BR9611957A - Di-hidrato de (2r,3s) -3- terc.- butoxicarbonilamino - 2 -hidroxi - 3 - fenilpropionato de 4,10 beta-diacetoxi - 2 - alfa-benzoiloxi-5beta, 20 - epoxi - 1 - hidroxi - 9 - oco - 19 - nor - ciclopropa[g]tax - 11eno - 13alfa - ila e processo para preparação do mesmo - Google Patents

Di-hidrato de (2r,3s) -3- terc.- butoxicarbonilamino - 2 -hidroxi - 3 - fenilpropionato de 4,10 beta-diacetoxi - 2 - alfa-benzoiloxi-5beta, 20 - epoxi - 1 - hidroxi - 9 - oco - 19 - nor - ciclopropa[g]tax - 11eno - 13alfa - ila e processo para preparação do mesmo

Info

Publication number
BR9611957A
BR9611957A BR9611957A BR9611957A BR9611957A BR 9611957 A BR9611957 A BR 9611957A BR 9611957 A BR9611957 A BR 9611957A BR 9611957 A BR9611957 A BR 9611957A BR 9611957 A BR9611957 A BR 9611957A
Authority
BR
Brazil
Prior art keywords
hydroxy
13alfa
11eno
5beta
cyclopropa
Prior art date
Application number
BR9611957A
Other languages
English (en)
Inventor
Michel Lavigne
Jean-Rene Authelin
Eric Didier
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9485512&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9611957(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of BR9611957A publication Critical patent/BR9611957A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
BR9611957A 1995-12-14 1996-12-09 Di-hidrato de (2r,3s) -3- terc.- butoxicarbonilamino - 2 -hidroxi - 3 - fenilpropionato de 4,10 beta-diacetoxi - 2 - alfa-benzoiloxi-5beta, 20 - epoxi - 1 - hidroxi - 9 - oco - 19 - nor - ciclopropa[g]tax - 11eno - 13alfa - ila e processo para preparação do mesmo BR9611957A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9514841A FR2742438B1 (fr) 1995-12-14 1995-12-14 Dihydrate du (2r,3s)-3-tert-butoxycarbonylamino-2-hydroxy- 3-phenylpropionate de 4,10beta-diacetoxy-2alpha-benzoyloxy- 5beta,2o-epoxy-1-hydroxy-9-oxo-19-nor-cyclopropa(g)tax-11- ene-13alpha-yle, et son procede de preparation
PCT/FR1996/001957 WO1997021695A1 (fr) 1995-12-14 1996-12-09 DIHYDRATE DU (2R,3S)-3-TERT-BUTOXYCARBONYLAMINO-2-HYDROXY-3-PHENYLPROPIONATE DE 4,10β-DIACETOXY-2α-BENZOYLOXY-5β,20-EPOXY-1-HYDROXY-9-OXO-19-NOR-CYCLOPROPA[G]TAX-11-ENE-13α-YLE, ET SON PROCEDE DE PREPARATION

Publications (1)

Publication Number Publication Date
BR9611957A true BR9611957A (pt) 1999-02-17

Family

ID=9485512

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9611957A BR9611957A (pt) 1995-12-14 1996-12-09 Di-hidrato de (2r,3s) -3- terc.- butoxicarbonilamino - 2 -hidroxi - 3 - fenilpropionato de 4,10 beta-diacetoxi - 2 - alfa-benzoiloxi-5beta, 20 - epoxi - 1 - hidroxi - 9 - oco - 19 - nor - ciclopropa[g]tax - 11eno - 13alfa - ila e processo para preparação do mesmo

Country Status (37)

