CN1273585A - 作为除草剂的取代的3－(1,2－苯并异噻唑或异噁唑－5－基)－取代的嘧啶 - Google Patents

作为除草剂的取代的3－(1,2－苯并异噻唑或异噁唑－5－基)－取代的嘧啶 Download PDF

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CN1273585A
CN1273585A CN98809898A CN98809898A CN1273585A CN 1273585 A CN1273585 A CN 1273585A CN 98809898 A CN98809898 A CN 98809898A CN 98809898 A CN98809898 A CN 98809898A CN 1273585 A CN1273585 A CN 1273585A
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比得·约翰·威普洛
马克·克里斯多夫·曼费迪
里查·安东尼·瑞普拉
麦克·佛奈·寇司提
麦克·安东尼·栝夏若
桂葛瑞·杰·海力
比利·金·布拉克
瑟吉奥·艾芬·欧法拉度
凯斯·道格拉斯·巴尼司
盖瑞·艾伦·梅尔
大卫·艾伦·杭特
玛利安·卡尔森
卡芬·大卫·海佛南
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Wyeth Holdings LLC
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American Cyanamid Co
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Abstract

本发明提供了式(Ⅰ)3－(1,2－苯并异噻唑—和异噁唑－5－基)－2,4－(1H,3H)－嘧啶二酮或硫酮化合物,及式Ⅱ3－(1,2－苯并异噻唑和异噁唑－5－基)－4(3H)－嘧啶酮或硫酮化合物。本发明进一步提供了用于防治不需要植物种类的包含这些化合物的组合物和方法。

Description

作为除草剂的取代的3-(1，2-苯并异噻唑或异噁唑-5-基)- 取代的嘧啶
发明背景
杂草因减少作物收成及降低作物品质而致全球经济损失。全球农作物必须与数百种杂草品种竞争。
尽管目前已有除草剂商品，但因杂草而损害作物的情形仍旧发生。因此仍需研究开发更有效和/或更具选择性的除草剂。
某些苯并异噁唑及苯并异噻唑除草剂已在美国专利Nos.5,484,763及5,523,278中加以说明。这些专利总的揭示了被22个特定基团之一的Q基团取代的苯并异噁唑及苯并异噻唑化合物。然而这些专利仅例举了一个Q基团(Q6)。此外，这些专利案并未揭示它们的化合物适用于在玉米和小麦存在下选择性地控制杂草。
现已惊人地发现，这些专利所一般揭示的某些化合物与其中Q为Q6的相应化合物相比是更有效和/或更具选择性的除草剂。
因此本发明的一个目的是提供对不要的植物品种能高度有效进行控制的化合物。
本发明另一个目的为控制不要的植物品种的方法。
本发明再一个目的是提供在作物的存在下选择性地控制不要的植物品种的方法。
本发明这些和其他目的与特征可由下文详细说明中作进一步了解。
发明概述
本发明揭示了用作除草剂的3-(1，2-苯并异噻唑-和异噁唑-5-基)-2，4(1H，3H)-嘧啶二酮或硫酮及3-(1，2-苯并异噻唑-和异噁唑-5-基)-4(3H)-嘧啶酮或硫酮化合物。
本发明化合物是由结构式I及II代表的化合物及其光学异构体，非对映异构体和/或互变异构体
Figure A9880989800621
其中
R为C1-C6烷基，C1-C6卤代烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR4或NR5R6；
R1与R2分别为氢，卤素，C1-C6烷基，C3-C7环烷基，C1-C6卤代烷基，C3-C6烯基，C3-C6卤代烯基，C3-C6炔基，OR7，S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，它们代表任选地被氧，硫或氮隔开，并任选地被1-3个甲基或一个或多个卤原子取代的4-到7-元饱和或不饱和环；
R3为卤素或A2R11；
X为氢，卤素或C1-C4烷基；
X1为氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素，氰基，R12，X2R12，X3R12，X2X3R12或X3X2R12；
X2为O，S(O)p或NR13；
X3为-C(＝A3)-，-C(＝NOR14)-或-C(＝N-NR13R50)；
R4，R5，R6，R7，R8，R9，R10，R11与R14分别为氢，C1-C6烷基，C3-C7环烷基，C2-C8烷氧基烷基，C2-C6烯基，C2-C6炔基或苄基；
R12为氢，
C1-C8烷基，C3-C7环烷基，C2-C8烯基，C5-C6环烯基或C2-C8炔基，其中各基团任选地被下列任何组合取代：1至6个卤原子，1至3个C1-C20烷氧基(它们可任选地被一个C1-C6烷氧基，苄氧基或C1-C6烷硫基取代)，1或2个C1-C10卤代烷氧基，1或2个NR15R16基团，1至3个S(O)qR17基团，1或2个氰基，1或2个C3-C7环烷基，1个硫氰基，1个O(SO2)R17基团，1个O(NO2)基团，1或2个C(O)R18基团，1或2个CO2R19基团，1或2个C(O)SR19基团，1或2个C(O)NR20R21基团，1至3个X4R22基团，1或2个P(O)(OR23)2基团，1或2个Si(R24)3基团，
1个4至10元单环或稠合双环、杂环(它任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1或2个苯基，其中每个苯基独立任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C3-C7环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团或1个X5R27基团，
任选地被下列任何组合取代的苯基：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基，1个C3-C6环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，或
任选地被下列任何组合取代的茚满：1或2个卤原子，1或2个C1-C4烷基，1个C1-C4烷氧基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，它们形成了任选地被一个或多个独立地选自卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基，或X4R22基团取代的5至12元单环或稠合双环、杂环；
R13为氢，C1-C8烷氧基烷基，C1-C6烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR23，氰基，SO2R51或1个任选地被一个或多个独立地选自卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基的基团取代的一个5至12元单环或稠合双环杂环；当R13及R12和它们所连接的氮原子结合在一起时，它们形成了任选地被一个或多个独立地选自卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团取代的5至12元单环或稠合双环、杂环；
R28为卤素；
R22与R27分别为氢，Si(R31)3，C(O)NR35R36，C(O)R33，SO2R47，
C1-C20烷基，它被下列基团取代：一个羟基，苄氧基，硝基，OC(O)R33，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，P(O)(OH)NH2，P(O)(OH)(OR23)，C(O)NR35OR23，氰基或2-二氧戊环基，
1个苯基，二氢呋喃酮或呋喃酮环，其中每个可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
任选地被一个或多个独立地选自卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基的基团取代的一个5至12元单环或稠合双环、杂环，
C3-C20烯基，它可任选地被下列基团取代：1至3个卤原子，1个羟基，1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中每个环可任选地被下列任何组合所取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它可任选地被下列基团取代：一个羟基，C1-C6烷氧基，C1-C4烷基，C2-C4烯基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环所取代，其中每个环任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个羟基，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中每个环任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，
苄基，它的苯环上任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团，或
4至10元杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个CO2R26基团，
C(O)R43，或
CO2R42；
R16与R21分别为氢，C1-C6烷基，C1-C4烷氧基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17，R18，R25，R30，R33，R45及R51分别为NR46R48，
-N＝CR46R48，C1-C8烷基，它可任选地被一个C1-C6烷氧基，噻吩或呋喃基取代，C1-C6卤代烷基，C3-C8环烷基，CO2R23，C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团，或
5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R19及R26分别为氢，C1-C20烷基，C1-C8卤代烷基，C3-C7环烷基，C3-C7卤代环烷基，C3-C20烯基，C3-C8卤代烯基，C5-C8环烯基，C5-C8卤代环烯基，C3-C8炔基，C3-C8卤代炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它可任选地被一个CO2R48，C1-C6烷氧基，C1-C6硫代烷基，C2-C20烷氧基烷氧基，苯基，OSi(R47)3，OC(O)R33，C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它可任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它可任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它可任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
2-，3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基，呋喃基，噻吩基，四氢呋喃基，C3-C8环烷基，二噁烷或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢，氰基，C1-C6烷基，SO2R51或苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50和它们所连接的氮原子结合在一起时，可为5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
m，n，p与q分别为0，1或2之整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R24，R31，R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R23，R39，R40，R42，R43，R44，R46及R48分别为氢，C2-C6烯基，C3-C8环烷基，
C1-C8烷基，它可任选地被一或二个C1-C4烷氧基取代；
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，且
当R46与R48及其所连接的原子结合在一起时，它们形成了5至12元单环或稠合双环、杂环或环烷基环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；及
A，A1，A2，A3，A4，X4及X5分别为O或S。
本发明也涉及含有这些化合物的组合物，及使用这些化合物及组合物的方法。已有利地发现本发明化合物和含所述化合物的组合物适用于控制不需要的植物品种。本发明化合物特别适用于在作物存在下选择性地控制不需要的植物品种。
发明详述
本发明提供一种控制不需要的植物品种的方法，该方法包括向所述植物的叶部或向含其种子或其他繁殖器官的土壤或水中施用除草有效量的式I 3-(1，2-苯并异噻唑-或异噁唑-5-基)-2，4-(1H，3H)-嘧啶二酮或硫酮化合物或式II 3-(1，2-苯并异噻唑-或异噁唑-5-基)-4(3H)-嘧啶酮或硫酮化合物。
本发明的除草化合物由结构式I及II代表其中R，R1，R2，R3，A，A1，X，X1，Y及Z均如上述式I与II的定义。
现已惊人地发现，本发明式I与II化合物与美国专利Nos.5,484,763及5,523,278中例举之相应化合物(其中Q为Q6)相比是更有效和/或更具选择性的除草剂。此外，我们已发现本发明式I化合物特别适用于在作物如：玉米，小麦，稻及大豆的存在下选择性地控制不需要的植物品种。
本发明优选化合物为这些由结构式I及II代表的化合物：
Figure A9880989800682
其中
R为C1-C6烷基，C1-C6卤代烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR4或NR5R6；
R1与R2分别为氢，卤素，C1-C6烷基，C3-C7环烷基，C1-C6卤代烷基，C3-C6烯基，C3-C6卤代烯基，C3-C6炔基，OR7，S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，它们代表4至7元饱和或不饱和环，它们可任选地穿插氧，硫或氮，且可任选地被一至三个甲基或一个或多个卤原子取代；
R3为卤素或A2R11；
X为氢，卤素或C1-C4烷基；
X1为氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素，氰基，R12，X2R12，X3R12，X2X3R12或X3X2R12；
X2为O，S(O)p或NR13；
X3为-C(＝A3)-或-C(＝NOR14)-；
R4，R5，R6，R7，R8，R9，R10，R11与R14分别为氢，C1-C6烷基，C3-C7环烷基，C2-C6烯基，C2-C6炔基或苄基；
R12为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基，C5-C6环烯基或C2-C6炔基，其中各基团可任选地被下列任何组合取代：1至6个卤原子，1至3个C1-C20烷氧基，1或2个C1-C10卤代烷氧基，1或2个NR15R16基团，1至3个S(O)qR17基团，1或2个氰基，1或2个C(O)R18基团，1或2个CO2R19基团，1或2个C(O)NR20R21基团，1至3个X4R22基团，1或2个P(O)(OR23)2基团，1或2个Si(R24)3基团，
1个4至10元杂环(它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C3-C7环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团或1个X5R27基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基，1个C3-C6环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
当R12与R13及其所连接的氮原子结合在一起时，它们形成了5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基，或X4R22基团；
R13为氢，C1-C6烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR23，氰基或SO2R51，且当R13及R12及其所连接的氮原子结合在一起时，它们形成了5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢，Si(R31)3，
C1-C20烷基，它被下列基团取代：一个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，P(O)(OH)NH2，P(O)(OH)(OR23)，C(O)NHOR23，氰基或2-二氧戊环基，
1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，或C1-C4卤代烷基磺酰基，
C3-C20烯基，它可任选地被下列基团取代：1至3个卤原子，1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NHOR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它可任选地被下列基团取代：一个C1-C6烷氧基，C1-C4烷基，C2-C4烯基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NHOR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它可任选地被下列基团取代：1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NHOR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，
苄基，其在苯环上可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团，或
4至10元杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
C(O)R43，
R16与R21分别为氢，C1-C6烷基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17，R18，R25，R30，R33，R45及R51分别为C1-C4烷基，C1-C4卤代烷基，CO2R23，C2-C6烯基，它们可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团，或
5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R19与R26分别为氢，C1-C20烷基，C1-C8卤代烷基，C3-C7环烷基，C3-C7卤代环烷基，C3-C20烯基，C3-C8卤代烯基，C5-C8环烯基，C5-C8卤代环烯基，C3-C8炔基，C3-C8卤代炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它可任选地被一个CO2R48，C1-C6烷氧基，或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，
C3-C8卤代环烷基，
C3-C20烯基，它可任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它可任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
2-，3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它可被一个吡啶基，呋喃基，噻吩基，四氢呋喃基或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢，氰基，C1-C6烷基，SO2R51或苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50及所连接的氮原子结合在一起时，可为5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
m，n，p与q分别为0，1或2之整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R24，R31，R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R23，R39，R40，R42，R43，R44，R46及R48分别为氢，C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，且
A，A1，A2，A3，A4，X4及X5分别为O或S；
及其光学异构体，非对映异构体和/或互变异构体。
本发明另一类较佳化合物为有结构式I的化合物：
Figure A9880989800731
其中
R为C1-C6烷基，C1-C6卤代烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR4或NR5R6；
R1与R2分别为氢，卤素，C1-C6烷基，C3-C7环烷基，C1-C6卤代烷基，C3-C6烯基，C3-C6卤代烯基，C3-C6炔基，OR7，S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它们可任选地穿插氧，硫或氮，且可任选地被一至三个甲基或一个或多个卤原子取代；
X为氢，卤素或C1-C4烷基；
X1为氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素，氰基，R12，X2R12，X3R12，X2X3R12或X3X2R12；
X2为O，S(O)p或NR13；
X3为-C(＝A3)-，-C(＝NOR14)-或-C(＝N-NR13R50)；
R4，R5，R6，R7，R8，R9，R10与R14分别为氢，C1-C6烷基，C3-C7环烷基，C2-C8烷氧基烷基，C2-C6烯基，C2-C6炔基或苄基；
R12为氢，
C1-C8烷基，C3-C7环烷基，C2-C8烯基，C5-C6环烯基或C2-C8炔基，其中各基团可任选地被下列任何组合取代：1至6个卤原子，1至3个C1-C20烷氧基(它们可任选地被一个C1-C6烷氧基，苄氧基或C1-C6烷硫基取代)，1或2个C1-C10卤代烷氧基，1或2个NR15R16基团，1至3个S(O)qR17基团，1或2个氰基，1或2个C3-C7环烷基，1个硫氰基，1个O(SO2)R17基团，1个O(NO2)基团，1或2个C(O)R18基团，1或2个CO2R19基团，1或2个C(O)SR19基团，1或2个C(O)NR20R21基团，1至3个X4R22基团，1或2个P(O)(OR23)2基团，1或2个Si(R24)3基团，
