BR0311538A - Pirazolopirimidinas - Google Patents

Pirazolopirimidinas

Info

Publication number
BR0311538A
BR0311538A BR0311538-0A BR0311538A BR0311538A BR 0311538 A BR0311538 A BR 0311538A BR 0311538 A BR0311538 A BR 0311538A BR 0311538 A BR0311538 A BR 0311538A
Authority
BR
Brazil
Prior art keywords
halo
optionally substituted
new
cycloalkyl
dihydroxy
Prior art date
Application number
BR0311538-0A
Other languages
English (en)
Inventor
Olaf Gebauer
Nico Joerg Greul
Herbert Gayer
Bernd-Wieland Kr Ger
Hans-Ludwig Elbe
Ralf Dunkel
Oliver Guth
Arnd Voerste
Stefan Hillebrand
Stefan Herrmann
Ulrich Heinemann
Ronald Ebbert
Karl-Heinz Kuck
Peter Loesel
Ulrike Wachendorff-Neumann
Astrid Mauler-Machnik
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR0311538A publication Critical patent/BR0311538A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

"PIRAZOLOPIRIMIDINAS". A presente invenção refere-se a novas pirazolopirimidinas de fórmula: em que: R^ 1^, R^ 2^, R^ 3^, X^ 1^ e X^ 2^ são como definidos na presente descrição; um processo para preparação dessas substâncias e seu uso para o controle de organismos nocivos. A invenção refere-se ainda a novos intermediários de fórmulas: e e aos processos para sua preparação.
BR0311538-0A 2002-05-29 2003-05-16 Pirazolopirimidinas BR0311538A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10223917A DE10223917A1 (de) 2002-05-29 2002-05-29 Pyrazolopyrimidine
PCT/EP2003/005159 WO2004000844A1 (de) 2002-05-29 2003-05-16 Pyrazolopyrimidine und ihre verwendung zur bekämpfung von schädlichen organismen

Publications (1)

Publication Number Publication Date
BR0311538A true BR0311538A (pt) 2005-03-01

Family

ID=29432434

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0311538-0A BR0311538A (pt) 2002-05-29 2003-05-16 Pirazolopirimidinas

Country Status (20)

