BR0113776A - Composição de pirrolocarbazóis selecionados fundidos e método para tratar e prevenir várias doenças usando a citada composição - Google Patents
Composição de pirrolocarbazóis selecionados fundidos e método para tratar e prevenir várias doenças usando a citada composiçãoInfo
- Publication number
- BR0113776A BR0113776A BR0113776-0A BR0113776A BR0113776A BR 0113776 A BR0113776 A BR 0113776A BR 0113776 A BR0113776 A BR 0113776A BR 0113776 A BR0113776 A BR 0113776A
- Authority
- BR
- Brazil
- Prior art keywords
- composition
- various diseases
- treating
- fused pyrrolocarbazoles
- preventing various
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 4
- 201000010099 disease Diseases 0.000 title abstract 3
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title abstract 3
- QNMMYUBZGLXCCK-UHFFFAOYSA-N pyrrolo[3,2-a]carbazole Chemical class N1=C2C=CC=CC2=C2C1=C1C=CN=C1C=C2 QNMMYUBZGLXCCK-UHFFFAOYSA-N 0.000 title abstract 3
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- AIDS & HIV (AREA)
- Ophthalmology & Optometry (AREA)
Abstract
"COMPOSIçãO DE PIRROLOCARBAZóIS SELECIONADOS FUNDIDOS E MéTODO PARA TRATAR E PREVENIR VáRIAS DOENçAS USANDO A CITADA COMPOSIçãO". A presente invenção se relaciona geralmente com pirrolocarbazóis fundidos selecionados, incluindo composições farmacêuticas dos mesmos e métodos para tratar doenças com os mesmos. A presente invenção também é dirigida a intermediários e processos para produzir estes pirrolocarbazóis fundidos.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22780300P | 2000-08-25 | 2000-08-25 | |
US27845501P | 2001-03-23 | 2001-03-23 | |
US09/935,285 US6630500B2 (en) | 2000-08-25 | 2001-08-22 | Selected fused pyrrolocarbazoles |
PCT/US2001/026266 WO2002017914A2 (en) | 2000-08-25 | 2001-08-23 | Fused pyrrolocarbazoles against inflammation |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0113776A true BR0113776A (pt) | 2004-02-03 |
Family
ID=27397767
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0113776-0A BR0113776A (pt) | 2000-08-25 | 2001-08-23 | Composição de pirrolocarbazóis selecionados fundidos e método para tratar e prevenir várias doenças usando a citada composição |
Country Status (26)
Country | Link |
---|---|
US (3) | US6630500B2 (pt) |
EP (1) | EP1311263B1 (pt) |
JP (1) | JP5399598B2 (pt) |
KR (1) | KR100810190B1 (pt) |
CN (1) | CN1298323C (pt) |
AR (1) | AR034143A1 (pt) |
AT (1) | ATE306920T1 (pt) |
AU (1) | AU8520501A (pt) |
BG (1) | BG66103B1 (pt) |
BR (1) | BR0113776A (pt) |
CA (1) | CA2420592C (pt) |
CZ (1) | CZ303707B6 (pt) |
DE (1) | DE60114215T2 (pt) |
DK (1) | DK1311263T3 (pt) |
EA (1) | EA006371B1 (pt) |
ES (1) | ES2250463T3 (pt) |
HK (1) | HK1053989A1 (pt) |
HU (1) | HU230128B1 (pt) |
IL (2) | IL154590A0 (pt) |
MX (1) | MXPA03001562A (pt) |
NO (1) | NO325689B1 (pt) |
NZ (1) | NZ524288A (pt) |
PL (1) | PL212956B1 (pt) |
SK (1) | SK287498B6 (pt) |
TW (1) | TWI299731B (pt) |
WO (1) | WO2002017914A2 (pt) |
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KR101254371B1 (ko) | 2003-07-18 | 2013-05-02 | 암젠 프레몬트 인코포레이티드 | 간세포 성장인자에 결합하는 분리된 항체 |
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