1个4至10元单环或稠合双环、杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1或2个苯基，其中各苯基分别可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C3-C7环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团或1个X5R27基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基，1个C3-C6环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，或
茚满基，它可任选地被下列任何组合取代：1或2个卤原子，1或2个C1-C4烷基，1个C1-C4烷氧基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，它们形成了可任选地被一个或多个分别选自下列之基团取代的5至12元单环或稠合双环、杂环：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基，或X4R22基团；
R13为氢，C1-C8烷氧基烷基，C1-C6烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR23，氰基，SO2R51或1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基，且当R13及R12及其所连接的氮原子结合在一起时，形成了5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢，Si(R31)3，C(O)NR35R36，C(O)R33，SO2R47，
C1-C20烷基，它被下列基团取代：一个羟基，苄氧基，硝基，OC(O)R33，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，P(O)(OH)NH2，P(O)(OH)(OR23)，C(O)NR35OR23，氰基或2-二氧戊环基，
1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基，
C3-Cx烯基，它可任选地被下列基团取代：1至3个卤原子，1个羟基，1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它可任选地被下列基团取代：一个羟基，C1-C6烷氧基，C1-C4烷基，C2-C4烯基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它可任选地被下列基团取代：1个羟基，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它们可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，
苄基，其苯环上可任选地经下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团，或
4至10元杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个CO2R26基团，
C(O)R43，或
CO2R42；
R16与R21分别为氢，C1-C6烷基，C1-C4烷氧基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17，R18，R25，R30，R33，R45及R51分别为NR46R48，
-N＝CR46R48，C1-C8烷基，它可任选地被一个C1-C6烷氧基，噻吩或呋喃基取代，C1-C6卤代烷基，C3-C8环烷基，CO2R23，C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团，或
5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R19及R26分别为氢，C1-C20烷基，C1-C8卤代烷基，C3-C7环烷基，C3-C7卤代环烷基，C3-C20烯基，C3-C8卤代烯基，C5-C8环烯基，C5-C8卤代环烯基，C3-C8炔基，C3-C8卤代炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它可任选地被一个CO2R48，C1-C6烷氧基，C1-C6硫烷基，C2-C20烷氧基烷氧基，苯基，OSi(R47)3，OC(O)R33，C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它可任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它可任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它可任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
2-，3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基，呋喃基，噻吩基，四氢呋喃基，C3-C8环烷基，二噁烷或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢，氰基，C1-C6烷基，SO2R51或苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
m，n，p与q分别为0，1或2之整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R24，R31，R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R23，R39，R40，R42，R43，R44，R46及R48分别为氢，C2-C6烯基，C3-C8环烷基，
C1-C8烷基，它可任选地被一或二个C1-C4烷氧基取代；
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，且
当R46与R48及其所连接的原子结合在一起时，形成了5至12元单环或稠合双环、杂环或环烷基环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；及
A，A1，A3，A4，X4及X5分别为O或S；
及其光学异构体，非对映异构体和/或互变异构体。
本发明更优选的式I除草剂为式中：
R为C1-C4烷基，C1-C4卤代烷基，C3-C4烯基，C3-C4炔基或苄基；
R1为卤素或C1-C4卤代烷基；
R2为氢，卤素或C1-C4卤代烷基；
X与X1分别为氢或卤素；
Z为O或S；
Y为氰基，R12，X2R12或X3X2R12；
X2为O，S或NR13；
X3为-C(＝A3)-，-C(＝NOR14)或-C(＝N-NR13R50)；
R12为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基，C5-C6环烯基或C2-C6炔基，其中各基团可任选地被下列任何组合取代：1至3个卤原子，1或2个C1-C20烷氧基，1或2个C1-C10卤代烷氧基，1个NR15R16基团，1个S(O)qR17基团，1或2个氰基，1或2个C(O)R18基团，1或2个CO2R19基团，1或2个C(O)SR19基团，1或2个C(O)NR20R21基团，1或2个X4R22基团，1个P(O)(OR23)2基团，1个Si(R24)3基团，
1个4至10元单环或稠合双环、杂环(它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它可任选地被下列任何组合取代：1至3个卤原子，1个C1-C6烷基，1个C1-C6烷氧基，1个C3-C7环烷基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团或1个X5R27基团，
苯基，它可任选地被下列任何组合取代：1或2个卤原子，1至3个C1-C4烷基，1或2个C1-C4烷氧基，1个C3-C6环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团；
R13为氢，C2-C6烷氧基烷基，C1-C4烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR23，氰基或SO2R51；
R28为卤素；
R22与R27分别为氢，Si(R31)3，C(O)NR35R36，C(O)R33，SO2R47，
C1-C20烷基，它被下列基团取代：一个羟基，苄氧基，硝基，OC(O)R33，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，P(O)(OH)NH2，P(O)(OH)(OR23)，C(O)NR35OR23，氰基或2-二氧戊环基，
1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，或C1-C4卤代烷基磺酰基，
C3-C20烯基，它可任选地被下列基团取代：1至3个卤原子，1个羟基，1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它可任选地被下列基团取代：一个羟基，C1-C6烷氧基，C1-C4烷基，C2-C4烯基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它可任选地被下列基团取代：1个羟基，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它们可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，
苄基，其苯环上可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团，或
4至10元杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个CO2R26基团，
C(O)R43，或
CO2R42；
R14为氢，C1-C6烷基，C3-C7环烷基，C2-C8烷氧基烷基，C2-C6烯基，C2-C6炔基或苄基；
R16与R21分别为氢，C1-C6烷基，C1-C4烷氧基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R17，R18，R25，R30，R33，R45及R51分别为NR46R48，
-N＝CR46R48，C1-C8烷基，它可任选地被一个C1-C6烷氧基，噻吩或呋喃基取代，C1-C6卤代烷基，C3-C8环烷基，CO2R23，C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团，或
5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R19与R26分别为氢，C1-C20烷基，C1-C8卤代烷基，C3-C7环烷基，C3-C7卤代环烷基，C3-C20烯基，C3-C8卤代烯基，C5-C8环烯基，C5-C8卤代环烯基，C3-C8炔基，C3-C8卤代炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
C1-C20烷基，它可任选地被一个CO2R48，C1-C6烷氧基，C1-C6硫烷基，C2-C20烷氧基烷氧基，苯基，OSi(R47)3，OC(O)R33，C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它可任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它可任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它可任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
C1-C4烷基，它被一个吡啶基，呋喃基，噻吩基，四氢呋喃基，C3-C8环烷基，二噁烷或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢，氰基，C1-C6烷基，SO2R51或可任选地被一个或多个分别选自下列之基团取代的苯基：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，形成了5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
q为0，1或2之整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R24，R31，R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R23，R39，R40，R42，R43，R44，R46及R48分别为氢，C2-C6烯基，C3-C8环烷基，
C1-C8烷基，它可任选地被一或二个C1-C4烷氧基取代；
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，且
A，A1，A3，A4，X4及X5分别为O或S；
及其光学异构体，非对映异构体和/或互变异构体。
另一类更优选的式I除草剂为式中：
R为C1-C4烷基；
R1为C1-C4卤代烷基；
R2为氢；
X与X1分别为氢或卤素；
Z为O或S；
Y为R12，OR12，C(O)NR13R12，C(O)R12，CO2R12，C(O)SR12或C(＝NOR14)；
R12为氢，
C1-C6烷基或C2-C6烯基，其中各基团可任选地被下列任何组合取代：1至3个卤原子，1或2个C1-C4烷氧基，1个C1-C10卤代烷氧基，1个NR15R16基团，1个S(O)qR17基团，1或2个氰基，1或2个C(O)R18基团，1或2个CO2R19基团，1或2个C(C)NR20R21基团，1个X4R22基团，1个P(O)(OR23)2基团，1个OC(O)R33基团，
1个咪唑环，它们可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
1个邻苯二甲酰亚胺环，它们可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
1个四元有机铵基团，或
1个苯基，它可任选地被下列任何组合取代：1至3个卤原子，1个C1-C4烷基，1个C1-C4烷氧基或1个X5R27基团，或
苯基，它可任选地被下列任何组合取代：1或2个卤原子，1至3个C1-C4烷基，1个C1-C4烷氧基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团或1个N(R29)SO2R30基团；
R13为氢，C1-C6烷氧基烷基，C1-C4烷基，OR23，氰基或SO2R51；
R28为卤素；
R22与R27分别为氢，C(O)R33，SO2R47，
被下列基团取代的C1-C4烷基：一个C1-C6烷氧基，CO2R32，C(O)R33，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NHOR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C6烯基，它可任选地被1个C1-C6烷氧基，CO2R32，C(O)R33或C(OR34)2基团取代，
C3-C6炔基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1或2个C1-C4烷基，1或2个C1-C4烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，或
苄基，其苯环上可任选地被下列任何组合取代：1至3个卤原子，1或2个C1-C4烷基，1或2个C1-C4烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团；
R20为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个CO2R26基团，
C(O)R43，或
CO2R42；
R14为氢，C1-C6烷基，C3-C7环烷基，C3-C8烷氧基烷基，C2-C6烯基，C2-C6炔基或苄基；
R15为氢，
C1-C4烷基，它可任选地被1个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
C(O)R43；
R16为氢，C1-C4烷基，P(O)(OR44)2，SO2R45，C(O)R46，或
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R21为氢，C1-C6烷基，C1-C4烷氧基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R17，R18，R25，R30，R33，R45及R51分别为NR46R48，C1-C4烷基，C1-C4卤代烷基，
C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团；
R19与R26分别为氢，C1-C4烷基，C3-C6烯基，C3-C6炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
C1-C4烷基，它可任选地被一个CO2R48，OC(O)R33或C1-C4烷氧基取代，
C1-C4卤代烷基，
C3-C8环烷基，
C3-C8卤代环烷基，
C3-C6烯基，它可任选地被一个苯基取代，
C3-C6卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C6炔基，它可任选地被一个苯基取代，
C3-C6卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
C1-C4烷基，它被一个吡啶基，呋喃基，噻吩基，四氢呋喃基，或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C4烷基，且R36与R50分别为氢，氰基，C1-C4烷基，SO2R51或苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
q为0，1或2之整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R39，R40，R42，R43，R44，R46及R48分别为氢，C2-C6烯基，C3-C8环烷基，
C1-C8烷基，它可任选地被一或二个C1-C4烷氧基取代；
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
A1，X4及X5分别为O或S；
R23为氢或C1-C4烷基；且
A为O。
第三类更优选的式I除草剂为式中：
R为甲基；
R1为三氟甲基；
R2与X1为氢；
X为氢或氟；
Z为O或S；
Y为R12，CO2R12，C(O)R12或C(O)NR13R12；
R12为氢，
C1-C6烷基，它可任选地被下列任何组合取代：1至3个卤原子，1个羟基，1或2个C1-C4烷氧基，1个C1-C4卤代烷氧基，1个SO2R17基团，1或2个氰基，1个C(O)R18基团，1或2个CO2R19基团，1或2个C(O)NR20R21基团，1个P(O)(OR23)2基团或1个OC(O)R33基团，
C2-C6烯基，它可任选地被下列任何组合取代：1个C(O)R18基团或1个CO2R19基团，
Figure A9880989800881
R13为氢，C1-C4烷基或SO2R51；
R14为氢，C1-C4烷基或苄基；
R18，R23，R56及R57分别为氢或C1-C3烷基；
R52，R53，R54及R55分别为氢，C1-C3烷基，C2-C3烯基，C1-C3烷氧基或卤素，但其限制条件为R52，R53，R54及R55中至少一个为氢；
R19为氢，C1-C4烷基，C3-C6烯基，C3-C6炔基，苄基，吡啶基或碱金属，碱土金属，铵或有机铵阳离子；
R20为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个CO2R26基团，
C(O)R43，或
CO2R42；
R21为氢，C1-C6烷基，C1-C4烷氧基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R22为氢，C(O)R33，SO2R47，
C1-C4烷基，它可任选地被一个氰基取代，
C3-C6烯基，或
C3-C6炔基；
R32为氢，
C1-C4烷基，它可任选地被一个CO2R48或C1-C4烷氧基取代，
C1-C4卤代烷基，
C3-C6烯基，它可任选地被1个苯基取代，
C3-C6炔基，它可任选地被1个苯基取代，
C1-C4烷基，它被1个吡啶基，呋喃基，噻吩基，四氢呋喃基或NR49R50基团取代，或
碱金属，碱土金属，铵或有机铵阳离子；
R35及R49分别为氢或C1-C4烷基；
R36为SO2R51或C1-C3烷氧基；
R17，R33及R51分别为C1-C4烷基，C1-C4卤代烷基，NR46R48，C3-C6环烷基或异噁唑环；
R45为NR46R48，C1-C4烷基，C1-C4卤代烷基，
C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团；
R26为氢，C1-C4烷基，C3-C6烯基，C3-C6炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R41为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R42，R43及R44分别为氢，
C2-C6烯基，C3-C8环烷基，
C1-C8烷基，它可任选地被1个或2个C1-C4烷氧基取代，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
X4为O或S；
R46与R48分别为氢，C1-C4烷基或苄基；
R47为C1-C4烷基；
R50为C1-C4烷基或
苯基，它可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；及
A与A1为O。
本发明之最佳式I化合物为这些化合物，其中：
R为甲基；
R1为三氟甲基；
R2与X1为氢；
X为氢或氟；
Z为O或S；
Y为C1-C3烷基，CO2R32，卤代甲基，氰基甲基，C(CH3)2CO2R32，C1-C3烷氧基乙基，C1-C3烷氧基甲基，羟甲基，CHO，C(O)CH3，CH(CH3)(C1-C4烷氧基)，C(CH3)2CN，CH[O(C1-C3烷基)]2，CH2SO2R17，C(O)NHSO2R51，
R53，R54，R55及R56分别为氢或甲基，但其限制条件为R53，R54及R55中至少一个为氢；
R22为氰基甲基，甲基，乙基，烯丙基，或炔丙基；
R32为氢，
C1-C4烷基，它可任选地被1个CO2R48基团取代，
C1-C4卤代烷基，
C3-C6烯基，或
C3-C6炔基；
R35为氢；
R36为SO2R51或C1-C3烷氧基；
R17与R51分别为C1-C4烷基，C1-C4卤代烷基，NR46R48，C3-C6环烷基或异噁唑环；
R46与R48分别为氢，C1-C4烷基或苄基；且
A与A1为O。
本发明3-(1，2-苯并异噻唑-及异噁唑-5-基)-2，4(1H，3H)-嘧啶二酮或硫二酮化合物中，特别有效的除草剂包括：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-(二甲氨基)乙酯；
