UY32835A - Proceso para la preparación de amidas de ácido pirazol carboxílico - Google Patents

Proceso para la preparación de amidas de ácido pirazol carboxílico

Info

Publication number
UY32835A
UY32835A UY0001032835A UY32835A UY32835A UY 32835 A UY32835 A UY 32835A UY 0001032835 A UY0001032835 A UY 0001032835A UY 32835 A UY32835 A UY 32835A UY 32835 A UY32835 A UY 32835A
Authority
UY
Uruguay
Prior art keywords
preparation
amidas
pirazol
carboxyl acid
steps
Prior art date
Application number
UY0001032835A
Other languages
English (en)
Inventor
Giordano Fanny
Mueller Adrian
Lagger Martin
Gribkov Denis
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of UY32835A publication Critical patent/UY32835A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/44—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups being part of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/62—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by hydrogenation of carbon-to-carbon double or triple bonds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/65—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups
    • C07C45/66—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups by dehydration
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/69—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by addition to carbon-to-carbon double or triple bonds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
    • C07C49/693—Unsaturated compounds containing a keto groups being part of a ring containing halogen polycyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
    • C07C49/743—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups having unsaturation outside the rings, e.g. humulones, lupulones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
    • C07D251/40—Nitrogen atoms
    • C07D251/42—One nitrogen atom
    • C07D251/44—One nitrogen atom with halogen atoms attached to the two other ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Proceso para la preparación de (9-diclorometileno-1,2,3,4-tetrahidro-1,4-metano-naftalen-5-i1)-a mida del ácido 3-difluormetil-1-metii-1 H-pirazol-4-carboxílico, que consiste de siete etapas que comprenden pasos de hidrogenación, reducción, deshidra tación, reacción con hidroxilamina, y acilación para obtener el producto de fórmula (I).
UY0001032835A 2009-08-06 2010-08-06 Proceso para la preparación de amidas de ácido pirazol carboxílico UY32835A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09167363 2009-08-06
EP09169501 2009-09-04

Publications (1)

Publication Number Publication Date
UY32835A true UY32835A (es) 2011-03-31

Family

ID=42670451

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032835A UY32835A (es) 2009-08-06 2010-08-06 Proceso para la preparación de amidas de ácido pirazol carboxílico

Country Status (28)

Country Link
US (1) US8507694B2 (es)
EP (1) EP2462108B1 (es)
JP (1) JP5667186B2 (es)
KR (1) KR101712083B1 (es)
CN (1) CN102574779B (es)
AR (1) AR077707A1 (es)
AU (1) AU2010280923B2 (es)
BR (1) BR112012002641B1 (es)
CA (1) CA2770144C (es)
CL (1) CL2012000272A1 (es)
CO (1) CO6430457A2 (es)
CR (1) CR20120056A (es)
DK (1) DK2462108T3 (es)
EA (1) EA019475B1 (es)
EC (1) ECSP12011647A (es)
EG (1) EG26957A (es)
ES (1) ES2417315T3 (es)
GE (1) GEP20146010B (es)
IL (1) IL217692A (es)
IN (1) IN2012DN00289A (es)
MX (1) MX2012001480A (es)
MY (1) MY161666A (es)
NZ (1) NZ597576A (es)
PL (1) PL2462108T3 (es)
TW (1) TWI441812B (es)
UY (1) UY32835A (es)
WO (1) WO2011015416A1 (es)
ZA (1) ZA201200413B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI534126B (zh) 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
TWI510472B (zh) * 2012-02-15 2015-12-01 Syngenta Participations Ag 立體選擇性製備吡唑羧醯胺之方法
GB201403438D0 (en) * 2014-02-27 2014-04-16 Syngenta Participations Ag Polymorphs
CR20160478A (es) 2014-03-20 2017-01-02 Mitsui Chemicals Agro Inc Composición de control de enfermedades de plantas y método para controlar enfermedades de plantas mediante su aplicación
WO2024017788A1 (en) 2022-07-22 2024-01-25 Syngenta Crop Protection Ag Solid form of a heterocyclic amide derivative
WO2024077487A1 (en) * 2022-10-11 2024-04-18 Syngenta Crop Protection Ag Process for the preparation of pyrazole carboxylic acid amides

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4370341A (en) * 1980-12-11 1983-01-25 Ayerst, Mckenna & Harrison, Ltd. 6,7,8,9-Tetrahydro-3H-benz[E]indol-8-amine derivatives
JPS58194853A (ja) * 1982-05-11 1983-11-12 Showa Denko Kk シクロヘキセン−アセチルオキシム誘導体
US5093347A (en) * 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US5932752A (en) * 1995-12-29 1999-08-03 Council Of Scientific And Industrial Research Process for the C-C bond forming reaction using solid acid catalysts
GB0224316D0 (en) * 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
CN1618783A (zh) * 2004-04-22 2005-05-25 复旦大学 一种多取代苯醌的制备方法
EP1940813B1 (en) * 2005-10-25 2010-11-24 Syngenta Participations AG Heterocyclic amide derivatives useful as microbiocides

Also Published As

Publication number Publication date
DK2462108T3 (da) 2013-07-08
JP2013501016A (ja) 2013-01-10
TW201107297A (en) 2011-03-01
MX2012001480A (es) 2012-02-22
TWI441812B (zh) 2014-06-21
AR077707A1 (es) 2011-09-14
EA201200246A1 (ru) 2012-08-30
CA2770144A1 (en) 2011-02-10
ES2417315T3 (es) 2013-08-07
JP5667186B2 (ja) 2015-02-12
CL2012000272A1 (es) 2012-09-28
KR20120043059A (ko) 2012-05-03
BR112012002641B1 (pt) 2018-05-22
US8507694B2 (en) 2013-08-13
GEP20146010B (en) 2014-01-10
CA2770144C (en) 2017-03-21
WO2011015416A1 (en) 2011-02-10
EG26957A (en) 2015-02-01
CR20120056A (es) 2012-03-06
PL2462108T3 (pl) 2013-09-30
CN102574779A (zh) 2012-07-11
MY161666A (en) 2017-04-28
AU2010280923A1 (en) 2012-02-09
IL217692A (en) 2015-07-30
CO6430457A2 (es) 2012-04-30
IN2012DN00289A (es) 2015-05-08
US20120136162A1 (en) 2012-05-31
ZA201200413B (en) 2012-10-31
EA019475B1 (ru) 2014-03-31
AU2010280923B2 (en) 2014-08-07
EP2462108B1 (en) 2013-04-17
KR101712083B1 (ko) 2017-03-03
EP2462108A1 (en) 2012-06-13
NZ597576A (en) 2013-01-25
CN102574779B (zh) 2014-10-15
ECSP12011647A (es) 2012-03-30
BR112012002641A2 (pt) 2016-03-22

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Effective date: 20210409