NZ323964A - 4,10beta-diacetoxy-2alpha-benzoyloxy-5beta,20-epoxy-1-hydroxy-9-oxo-19-nor-cy clopropa[g]tax-11-ene-13alpha-yl - Google Patents

4,10beta-diacetoxy-2alpha-benzoyloxy-5beta,20-epoxy-1-hydroxy-9-oxo-19-nor-cy clopropa[g]tax-11-ene-13alpha-yl

Info

Publication number
NZ323964A
NZ323964A NZ323964A NZ32396496A NZ323964A NZ 323964 A NZ323964 A NZ 323964A NZ 323964 A NZ323964 A NZ 323964A NZ 32396496 A NZ32396496 A NZ 32396496A NZ 323964 A NZ323964 A NZ 323964A
Authority
NZ
New Zealand
Prior art keywords
hydroxy
diacetoxy
benzoyloxy
tax
ene
Prior art date
Application number
NZ323964A
Inventor
Eric Didier
Michel Lavigne
Jean-Rene Authelin
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9485512&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ323964(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of NZ323964A publication Critical patent/NZ323964A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

4,10Ô-diacetoxy-2ß-benzoyloxy-5Ô,20-epoxy-1-hydroxy-9-oxo-19-nor-cyclopropa[g]tax-11-ene-13ß-ßyl (2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate dihydrate is disclosed. Also encompassed is the preparation thereof by crystallisation from a water-alcohol or water-ketone solution.
NZ323964A 1995-12-14 1996-12-09 4,10beta-diacetoxy-2alpha-benzoyloxy-5beta,20-epoxy-1-hydroxy-9-oxo-19-nor-cy clopropa[g]tax-11-ene-13alpha-yl NZ323964A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9514841A FR2742438B1 (en) 1995-12-14 1995-12-14 (2R, 3S) DIHYDRATE -3-TERT-BUTOXYCARBONYLAMINO-2-HYDROXY- 3-PHENYLPROPIONATE OF 4,10BETA-DIACETOXY-2ALPHA-BENZOYLOXY- 5BETA, 2O-EPOXY-1-HYDROX CYCLOPROPA (G) TAX-11- ENE-13ALPHA-YLE, AND PREPARATION METHOD THEREOF
PCT/FR1996/001957 WO1997021695A1 (en) 1995-12-14 1996-12-09 4,10β-DIACETOXY-2α-BENZOYLOXY-5β,20-EPOXY-1-HYDROXY-9-OXO-19-NOR-CYCLOPROPA[G]TAX-11-ENE-13α-YL (2R,3S)-TERT-BUTOXYCARBONYLAMINO-2-HYDROXY-3-PHENYLPROPIONATE DIHYDRATE, AND METHOD FOR PREPARING SAME

Publications (1)

Publication Number Publication Date
NZ323964A true NZ323964A (en) 2000-01-28

Family

ID=9485512

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ323964A NZ323964A (en) 1995-12-14 1996-12-09 4,10beta-diacetoxy-2alpha-benzoyloxy-5beta,20-epoxy-1-hydroxy-9-oxo-19-nor-cy clopropa[g]tax-11-ene-13alpha-yl

Country Status (37)

Country Link
EP (1) EP0876361B1 (en)
JP (1) JP4059351B2 (en)
KR (1) KR100429330B1 (en)
CN (1) CN101113143A (en)
AR (1) AR004380A1 (en)
AT (1) ATE204573T1 (en)
AU (1) AU713086C (en)
BG (1) BG63010B1 (en)
BR (1) BR9611957A (en)
CA (1) CA2236545C (en)
CO (1) CO4810227A1 (en)
CZ (1) CZ288998B6 (en)
DE (1) DE69614716T2 (en)
DK (1) DK0876361T3 (en)
DZ (1) DZ2140A1 (en)
EA (1) EA000668B1 (en)
ES (1) ES2162123T3 (en)
FR (1) FR2742438B1 (en)
GR (1) GR3036437T3 (en)
HU (1) HU224962B1 (en)
IL (1) IL124766A (en)
IN (1) IN185809B (en)
MY (1) MY115886A (en)
NO (1) NO317356B1 (en)
NZ (1) NZ323964A (en)
OA (1) OA11012A (en)
PL (1) PL187613B1 (en)
PT (1) PT876361E (en)
RO (1) RO115880B1 (en)
SK (1) SK282512B6 (en)
TN (1) TNSN96157A1 (en)
TR (1) TR199801087T2 (en)
TW (1) TW358093B (en)
UA (1) UA55401C2 (en)
UY (1) UY24387A1 (en)
WO (1) WO1997021695A1 (en)
ZA (1) ZA9610200B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102851740A (en) * 2011-06-30 2013-01-02 复旦大学 Fluorinated docetaxel crystal and its preparation method

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2698871B1 (en) * 1992-12-09 1995-02-24 Rhone Poulenc Rorer Sa New taxoids, their preparation and the pharmaceutical compositions containing them.

Also Published As

Publication number Publication date
DZ2140A1 (en) 2002-07-23
GR3036437T3 (en) 2001-11-30
EP0876361A1 (en) 1998-11-11
BR9611957A (en) 1999-02-17
AR004380A1 (en) 1998-11-04
CO4810227A1 (en) 1999-06-30
DE69614716T2 (en) 2002-06-27
AU1101397A (en) 1997-07-03
EP0876361B1 (en) 2001-08-22
EA000668B1 (en) 2000-02-28
CA2236545C (en) 2007-01-30
FR2742438A1 (en) 1997-06-20
DE69614716D1 (en) 2001-09-27
OA11012A (en) 2003-03-06
SK282512B6 (en) 2002-10-08
FR2742438B1 (en) 1998-01-16
ATE204573T1 (en) 2001-09-15
MY115886A (en) 2003-09-30
HUP9904048A1 (en) 2001-04-28
MX9804604A (en) 1998-10-31
ZA9610200B (en) 1997-06-23
NO982561D0 (en) 1998-06-04
JP2000501722A (en) 2000-02-15
UY24387A1 (en) 2001-08-27
TW358093B (en) 1999-05-11
CZ288998B6 (en) 2001-10-17
KR19990072107A (en) 1999-09-27
NO317356B1 (en) 2004-10-18
CZ183098A3 (en) 1998-09-16
HU224962B1 (en) 2006-04-28
KR100429330B1 (en) 2005-01-13
PL187613B1 (en) 2004-08-31
AU713086B2 (en) 1999-11-25
AU713086C (en) 2002-09-19
EA199800452A1 (en) 1998-12-24
BG63010B1 (en) 2001-01-31
BG102535A (en) 1999-08-31
ES2162123T3 (en) 2001-12-16
NO982561L (en) 1998-06-04
JP4059351B2 (en) 2008-03-12
PT876361E (en) 2001-11-30
CN101113143A (en) 2008-01-30
DK0876361T3 (en) 2001-10-08
WO1997021695A1 (en) 1997-06-19
IL124766A0 (en) 1999-01-26
CA2236545A1 (en) 1997-06-19
IN185809B (en) 2001-05-05
HUP9904048A3 (en) 2001-08-28
TR199801087T2 (en) 1998-09-21
UA55401C2 (en) 2003-04-15
RO115880B1 (en) 2000-07-28
SK79098A3 (en) 1998-11-04
TNSN96157A1 (en) 2005-03-15
IL124766A (en) 2001-03-19
PL327451A1 (en) 1998-12-07

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