2-{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(6-甲氧基间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-(对-乙苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}丙酸甲酯；
{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}乙酸甲酯；
3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-(6-氟-3-甲基-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸乙酯；
1-甲基-3-{3-[6-(2-丙炔氧基)-间-甲苯基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-{3-{6-[(1-苯并咪唑基羰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-{3-{6-{[(间-氰基苯基)氨基甲酰基]甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸烯丙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸3-苯基-2-丙炔酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸1-甲基-2-丙炔酯；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸2-氯乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2，2，2-三氟乙酯；
3-[3-(2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-[3-(6-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，4-二甲苯基}氧基}乙酸甲酯；
3-{3-{6-{[(间-氰基苯基)氨基甲酰基]甲氧基}-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
1-甲基-3-{3-[(甲磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(邻-甲氧苯基)-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酰基}甲磺酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}丙酸2-丙炔酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈；
3-[3-[(烯丙基氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲基磺酰基)-1，2-苯并异噻唑-3-甲酰胺(carboxamide)；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}丙酸；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲氧乙酰胺；
2-{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧苯氧基}丙酸甲酯；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-(甲基磺酰基)乙酰胺；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-(甲基磺酰基)丙酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲基-N-(甲基磺酰基)乙酰胺；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-甲基-N-(甲基磺酰基)乙酰胺；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-(乙基磺酰基)乙酰胺；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-噻吩羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，苯甲酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲氧基乙酸酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二乙基-1，2-苯并异噻唑-3-乙腈；
3-[6-氟-3-(甲氧基甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，5-异噁唑羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，环丙烷羧酸酯；
3-(乙酰基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-(1-甲氧基乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
N-(苄基磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸苄酯；
N-(苄基磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(对-甲苄基)磺酰基]-1，2-苯并异噻唑-3-甲酰胺；
N-(苄基磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲酰胺；
3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(carboxaldehyde)，3-(二甲基缩醛)；
3-(6-氟-3-甲基-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲醛(carboxaldehyde)，3-(二甲基缩醛)；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-羧酸；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-甲基-1，2-苯并异噻唑-3-乙腈；
N-(苄基磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙氧基甲基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸甲酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-糠酸酯；
N-[(间-氯苄基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；与
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲基氨基甲酸酯。
上述卤素实施例为氟，氯，溴及碘。说明书和权利要求书中使用的术语卤代烷基，卤代环烷基，卤代烷氧基，卤代烯基，卤代环烯基及卤代炔基等名词指分别被一个或多个卤原子取代的烷基，环烷基，烷氧基，烯基，环烯基及炔基。上式I与II中，碱金属包括：钠，钾与锂。式I与II的碱土金属包括镁与钙。此外，术语″有机铵″被定义为由带正电价的氮原子连接至一至四个各含1至16个碳原子的脂族基团构成的基团。
上式I与II中，5至12元单环或稠合双环、杂环包括(但不限于)：苯并咪唑，咪唑，咪唑-2-硫酮，吲哚，N-羧氨基苯甲酸酐，吗啉，哌嗪，哌啶，嘌呤，吡唑，吡咯，吡咯烷，及1，2，4-三唑环，其中各环可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基。
上式I与II中，4至10元杂环包括(但不限于)：咪唑与邻苯二甲酰亚胺环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团。
本发明式I与II化合物为用于防治各种不要的植物品种的有效除草剂。这些化合物可有效防治干地及湿地的本土杂草。当化合物施用至上述植物的叶部或含其种子或其他繁殖器官如：匍匐枝，块根或根基的土壤或水中，施用率为约0.001公斤/公顷至4公斤/公顷，以约0.001公斤/公顷至1公斤/公顷较佳时，可有效地防治上述植物。
已有利地发现，本发明式I与II化合物特别适合在作物，作物种子或其他作物繁殖器官存在下选择性地防治不要的植物品种。特别是，本发明有些化合物在芽前和/或芽后施加时，在大豆和/或诸如玉米，小麦和稻的谷类作物中有选择性。
此外并发现，本发明式I与II化合物可这样在移植的稻培养物中选择性地控制不要的植物品种：在稻移植后，向含有所述不要的植物品种的种子或其他繁殖器官的土壤或水中施用除草有效量的式I化合物。
在玉米存在下选择性地控制不要的植物品种的特别有用的本发明式I化合物包括：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-(二甲氨基)乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(对-乙苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}乙酸甲酯；
3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸1-甲基-2-丙炔酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
1-甲基-3-{3-[(甲磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(邻-甲氧苯基)-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酰基}甲磺酰胺；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈；
3-[3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲基-N-(甲磺酰基)乙酰胺；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲基氨基甲酸酯；
N-(苄基磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-羧酸；与
N-(苄基磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲酰胺。
在小麦存在下选择性控制不要的植物品种的特别适用的本发明式I化合物包括：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对甲苯基}氧基}乙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-(二甲氨基)乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}丙酸甲酯；
3-(6-氟-3-甲基-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-{3-{6-[(1-苯并咪唑羰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸烯丙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸3-苯基-2-丙炔酯；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸2氯乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2，2，2-三氟乙酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，4-二甲苯基}氧基}乙酸甲酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲氧乙酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲基-N-(甲磺酰基)乙酰胺；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯；
3-(3-乙酰基-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酰甲酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
N-[(间-氯苄基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；与
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺。
在稻存在下选择性控制不要的植物品种的特别适用的本发明3-(1，2-苯并异噻唑-5-基]-2，4(1H，3H)-嘧啶二酮化合物包括：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸乙酯；
1-甲基-3-[3-(6-(2-丙炔氧基)-间-甲苯基]-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-{6-{[(间-氰苯基)氨基甲酰基]甲氧基}-间-甲苯基}-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-(2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-[3-(6-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-{6-{[(间-氰苯基)氨基甲酰基]甲氧基}-间-甲苯基}-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{邻-[5-(3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
3-[3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二乙基-1，2-苯并异噻唑-3-乙腈；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，5-异噁唑羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，环丙烷羧酸酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸苄酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；与
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺。
在大豆存在下选择性控制不要植物生长的特别适用的本发明式I化合物包括：
2-{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(邻-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}丙酸2-丙炔酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
3-[3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，苯甲酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-噻吩羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲氧乙酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，环丙烷羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-糠酸酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；与
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺。
虽然本发明化合物单独使用时可有效控制不要的植物品种，但亦可与其他生物化学物质(包括除草剂)组合使用。
本发明化合物可为固体或液体除草剂组合物形式施加到含不要植物的叶部或含其种子或其它繁殖器官的土壤或水里，所述的组合物包含除草有效量的所需化合物，它分散或溶于农业上可接受的惰性固体或液体载体。该组合物可在芽前或芽后处理施用。
本发明式I与II化合物可配制成乳化浓缩物，可湿化粉末，颗粒制剂，悬浮浓缩物，可流动浓缩物，等等。
式I中Z为S之化合物可依流程图I制备：用硫和氢氧化铵或氨使式III酮环化，形成式IV硝基苯并异噻唑，采用一般还原剂如：铁，于乙酸中，还原式IV化合物，形式V氨基苯并异噻唑，由式V化合物与光气或光气同等物反应，形成式VI异氰酸酯，使异氰酸酯与式VII 3-氨基丙烯酸酯，于碱(如：氢化钠)存在下反应，形成式VIII中间化合物，使式III化合物与式IX亲电子物于碱(如：碳酸钾)之存在下反应。
                        流程I
Figure A9880989801061
                      流程I(续)
Figure A9880989801071
式I中Z为S的化合物亦可依流程II制备：使式V氨基苯并异噻唑与式X 1，3-丙二酮于诸如三乙胺的碱存在下反应，形成式XI中间化合物，并使式XI化合物与光气或硫光气或其同等物质反应，然后与式XII胺于诸如三乙胺或吡啶的碱存在下反应。
                          流程II
或者，式I中Z为S之化合物可依流程III制备：使式V氨基苯并异噻唑与式XIII 2-二烷氨基-6H-1，3-噁嗪-6-酮于诸如乙酸的有机酸存在下反应，形成式VIII中间化合物，使式VIII化合物与式IX亲电子物于碱(如：碳酸钾)存在下反应。
                              流程III
Figure A9880989801091
可这样制备式I中Y为被一个X4R22基团取代的苯基的化合物：使式I中Y为被一个C1-C4烷氧基或C1-C4烷硫基取代的苯基的化合物与三溴化硼反应，形成式中Y为被一个羟基或硫代基团取代的苯基的相应化合物，使所形成所化合物与式Z1R22亲电子物(Z1＝Cl，Br或I)于诸如氢氧化钾的碱存在下反应。
式I中Z为O之化合物可依流程IV制备：使式III酮与羟胺盐酸盐，任选地在乙酸钠存在下反应，形成式XIV的肟，使式XIV化合物用诸如氢氧化钾的碱使式XIV化合物环化，形成式XV硝基苯并异噁唑，采用一般还原剂(如：氯化亚锡(II))，于乙酸中还原式XV化合物，形成式XVI氨基苯并异噁唑，使式XVI化合物与式XIII2-二烷氨基-6H-1，3-噁嗪-6-酮于有机酸(如：乙酸)存在下反应，形成式XVII中间化合物，使式XVII化合物与式IX亲电子物于碱(如：碳酸钾)存在下反应。
                       流程IV
                         流程IV(续)
Figure A9880989801121
                         流程IV(续)
Figure A9880989801131
或者，式XV硝基苯并异噁唑化合物可依流程图V所示制备：使式XVIII酮与羟胺盐酸盐，任选地在诸如乙酸钠的碱存在下反应，形成式XIX肟，用1，1’-羰基二咪唑于诸如三乙胺的碱存在下使式XIX环化，形成式XX苯并异噁唑，并使用一般方法，如：硝酸/硫酸混合物，硝化式XX化合物。
                           流程V
                         流程V(续)
Figure A9880989801141
式I中Y为卤甲基的化合物可依流程图VI制备：用如N-溴琥珀酰亚胺，N-氯琥珀酰亚胺，N-碘琥珀酰亚胺，溴，氯，硫酰氯，硫酰溴等等的卤化剂卤化式I中Y为甲基的化合物。
                         流程VI
(Z3＝CH2Br或CHBr2)
式I中Y为C1-C20烷氧基甲基的化合物可依流程VII制备：使式I中Y为溴甲基的化合物与C1-C20醇于三氟甲磺酸银存在下反应。
                         流程VII
Figure A9880989801161
式I中Y为被一个X4R22基团取代的甲基的化合物可依流程图VIII所示制备：使式I中Y为溴甲基的化合物与式XXI醇或硫醇，于诸如氢化钠的碱存在下反应。
                         流程VIII
式I中Y为C1-C4烷硫甲基的化合物可依流程图IX制备：使式I中Y为溴甲基的化合物与碱金属硫醇盐反应。
                            流程IX
Figure A9880989801171
式V中Y为OR12的中间化合物可依流程图X制备：用诸如硝酸/硫酸混合物的常规硝化剂硝化式XXII苯并异噁唑-3-醇或苯并异噻唑-3-醇，形成式XXIII 5-硝基苯并异噁唑-3-醇或5-硝基苯并异噻唑-3-醇，使式XXIII化合物与式XXIV亲电子物于诸如碳酸钾的碱存在下反应，形成式XXV中间化合物，并使用常规还原剂还原式XXV化合物。
                         流程X
式V中Y为Cl或Br的中间化合物可依流程图XI制备：使式XXIII 5-硝基苯并异噁唑-3-醇或5-硝基苯并异噻唑-3-醇与磷酰氯，磷酰溴或五溴化磷反应，形成式XXVI 3-卤-5-硝基苯并异噁唑或3-卤-5-硝基苯并异噻唑，并采用常规还原剂还原式XXVI化合物。
                              流程XI
Figure A9880989801191
式I中A为O且A1为S的化合物可依流程XII制备：使式I中A与A1为O的化合物与Lawesson试剂(2，4-双(4-甲氧苯基)-1，3-二硫杂-2，4-二磷烷-2，4-二硫化物)，于诸如碳酸氢钠的碱存在下反应。
                        流程XII
式I中A与A1为S的化合物可依流程图XIII制备：使式I中A为S且A1为O的化合物与Lawesson试剂于碱存在下反应。
                        流程XIII
Figure A9880989801211
式I中R19，R26与R32为氢的化合物可由相应的式I酯经酸(如：三氟乙酸)水解制得。所得式I酸再与亚硫酰氯或草酰氯反应，形成的酰基氯再与R19OH，R26OH或R32OH醇或HNR20R21，HNR35R36或HNR49R50胺反应，形成另一种式I化合物。
式I中R19，R26与R32为碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子的化合物可由式I中R19，R26及R32为氢的化合物用常规方法制备。
