975
- 1975-08-06 IL IL47885A patent/IL47885A/xx unknown
- 1975-08-18 CA CA233,620A patent/CA1064040A/en not_active Expired
- 1975-08-19 AU AU84081/75A patent/AU496881B2/en not_active Expired
- 1975-08-20 MX MX755341U patent/MX4832E/es unknown
- 1975-08-28 GB GB35569/75A patent/GB1485719A/en not_active Expired
- 1975-08-29 NL NLAANVRAGE7510224,A patent/NL174462C/xx not_active IP Right Cessation
- 1975-09-03 AR AR260311A patent/AR224222A1/es active
- 1975-09-05 YU YU2244/75A patent/YU39746B/xx unknown
- 1975-09-05 NO NO753048A patent/NO144345C/no unknown
- 1975-09-19 JP JP50113538A patent/JPS5910344B2/ja not_active Expired
- 1975-09-19 FI FI752614A patent/FI64583C/fi not_active IP Right Cessation
- 1975-09-19 DE DE19752541833 patent/DE2541833A1/de active Granted
- 1975-09-19 IE IE2061/75A patent/IE43267B1/en unknown
- 1975-09-22 CH CH1225575A patent/CH623813A5/de not_active IP Right Cessation
- 1975-09-22 SE SE7510595A patent/SE428471B/xx not_active IP Right Cessation
- 1975-09-22 FR FR7529009A patent/FR2285126A1/fr active Granted
- 1975-09-23 DK DK427075A patent/DK155283C/da active
-
1980
- 1980-03-06 HK HK83/80A patent/HK8380A/xx unknown
- 1980-12-31 MY MY1980270A patent/MY8000270A/xx unknown
-
1981
- 1981-09-21 YU YU02269/81A patent/YU226981A/xx unknown
- 1981-09-21 YU YU02270/81A patent/YU227081A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO753048L (fi) | 1976-03-24 |
| IE43267L (en) | 1976-03-23 |
| DK155283B (da) | 1989-03-20 |
| DK155283C (da) | 1989-07-24 |
| YU226981A (en) | 1982-02-28 |
| FI752614A (fi) | 1976-03-24 |
| DK427075A (da) | 1976-03-24 |
| YU39746B (en) | 1985-04-30 |
| GB1485719A (en) | 1977-09-14 |
| YU224475A (en) | 1982-02-28 |
| CA1064040A (en) | 1979-10-09 |
| FR2285126A1 (fr) | 1976-04-16 |
| NO144345C (no) | 1981-08-12 |
| JPS5157828A (en) | 1976-05-20 |
| FI64583C (fi) | 1983-12-12 |
| FR2285126B1 (fi) | 1979-09-14 |
| MY8000270A (en) | 1980-12-31 |
| NL174462B (nl) | 1984-01-16 |
| YU227081A (en) | 1982-02-28 |
| NL7510224A (nl) | 1976-03-25 |
| NL174462C (nl) | 1984-06-18 |
| MX4832E (es) | 1982-10-26 |
| IL47885A (en) | 1979-01-31 |
| DE2541833C2 (fi) | 1989-09-14 |
| AU8408175A (en) | 1977-02-24 |
| IE43267B1 (en) | 1981-01-28 |
| FI64583B (fi) | 1983-08-31 |
| DE2541833A1 (de) | 1976-04-01 |
| IL47885A0 (en) | 1975-11-25 |
| AU496881B2 (en) | 1978-11-09 |
| SE428471B (sv) | 1983-07-04 |
| JPS5910344B2 (ja) | 1984-03-08 |
| HK8380A (en) | 1980-03-14 |
| SE7510595L (sv) | 1976-03-24 |
| NO144345B (no) | 1981-05-04 |
| AR224222A1 (es) | 1981-11-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PL | Patent ceased |