BR0210016A - Heterociclos bicìclicos contendo nitrogênio, para uso como antibacterianos - Google Patents

Heterociclos bicìclicos contendo nitrogênio, para uso como antibacterianos

Info

Publication number
BR0210016A
BR0210016A BR0210016-9A BR0210016A BR0210016A BR 0210016 A BR0210016 A BR 0210016A BR 0210016 A BR0210016 A BR 0210016A BR 0210016 A BR0210016 A BR 0210016A
Authority
BR
Brazil
Prior art keywords
antibacterials
nitrogen
bicyclic heterocycles
containing bicyclic
derivatives
Prior art date
Application number
BR0210016-9A
Other languages
English (en)
Inventor
Gerald Brooks
David Thomas Davies
Graham Elgin Jones
Roger Edward Markwell
Neil David Pearson
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of BR0210016A publication Critical patent/BR0210016A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"HETEROCICLOS BICìCLICOS CONTENDO NITROGêNIO, PARA USO COMO ANTIBACTERIANOS". Descreve-se derivados de ciclo-hexano e ciclo-hexeno, e seus derivados de uso farmacêutico, úteis em métodos de tratamento de infecções bacterianas em mamíferos, particularmente humanos.
BR0210016-9A 2001-05-25 2002-05-24 Heterociclos bicìclicos contendo nitrogênio, para uso como antibacterianos BR0210016A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0112834.7A GB0112834D0 (en) 2001-05-25 2001-05-25 Medicaments
PCT/EP2002/005708 WO2003087098A1 (en) 2001-05-25 2002-05-24 Nitrogen-containing bicyclic heterocycles for use as antibacterials

Publications (1)

Publication Number Publication Date
BR0210016A true BR0210016A (pt) 2004-06-15

Family

ID=9915342

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0210016-9A BR0210016A (pt) 2001-05-25 2002-05-24 Heterociclos bicìclicos contendo nitrogênio, para uso como antibacterianos

Country Status (23)

Country Link
US (2) US7141564B2 (pt)
EP (1) EP1399443B1 (pt)
JP (2) JP4463565B2 (pt)
KR (1) KR20040010654A (pt)
CN (1) CN1535272A (pt)
AR (1) AR038172A1 (pt)
AT (1) ATE380812T1 (pt)
AU (1) AU2002367697A1 (pt)
BR (1) BR0210016A (pt)
CA (1) CA2448525A1 (pt)
CO (1) CO5540344A2 (pt)
CZ (1) CZ20033202A3 (pt)
DE (1) DE60224039T2 (pt)
ES (1) ES2298439T3 (pt)
GB (1) GB0112834D0 (pt)
HU (1) HUP0400017A2 (pt)
IL (1) IL158869A0 (pt)
MX (1) MXPA03010790A (pt)
NO (1) NO20035190D0 (pt)
PL (1) PL367079A1 (pt)
TW (1) TWI232219B (pt)
WO (1) WO2003087098A1 (pt)
ZA (1) ZA200308696B (pt)

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CN1535272A (zh) 2004-10-06
CZ20033202A3 (cs) 2004-08-18
EP1399443A1 (en) 2004-03-24
GB0112834D0 (en) 2001-07-18
JP2010031057A (ja) 2010-02-12
CO5540344A2 (es) 2005-07-29
AU2002367697A1 (en) 2003-10-27
ES2298439T3 (es) 2008-05-16
NO20035190D0 (no) 2003-11-21
MXPA03010790A (es) 2004-03-02
JP2005519981A (ja) 2005-07-07
ATE380812T1 (de) 2007-12-15
EP1399443B1 (en) 2007-12-12
DE60224039T2 (de) 2008-11-27
CA2448525A1 (en) 2003-10-23
KR20040010654A (ko) 2004-01-31
WO2003087098A1 (en) 2003-10-23
JP4463565B2 (ja) 2010-05-19
PL367079A1 (en) 2005-02-21
US20070135422A1 (en) 2007-06-14
TWI232219B (en) 2005-05-11
AR038172A1 (es) 2005-01-05
DE60224039D1 (de) 2008-01-24
IL158869A0 (en) 2004-05-12

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