BR112012002641B1 - Processo de preparação de amidas de ácido carboxílico pirazol, bem como compostos intermediários - Google Patents
Processo de preparação de amidas de ácido carboxílico pirazol, bem como compostos intermediários Download PDFInfo
- Publication number
- BR112012002641B1 BR112012002641B1 BR112012002641-0A BR112012002641A BR112012002641B1 BR 112012002641 B1 BR112012002641 B1 BR 112012002641B1 BR 112012002641 A BR112012002641 A BR 112012002641A BR 112012002641 B1 BR112012002641 B1 BR 112012002641B1
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- BR
- Brazil
- Prior art keywords
- compound
- formula
- reaction
- viii
- mol
- Prior art date
Links
- OWUJELSBTKCQMP-FOWTUZBSSA-N C=CCC(C(C1)=C(Cl)Cl)C(CCC2)=C1/C2=N/O Chemical compound C=CCC(C(C1)=C(Cl)Cl)C(CCC2)=C1/C2=N/O OWUJELSBTKCQMP-FOWTUZBSSA-N 0.000 description 1
- MSYUKIDLEBQGOU-UHFFFAOYSA-N NC(N)=C1C2C(C(CCC3)=O)=C3C1CC2 Chemical compound NC(N)=C1C2C(C(CCC3)=O)=C3C1CC2 MSYUKIDLEBQGOU-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/32—Oximes
- C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C251/44—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups being part of a ring other than a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/62—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by hydrogenation of carbon-to-carbon double or triple bonds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/65—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups
- C07C45/66—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups by dehydration
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
- C07C45/69—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by addition to carbon-to-carbon double or triple bonds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
- C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
- C07C49/693—Unsaturated compounds containing a keto groups being part of a ring containing halogen polycyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
- C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
- C07C49/743—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups having unsaturation outside the rings, e.g. humulones, lupulones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
- C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
- C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
- C07D251/40—Nitrogen atoms
- C07D251/42—One nitrogen atom
- C07D251/44—One nitrogen atom with halogen atoms attached to the two other ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/56—Ring systems containing bridged rings
- C07C2603/58—Ring systems containing bridged rings containing three rings
- C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
- C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09167363 | 2009-08-06 | ||
| EP09167363.2 | 2009-08-06 | ||
| EP09169501 | 2009-09-04 | ||
| EP091695501.5 | 2009-09-04 | ||
| PCT/EP2010/059703 WO2011015416A1 (en) | 2009-08-06 | 2010-07-07 | Process for the preparation of pyrazole carboxylic acid amides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BR112012002641A2 BR112012002641A2 (pt) | 2016-03-22 |
| BR112012002641B1 true BR112012002641B1 (pt) | 2018-05-22 |
Family
ID=42670451
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012002641-0A BR112012002641B1 (pt) | 2009-08-06 | 2010-07-07 | Processo de preparação de amidas de ácido carboxílico pirazol, bem como compostos intermediários |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US8507694B2 (https=) |
| EP (1) | EP2462108B1 (https=) |
| JP (1) | JP5667186B2 (https=) |
| KR (1) | KR101712083B1 (https=) |
| CN (1) | CN102574779B (https=) |
| AR (1) | AR077707A1 (https=) |
| AU (1) | AU2010280923B2 (https=) |
| BR (1) | BR112012002641B1 (https=) |
| CA (1) | CA2770144C (https=) |
| CL (1) | CL2012000272A1 (https=) |
| CO (1) | CO6430457A2 (https=) |
| CR (1) | CR20120056A (https=) |
| DK (1) | DK2462108T3 (https=) |
| EA (1) | EA019475B1 (https=) |
| EC (1) | ECSP12011647A (https=) |
| EG (1) | EG26957A (https=) |
| ES (1) | ES2417315T3 (https=) |
