BR112015006848A2 - formulação farmacêutica, método de indução de perda de peso, método de redução de gordura corporal, método de redução de ingesta de comida, método para melhorar homeostase de glicose e método para prevenir um aumento do índice de massa corporal de um paciente normal, pré-obeso, obeso ou obeso mórbido. - Google Patents

formulação farmacêutica, método de indução de perda de peso, método de redução de gordura corporal, método de redução de ingesta de comida, método para melhorar homeostase de glicose e método para prevenir um aumento do índice de massa corporal de um paciente normal, pré-obeso, obeso ou obeso mórbido.

Info

Publication number
BR112015006848A2
BR112015006848A2 BR112015006848A BR112015006848A BR112015006848A2 BR 112015006848 A2 BR112015006848 A2 BR 112015006848A2 BR 112015006848 A BR112015006848 A BR 112015006848A BR 112015006848 A BR112015006848 A BR 112015006848A BR 112015006848 A2 BR112015006848 A2 BR 112015006848A2
Authority
BR
Brazil
Prior art keywords
obese
reduction method
preterm
patient
preventing
Prior art date
Application number
BR112015006848A
Other languages
English (en)
Portuguese (pt)
Inventor
Cakir Isin
Majzoub Joseph
Mazitschek Ralph
Cabi Serkan
Ozcan Umut
Original Assignee
Childrens Medical Ct Corp
The Massachusetts General Hospital
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49304418&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112015006848(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Childrens Medical Ct Corp, The Massachusetts General Hospital filed Critical Childrens Medical Ct Corp
Publication of BR112015006848A2 publication Critical patent/BR112015006848A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/194Carboxylic acids, e.g. valproic acid having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/2264Obesity-gene products, e.g. leptin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
BR112015006848A 2012-09-27 2013-09-26 formulação farmacêutica, método de indução de perda de peso, método de redução de gordura corporal, método de redução de ingesta de comida, método para melhorar homeostase de glicose e método para prevenir um aumento do índice de massa corporal de um paciente normal, pré-obeso, obeso ou obeso mórbido. BR112015006848A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261706153P 2012-09-27 2012-09-27
PCT/US2013/061911 WO2014052583A1 (en) 2012-09-27 2013-09-26 Compounds for the treatment of obesity and methods of use thereof

Publications (1)

Publication Number Publication Date
BR112015006848A2 true BR112015006848A2 (pt) 2018-05-22

Family

ID=49304418

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015006848A BR112015006848A2 (pt) 2012-09-27 2013-09-26 formulação farmacêutica, método de indução de perda de peso, método de redução de gordura corporal, método de redução de ingesta de comida, método para melhorar homeostase de glicose e método para prevenir um aumento do índice de massa corporal de um paciente normal, pré-obeso, obeso ou obeso mórbido.

Country Status (21)

Country Link
US (6) US9968575B2 (enExample)
EP (3) EP3434268B1 (enExample)
JP (2) JP6480864B2 (enExample)
CN (3) CN111529535A (enExample)
AU (3) AU2013323528B2 (enExample)
BR (1) BR112015006848A2 (enExample)
CA (2) CA3030272C (enExample)
CY (1) CY1121166T1 (enExample)
DK (1) DK2900230T3 (enExample)
ES (1) ES2696626T3 (enExample)
HR (1) HRP20181879T1 (enExample)
HU (1) HUE040496T2 (enExample)
LT (1) LT2900230T (enExample)
PL (1) PL2900230T3 (enExample)
PT (1) PT2900230T (enExample)
RS (1) RS58010B1 (enExample)
RU (2) RU2768868C2 (enExample)
SI (1) SI2900230T1 (enExample)
SM (1) SMT201800604T1 (enExample)
TR (1) TR201815668T4 (enExample)
WO (1) WO2014052583A1 (enExample)

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CN106905404B (zh) * 2017-01-13 2019-08-27 广东工业大学 熊果酸衍生物及其制备方法和应用
CN116509842B (zh) * 2021-09-09 2024-09-20 厦门君德医药科技有限公司 药物组合物及其制备方法和应用
KR102470686B1 (ko) * 2022-06-07 2022-11-23 서울대학교산학협력단 디메틸제일아스테럴을 포함하는 대사성 질환 예방 또는 치료용 약학 조성물
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Also Published As

Publication number Publication date
US20210275482A1 (en) 2021-09-09
EP2900230B1 (en) 2018-08-15
RU2650646C2 (ru) 2018-04-16
US20180185314A1 (en) 2018-07-05
CA2886393A1 (en) 2014-04-03
CN111529534A (zh) 2020-08-14
HK1213190A1 (en) 2016-06-30
RU2018112067A3 (enExample) 2021-06-24
AU2018256619A1 (en) 2018-11-22
TR201815668T4 (tr) 2018-11-21
AU2016247206A1 (en) 2016-11-10
SI2900230T1 (sl) 2019-01-31
RU2768868C2 (ru) 2022-03-25
WO2014052583A1 (en) 2014-04-03
EP2900230A1 (en) 2015-08-05
AU2013323528A1 (en) 2015-04-09
JP2015531376A (ja) 2015-11-02
CA3030272C (en) 2021-09-28
US12064408B2 (en) 2024-08-20
ES2696626T3 (es) 2019-01-17
US20250161252A1 (en) 2025-05-22
CN111529535A (zh) 2020-08-14
PL2900230T3 (pl) 2019-02-28
US20210008019A1 (en) 2021-01-14
US11045439B2 (en) 2021-06-29
EP3434268B1 (en) 2022-04-20
SMT201800604T1 (it) 2019-01-11
CA2886393C (en) 2019-02-26
HRP20181879T1 (hr) 2019-02-08
PT2900230T (pt) 2018-11-26
EP3434268A1 (en) 2019-01-30
JP2019070052A (ja) 2019-05-09
JP6743211B2 (ja) 2020-08-19
CY1121166T1 (el) 2020-05-29
AU2018256619B2 (en) 2020-07-23
US9968575B2 (en) 2018-05-15
CA3030272A1 (en) 2014-04-03
AU2013323528B2 (en) 2016-11-10
RU2015115696A (ru) 2016-11-20
RS58010B1 (sr) 2019-02-28
US9925161B2 (en) 2018-03-27
US20150250753A1 (en) 2015-09-10
CN104822374A (zh) 2015-08-05
LT2900230T (lt) 2019-01-10
AU2016247206B2 (en) 2018-08-02
EP4082541A1 (en) 2022-11-02
DK2900230T3 (en) 2018-11-12
HUE040496T2 (hu) 2019-03-28
JP6480864B2 (ja) 2019-03-13
RU2018112067A (ru) 2019-03-07
US20170304245A1 (en) 2017-10-26
US10653654B2 (en) 2020-05-19

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