HUP0004477A2 - Herbicid hatású 3-(1,2-benzizotiazol- vagy-izoxazol-5-il)-csoporttal helyettesített pirimidinszármazékok, intermedierjeik, előállításuk és alkalmazásuk - Google Patents

Herbicid hatású 3-(1,2-benzizotiazol- vagy-izoxazol-5-il)-csoporttal helyettesített pirimidinszármazékok, intermedierjeik, előállításuk és alkalmazásuk

Info

Publication number
HUP0004477A2
HUP0004477A2 HU0004477A HUP0004477A HUP0004477A2 HU P0004477 A2 HUP0004477 A2 HU P0004477A2 HU 0004477 A HU0004477 A HU 0004477A HU P0004477 A HUP0004477 A HU P0004477A HU P0004477 A2 HUP0004477 A2 HU P0004477A2
Authority
HU
Hungary
Prior art keywords
group
atom
halogen atom
oxygen
alkyl
Prior art date
Application number
HU0004477A
Other languages
English (en)
Inventor
Sergio Ivan Alvarado
Keith Douglas Barnes
Billy Gene Bullock
Marianne Carlsen
Michael Vernie Cossette
Michael Anthony Guaciaro
Gregory Jay Haley
Gavin David Heffernan
David Allen Hunt
Mark Christopher Manfredi
Gary Allen Meier
Richard Anthony Rampulla
Peter John Wepplo
Original Assignee
American Cyanamid Co.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co. filed Critical American Cyanamid Co.
Publication of HUP0004477A2 publication Critical patent/HUP0004477A2/hu
Publication of HUP0004477A3 publication Critical patent/HUP0004477A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6536—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms
    • C07F9/6539—Five-membered rings
    • C07F9/6541—Five-membered rings condensed with carbocyclic rings or carbocyclic ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

A találmány szerinti vegyületek (I) és (II) általános képletében R jelentése alkil-, halogén-alkil-, cikloalkil-, alkenil-, alkinil-,benzilcsoport vagy -OR4 vagy -NR5R6 általános képletű csoport, R1, R2 jelentése hidrogén-, halogénatom, alkil-, cikloalkil-,alkenil-, alkinilcsoport, -OR7, S(O)nR8 vagy -NR9R10 általános képletűcsoport vagy R1 és R2 a közbezárt szénatomokkal telített vagytelítetlen gyűrűt alkot, amely heteroatomként oxigén-, kén vagynitrogén heteroatomot tartalmazhat, R3 jelentése halogénatom vagy oxigén- vagy kénatomon keresztülkapcsolódó hidrogénatom vagy szerves csoport, Z jelentése oxigénatom vagy S(O)m általános képletű csoport, Y jelentése halogénatom, cianocsoport, R12, X2R12, X3R12, X2X3R12 vagyX3X2R12 általános képletű csoport, X jelentése hidrogén-, halogénatom, alkilcsoport, X1 jelentése hidrogén-, halogénatom, adott esetben halogénatommalszubsztituált alkil- vagy alkoxicsoport, X2 jelentése oxigénatom, S(O)P vagy NR13 általános képletű csoport, X3 jelentése -C(=A3)-, -C(=NOR14)- vagy -C(=N-NR13R50)- általánosképletű csoport, R4, R5, R6, R7, R8, R9, R10 és R14 jelentésehidrogénatom, alkil-, cikloalkil-, alkoxi-alkil-, alkenil-, alkinil-vagy benzilcsoport, R12, R13 és R50 jelentése az 1. igénypontban megadott, A, A1, A3 jelentése egymástól függetlenül oxigén- vagy kénatom, p, m, n értéke 0, 1 vagy 2. Ó
HU0004477A 1997-09-17 1998-09-15 Herbicidal 3(-1,2-benzisothiazol or isoxazol-5 yl)-substituted pyrimidine derivatives, intermediates, preparation and use thereof HUP0004477A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93145197A 1997-09-17 1997-09-17
US12883198A 1998-08-04 1998-08-04

Publications (2)

Publication Number Publication Date
HUP0004477A2 true HUP0004477A2 (hu) 2001-02-28
HUP0004477A3 HUP0004477A3 (en) 2002-01-28

Family

ID=26826981

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0004477A HUP0004477A3 (en) 1997-09-17 1998-09-15 Herbicidal 3(-1,2-benzisothiazol or isoxazol-5 yl)-substituted pyrimidine derivatives, intermediates, preparation and use thereof

Country Status (24)

