BG108039A - Thiazolyl-, oxazolyl-, pyrrolyl- and amidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes - Google Patents

Thiazolyl-, oxazolyl-, pyrrolyl- and amidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes

Info

Publication number
BG108039A
BG108039A BG108039A BG10803903A BG108039A BG 108039 A BG108039 A BG 108039A BG 108039 A BG108039 A BG 108039A BG 10803903 A BG10803903 A BG 10803903A BG 108039 A BG108039 A BG 108039A
Authority
BG
Bulgaria
Prior art keywords
alkyl
inhibitors
given
formula
description
Prior art date
Application number
BG108039A
Other languages
Bulgarian (bg)
English (en)
Inventor
Anthony Marfat
Michael W. Mckechney
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG108039A publication Critical patent/BG108039A/xx

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
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    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
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  • Virology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
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  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • AIDS & HIV (AREA)
  • Otolaryngology (AREA)
  • Vascular Medicine (AREA)
  • Transplantation (AREA)
BG108039A 2001-01-31 2003-07-28 Thiazolyl-, oxazolyl-, pyrrolyl- and amidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes BG108039A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26548601P 2001-01-31 2001-01-31
PCT/IB2001/002728 WO2002060898A1 (en) 2001-01-31 2001-12-24 Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes

Publications (1)

Publication Number Publication Date
BG108039A true BG108039A (en) 2004-07-30

Family

ID=23010641

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108039A BG108039A (en) 2001-01-31 2003-07-28 Thiazolyl-, oxazolyl-, pyrrolyl- and amidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes

Country Status (24)

Country Link
US (3) US6559168B2 (es)
EP (1) EP1355907A1 (es)
JP (1) JP2004518691A (es)
KR (1) KR20030072614A (es)
CN (1) CN1489588A (es)
BG (1) BG108039A (es)
BR (1) BR0116850A (es)
CA (1) CA2436551A1 (es)
CR (1) CR7038A (es)
CZ (1) CZ20031903A3 (es)
EA (1) EA200300622A1 (es)
EC (1) ECSP034683A (es)
EE (1) EE200300362A (es)
HU (1) HUP0401305A2 (es)
IL (1) IL156412A0 (es)
IS (1) IS6844A (es)
MA (1) MA26985A1 (es)
MX (1) MXPA03006886A (es)
NO (1) NO20033398L (es)
OA (1) OA12542A (es)
PL (1) PL365443A1 (es)
TN (1) TNSN03050A1 (es)
WO (1) WO2002060898A1 (es)
ZA (1) ZA200305769B (es)

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