Country Link
US (1) US20060089499A1 (pt)
EP (1) EP1513843B1 (pt)
JP (1) JP2005533070A (pt)
KR (1) KR20050004234A (pt)
CN (1) CN1671709A (pt)
AT (1) ATE366253T1 (pt)
AU (1) AU2003240258A1 (pt)
BR (1) BR0311538A (pt)
CA (1) CA2487544A1 (pt)
DE (2) DE10223917A1 (pt)
DK (1) DK1513843T3 (pt)
ES (1) ES2289300T3 (pt)
IL (1) IL165348A0 (pt)
MX (1) MXPA04011824A (pt)
PL (1) PL373467A1 (pt)
PT (1) PT1513843E (pt)
RU (1) RU2331643C2 (pt)
UA (1) UA77546C2 (pt)
WO (1) WO2004000844A1 (pt)
ZA (1) ZA200409618B (pt)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1534712B1 (en) 2002-09-04 2007-05-16 Schering Corporation Pyrazolo[1,5-a]pyrimidine compounds as cyclin dependent kinase inhibitors
US7196078B2 (en) 2002-09-04 2007-03-27 Schering Corpoartion Trisubstituted and tetrasubstituted pyrazolopyrimidines as cyclin dependent kinase inhibitors
US7205308B2 (en) 2002-09-04 2007-04-17 Schering Corporation Trisubstituted 7-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors
US7119200B2 (en) 2002-09-04 2006-10-10 Schering Corporation Pyrazolopyrimidines as cyclin dependent kinase inhibitors
EP1534710B1 (en) 2002-09-04 2007-10-24 Schering Corporation Pyrazolopyrimidines as cyclin dependent kinase inhibitors
KR20050057072A (ko) 2002-09-04 2005-06-16 쉐링 코포레이션 사이클린 의존성 키나제 억제제로서의 피라졸로피리미딘
US7161003B1 (en) 2002-09-04 2007-01-09 Schering Corporation Pyrazolopyrimidines as cyclin dependent kinase inhibitors
WO2004022559A1 (en) 2002-09-04 2004-03-18 Schering Corporation Pyrazolopyrimidines as cyclin dependent kinase inhibitors
US8580782B2 (en) 2002-09-04 2013-11-12 Merck Sharp & Dohme Corp. Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors
US8673924B2 (en) 2002-09-04 2014-03-18 Merck Sharp & Dohme Corp. Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase inhibitors
KR20050115252A (ko) 2003-02-28 2005-12-07 데이진 화-마 가부시키가이샤 피라졸로[1,5-ａ]피리미딘 유도체
EP1608652A1 (en) * 2003-03-31 2005-12-28 Vernalis (Cambridge) Limited Pyrazolopyrimidine compounds and their use in medicine
CA2527136A1 (en) * 2003-06-03 2004-12-09 Basf Aktiengesellschaft Substituted pyrazolopyrimidines, methods for the production thereof, use of the same for controlling pathogenic fungi, and agents containing said compounds
KR20060027809A (ko) * 2003-06-27 2006-03-28 바이엘 크롭사이언스 아게 피라졸로피리미딘
DE10357565A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357568A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE10357567A1 (de) * 2003-12-10 2005-07-07 Bayer Cropscience Ag Pyrazolopyrimidine
DE102004008807A1 (de) 2004-02-20 2005-09-08 Bayer Cropscience Ag Pyrazolopyrimidine
EP1720879A2 (de) * 2004-02-25 2006-11-15 Basf Aktiengesellschaft Azolopyrimidin-verbindungen und ihre verwendung zur bekämpfung von schadpilzen
DE102005007534A1 (de) * 2005-02-17 2006-08-31 Bayer Cropscience Ag Pyrazolopyrimidine
BRPI0608712A2 (pt) * 2005-03-18 2010-12-07 Basf Ag processo para a preparação de composto, e, uso do composto
JP2007008864A (ja) * 2005-06-30 2007-01-18 Bayer Cropscience Ag ピラゾロピリミジン誘導体及び農園芸用殺菌剤
WO2007012599A1 (de) * 2005-07-27 2007-02-01 Basf Aktiengesellschaft Fungizide 5-methyl-6-phenyl-pyrazolopyrimidin-7-ylamine
CN101228170A (zh) * 2005-07-27 2008-07-23 巴斯福股份公司 杀真菌的5-烷基-6-苯基吡唑并嘧啶-7-基胺
CN101321760A (zh) 2005-10-06 2008-12-10 先灵公司 作为蛋白激酶抑制剂的吡唑并嘧啶
WO2007101804A1 (de) * 2006-03-07 2007-09-13 Basf Se Substituierte pyrazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
WO2007101859A1 (de) * 2006-03-07 2007-09-13 Basf Se Substituierte pyrazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
WO2008046856A2 (de) * 2006-10-18 2008-04-24 Basf Se Fungizide zusammensetzungen
WO2008084082A1 (de) * 2007-01-11 2008-07-17 Basf Se Verfahren zur herstellung arylsubstituierter anellierter pyrimidine
JP7179161B2 (ja) 2018-09-10 2022-11-28 イーライ リリー アンド カンパニー 乾癬および全身性エリテマトーデスの処置に有用なピラゾロ［１，５－ａ］ピリミジン－３－カルボキサミド誘導体
TWI800696B (zh) 2018-12-10 2023-05-01 美商美國禮來大藥廠 7-(甲基胺基)吡唑并[1,5-a]嘧啶-3-甲醯胺衍生物
CN110016036B (zh) * 2019-05-16 2022-06-03 辽宁大学 吡唑并[1,5-a]嘧啶类化合物及其制备方法和应用
AR121251A1 (es) 2020-02-12 2022-05-04 Lilly Co Eli Compuestos de 7-(metilamino)pirazolo[1,5-a]pirimidina-3-carboxamida
KR20230033708A (ko) * 2020-06-26 2023-03-08 니혼노야쿠가부시키가이샤 아릴테트라히드로피리다진 유도체 또는 그의 염류 및 해당 화합물을 함유하는 살충제 그리고 그 사용 방법
CN113287620B (zh) * 2021-06-18 2021-11-19 浙江大学 1H-吡唑并[3,4-d]嘧啶类化合物在制备禾谷镰刀菌杀菌剂中的应用
TW202342432A (zh) * 2021-12-28 2023-11-01 日商日本農藥股份有限公司 芳基四氫嗒𠯤衍生物或其鹽類及含有該化合物的殺蟲劑和其使用方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3130633A1 (de) * 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
US5817663A (en) * 1996-10-07 1998-10-06 American Cyanamid Company Pentafluorophenylazolopyrimidines
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
JP2001019693A (ja) * 1999-06-14 2001-01-23 American Cyanamid Co 殺菌・殺カビ性６−フェニル−ピラゾロピリミジン
US6552026B2 (en) * 1999-06-14 2003-04-22 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines

Also Published As

Publication number Publication date
RU2004139028A (ru) 2005-07-10
UA77546C2 (en) 2006-12-15
IL165348A0 (en) 2006-01-15
ZA200409618B (en) 2006-03-29
EP1513843A1 (de) 2005-03-16
PL373467A1 (en) 2005-09-05
KR20050004234A (ko) 2005-01-12
MXPA04011824A (es) 2005-03-31
CN1671709A (zh) 2005-09-21
US20060089499A1 (en) 2006-04-27
WO2004000844A1 (de) 2003-12-31
AU2003240258A1 (en) 2004-01-06
ATE366253T1 (de) 2007-07-15
JP2005533070A (ja) 2005-11-04
RU2331643C2 (ru) 2008-08-20
EP1513843B1 (de) 2007-07-04
DE10223917A1 (de) 2003-12-11
CA2487544A1 (en) 2003-12-31
PT1513843E (pt) 2007-09-26
ES2289300T3 (es) 2008-02-01
DE50307615D1 (de) 2007-08-16
DK1513843T3 (da) 2007-11-05

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A E 7A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 2064 DE 27/07/2010.