式IV中Y为被一个CO2R19基团取代的烷基的中间化合物可依流程图XIV制备：式XXVI中间化合物与式XXVII草酸酯于碱存在下反应，形成中间化合物，使尿素与中间化合物反应，形成式XXVIII中Y为被一个CO2R19基团取代的甲基的化合物，并任选地使式XXVIII化合物与C1-C5烷基卤化物于碱(如：氢化钠)之存在下反应，形成式XXIX化合物。此外，可由式XXVIII及XXIX化合物皂化，形成式中R19为氢的化合物。
                         流程XIV
Figure A9880989801221
或者，式III中Y为α-甲基乙酸酯的化合物可依流程图XV制备。
                     流程XV
可这样制备式III中Y为被一个CO2R19基团取代的甲基的中间化合物：使式XXX酰基氯与式XXXI乙酸酯于碱(如：氢化钠)之存在下反应，任选地使式III中Y为经一个CO2R19基团取代的甲基的化合物与C1-C5烷基卤化物于碱如：氢化钠存在下反应，形成式III中Y为α-烷基乙酸酯的化合物。该反应如流程XVI所示。
                      流程XVI
Figure A9880989801241
可这样制备式IV与XV中Y为被一个C(O)R18或C(O)R25基团取代的烷基或苯基的化合物：使相应的酰基氯与适当取代的溴化镁化合物，溴化铜化合物或锂化合物反应。该反应流程以式中Y为被一个C(O)R25基团取代的苯基为例说明。
                      流程XVII
Figure A9880989801251
可这样制备式I，IV与XV中Y为被一个CHO基团取代的烷基，环烷基，烯基，环烯基，炔基或苯基的化合物：用诸如硼烷-四氢呋喃配位物的常规的还原剂使式I，IV或XV中Y为被一个CO2H基团取代的烷基，环烷基，烯基，环烯基，炔基或苯基的化合物还原形成式I，IV或XV中Y为CH2O基团取代的烷基，环烷基，烯基，环烯基，炔基或苯基的化合物，所得的醇经常规氧化剂如：氧化铬(VI)氧化。反应流程以Y为经一个CHO基团取代的苯基为例说明于流程XVIII中。
                    流程XVIII
Figure A9880989801261
可这样制备式IV与XV中Y为被C(O)R18基团取代的烷基或环烷基的化合物：使式IV或XV中Y为卤代烷基或卤代环烷基的化合物与式XXXII锂试剂反应，形成中间化合物，该中间化合物再与路易士酸(如：三氟化硼)，于水存在下反应，该反应流程以式中Y为经一个C(O)R18基团取代的甲基为例说明于流程XIX中。
                        流程XIX
Figure A9880989801271
式I中Y为甲酰基的化合物也可如流程XX所示制备。
                      流程XX
Figure A9880989801281
式IV与XV中Y为X2R12且R12为可任选地被取代的苯基的化合物可依流程XXI制备：使式IV或XV中Y为Br的化合物与R12X2H化合物，于碱(如：碳酸钾)存在下反应。
                      流程XXI
Figure A9880989801282
式IV与XV中Y为三氟甲基的化合物可依流程图XXII制备：使式IV或XV中Y为Br的化合物与式XXXIII甲硅烷基化合物，于碘化亚酮(I)及碘化钾存在下反应。
                         流程XXII
Figure A9880989801291
或者，可这样制备式III与XIV中Y为三氟甲基的化合物：使式IV或XV中Y为Br的化合物与三氟乙酸钠于诸如四取代的钯催化剂的催化剂存在下反应。该反应流程如流程XXIII所示。
                        流程XXIII
Figure A9880989801292
式I中Y为CH2CN的化合物可依流程XXIV所示制备：式I中Y为CH2Br的化合物与氰化钾反应。
                      流程XXIV
Figure A9880989801301
可这样制备式I中Y为R12或X2R12且R12为氯烷基，氟烷基或碘烷基的化合物：使式I中R12为溴烷基的相应化合物与氯化锂，碘化钠，氟化钾或氟化银(I)反应。在下面的流程XXV中，该反应流程以式中Y为氟甲基，碘甲基及氯甲基为例说明。
                        流程XXV
Figure A9880989801311
式I中A为S且A1为O的化合物可依流程XXVI所示制备：使式V或XVI胺与硫光气或硫光气同等物，于碱(如：三乙胺)存在下反应，形成式XXXIV异硫氰酸酯，使式XXXIV化合物与式XXXV烯于碱(如：氢化钠)存在下反应。
                   流程XXVI
式I中A与A1为O的化合物可依流程图XXVII所示制备：使式XXXVI异氰酸酯与式XXXVII烯于碱(如：氢化钠)存在下反应，形成式XXXVIII脲类，式XXXVIII化合物再用酸环化，形成式XXXIX中间化合物，使式XXXIX化合物与式XL亲电子物于碱(如：碳酸钾)存在下反应。
                             流程XXVII
可这样制备式III中Y为被α-(C1-C6-烷基)或α，α-双(C1-C6-烷基)取代的乙酸酯的化合物：使式XLI酰基氯经锌及式XLII α-卤酯处理，形成式XLIII酮基酯中间物，其再硝化形成式III中间物。该反应图示于流程XXVIII。
                         流程XXVIII
Figure A9880989801341
式V中Y为Cl或Br的中间化合物亦可依流程XXIX制备：使式XLIV 5-硝基苯并异噻唑或5-硝基苯并异噁唑与氯或溴于酸(如：乙酸)中反应。该反应图示于下列流程图XXIX。
                        流程XXIX
Figure A9880989801351
式I中Y为C(O)X2R12且X2为O或S的化合物可依流程XXX制备。
                        流程XXX
Figure A9880989801352
                      流程XXX(续)
Figure A9880989801361
式I中Y为C(O)NR12R13的化合物可依下列流程XXXI制备。
                        流程XXXI
Figure A9880989801362
式I中Y为C(O)NR13SO2NR46R48的化合物可依下列流程XXXII制备。
                         流程XXXII
Figure A9880989801371
式I中Y为C(O)N(R12)OR23的化合物可依下列流程XXXIV制备。
                         流程XXXIV
式I中Y为CH(OH)R23，C(O)R23，CH(OR22)R23及CH(R23)OC(O)R33的化合物可依下列流程XXXV制备。
                     流程XXXV
其他制备式I化合物的方法及制备式II化合物之方法可从下列实施例中得以明了。此外，某些式I与II化合物可使用本技术领域公知的常规方法转化成其他式I与II化合物。
本发明也涉及如结构式XLV的中间化合物
Figure A9880989801391
其中R1，R2，A，A1，X，X1，Y与Z如上式I的定义。
较佳式XLV中间化合物为这些化合物，其中
R1与R2分别为氢，卤素，C1-C6烷基，C3-C7环烷基，C1-C6卤代烷基，C3-C6烯基，C3-C6卤代烯基，C3-C6炔基，OR7，S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它们可任选地穿插氧，硫或氮，且可任选地被一至三个甲基或一个或多个卤原子取代；
X为氢，卤素或C1-C4烷基；
X1为氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素，氰基，R12，X2R12，X3R12，X2X3R12或X3X2R12；
X2为O，S(O)p或NR13；
X3为-C(＝A3)-或-C(＝NOR14)-；
R4，R5，R6，R7，R8，R9，R10与R14分别为氢，C1-C6烷基，C3-C7环烷基，C2-C6烯基，C2-C6炔基或苄基；
R12为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基，C5-C6环烯基或C2-C6炔基，其中各基团可任选地被下列任何组合取代：1至6个卤原子，1至3个C1-C20烷氧基，1或2个C1-C10卤代烷氧基，1或2个NR15R16基团，1至3个S(O)qR17基团，1或2个氰基，1或2个O(O)R18基团，1或2个CO2R19基团，1或2个C(O)NR20R21基团，1至3个X4R22基团，1或2个P(O)(OR23)2基团，1或2个Si(R24)3基团，
1个4至10元杂环(它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C3-C7环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团或1个X5R27基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基，1个C3-C6环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，形成了5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列的基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基，或X4R22基团；
R13为氢，C1-C6烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR23，氰基或SO2R51，且当R13及R12及其所连接的氮原子结合在一起时，形成了5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢，Si(R31)3，
C1-C20烷基，其被下列基团取代：一个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，P(O)(OH)NH2，P(O)(OH)(OR23)，C(O)NHOR23，氰基或2-二氧戊环基，
1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，或C1-C4卤代烷基磺酰基，
C3-C20烯基，它可任选地被下列基团取代：1至3个卤原子，1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NHOR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它可任选地被下列基团取代：一个C1-C6烷氧基，C1-C4烷基，C2-C4烯基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NHOR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它可任选地被下列基团取代：1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NHOR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它们可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，
苄基，其苯环上可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团，或
4至10元杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
C(O)R43；
R16与R21分别为氢，C1-C6烷基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17，R18，R25，R30，R33，R45及R51分别为C1-C4烷基，C1-C4卤代烷基，CO2R23，C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团，或
5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R19与R26分别为氢，C1-C20烷基，C1-C8卤代烷基，C3-C7环烷基，C3-C7卤代环烷基，C3-C20烯基，C3-C8卤代烯基，C5-C8环烯基，C5-C8卤代环烯基，C3-C8炔基，C3-C8卤代炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它可任选地被一个CO2R48，C1-C6烷氧基，或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，
C3-C8卤代环烷基，
C3-C20烯基，它可任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它可任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
2-，3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，其被一个吡啶基，呋喃基，噻吩基，四氢呋喃基或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢，氰基，C1-C6烷基，SO2R51或苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
m，n，p与q分别为0，1或2的整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R24，R31，R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R23，R39，R40，R42，R43，R44，R46及R48分别为氢，C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，且
A，A1，A3，A4，X4及X5分别为O或S；
及其光学异构体，非对映异构体和/或互变异构体。
另一类较佳式XLV中间化合物为这些化合物，式中：
R1与R2分别为氢，卤素，C1-C6烷基，C3-C7环烷基，C1-C6卤代烷基，C3-C6烯基，C3-C6卤代烯基，C3-C6炔基，OR7，S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它可任选地穿插氧，硫或氮，且可任选地被一至三个甲基或一个或多个卤原子取代；
X为氢，卤素或C1-C4烷基；
X1为氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素，氰基，R12，X2R12，X3R12，X2X3R12或X3X2R12；
X2为O，S(O)p或NR13；
X3为-C(＝A3)-，-C(＝NOR14)-或-C(＝N-NR13R50)；
R4，R5，R6，R7，R8，R9，R10与R14分别为氢，C1-C6烷基，C3-C7环烷基，C2-C8烷氧基烷基，C2-C6烯基，C2-C6炔基或苄基；
R12为氢，
C1-C8烷基，C3-C7环烷基，C2-C8烯基，C5-C6环烯基或C2-C8炔基，其中各基团可任选地被下列任何组合取代：1至6个卤原子，1至3个C1-C20烷氧基(它们可任选地被一个C1-C6烷氧基，苄氧基或C1-C6烷硫基取代)，1或2个C1-C10卤代烷氧基，1或2个NR15R16基团，1至3个S(O)qR17基团，1或2个氰基，1或2个C3-C7环烷基，1个硫氰基，1个O(SO2)R17基团，1个O(NO2)基团，1或2个C(O)R18基团，1或2个CO2R19基团，1或2个C(O)SR19基团，1或2个C(O)NR20R21基团，1至3个X4R22基团，1或2个P(O)(OR23)2基团，1或2个Si(R24)3基团，
1个4至10元单环或稠合双环、杂环(它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1或2个苯基，其中各苯基分别可需要经下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C3-C7环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团或1个X5R27基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基，1个C3-C6环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，或
茚满基，它可任选地被下列任何组合取代：1或2个卤原子，1或2个C1-C4烷基，1个C1-C4烷氧基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，当5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基，或X4R22基团；
R13为氢，C1-C8烷氧基烷基，C1-C6烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR23，氰基，SO2R51或1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基，且当R13及R12及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢，Si(R31)3，C(O)NR35R36，C(O)R33，SO2R47，
C1-C20烷基，其被下列基团取代：一个羟基，苄氧基，硝基，OC(O)R33，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，P(O)(OH)NH2，P(O)(OH)(OR23)，C(O)NR35OR23，氰基或2-二氧戊环基，
1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，或C1-C4卤代烷基磺酰基，
C3-C20烯基，它可任选地被下列基团取代：1至3个卤原子，1个羟基，1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它可任选地被下列基团取代：一个羟基，C1-C6烷氧基，C1-C4烷基，C2-C4烯基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它可任选地被下列基团取代：1个羟基，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它们可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，
苄基，其苯环上可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团，或
4至10元杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个CO2R26基团，
C(O)R43，或
CO2R42；
R16与R21分别为氢，C1-C6烷基，C1-C4烷氧基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17，R18，R25，R30，R33，R45及R51分别为NR46R48，-N＝CR46R48，C1-C8烷基，它可任选地被一个C1-C6烷氧基，噻吩或呋喃基取代，C1-C6卤代烷基，C3-C8环烷基，CO2R23，C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团，或
5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R19与R26分别为氢，C1-C20烷基，C1-C8卤代烷基，C3-C7环烷基，C3-C7卤代环烷基，C3-C20烯基，C3-C8卤代烯基，C5-C8环烯基，C5-C8卤代环烯基，C3-C8炔基，C3-C8卤代炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它可任选地被一个CO2R48，C1-C6烷氧基，C1-C6硫代烷基，C2-C20烷氧基烷氧基，苯基，OSi(R47)3，OC(O)R33，C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它可任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它可任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它可任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
2-，3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基，呋喃基，噻吩基，四氢呋哺基，C3-C8环烷基，二噁烷或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢，氰基，C1-C6烷基，SO2R51或苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，形成了5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
m，n，p与q分别为0，1或2的整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R24，R31，R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R23，R39，R40，R42，R43，R44，R46及R48分别为氢，C2-C6烯基，C3-C8环烷基，
C1-C8烷基，它可任选地被一或二个C1-C4烷氧基取代；
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，且
当R46与R48及其所连接的原子结合在一起时，为5至12元单环或稠合双环、杂环或环烷基环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；及
A，A1，A3，A4，X4及X5分别为O或S；
及其光学异构体，非对映异构体和/或互变异构体。
更佳的本发明式XLV中间化合物为这些，其中：
R1为卤素或C1-C4卤代烷基；
R2为氢，卤素或C1-C4卤代烷基；
X与X1分别为氢或卤素；
Z为O或S；
Y为氰基，R12，X2R12或X3X2R12；
X2为O，S或NR13；
X3为-C(＝A3)-，-C(＝NOR14)或-C(＝N-NR13R50)；
R12为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基，C5-C6环烯基或C2-C6炔基，其中各基团可任选地被下列任何组合取代：1至3个卤原子，1或2个C1-C20烷氧基，1或2个C1-C10卤代烷氧基，1个NR15R16基团，1个S(O)qR17基团，1或2个氰基，1或2个C(O)R18基团，1或2个CO2R19基团，1或2个C(O)SR19基团，1或2个C(O)NR20R21基团，1或2个X4R22基团，1个P(O)(OR23)2基团，1个Si(R24)3基团，