Country Link
EP (1) EP0908457B1 (hu)
JP (1) JP2001516758A (hu)
KR (1) KR20010030612A (hu)
CN (1) CN1273585A (hu)
AR (3) AR015168A1 (hu)
AT (1) ATE227721T1 (hu)
AU (2) AU737864B2 (hu)
BG (1) BG104336A (hu)
BR (1) BR9813017A (hu)
CA (1) CA2246221A1 (hu)
CZ (1) CZ2000861A3 (hu)
DE (1) DE69809370T2 (hu)
ES (1) ES2185118T3 (hu)
HU (1) HUP0004477A3 (hu)
IL (1) IL125947A0 (hu)
MX (1) MXPA00002661A (hu)
NZ (1) NZ331825A (hu)
PL (1) PL339350A1 (hu)
SK (1) SK3552000A3 (hu)
TR (1) TR200000679T2 (hu)
TW (1) TW474927B (hu)
WO (1) WO1999014216A1 (hu)
YU (1) YU15800A (hu)
ZA (1) ZA988435B (hu)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6140270A (en) * 1998-09-14 2000-10-31 American Cyanamid Company Process for the preparation of 6-(perfluoroalkyl) uracil compounds from 2-(N,N-disubstituted) amino-4-(perfluoroalkyl)-1,3-oxazin-6-one compounds
IL144776A0 (en) * 1999-02-16 2002-06-30 Basf Ag Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils
WO2001079203A1 (en) * 2000-04-17 2001-10-25 Basf Aktiengesellschaft Herbicidal 3-heterocyclic substituted benzisothiazole and benzisoxazole compounds
AU2001291836A1 (en) * 2000-09-08 2002-03-22 Basf Aktiengesellschaft Method for producing anellated tetrahydro-(1h)-triazoles
EP1446125B1 (en) 2001-08-30 2009-04-29 Alizyme Therapeutics Limited Thieno-(1,3)-oxazin-4-ones with lipase inhibiting activity
WO2003087072A1 (fr) * 2002-03-29 2003-10-23 Mochida Pharmaceutical Co., Ltd. Agent therapeutique destine a des troubles endotheliaux
KR101055954B1 (ko) 2002-10-30 2011-08-09 바스프 에스이 이관능성 페닐이소(티오)시아네이트, 그의 제조 방법 및그의 제조를 위한 중간체 생성물
ES2770550T3 (es) 2011-05-17 2020-07-02 Univ California Inhibidores de quinasa
CA2836410C (en) 2011-05-17 2019-08-20 Principia Biopharma Inc. Tyrosine kinase inhibitors
US9376438B2 (en) 2011-05-17 2016-06-28 Principia Biopharma, Inc. Pyrazolopyrimidine derivatives as tyrosine kinase inhibitors
PL2892900T3 (pl) 2012-09-10 2018-02-28 Principia Biopharma Inc. Związki pyrazolopirymidonowe jako inhibitory kinazy
US8957080B2 (en) 2013-04-09 2015-02-17 Principia Biopharma Inc. Tyrosine kinase inhibitors
DE102013226249A1 (de) * 2013-12-17 2015-06-18 Wacker Chemie Ag Polyetherreste aufweisende Organopolysiloxangele
JP6504548B2 (ja) 2014-02-21 2019-04-24 プリンシピア バイオファーマ インコーポレイテッド Ｂｔｋ阻害剤の塩および固体形態
CA2970723C (en) 2014-12-18 2023-09-05 Principia Biopharma Inc. Treatment of pemphigus
WO2016210165A1 (en) 2015-06-24 2016-12-29 Principia Biopharma Inc. Tyrosine kinase inhibitors
MX390619B (es) 2016-06-29 2025-03-21 Principia Biopharma Inc Formulaciones de liberacion modificada de 2-[3-[4-amino-3-(2-fluoro-4-fenoxi-fenil)pirazolo[3,4-d]pirimidin-1-il]piperidina-1-carbonil]-4-metil-4-[4-(oxetan-3-il)piperazin-1-il]pent-2-enenitrilo
EP3648605A1 (en) * 2017-07-03 2020-05-13 Bayer CropScience Aktiengesellschaft Novel isothiazolo-based bicycles, processes for their preparation and their use as herbicides and/or plant growth regulators
CN109776302A (zh) * 2017-11-13 2019-05-21 中国科学院化学研究所 一种由木质素为甲基源制备重要化学品的方法
CA3154257A1 (en) 2019-10-14 2021-04-22 Principia Biopharma Inc. Methods for treating immune thrombocytopenia by administering (r)-2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile
CN114276287B (zh) * 2021-12-27 2023-10-03 浙江工业大学 N-(取代苄氧基)酰胺类化合物及其制备方法和应用
CN116354953B (zh) * 2022-12-31 2024-07-16 西北农林科技大学 含苯并噻唑类化合物的除草组合物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU627906B2 (en) * 1989-07-14 1992-09-03 Nissan Chemical Industries Ltd. Uracil derivatives and herbicides containing the same as active ingredient
IL97102A0 (en) * 1990-02-16 1992-03-29 Ici Plc Heterocyclic compounds
US5484763A (en) * 1995-02-10 1996-01-16 American Cyanamid Company Substituted benzisoxazole and benzisothiazole herbicidal agents
US5753595A (en) * 1995-08-31 1998-05-19 Fmc Corporation Herbicidal 3-(substituted benzoxazol-7-yl) and 3-(Substituted benzothiazol-7-yl)-1-substituted-6-trifluoromethyl-2 4-(1h 3h)pyrimidinediones
BR9610772A (pt) * 1995-10-04 1999-07-13 Fmc Corp Composto composição herbicida e processos para preparação dos compostos e para o controle do crescimento de plantas indesejadas

