BR112012033253A2 - novos derivados de pirimidina fundidos para inibição da atividade de tirosina quinase - Google Patents

novos derivados de pirimidina fundidos para inibição da atividade de tirosina quinase

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Publication number
BR112012033253A2
BR112012033253A2 BR112012033253A BR112012033253A BR112012033253A2 BR 112012033253 A2 BR112012033253 A2 BR 112012033253A2 BR 112012033253 A BR112012033253 A BR 112012033253A BR 112012033253 A BR112012033253 A BR 112012033253A BR 112012033253 A2 BR112012033253 A2 BR 112012033253A2
Authority
BR
Brazil
Prior art keywords
inhibition
tyrosine kinase
kinase activity
pyrimidine derivatives
fused pyrimidine
Prior art date
Application number
BR112012033253A
Other languages
English (en)
Portuguese (pt)
Inventor
Eun Joo Kwak
Ji Young Jeon
Ju Yeon Lee
Kwang Ok Lee
Kwee Hyun Suh
Maeng Sup Kim
Mi Ra Kim
Mi Young Cha
Myoung Gi Jo
Seok Jong Kang
Tae Hee Ha
Original Assignee
Hanmi Science Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45371929&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112012033253(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hanmi Science Co Ltd filed Critical Hanmi Science Co Ltd
Priority to BR122014012788-0A priority Critical patent/BR122014012788B1/pt
Publication of BR112012033253A2 publication Critical patent/BR112012033253A2/pt

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    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
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    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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BR112012033253A 2010-06-23 2011-06-20 novos derivados de pirimidina fundidos para inibição da atividade de tirosina quinase BR112012033253A2 (pt)

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Application Number Priority Date Filing Date Title
BR122014012788-0A BR122014012788B1 (pt) 2010-06-23 2011-06-20 Derivados de pirimidina fundidos, seus usos, e composição farmacêutica para inibição da atividade de tirosina quinase

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