1个4至10元单环或稠合双环杂环(它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它可任选地被下列任何组合取代：1至3个卤原子，1个C1-C6烷基，1个C1-C6烷氧基，1个C3-C7环烷基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团或1个X5R27基团，或
苯基，它可任选地被下列任何组合取代：1或2个卤原子，1至3个C1-C4烷基，1或2个C1-C4烷氧基，1个C3-C6环烷基，1个C1-C4卤代烷基，1个C1-C4烷硫基，1个氰基，1个硝基，1个C(O)R25基团，1个CO2R26基团，1个X4R22基团，1个CH＝CHR22基团，1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
R13为氢，C2-C6烷氧基烷基，C1-C6烷基，C3-C7环烷基，C3-C6烯基，C3-C6炔基，苄基，OR23，氰基或SO2R51；
R28为卤素；
R22与R27分别为氢，Si(R31)3，C(O)NR35R36，C(O)R33，SO2R47，
C1-C20烷基，它被下列基团取代：一个羟基，苄氧基，硝基，OC(O)R33，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，P(O)(OH)NH2，P(O)(OH)(OR23)，C(O)NR35OR23，氰基或2-二氧戊环基，
1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
1个5至12元单环或稠合双环、杂环，它们可任选地被1个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，或C1-C4卤代烷基磺酰基，
C3-C20烯基，它可任选地被下列基团取代：1至3个卤原子，1个羟基，1个C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或1个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它可任选地被下列基团取代：一个羟基，C1-C6烷氧基，C1-C4烷基，C2-C4烯基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它可任选地被下列基团取代：1个羟基，C1-C6烷氧基，CO2R32，C(O)R33，C(A4R34)2，C(O)NR35R36，C(O)ON＝CR37R38，C(O)NR35OR23，氰基或2-二氧戊环基，或一个苯基，二氢呋喃酮或呋喃酮环，其中各环可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它们可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团或1个C(O)R33基团，
苄基，其苯环上可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C6烷基，1至3个C1-C6烷氧基，1个C1-C4卤代烷基，1个C1-C4卤代烷氧基，1个氰基，1个硝基，1个NR39R40基团，或1个C(O)R33基团，或
4至10元杂环，它们可任选地被下列任何组合取代：1或2个氧代基，1或2个硫代基，1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢，
C1-C6烷基，C3-C7环烷基，C2-C6烯基或C2-C6炔基，其中各基团可任选地被一个CO2R42基团取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个CO2R26基团，
C(O)R43，或
CO2R42；
R14为氢，C1-C6烷基，C3-C7环烷基，C2-C8烷氧基烷基，C2-C6烯基，C2-C6炔基或苄基；
R16与R21分别为氢，C1-C6烷基，C1-C4烷氧基，C3-C7环烷基，C2-C6烯基，C3-C7环烯基，C2-C6炔基，P(O)(OR44)2，SO2R45，C(O)R46，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R17，R18，R25，R30，R33，R45及R51分别为NR46R48，
-N＝CR46R48，C1-C8烷基，它可任选地被一个C1-C6烷氧基，噻吩或呋喃基取代，C1-C6卤代烷基，C3-C8环烷基，CO2R23，C2-C6烯基，它可任选地被苯基取代，
苄基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基或1个X4R22基团，
苯基，它可任选地被下列任何组合取代：1至3个卤原子，1至3个C1-C4烷基，1至3个C1-C4卤代烷基，1至3个C1-C4烷氧基，1至3个C1-C4卤代烷氧基，1个硝基，1个氰基，或1个X4R22基团，或
5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基磺酰基或X4R22基团；
R19与R26分别为氢，C1-C20烷基，C1-C8卤代烷基，C3-C7环烷基，C3-C7卤代环烷基，C3-C20烯基，C3-C8卤代烯基，C5-C8环烯基，C5-C8卤代环烯基，C3-C8炔基，C3-C8卤代炔基，Si(R41)3，苄基，苯基，糠基，吡啶基，噻吩基，羟亚氨基，或碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R32为氢，
Si(R47)3，
C1-C20烷基，它可任选地被一个CO2R48，C1-C6烷氧基，C1-C6硫烷基，C2-C20烷氧基烷氧基，苯基，OSi(R47)3，OC(O)R33，C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它可任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它可任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它可任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，
C1-C4烷基，它被一个吡啶基，呋喃基，噻吩基，四氢呋喃基，C3-C8环烷基，二噁烷或NR49R50基团取代，或
碱金属，碱土金属，锰，铜，锌，钴，银，镍，铵或有机铵阳离子；
R34，R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢，氰基，C1-C6烷基，SO2R51或苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环、杂环，它们可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，氨基，羟基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C1-C4卤代烷基磺酰基；
q为0，1或2的整数；
R29为氢，C1-C4烷基或C1-C4卤代烷基；
R24，R31，R41及R47分别为C1-C4烷基，
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基；
R23，R39，R40，R42，R43，R44，R46及R48分别为氢，C2-C6烯基，C3-C8环烷基，
C1-C8烷基，它可任选地被一或二个C1-C4烷氧基取代；
苄基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它可任选地被一个或多个分别选自下列之基团取代：卤素，氰基，硝基，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基及C1-C4卤代烷氧基，且
A，A1，A3，A4，X4及X5分别为O或S；及其光学异构体，非对映异构体和/或互变异构体。
为了帮助进一步了解本发明，现提出下列实施例作更详尽的阐述。除了权利要求书的界定外，本发明并不受这些实施例的限制。
实施例1
2’-氯-2-甲氧基-5-甲基-5’-硝基苯酮的制备
使氯化铝(33.3克，25.0毫摩尔)在二氯甲烷里的混合物冷却至约5℃，用对-甲基苯甲醚(31.6克，25.0毫摩尔)处理1小时，同时保持反应混合物温度在10℃以下，以20分钟时间，用2-氯-5-硝基苯甲酰氯(50.0克，22.7毫摩尔)的二氯甲烷溶液处理20分钟，同时保持反应混合物温度在10℃以下，温热到室温并搅拌60分钟，倒至冰上。所得水性混合物经浓盐酸(50毫升)处理，以二氯甲烷萃取。有机萃取液经无水硫酸镁干燥，真空浓缩，产生黄色固体。此固体置入40℃的球形管(Kugelrohr)中，以除去残留的对-甲基苯甲醚，得到标题化合物的米色固体(68.8克，99.1％)，经NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：W    W1    W2              W3       W4     mp℃H    I      H                H         OCH3   115-116.5H    H      CH3             H         OCH3H    H      C2H5           H         HH    CH3   CH3             H         OCH3H    H      OCH3            H         H       108-112H    C2H5H                 H         OCH3   98-99.5H    H      OCH3            H         CH3    91-92H    H      CH3             H         H       95.5-96.5H    H      SCH3            H         H       127-128H    H      CH3             H         OCH3   91-92.5H    H      C2H5          H         HH    H      Cl               H         H       88.5-90.5H    H      F                H         H       68-69.5H    Cl     H                H         OCH3   124-126H    OCH3  H                H         OCH3   71-73H    H      OCH3            H         OCH3   98-100H    CH3   CH3             H         OCH3  127-129H    H      Cl               H         OCH3   96-99CH3 H      CH3            H         OCH3   108.5-110H    H      H                CH3      OCH3   71-74H    H      N(CH3)SO2CH3 H         H       126-128H    CH3   Cl               H         OCH3   110-112 H    CH3          H        CH3   OCH3   104-106CH3  CH3          CH3     H      OCH3   69-71H    CH(CH3)2    H        H      OCH3H    CH3          H        H      HH    H             H        H      CNH    H             H        H      OCH3H    OCH3         H        H      HH    F             H        H      OCH3H    H             F        H      OCH3H    H             H        H      SCH3H    H             H        H      OCH3H    H             H        H      FH    SCH3         H        H      HH    H             OCH3    H      HH        -(CH2)3-         H      OCH3
实施例2
3-(6-甲氧基-间-甲苯基)-5-硝基-1，2-苯并异噻唑的制备
将氢氧化铵(350毫升30％溶液，270毫摩尔)加到2’-氯-2-甲氧基-5-甲基-5’-硝基苯酮(68.7克，22.5毫摩尔)与硫(7.57克，23.6毫摩尔)在N，N-二甲基甲酰胺里的混合物中。所得反应混合物于80℃下搅拌19.5小时，冷却至40℃，再用氢氧化铵(50毫升30％溶液)处理，于80℃下搅拌25小时，冷却，倒至冰上，所得水性混合物过滤，得到标题产物的黄色固体(63.5克，93.9％)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989801571
W       W1      W2      W3     W4     mp℃H       H        CH3     H       OCH3   201-203H       CH3     CH3     H       OCH3   199-200H       CH3     H        H       H       116.5-117.5H       H        Cl       H       OCH3   229-231H       H        H        CH3    OCH3   134-136H       H        H        H       CN      187.5-189H       H        H        H       OCH3   193-198H       H        OCH3    H       H       201-203H       OCH3    H        H       H       174-175H       F        H        H       OCH3   224-226H       C2H5  H        H       OCH3   153-154.5H       H        CH3     H       H       188-189 W    W1         W2             W3  W4     mp℃H    H           N(CH3)SO2CH3 H    HH    CH3        Cl              H    OCH3   230-234H    I           H               H    OCH3H    H           SCH3           H    H       177.5-178.5H    H           OCH3           H    CH3    131-135H    H           F               H    H       226-228H    H           Cl              H    H       217.5-219H    H           F               H    OCH3   224-225H    H           H               H    SCH3   114.5-115.5H    H           CH3            H    OCH3   201-203H    OCH3       H               H    OCH3   195-196H    H           H               H    CH3    145-146H    H           H               H    F       181-182H    H           OCH3           H    OCH3   171-172.5H    SCH3       H               H    H       139-140.5H    CH3        H               CH3 OCH3H    CH3        CH3            H    OCH3CH3  CH(CH3)2 H               H    OCH3H    H           CH3            CH3 OCH3H      -(CH2)3-               H    OCH3
实施例3
3-甲基-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989801581
将氨(45克，2，642毫摩尔)通入-40℃之不锈钢桶中的甲醇内。然后加入硫(30.5克，95.0毫摩尔)及2’-氯-5’-硝基乙酰苯(19克，95.0毫摩尔)。密封不锈钢桶，于约90℃下加热过夜。冷却后，自桶中取出反应混合物，真空浓缩，得到残留物。残留物用二氯甲烷稀释，通过硅胶管塞，真空浓缩，产生标题化合物的橙色固体(12.0克)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
实施例4
5-氨基-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑的制备
Figure A9880989801592
使3-(6-甲氧基-间-甲苯基)-5-硝基-1，2-苯并异噻唑(63.0克，0.210摩尔)，5％乙酸(1.52升，1.21摩尔)及乙酸乙酯(975毫升)的混合物加热至65℃，用铁粉(58.6克，1.05摩尔)分批处理，于65℃下搅拌，经石英滤纸过滤。分离滤液相，用乙酸乙酯萃取水相。合并有机相与萃取液，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到标题产物的橙色油(55.7克，98.1％)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：X                      Y                       mp℃H                      HH                      CN                      118.5-120H                      CH3                    112-113.5H                      C2H5H                     
Figure A9880989801602
        179-181H                     
Figure A9880989801603
       90-91F                     
Figure A9880989801604
H                                    130-130.5X                       Y                             mp℃H                                  152-153H                                       121.5-123H             
Figure A9880989801613
                         108.5-109.5H             
Figure A9880989801614
                         158.5-161H             
Figure A9880989801615
                          101.5-102.5H                                        104-105H                                191-192.5X                        Y                            mp℃H                  
Figure A9880989801621
H                   H                                    128-129H                   H                                         64H                  
Figure A9880989801626
               108.5-109.5H                                     133-134H                  
Figure A9880989801628
                   114.5-115X                   Y                                 mp℃H                                  152-153.5H           
Figure A9880989801632
                            146-147H           
Figure A9880989801633
                            60-65H           
Figure A9880989801634
                          143-145H           
Figure A9880989801635
                              100-101H            H           
Figure A9880989801637
                      125-127X                      Y                              mp℃H            
Figure A9880989801641
                       172-174H            
Figure A9880989801642
                            146-147H                                  161-162H            
Figure A9880989801644