Also Published As

Publication number Publication date
JP2001516758A (ja) 2001-10-02
TW474927B (en) 2002-02-01
BG104336A (en) 2001-09-28
SK3552000A3 (en) 2001-01-18
AU8423998A (en) 1999-04-01
DE69809370D1 (de) 2002-12-19
WO1999014216A1 (en) 1999-03-25
ES2185118T3 (es) 2003-04-16
ZA988435B (en) 2000-03-15
YU15800A (sh) 2002-11-15
AR021081A2 (es) 2002-06-12
BR9813017A (pt) 2000-08-15
EP0908457A1 (en) 1999-04-14
TR200000679T2 (tr) 2000-08-21
PL339350A1 (en) 2000-12-18
ATE227721T1 (de) 2002-11-15
AU737864B2 (en) 2001-08-30
CN1273585A (zh) 2000-11-15
IL125947A0 (en) 1999-04-11
KR20010030612A (en) 2001-04-16
AU9392598A (en) 1999-04-05
DE69809370T2 (de) 2003-03-27
MXPA00002661A (es) 2001-10-31
CZ2000861A3 (cs) 2000-08-16
CA2246221A1 (en) 1999-03-17
AR021500A2 (es) 2002-07-24
EP0908457B1 (en) 2002-11-13
HUP0004477A3 (en) 2002-01-28
NZ331825A (en) 2000-04-28
AR015168A1 (es) 2001-04-18

Similar Documents

Publication Publication Date Title
HUP0004477A2 (hu) Herbicid hatású 3-(1,2-benzizotiazol- vagy-izoxazol-5-il)-csoporttal helyettesített pirimidinszármazékok, intermedierjeik, előállításuk és alkalmazásuk
ATE353870T1 (de) Dibenzylaminverbindung und deren medizinische verwendung
IL147651A0 (en) Isoxazoline derivative and herbicide containing the same as the active ingredient
HUP0401335A2 (hu) Herbicid hatású [(piridil-propinil)-oxi]-fenil-származékok, előállításuk és alkalmazásuk
CY1105863T1 (el) Παραγωγα εποθιλονης και η συνθεση και η χρηση τους
ATE286026T1 (de) Amid-derivate und deren medizinische verwendung
NO972666L (no) Anilinderivater med nitrogenmonoksyd-synteseinhiberende aktivitet
EP1206937A4 (en) EXTERNAL NITROIMIDAZOLE PREPARATIONS FOR TREATING DERMATOSIS
HUP0004212A2 (hu) Inszekticid hatású szubsztituált aminokinazolinon(tion)-származékok, intermedierjeik, előállításuk és alkalmazásuk
MXPA02011417A (es) 1-aminoalquil-lactamas sustituidas y su uso como antagonistas de receptores muscarinicos.
BG104287A (en) Halogensubstituted tetracyclic derivatives of tetrahydrofuran
BG104853A (en) Thienylazolylalcoxyethanamines, their preparation and their application as medicaments
BR9509629A (pt) Derivados de aminotetrazol úteis como inibidores de óxido nítrico sintase
BR0308759A (pt) Derivados de fenil amidas siliconadas utilizáveis como microbiocida
EP1357124A4 (en) HETEROCYCLIC COMPOUNDS AND COMPOSITIONS IMPROVING CEREBRAL FUNCTIONS CONTAINING THESE AS ACTIVE INGREDIENTS
MXPA02011464A (es) Derivados 1,4-diazepan-2,5-diona y su uso como antagonistas del receptor de la nk-1.
ATE283840T1 (de) Chondrogonese promotoren und indolin-2-on derivate
DE60037766D1 (de) Verfahren zur Herstellung von 2-Alkyl-3-aminothiophen Derivate und 3-Aminothiophen Derivate
HUP9700983A2 (hu) 1,4-Diaril-2-fluor-2-butén-származékok, intermedierjeik, előállításuk és alkalmazásuk, valamint hatóanyagként ezeket a vegyületeket tartalmazó inszekticid és akaricid készítmények
HUP0001009A2 (hu) Herbicid hatású 3-karbamoil/3-tiokarbamoil-szubsztituált 2-benzoil-ciklohexán-1,3-dionok, intermedierjeik, előállításuk és alkalmazásuk
ATE397609T1 (de) Corticotropinfreisetzungsfaktor antagonisten
ATE229538T1 (de) 22r-hydroxycholesta-8,14-diene derivate zur hemmung der meiose
TW200504071A (en) 7-(alkenylamino)triazolopyrimidines, their preparation and their use in the control of harmful fungi, and preparations comprising them
DE69832614D1 (de) Benzopyranderivate zur behandlung von perihperer gefässerkrankung
DE69124017D1 (de) Heterocyclische Derivate