Country Link
EP (1) EP0876361B1 (pt)
JP (1) JP4059351B2 (pt)
KR (1) KR100429330B1 (pt)
CN (1) CN101113143A (pt)
AR (1) AR004380A1 (pt)
AT (1) ATE204573T1 (pt)
AU (1) AU713086C (pt)
BG (1) BG63010B1 (pt)
BR (1) BR9611957A (pt)
CA (1) CA2236545C (pt)
CO (1) CO4810227A1 (pt)
CZ (1) CZ288998B6 (pt)
DE (1) DE69614716T2 (pt)
DK (1) DK0876361T3 (pt)
DZ (1) DZ2140A1 (pt)
EA (1) EA000668B1 (pt)
ES (1) ES2162123T3 (pt)
FR (1) FR2742438B1 (pt)
GR (1) GR3036437T3 (pt)
HU (1) HU224962B1 (pt)
IL (1) IL124766A (pt)
IN (1) IN185809B (pt)
MY (1) MY115886A (pt)
NO (1) NO317356B1 (pt)
NZ (1) NZ323964A (pt)
OA (1) OA11012A (pt)
PL (1) PL187613B1 (pt)
PT (1) PT876361E (pt)
RO (1) RO115880B1 (pt)
SK (1) SK282512B6 (pt)
TN (1) TNSN96157A1 (pt)
TR (1) TR199801087T2 (pt)
TW (1) TW358093B (pt)
UA (1) UA55401C2 (pt)
UY (1) UY24387A1 (pt)
WO (1) WO1997021695A1 (pt)
ZA (1) ZA9610200B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102851740A (zh) * 2011-06-30 2013-01-02 复旦大学 一种氟代多烯紫杉醇晶体及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2698871B1 (fr) * 1992-12-09 1995-02-24 Rhone Poulenc Rorer Sa Nouveau taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
PL187613B1 (pl) 2004-08-31
DE69614716T2 (de) 2002-06-27
PL327451A1 (en) 1998-12-07
FR2742438B1 (fr) 1998-01-16
CA2236545A1 (fr) 1997-06-19
AU1101397A (en) 1997-07-03
NO982561L (no) 1998-06-04
NO317356B1 (no) 2004-10-18
EP0876361A1 (fr) 1998-11-11
CN101113143A (zh) 2008-01-30
JP4059351B2 (ja) 2008-03-12
MX9804604A (es) 1998-10-31
SK79098A3 (en) 1998-11-04
EA199800452A1 (ru) 1998-12-24
RO115880B1 (ro) 2000-07-28
BG63010B1 (bg) 2001-01-31
ZA9610200B (en) 1997-06-23
UY24387A1 (es) 2001-08-27
SK282512B6 (sk) 2002-10-08
BG102535A (en) 1999-08-31
JP2000501722A (ja) 2000-02-15
MY115886A (en) 2003-09-30
CA2236545C (fr) 2007-01-30
OA11012A (fr) 2003-03-06
ATE204573T1 (de) 2001-09-15
AU713086B2 (en) 1999-11-25
AU713086C (en) 2002-09-19
DK0876361T3 (da) 2001-10-08
AR004380A1 (es) 1998-11-04
HU224962B1 (en) 2006-04-28
KR100429330B1 (ko) 2005-01-13
DZ2140A1 (fr) 2002-07-23
GR3036437T3 (en) 2001-11-30
EP0876361B1 (fr) 2001-08-22
NZ323964A (en) 2000-01-28
EA000668B1 (ru) 2000-02-28
CZ288998B6 (cs) 2001-10-17
ES2162123T3 (es) 2001-12-16
HUP9904048A3 (en) 2001-08-28
NO982561D0 (no) 1998-06-04
KR19990072107A (ko) 1999-09-27
UA55401C2 (uk) 2003-04-15
IL124766A (en) 2001-03-19
DE69614716D1 (de) 2001-09-27
CZ183098A3 (cs) 1998-09-16
IL124766A0 (en) 1999-01-26
IN185809B (pt) 2001-05-05
HUP9904048A1 (hu) 2001-04-28
TW358093B (en) 1999-05-11
TNSN96157A1 (fr) 2005-03-15
CO4810227A1 (es) 1999-06-30
WO1997021695A1 (fr) 1997-06-19
FR2742438A1 (fr) 1997-06-20
PT876361E (pt) 2001-11-30
TR199801087T2 (xx) 1998-09-21

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BR9611957A (pt) Di-hidrato de (2r,3s) -3- terc.- butoxicarbonilamino - 2 -hidroxi - 3 - fenilpropionato de 4,10 beta-diacetoxi - 2 - alfa-benzoiloxi-5beta, 20 - epoxi - 1 - hidroxi - 9 - oco - 19 - nor - ciclopropa[g]tax - 11eno - 13alfa - ila e processo para preparação do mesmo
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Legal Events

Date Code Title Description
TC Change of name
FB36 Technical and formal requirements: requirement - article 36 of industrial property law
HJEG Technical examination (opinion): technical examination (opinion) related to article 229 of industrial property law
FF Decision: intention to grant
HHFI Decision: rectification
FF Decision: intention to grant
HKFF Publication of grant (deleted)
FG9A Patent or certificate of addition granted
B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 17A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2258 DE 15-04-2014 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.