                 173-175H            
Figure A9880989801645
H            
Figure A9880989801646
X                                Y                      mp℃H                   
Figure A9880989801651
H                   
Figure A9880989801652
实施例5
3-[3-(6-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使5-氨基-3-(6-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑(8.53克，30.0毫摩尔)，2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(6.87克，33.0毫摩尔)及乙酸的混合物回流2小时，冷却，并倒入水中。所得水性混合物过滤得到固体。含此固体的二氯甲烷溶液依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到油状物。此油状物用硅胶及5％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的黄色泡沫物(8.37克，62.0％)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：X    X    R1     Y                    mp℃H    H    CF3    CN                   255-258H    H    CF3    H                    ＞260H    H    CF3    CH3                 273-274H    H    CF3    C2H5H    H    CF3   
Figure A9880989801662
    230-231H    H    CF3   
Figure A9880989801663
X    X1    R1           Y                  mp℃H    H     CF3    
Figure A9880989801671
             125-130H    H     CF3                   ＞280H    H     CF3    
Figure A9880989801673
       253-254H    H     CF3    
Figure A9880989801674
        149-152H    H     CF3     H    H     CH3    
Figure A9880989801676
            ＞250H    H     CF3     X    X1   R4            Y       mp℃H    H    CF3     H    H    CF3    
Figure A9880989801682
H    H    CF3     H    H    CF3    
Figure A9880989801684
H    H    CF3     H    H    CF3    
Figure A9880989801686
X    X1    R1            Y              mp℃H    H    CF3     
Figure A9880989801691
H    H    CF3   
Figure A9880989801692
      208-210H    H    CF3    H    H    CF3   
Figure A9880989801694
H    H    CF3   
Figure A9880989801695
F    Br   CF3      CH3X    X1  R1            Y               mp℃F    H    CF3   
Figure A9880989801696
F    H    CF3      CH3
实施例6
3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基异氰酸酯的制备
Figure A9880989801701
用光气(1.074毫升20％甲苯溶液，2.06摩尔)处理5-氨基-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑(157克，0.581摩尔)的甲苯溶液，加热及搅拌至回流5小时，再用光气(100毫升20％甲苯溶液)处理，回流过夜，真空浓缩，产生的标题产物为黄橙色固体(169克，98.2％)，用NMR光谱分析法鉴定。
基本上采用相同方法，但改用光气或硫光气，得到下列化合物：
Figure A9880989801711
A                      YO                      CH3O                 
Figure A9880989801712
O                 
Figure A9880989801713
O                  O                 
Figure A9880989801715
A                      YS                  实施例73-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989801721
将60％氢化钠在矿物油(15.9克，0.397摩尔)和N，N-二甲基甲酰胺里的混合物冷却至-10℃，用3-氨基-4，4，4-三氟巴豆酸乙酯(72.7克，0.397摩尔)的醚溶液处理1小时，温热至室温并搅拌90分钟，冷却至-70℃，用3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基异氰酸酯(107克，0.361摩尔)的N，N-二甲基甲酰胺溶液处理80分钟，同时保持约-65℃以下的温度，慢慢温热到室温并搅拌过夜，倒至冰上。所得水性混合物用乙酸乙酯洗涤，用浓盐酸酸化至pH 2，用乙醚萃取。有机萃取液经无水硫酸镁干燥，真空浓缩，产生标题产物的橙色油(110克，70.5％)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989801731
R1          A             Y                  mp℃CF3         O             CH3               273-274CF3         O        
Figure A9880989801732
R1          A             Y                  mp℃CF3         O        
Figure A9880989801733
    253-254CF3         O                    ＞280CH3         O        
Figure A9880989801735
          ＞250CF3         S                   213-216
实施例8
3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989801741
使3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(160克，0.369摩尔)，碳酸钾(76.6克，0.554摩尔)与碘甲烷(34.5毫升，0.544摩尔)在N，N-二甲基甲酰胺里的混合物于室温下搅拌4小时，并倒至冰上。所得水性混合物用二氯甲烷萃取。有机萃取液用己烷稀释，以水洗涤，用无水硫酸镁干燥，真空浓缩，得到标题产物的橙色泡沫状物(163克，98.8％)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989801751
X    X1  R            R1     Y                       mp℃H    H    CH3         CF3    H                       223-225H    H    CH3         CF3    CN                      239-240H    H    CH3         CF3    CH3                    244-245H    H    CH2C≡CH    CF3    CH3H    H    CH3         CF3    CH2OCH2CO2CH3      143-144H    H    CH2C6H5  CF3    CH3H    H    CH2CN       CF3    CH3H    H    CH2CH2F    CF3    CH3H    H    CH3         CF3    C2H5                 171-172H    H    CH3         CF3    
Figure A9880989801752
      198-200H    H    CH3         CF3          170.5-172H    H    CH3         CF3    
Figure A9880989801754
            175.5-180X    X1  R            R1           Y                     mp℃H    H    CH3         CF3    
Figure A9880989801761
              173-175H    H    CH3         CF3    
Figure A9880989801762
         225-227H    H    CH3         CF3    
Figure A9880989801763
         185-187H    H    CH(CH3)2   CF3     H    H    CH3         CF3    
Figure A9880989801765
X    X1  R       R1             Y                   mp℃H    H    CH3    CF3         187-190H    H    CH3    CF3                   83-86H    H    CH3    CF3    
Figure A9880989801773
           299H    H    CH3    CF3    
Figure A9880989801774
  220-225H    H    CH3    CF3    
Figure A9880989801775
              216-217X    X1  R            R1             Y              mp℃H    H    CH3         CF3         103-105H    H    CH3CH＝CH2 CF3   
Figure A9880989801782
H    H    CH3CH3     CF3    H    H    CH3         CH3   
Figure A9880989801784
          210-213H    H    C2H5       CF3   
Figure A9880989801785
         105-107X    X4   R            R1             Y                mp℃H    H    C2H5        CH3    H    H    CH2CH＝CH2  CF3   
Figure A9880989801792
            122-127H    H    CH3          CF3   
Figure A9880989801793
H    H    CH3          CF3   
Figure A9880989801794
H    H    CH3          CF3   
Figure A9880989801795
     147-149X    X1  R            R1          Y             mp℃H    H    CH3         CF3   
Figure A9880989801801
      170-172H    H    CH(CH3)2   CF3   
Figure A9880989801802
     151-154H    H    CH3         CF3   
Figure A9880989801803
H    H    CH3         CF3   
Figure A9880989801804
  227-228F    H    CH3         CF3       CH3Cl   H    CH3         CF3   
Figure A9880989801805
F    Br   CH3         CF3       CH3         211-213X    X1  R    R1         Y              mp℃F    H    CH3 CF3  
Figure A9880989801811
此外，当R为CF3且Y为甲基时，在氮和氧上均发生烷化，得到下列混合物：
Figure A9880989801812
R                ％A                 ％BCH2CH3            50                 50CH2CH(CH3)2        55                 45CH2CH＝CH2          85                 15
相似的是，分离出下列O-烷化及N-烷化化合物的混合物，随后利用柱层析分离：
Figure A9880989801813
R                        mp℃CH2CH3                  105-107CH2CH＝CH2               122-127
Figure A9880989801821
R                          mp℃CH2CH3                  143-146CH2CH＝CH2               129-133此外，当A为硫时，得到下列S-烷化产物：
实施例9
3-[3-(6-羟基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(111克，0.248摩尔)的二氯甲烷溶液冷却至-5℃，用1M三溴化硼的二氯甲烷溶液(322毫升，0.322摩尔)处理1小时，搅拌1小时，依次用水和盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生标题产物的黄色固体(105克，98.1％)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989801831
X    R            R1     W1         W2    W3   W4   mp℃H    CH3         CF3    I           H      H     OHH    CH3         CF3    H           CH3   H     OHH    CH3         CF3    CH3        CH3   H     OH    265-266H    CH3         CH3    CH3        H      H     OH    ＞250H    CH3         CF3    CH3        H      H     OHH    CH2CH＝CH2 CF3    CH3        H      H     OHH    CH3         CF3    CH3        H      CH3  OHH    CH3         CF3    C2H5      H      H     OHH    CH3         CF3    CH(CH3)2  H      H     OHH    C2H5       CH3    CH3        H      H     OHH    CH3         CF3    H           H      H     OHH    CH3         CF3    H           OH     H     HH    CH3         CF3    CHO         H      H     OHH    CH3         CF3    H           CH3   CH3  OH    ＞260H    CH3         CF3    H           H      OH    H     200-202H    CH3         CF3    I           CH3   H     OH    ＞250H    CH3         CF3    -(CH2)3-        H     OH    244-247H    CH3         CF3    OH          H      H     OH    239-242H    CH3         CF3    OCH3       H      H     OH    180-182H    CH3         CF3    CH3        H      Cl    OH    232-235F    CH3         CF3    CH3        H      H     OH
实施例10
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-5-基}-对-甲苯基}氧基}乙酸甲酯的制备
使3-[3-(6-羟基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(70.6克，0.163摩尔)，碳酸钾(27.1克，0.196摩尔)及溴乙酸甲酯在N，N-二甲基甲酰胺里的混合物于室温下搅拌39小时，用乙酸乙酯稀释，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到黄色泡沫状物。此黄色泡沫状物使用硅胶及39∶1至9∶1二氯甲烷的乙醚溶液进行快速柱层析，产生标题产物的白色泡沫状物(67.9克，82.4％)，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：R      R1    W1    W2  W3   W5         W6       W7  mp℃CH3   CF3   CH3   H    H        HCH3   CF3   CH3   H    H             CO2CH3      H    100-110CH3   CF3   H      CH3 H             CO2CH3      H    160-162CH3   CF3   H      CH3 H             CO2CH3      H    162-163.5CH3   CF3   CH3   CH3 H             CO2CH3      H    128-130 R      R1     W1    W2   W3   W5   W6       W7   mp℃CH3    CH3    CH3   H     I     H     CO2CH3  HCH3    CH3    CH3   CH3  H     CH3  CO2CH3  HCH3    CH3    CH3   Cl    H     H     CO2CH3  H    165-167CH3    CH3    I      H     H     CH3  CO2CH3  H    178-180CH3    CH3    I      H     H     H     CO2CH3  H    183-184CH3    CH3    I      CH3  H     H     CO2CH3  H    203-206CH3    CH3    I      CH3  H     CH3  CO2CH3  H    179-181CH3    CH3    CH3   H     H     CH3  CO2CH3  H    100-1061CH3    CH3    CH3   H     H     CH3  CO2CH3  H    99-1042
1R-异构体
2S-异构体 R      R1     W1           W2  W3  W5    W6       W7  mp℃CH3    CF3    CH3          H    CH3 H      CO2CH3  H    139-141CH3    CF3    CH3          H    CH3 CH3   CO2CH3  H    88CH3    CF3    C2H5        H    H    CH3   CO2CH3  H    75-77CH3    CF3    CH3          H    H    C2H5 CO2CH3  HCH3    CF3    CH(CH3)2    H    H    CH3   CO2CH3  H    90-92.5CH3    CH3    CH3          H    H    H      CO2CH3  H     117-125CH3    CH3    CH3          H    H    CH3   CO2CH3  H     112-115C2H5  CH3    CH3          H    H    H      CO2CH3  H     77-85CH3    CF3    CH3          H    H    CH3   CO2CH3  HCH3    CF3    CH3          H    H    H      C≡CH      H R      R1     W1     W2  W3  W5  W6                W7   mp℃CH3    CF3    CH3    H    H    H    CN                  HCH3    CF3    CH3    H    H    CH3 CN                  HCH3    CF3    CH3    H    H    CH3 CH3                HCH3    CF3    CH3    H    H    H    CH3                HCH3    CF3    CH3    H    H    H  
