NO20065902L - 3-{4-(pyridin-3-yl)fenyl}-5-(1H-,1,2,3-triazol-1-ylmetyl)-1,3-oksazolidin-2-oner som antibakterielle midler - Google Patents
3-{4-(pyridin-3-yl)fenyl}-5-(1H-,1,2,3-triazol-1-ylmetyl)-1,3-oksazolidin-2-oner som antibakterielle midlerInfo
- Publication number
- NO20065902L NO20065902L NO20065902A NO20065902A NO20065902L NO 20065902 L NO20065902 L NO 20065902L NO 20065902 A NO20065902 A NO 20065902A NO 20065902 A NO20065902 A NO 20065902A NO 20065902 L NO20065902 L NO 20065902L
- Authority
- NO
- Norway
- Prior art keywords
- oxazolidin
- triazol
- ylmethyl
- pyridin
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Forbindelser med formel I, samt farmasøytisk akseptable salter og prodrugs derav, er beskrevet, hvor R1, R2, R3 og R4 er som definert heri. Også beskrevet er fremgangsmåter for fremstilling av forbindelser med formel I samt fremgangsmåter for anvendelse av forbindelser med formel I for behandling av bakterielle infeksjoner.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0411592A GB0411592D0 (en) | 2004-05-25 | 2004-05-25 | Chemical compounds |
GB0500053A GB0500053D0 (en) | 2005-01-05 | 2005-01-05 | Chemical compounds |
PCT/GB2005/002055 WO2005116023A1 (en) | 2004-05-25 | 2005-05-24 | 3- {4- (pyridin-3-yl) phenyl} -5- (1h-1, 2, 3-triazol-1-ylmethyl) -1, 3-oxazolidin-2-ones as antibacterial agents |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20065902L true NO20065902L (no) | 2007-02-20 |
Family
ID=34968777
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20065902A NO20065902L (no) | 2004-05-25 | 2006-12-19 | 3-{4-(pyridin-3-yl)fenyl}-5-(1H-,1,2,3-triazol-1-ylmetyl)-1,3-oksazolidin-2-oner som antibakterielle midler |
Country Status (9)
Country | Link |
---|---|
US (1) | US20080021071A1 (no) |
EP (1) | EP1753755A1 (no) |
JP (1) | JP2008500318A (no) |
AU (1) | AU2005247670A1 (no) |
BR (1) | BRPI0511524A (no) |
CA (1) | CA2567929A1 (no) |
IL (1) | IL179347A0 (no) |
NO (1) | NO20065902L (no) |
WO (1) | WO2005116023A1 (no) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100854211B1 (ko) | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
WO2010042887A2 (en) | 2008-10-10 | 2010-04-15 | Trius Therapeutics | Methods for preparing oxazolidinones and compositions containing them |
PE20120585A1 (es) | 2009-02-03 | 2012-06-13 | Trius Therapeutics | Forma cristalina del fosfato de dihidrogeno r)-3-(4-(2-(2-metiltetrazol-5-il) piridin-5-il)-3-fluorofensil)-5-hidroximetil oxazolidin-2-ona |
US8580767B2 (en) * | 2009-05-28 | 2013-11-12 | Trius Therapeutics, Inc. | Oxazolidinone containing dimer compounds, compositions and methods to make and use |
CN102260277B (zh) * | 2010-05-24 | 2013-07-24 | 中国科学院上海药物研究所 | 新型苯并噁嗪噁唑烷酮类化合物及其制备方法和用途 |
US9365530B2 (en) | 2012-05-07 | 2016-06-14 | The University Of North Carolina At Chapel Hill | Direct anti-markovnikov addition of acids to alkenes |
US10017441B2 (en) | 2013-05-02 | 2018-07-10 | The University Of North Carolina At Chapel Hill | Direct anti-markovnikov addition of acids to alkenes |
WO2016061772A1 (en) | 2014-10-22 | 2016-04-28 | Merck Sharp & Dohme Corp. | Nargenicin compounds and uses thereof as antibacterial agents |
EP3436434B1 (en) | 2016-03-31 | 2020-07-08 | Oncternal Therapeutics, Inc. | Indoline analogs and uses thereof |
AU2021292747A1 (en) | 2020-06-18 | 2023-02-23 | Akagera Medicines, Inc. | Oxazolidinone compounds, liposome compositions comprising oxazolidinone compounds and methods of use thereof |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5254577A (en) * | 1988-07-29 | 1993-10-19 | The Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
HUP0301562A2 (hu) * | 2000-06-05 | 2003-12-29 | Dong A Pharm. Co., Ltd. | Új oxazolidinonszármazékok és eljárás ezek előállítására, ezeket tartalmazó gyógyszerkészítmények |
KR20040087329A (ko) * | 2002-02-28 | 2004-10-13 | 아스트라제네카 아베 | 3-시클릴-5-(질소-함유 5-원 고리) 메틸-옥사졸리디논유도체 및 그의 항균제로서의 용도 |
KR20050084010A (ko) * | 2002-11-28 | 2005-08-26 | 아스트라제네카 아베 | 항균제로서의 옥사졸리디논 |
AR045690A1 (es) * | 2003-06-03 | 2005-11-09 | Rib X Pharmaceuticals Inc | Compuestos biaril heterociclicos y metodos para preparar y utilizar los mismos |
CA2529293A1 (en) * | 2003-07-02 | 2005-01-20 | Merck & Co., Inc. | Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof |
WO2005061468A1 (en) * | 2003-12-17 | 2005-07-07 | Rib-X Pharmaceuticals, Inc. | Halogenated biaryl heterocyclic compounds and methods of making and using the same |
-
2005
- 2005-05-24 JP JP2007514088A patent/JP2008500318A/ja active Pending
- 2005-05-24 CA CA002567929A patent/CA2567929A1/en not_active Abandoned
- 2005-05-24 BR BRPI0511524-8A patent/BRPI0511524A/pt not_active Application Discontinuation
- 2005-05-24 AU AU2005247670A patent/AU2005247670A1/en not_active Abandoned
- 2005-05-24 EP EP05746538A patent/EP1753755A1/en not_active Withdrawn
- 2005-05-24 WO PCT/GB2005/002055 patent/WO2005116023A1/en active Application Filing
- 2005-05-24 US US11/569,208 patent/US20080021071A1/en not_active Abandoned
-
2006
- 2006-11-16 IL IL179347A patent/IL179347A0/en unknown
- 2006-12-19 NO NO20065902A patent/NO20065902L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
US20080021071A1 (en) | 2008-01-24 |
JP2008500318A (ja) | 2008-01-10 |
EP1753755A1 (en) | 2007-02-21 |
IL179347A0 (en) | 2007-03-08 |
WO2005116023A8 (en) | 2007-01-11 |
BRPI0511524A (pt) | 2007-12-26 |
CA2567929A1 (en) | 2005-12-08 |
AU2005247670A1 (en) | 2005-12-08 |
WO2005116023A1 (en) | 2005-12-08 |
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Legal Events
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FC2A | Withdrawal, rejection or dismissal of laid open patent application |