| GE (1) | GEP20146010B (https=) |
| IL (1) | IL217692A (https=) |
| IN (1) | IN2012DN00289A (https=) |
| MX (1) | MX2012001480A (https=) |
| MY (1) | MY161666A (https=) |
| NZ (1) | NZ597576A (https=) |
| PL (1) | PL2462108T3 (https=) |
| TW (1) | TWI441812B (https=) |
| UY (1) | UY32835A (https=) |
| WO (1) | WO2011015416A1 (https=) |
| ZA (1) | ZA201200413B (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI534126B (zh) | 2011-01-25 | 2016-05-21 | 先正達合夥公司 | 用於製備吡唑羧酸醯胺之方法 |
| TWI510472B (zh) * | 2012-02-15 | 2015-12-01 | Syngenta Participations Ag | 立體選擇性製備吡唑羧醯胺之方法 |
| GB201403438D0 (en) * | 2014-02-27 | 2014-04-16 | Syngenta Participations Ag | Polymorphs |
| RU2673722C2 (ru) | 2014-03-20 | 2018-11-29 | Мицуи Кемикалз Агро, Инк. | Композиция для борьбы с болезнями растений и способ борьбы с болезнями растений путем ее применения |
| KR20250036910A (ko) | 2022-07-22 | 2025-03-14 | 신젠타 크롭 프로텍션 아게 | 이종환식 아미드 유도체의 고체 형태 |
| CN120835879A (zh) * | 2022-10-11 | 2025-10-24 | 先正达农作物保护股份公司 | 用于制备吡唑羧酸酰胺的方法 |
| CN117362179B (zh) * | 2023-09-22 | 2025-07-08 | 浙江工业大学 | 一种苯并烯氟菌唑中间体9-二氯亚甲基-1,4-二氢-5-硝基-1,4-甲桥萘的制备方法 |
| PY2503719A (es) | 2024-01-26 | 2025-08-05 | Syngenta Crop Protection Ag | Proceso químico |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4370341A (en) * | 1980-12-11 | 1983-01-25 | Ayerst, Mckenna & Harrison, Ltd. | 6,7,8,9-Tetrahydro-3H-benz[E]indol-8-amine derivatives |
| JPS58194853A (ja) * | 1982-05-11 | 1983-11-12 | Showa Denko Kk | シクロヘキセン−アセチルオキシム誘導体 |
| US5093347A (en) * | 1991-01-28 | 1992-03-03 | Monsanto Company | 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use |
| US5932752A (en) * | 1995-12-29 | 1999-08-03 | Council Of Scientific And Industrial Research | Process for the C-C bond forming reaction using solid acid catalysts |
| GB0224316D0 (en) * | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| CN1618783A (zh) * | 2004-04-22 | 2005-05-25 | 复旦大学 | 一种多取代苯醌的制备方法 |
| US7732469B2 (en) * | 2005-10-25 | 2010-06-08 | Syngenta Crop Protection, Inc. | Heterocyclic amide derivatives useful as microbiocides |
-
2010
- 2010-07-07 AU AU2010280923A patent/AU2010280923B2/en active Active
- 2010-07-07 BR BR112012002641-0A patent/BR112012002641B1/pt active IP Right Grant
- 2010-07-07 CA CA2770144A patent/CA2770144C/en active Active
- 2010-07-07 WO PCT/EP2010/059703 patent/WO2011015416A1/en not_active Ceased
- 2010-07-07 GE GEAP201012617A patent/GEP20146010B/en unknown
- 2010-07-07 PL PL10729880T patent/PL2462108T3/pl unknown
- 2010-07-07 ES ES10729880T patent/ES2417315T3/es active Active
- 2010-07-07 EA EA201200246A patent/EA019475B1/ru not_active IP Right Cessation
- 2010-07-07 NZ NZ597576A patent/NZ597576A/xx unknown
- 2010-07-07 DK DK10729880.4T patent/DK2462108T3/da active
- 2010-07-07 MX MX2012001480A patent/MX2012001480A/es active IP Right Grant
- 2010-07-07 CN CN201080034393.8A patent/CN102574779B/zh active Active
- 2010-07-07 US US13/389,000 patent/US8507694B2/en active Active
- 2010-07-07 IN IN289DEN2012 patent/IN2012DN00289A/en unknown
- 2010-07-07 JP JP2012523260A patent/JP5667186B2/ja active Active
- 2010-07-07 KR KR1020127005767A patent/KR101712083B1/ko active Active
- 2010-07-07 MY MYPI2012000229A patent/MY161666A/en unknown
- 2010-07-07 EP EP10729880.4A patent/EP2462108B1/en active Active
- 2010-08-04 AR ARP100102863A patent/AR077707A1/es active IP Right Grant
- 2010-08-04 TW TW099125901A patent/TWI441812B/zh active
- 2010-08-06 UY UY0001032835A patent/UY32835A/es active IP Right Grant
-
2012
- 2012-01-18 ZA ZA2012/00413A patent/ZA201200413B/en unknown
- 2012-01-22 EG EG2012010118A patent/EG26957A/xx active
- 2012-01-23 IL IL217692A patent/IL217692A/en active IP Right Grant
- 2012-02-01 CR CR20120056A patent/CR20120056A/es unknown
- 2012-02-02 EC ECSP12011647 patent/ECSP12011647A/es unknown
- 2012-02-02 CL CL2012000272A patent/CL2012000272A1/es unknown
- 2012-02-03 CO CO12019264A patent/CO6430457A2/es active IP Right Grant
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] | ||
| B25G | Requested change of headquarter approved | ||
| B25A | Requested transfer of rights approved |