Figure A9880989801881
            HCH3    CF3            H    H    H    CH＝CHCO2CH3      HCH3    CF3    CH3    H    H    H    (CH2)2CO2C2H5 HCH3    CF3    CH3    H    H    H    CH2CO2CH3        HCH3    CF3    CH3    H    H    H    CO2C(CH3)3       H
R          R1     W1        W2     W3     W5       W6            W7       mp℃
CH3       CF3    CH3       H       H       H         CH(CH3)2     H
CH3       CF3    CH3       H       H       H         CH＝CH2        H
CH3       CF3    CH3       H       H       CH3      CO2C(CH3)3  H
CH3       CF3    CH3       H       H       C2H5    CO2CH3       H
CH3       CF3    CH3       H       H       CH3      CO2CH3       CH3
CH3       CF3    CH3       H       H       n-C3H7  CO2CH3       H
CH3       CF3    CH3       H       H       CH3      CO2C(CH3)3  CH3
CH3       CF3    H          CH3    H       H         CO2CH2C≡CH  H         192-195CH2CH＝CH2   CF3    CH3       H       H       H         CO2CH2C≡CH  H         138-145
CH3       CF3    CH3       CH3    H       H         CO2CH2C≡CH  H         188.5-190 R      R1     W1    W2   W3        W5          W6             W7       mp℃C2H5  CF3    CH3   H     H          H            CO2CH3        HCH3    CF3    CH3   H     H          H            CH＝CHCO2CH3  HCH3    CF3    CH3   H     H          n-C3H7    CO2C2H5      HCH3    CF3    H      H     H          H            CO2CH3        H         154-156CH3    CF3    H      H     H          CH3         CO2CH3        H         174-175CH3    CF3    H      H     H          H            CO2CH2C≡CH   H         148-150CH3    CF3    CH3   Cl    H          CH3         CO2CH3       H         93-104CH3    CF3    CHO    H     H          H            CO2CH3        H         78-81CH3    CF3    CH3   H     H          H            C(O)C6H5      HR       R1     W1    W2  W3  W5    W6                 W7   mp℃CH3    CF3    CH3   H    H    H    
Figure A9880989801911
   HCH3    CF3    CH3   H    H    H      C(O)C(CH3)3       HCH3    CF3    H      H    H    H      C(O)C(CH3)3       HCH3    CF3    H      H    H    CH3 
Figure A9880989801912
   HCH3    CF3    CH3   H    H    H      CH2CH(OCH3)2      H    70-75CH3    CF3    H      CH3 CH3 H      CO2CH3            H    96-98CH3    CF3    H      CH3 CH3 CH3   CO2CH3            HCH3    CF3    H      CH3 CH3 H      CO2CH2C≡CH       H    155-156CH3    CF3    OCH3  H    H    H      CO2CH3            H    148-151CH3    CF3      -(CH2)3-   H    H    CO2CH3                        H     166-167CH3    CF3      -(CH2)3-   H    CH3 CO2CH3                        H    108-113CH3    CF3      -(CH2)3-   H    H    CO2CH2C≡CH                   H     188-190CH3    CF3    CH3      H    H    F    CO2CH3                        FCH3    CF3    CH3      H    H    CH3 
Figure A9880989801921
       HCH3    CF3    CH3      H    H    H    
Figure A9880989801922
    HX       W1     W2     W3     W4                mp℃Cl       CH3    H       H       OCH2CO2CH3F       CH3    H       H       OCH2CO2CH3F       H       H       H       OCH2CO2CH3F       H       H       H       OCH(CH3)CO2CH3F       CH3    H       H       OCH(CH3)CO2CH3X         W1            W2                   W3            W4          mp℃H         H              H                  OCH2CH3         H         173-174H         H              H                  OCH(CH3)2       H         189-190H         H         OCH2CO2CH3              H              H         164-166H         H         OCH(CH3)CO2CH3          H              H         149-153H         H         OCH2CO2CH2C≡CH         H              H         144-146H         H         OCH2CO2C(CH3)3         H              H         150-152H         H              H               OCH(CH3)CO2CH3    H         119-121H         H              H               OCH2CO2CH2C≡CH   H         178.5-180H         H              H               OCH2CO2CH3        H         201.5-202
实施例11
2-氯-2’-甲氧基-5’-甲基-5-硝基苯酮肟的制备
Figure A9880989801951
用羟胺盐酸盐(102.3克，1.47摩尔)的水溶液处理2-氯-2’-甲氧基-5’-甲基-5-硝基苯酮(90.0克，0.294摩尔)在乙醇中的混合物，回流过夜，倒至冰上。所得的水性混合物过滤得到固体。以水洗涤固体，在热真空的烘箱中干燥过夜，产生标题产物的白色固体(84.2克)，以1H NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：X         W            W2              W3        mp℃H         OCH3        H                H          173-178H         H            H                H          143-145H         H            OCH3            H          191-192.5H         OCH3        H                FH         H            OCH2CO2CH3   H           150-155H         OCH3        H                CH3       185.5-186.5F         OCH3        H                CH3
实施例12
3-(6-甲氧基-间-甲苯基)-5-硝基-1，2-苯并异噁唑的制备
Figure A9880989801961
将2-氯-2’-甲氧基-5’-甲基-5-硝基-苯酮肟(84.0克，0.262摩尔)在乙醇中的混合物温热到65℃，用150毫升10％氢氧化钾溶液处理25分钟，加热至78℃达1小时，冷却并倒至冰上。所得水性混合物过滤得到固体。固体以水洗涤，干燥，用N，N-二甲基甲酰胺重结晶，依次用N，N-二甲基甲酰胺及乙醇洗涤，在80℃的真空烘箱中干燥，产生标题产物的固体(mp 225-226℃)，以1H NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989801962
X         W       W1       W2        mp℃H         OCH3   H         H          170-171H         H       H         H          138-139H         H       H         OCH3      205-207F         OCH3   CH3      H
实施例13
5-氨基-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑和5-氨基-4-氯-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑的制备
Figure A9880989801971
温热3-(6-甲氧基-间-甲苯基)-5-硝基-1，2-苯并异噁唑(20.0克，0.0703摩尔)在乙酸(380毫升)中的混合物，用氯化亚锡(II)二水合物(47.4克，0.210摩尔)在浓盐酸(110毫升)中的温溶液处理，回流1小时，冷却至10℃，真空浓缩，得到胶状物。搅拌下将此胶状物加到水中，得到浆状物。此浆状物用80克50％氢氧化钠溶液处理，在60℃至80℃下搅拌1小时，冷却并倾析得到残留物。用氢氧化钾(10克)处理该残留物在乙醇中的混合物，加热过夜，冷却至室温，以盐酸中和，真空浓缩，得到残留物。用乙酸乙酯稀释残留物，过滤。滤液经真空浓缩，使用硅胶及2％乙酸乙酯的二氯甲烷溶液层析，产生标题产物的半固体，以元素分析法及质谱分析法鉴定。
基本上采用相同方法，但改用5-硝基-3-苯基-1，2-苯并异噁唑替代3-(6-甲氧基-间-甲苯基)-5-硝基-1，2-苯并异噁唑，得到5-氨基-3-苯基-1，2-苯并异噁唑。
实施例14
3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989801981
使5-氨基-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑(8.40克，0.033摩尔)，2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(7.60克，0.036摩尔)和乙酸的混合物回流3小时，冷却，倒至冰上，加水稀释。所得水性混合物过滤得到固体。以水洗涤固体，干燥，产生标题产物的粉红色固体，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989801982
X         X1        W       W3     mp℃H         H          OCH3   H       214-216H         H          H       HH         Cl         OCH3   CH3F         H          OCH3   CH3
实施例15
3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(10.5克，0.0255摩尔)与碳酸钾(7.04克，0.051摩尔)在N，N-二甲基甲酰胺中的混合物搅拌15分钟，用甲基碘(7.24克，0.051摩尔)处理，搅拌过夜，倒至冰上。所得水性混合物用二氯甲烷萃取。合并有机萃取液，用水洗涤，用无水硫酸镁干燥，真空浓缩，得到褐色玻璃状物。采用硅胶及己烷/乙酸乙酯溶液(3∶1)对玻璃状物进行无水柱层析，产生标题产物的灰白色固体，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989801992
X         X1        W            W1        mp℃H         H          OCH3        HH         H          H            H         225-226.5H         Cl         OCH3        CH3F         H          OCH3        CH3F         H          OCH3        H
实施例16
3-[3-(6-羟基-间-甲苯基)-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮的制备
Figure A9880989802001
使3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(5.00克，0.0116摩尔)在二氯甲烷中的混合物冷却至-10℃，用15.1毫升1M三溴化硼的二氯甲烷溶液滴加处理，同时保持反应混合物温度在-15℃至0℃，温热至室温，滴加5毫升三溴化硼溶液，在室温下搅拌1小时，倒至稀盐酸中。所得水性混合物用丙酮稀释，真空浓缩，加水稀释，过滤得到固体。用水洗涤固体，在60℃的真空烘箱中干燥，产生标题产物的黄色固体，以质谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802002
X                  X1                     W3H                  H                       HH                  Cl                      CH3F                  H                       CH3F                  H                       H
实施例17
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-5-基}-对-甲苯基}氧基}乙酸甲酯的制备
Figure A9880989802011
使3-[3-(6-羟基-间-甲苯基)-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮(2.25克，0.00540摩尔)及碳酸钾(1.50克，0.0108摩尔)在N，N-二甲基甲酰胺中的混合物搅拌数分钟，用溴乙酸甲酯(0.903克，0.00590摩尔)处理，在室温下搅拌，倒至冰-水混合物中。所得水性混合物过滤得到固体。使用硅胶和4％醚的二氯甲烷溶液进行固体的无水柱层析，产生标题产物的玻璃状物，用NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802021
X        X1      W3        W5        W6                  mp℃H        H        H          H          CH3H        H        H          CH3       CH3H        H        CH3       CH3       CH3H        H        CH3       H          CH3H        H        CH3       H          CH2C≡CHH        H        CH3       CH3       CH2C≡CHH        Cl       CH3       CH3       C(CH3)3H        Cl       CH3       H          C(CH3)3F        H        CH3       CH3       CH3                97-99F        H        CH3       CH3       CH2CH3            118-120F        H        CH3       H          CH2CH3            88-91F        H        CH3       H          CH(CH3)2          152-155F        H        CH3       H          C(CH3)3           89-91H        Cl       CH3       H          CH3                105-150F        H        CH3       H          CH3                129-131F        H        H          H          CH3F        H        H          CH3       CH3F        H        H          H          CH(CH3)2F        H        H          CH3       CH(CH3)2F        H        CH3       H          CH2CH＝CH2F        H        CH3       H          CH2C≡CHF        H        H          H          CH2CH＝CH2F        H        H          H          CH2C≡CHF        H        CH3       CH3      CH2CH＝CH2X        X1       W3        W5        W6                  mp℃F        H         H          CH3       CH2CH＝CH2F        H         CH3       CH3       CH2C≡CHF        H         H          CH3       CH2C≡CHF        H         CH3       H         
Figure A9880989802031
F        H         CH3       CH3        F        H         H          H          F        H         H          CH3      
Figure A9880989802034
F        H         CH3       H          CH2C6H5F        H         CH3       CH3       CH2C6H5F        H         H          H          CH2C6H5F        H         H          CH3       CH2C6H5
实施例18
3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮和3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802035
使1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(16.6克，48.8毫摩尔)，N-溴琥珀酰亚胺(34.8克，195毫摩尔)及苯甲酰过氧化物(0.295克，1.22毫摩尔)在1，2-二氯乙烷中的混合物回流1小时，再用苯甲酰过氧化物(0.30克)处理，回流3.5小时，冷却至室温。冷却的反应混合物使用硅胶及二氯甲烷/己烷溶液(1∶1)进行柱层析，产生标题产物混合物，将它溶于二氯甲烷。所得有机溶液依次用15％亚硫酸氢钠溶液及水洗涤，用无水硫酸镁干燥，真空浓缩，得到黄色固体。此黄色固体使用硅胶及1％叔丁基甲基醚的二氯甲烷溶液进行柱层析，产生3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的灰白色固体，mp203-204℃，和3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的灰白色固体，mp107-110℃。
基本上采用相同方法，由1-甲基-3-(3-甲基-6-氟-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮制得下列化合物：
Figure A9880989802041
X1                 X2                 mp℃H                   Br                  185-187Br                  Br                  239-240
实施例19
3-[3-(甲氧甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
用甲醇稀释3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.750克，1.79毫摩尔)的1，2-二氯乙烷溶液，用三氟甲磺酸银(0.610克，2.37毫摩尔)处理，于室温下搅拌过夜，经硅藻土过滤。所得滤液用饱和碳酸氢钠溶液洗涤，用无水硫酸镁干燥，真空浓缩，得到固体。此固体使用硅胶及2％及5％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的白色固体(0.600克，mp 161-163℃)，以1H NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802061
X1                  W4                        mp℃H                    HH                    CH3H                    CH(CH3)2H                    CH2C6H5H                    CH2CH＝CH2H                    CH(CH2Cl)2H                    CH2CF3H                    (CH2)3CH3H                    CH(CH3)CH＝CH2H                    CH(CH3)CF3H                    HC2CH＝C(CH3)2H                    H                    (CH2)3CH＝CH2H                    CH2CH2CH＝CH2H                    C(O)CH3H                    CH2CH2FH                    C2H5H                    CH2CH2ClH                    CH2CH2OCH2CH3H                    CH2CHF2H                    HC2CH＝CHCH3H                    CH(CH2F)2H                    CH2CH2CH＝CHCH2CH3H                    HC2CH2CH2ClX                  W4                    mp℃H             H            
Figure A9880989802072
H             H            
Figure A9880989802074
H            
Figure A9880989802075
H            
Figure A9880989802076
H             H            
Figure A9880989802078
H            
Figure A9880989802079
X                   W4                   mp℃H            
Figure A9880989802081
H            
Figure A9880989802082
H            
Figure A9880989802083
H            
Figure A9880989802084
H            
Figure A9880989802085
H            
Figure A9880989802086
H            
Figure A9880989802087
H            
Figure A9880989802088
H            
Figure A9880989802089
X                 W4                      mp℃H            
Figure A9880989802091
H             H            
Figure A9880989802093
F                CH2OCH3                134-135
实施例20
{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫代}乙酸甲酯的制备
Figure A9880989802094
用硫代乙醇酸甲酯(90.0毫升，1.00毫摩尔)处理经已烷洗涤的氢化钠(0.0360克，60％油分散液，0.900毫摩尔)在四氢呋喃中的混合物，搅拌至气体停止释出为止，用3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.300克，0.710毫摩尔)的四氢呋喃溶液滴加处理，搅拌10分钟，真空浓缩，得到残留物。残留物用二氯甲烷及水稀释。分离有机相，用无水硫酸镁干燥，真空浓缩，得到油状物。此油状物使用硅胶及5％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的澄清油，以1H NMR光谱分法析鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802101
实施例21
1-甲基-3-{3-[(甲硫基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802102
用硫甲醇钠(0.332克，4.74毫摩尔)处理含3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.66克，3.95毫摩尔)的乙腈溶液，于室温下搅拌过夜，再用硫甲醇钠(约15毫克)处理，搅拌1小时，真空浓缩，得到残留物。残留物加二氯甲烷及水稀释。分离有机相，用盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到固体，此固体使用硅胶及2％乙醚的二氯甲烷溶液进行柱层析，产生标题化合物的白色固体，以1H NMR光谱分析法鉴定。
实施例22
间-氟苯基乙酸酯的制备
Figure A9880989802111
将3-氟苯酚(100克，0.890摩尔)的二氯甲烷溶液冷却至0℃至5℃，用吡啶(75.0毫升，0.930摩尔)处理，搅拌数分钟，滴加乙酰氯(66.0毫升，0.930摩尔)处理，同时保持反应混合物温度在17℃以下，在冰浴温度下搅拌2小时，温热至室温，倒至冰-水混合物中。分离有机相，用盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到标题产物的黄色油，以1H NMR光谱分析法鉴定。
实施例23
4’-氟-2’-羟基乙酰苯的制备
Figure A9880989802112
在冰浴中冷却乙酸间-氟苯基酯(123克，0.798摩尔)于冰浴中冷却，分批加入氯化铝(150克，1.12摩尔)，在190℃下搅拌1小时，冷却得到固体。向固体中加入冰、水和盐酸的混合物及二氯甲烷。所得混合物搅拌数分钟，分离各相。有机相依次用水、饱和碳酸氢钠溶液及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到标题产物(99.0克)，以1H NMR光谱分析法鉴定。
实施例24
4’-氟-2’-羟基乙酰苯，肟的制备
Figure A9880989802121
使4’-氟-2’-羟基乙酰苯(99.0克，0.640摩尔)、羟胺盐酸盐(89.0克，1.28摩尔)及乙酸钠(79.0克，0.960摩尔)在甲醇中的混合物回流1小时，倒至冰-水混合物中。所得水性混合物过滤得到固体。此固体溶于二氯甲烷中，所得有机溶液经无水硫酸镁干燥，真空浓缩，用己烷稀释，过滤，得到标题产物的固体(55.0克，mp 112-114℃)，以1H NMR光谱分析法鉴定。
实施例25
6-氟-3-甲基-1，2-苯并异噁唑的制备
将4’-氟-2’-羟基乙酰苯肟(47.0克，0.278摩尔)在四氢呋喃里的混合物加热至恰好回流为止，用1，1’-羰基二咪唑(55.0克，0.340摩尔)与三乙胺(39.0克，0.390摩尔)的四氢呋喃溶液处理，回流1小时，冷却，真空浓缩，倒至冰-水混合物中。所得水性混合物用醚萃取。合并有机萃取液，依次用饱和氯化铵溶液及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到油状物。此油状物使用硅胶及二氯甲烷/己烷溶液(1∶1)进行柱层析，产生标题产物的黄色油，以1H NMR光谱分析法鉴定。
实施例26
6-氟-3-甲基-5-硝基-1，2-苯并异噁唑的制备
用冰浴冷却6-氟-3-甲基-1， 2-苯并异噁唑(23.5克，0.156摩尔)在浓硫酸中的混合物，滴加90％硝酸(8.50毫升)处理，同时保持反应混合物温度在15℃以下，于冰浴温度下搅拌1小时，再以90％硝酸(5.80毫升)处理，温热到室温并搅拌过夜，倒至冰上。所得水性混合物过滤得到固体。固体风干，溶于二氯甲烷中。所得有机溶液经无水硫酸镁干燥，以己烷稀释，过滤，得到标题产物的紫色固体，以1H NMR光谱分析法鉴定。
实施例27
5-氨基-6-氟-3-甲基-1，2-苯并异噁唑及5-氨基-4-氯-6-氟-3-甲基-1，2-苯并异噁唑的制备
Figure A9880989802132
将6-氟-3-甲基-5-硝基-1，2-苯并异噁唑(3.00克，0.0153摩尔)及乙酸(85.0毫升)的混合物加热至40℃，用氯化亚锡(II)二水合物(9.70克，0.0430摩尔)及浓盐酸(45.0毫升)的溶液处理，回流90分钟，真空浓缩，用2N氢氧化钠溶液中和，过滤得到固体。此固体使用硅胶及二氯甲烷进行柱层析，得到标题产物的固体，以NMR光谱分析法鉴定
基本上采用相同方法，但改用乙酸乙酯/乙醇混合物替代乙酸，得到下列化合物：
Figure A9880989802141
X                          YH                          CH3H                          ClH                          OCH2CO2CH3H                          OCH(CH3)2H                          OCH(CH3)CO2CH3F                          OCH2CO2CH3H                          OCH3
实施例28
3-(-6-氟-3-甲基-1，2-苯并异噁唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使5-氨基-6-氟-3-甲基-1，2-苯并异噁唑(4.85克，0.029摩尔)与2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(6.70克，0.0320摩尔)在乙酸中的混合物回流90分钟，冷却至室温，倒至冰-水混合物中。所得水性混合物过滤得到固体。此固体风干，溶于乙酸乙酯中。所得有机溶液用盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生标题产物的黄色固体(7.00克，mp235-237℃)，以NMR光谱分析法鉴定。基本上采用相同方法，得到下列化合物：
Figure A9880989802151
X            X1           Y                     mp℃H            H             CH3                  283-182H            H             ClH            H             OCH2CO2CH3        180-182H            H             OCH(CH3)2           213-215H            H             OCH3                 230-235F            Cl            CH3                  125-130
实施例29
3-(6-氟-3-甲基-1，2-苯并异噁唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802152
使3-(6-氟-3-甲基-1，2-苯并异噁唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(3.00克，9.12毫摩尔)及碳酸钾(2.52克，18.2毫摩尔)在N，N-二甲基甲酰胺里的混合物搅拌15分钟，用甲基碘(2.58克，18.2毫摩尔)处理，在室温下搅拌过夜，倒至冰-水混合物中。所得水性混合物过滤，得到的固体用二氯甲烷/己烷溶液重结晶，得到标题产物的白色固体(mp 158-159℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802161
X            X1          Y                     mp℃H            H            CH3                  196-198H            H            Cl                    168.5-170H            H            OCH2CO2CH3        156-157H            H            OCH(CH3)2H            H            OCH3                 160-161F            Cl           CH3                  154-155
实施例30
2’-氯-5’-硝基乙酰苯，肟的制备
Figure A9880989802162
用羟胺盐酸盐(83.0克，1.19摩尔)的水溶液处理2’-氯-5’-硝基乙酰苯(50.0克，0.250摩尔)在乙醇中的混合物，回流过夜，冷却至室温，过滤，产生标题产物的固体(mp 165-167℃)，以NMR光谱分析法鉴定。
实施例31
3-甲基-5-硝基-1，2-苯并异噁唑的制备
用10％氢氧化钾溶液(7.86克KOH)滴加处理2’-氯-5’-硝基乙酰苯，肟(30.0克，0.140摩尔)的乙醇混合物，在室温下搅拌1小时，回流过夜，冷却，倒至水中。所得水性混合物过滤得到固体。此固体使用硅胶及二氯甲烷进行柱层析，产生标题产物的黄色固体(mp84.5-86.5℃)，以NMR光谱分析法鉴定。
实施例32
5-硝基-1，2-苯并异噁唑-3-醇的制备
Figure A9880989802171
向浓硫酸中分批加入1，2-苯并异噁唑-3-醇(19.7克，0.146摩尔)，在所得反应混合物中滴加70％硝酸(11.3毫升)处理，搅拌90分钟，倒至冰上。所得水性混合物过滤，得到蜡状糊状物。此糊状物用甲醇/水混合物重结晶，产生标题产物的固体，以1H NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802172
实施例33
[(5-硝基-1，2-苯并异噁唑-3-基)氧基]乙酸甲酯的制备
Figure A9880989802173
使5-硝基-1，2-苯并异噁唑-3-醇(3.90克，0.0220摩尔)与碳酸钾(4.17克，0.0300摩尔)在N，N-二甲基甲酰胺中的混合物搅拌30分钟，用溴乙酸甲酯(3.96克，0.0260摩尔)处理，在室温下搅拌过夜，倒至酸性冰-水混合物中。所得水性混合物用乙酸乙酯萃取。合并有机萃取液，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到黄色油。此油使用硅胶及(1∶1)到(4∶1)二氯甲烷/己烷梯度进行柱层析，产生标题产物的白色固体(2.80克，mp 72-73.5℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：X                 Y                 mp℃H              OCH(CH3)2         81-83H              OCH2CH＝CH2       70-72H              OCH3               101.5-103Cl             OCH(CH3)CO2CH3  98-100F              OCH2CO2CH3      104-106
实施例34
3-氯-5-硝基-1，2-苯并异噁唑的制备
Figure A9880989802182
在玻璃圆桶中放入5-硝基-1，2-苯并异噁唑-3-醇(4.00克，0.0220摩尔)及磷酰氯(40.0毫升，65.8克，0.429摩尔)的混合物，于150-155℃下加热2小时，冷却过夜，真空浓缩，用二氯甲烷稀释，用碳酸氢钠溶液调至约pH8。分离各相。有机相依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到残留物。残留物使用硅胶及二氯甲烷/己烷溶液(1∶1)进行柱层析，产生标题产物的琥珀色油，以NMR光谱分析法鉴定。
实施例35
2-{{2-{5-[3，6-二氢-3-甲基-2-氧基-6-硫代-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-丙酸甲酯的制备
Figure A9880989802191
使2-{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯(2.00克，3.80毫摩尔)、碳酸氢钠(1.24克，14.8毫摩尔)与Lawesson试剂(2，4-双(4-甲氧苯基)-1，3-二硫杂-2，4-二磷烷-2，4-二硫化物，1.70克，4.20毫摩尔)在甲苯中的混合物回流2小时，过滤除去固体，真空浓缩，得到橙色泡沫状物。此泡沫状物使用硅胶及0％与1％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的橙色泡沫状物(1.45克，mp110-112℃)，以NMR光谱分析法鉴定。
实施例36
2-氯-2’-甲氧基-5-硝基苯酮的制备
Figure A9880989802201
使2-溴苯甲醚(27.9克，145毫摩尔)的乙醚溶液冷却至-70℃，用丁基锂(64.0毫升，160毫摩尔)处理，于-70℃下搅拌1小时，用0.5M氯化锌的四氢呋喃溶液(320毫升，160毫摩尔)处理，于-70℃下搅拌1小时，加温至约0℃，真空浓缩，得到黄绿色油。该油的四氢呋喃溶液依次用四(三苯基膦)钯(O)(5.00克，4.35毫摩尔)及2-氯-5-硝基苯甲酰氯(35.0克，159毫摩尔)的四氢呋喃溶液洗涤，搅拌3天，倒至10％盐酸中，所得水性混合物用二氯甲烷萃取。合并有机萃取液，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到半固体。此固体与乙醚研磨，产生标题产物的黄色固体，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802211
W1          W2             W3           W4            mp℃H            Cl              H             OCH3          96-99H            H               CH3          OCH3          71-74F            H               H             OCH3Cl           H               H             OCH3          124-126OCH3        H               H             OCH3          71-73H            OCH3           H             OCH3          98-100H            F               H             OCH3W1          W2            W3           W4            mp℃H            H               CH3          H              65-66.5H            H               SCH3         H              87-88H            H               H             F              118-120H            H               H             CH3           78-79.5H            H               H             SCH3          123-124.5H            F               H             HH            H               OCH3         HH            H               H             OCH3H            CH3            CH3         OCH3
实施例37
2-氯-2’-甲氧基-5-硝基二苯基甲醇的制备
向镁(7.10克，0.293摩尔)在醚中的混合物里分批加入2-溴苯甲醚(50.0克，0.267摩尔)的醚溶液。添加完毕后，使反应混合物加热回流1小时，用醚稀释，冷却至0℃，用2-氯-5-硝基苯甲醛(39.0克，0.210摩尔)的四氢呋喃溶液处理，温热到室温，用冰-水混合物稀释。以盐酸(pH2-pH3)酸化水性混合物后，分离有机相，以醚萃取水相。合并有机相，依次用10％碳酸氢钠溶液及盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生标题产物的褐色胶状物。
基本上采用相同方法，得到下列化合物：
Figure A9880989802221
W                          W3                         W4OCH3                      H                           OCH3CH3                       H                           OCH3F                          H                           OCH3H                          OCH3                       H
实施例38
2-氯-2’-甲氧基-5-硝基苯酮的制备
Figure A9880989802222
向2-氯-2’-甲氧基-5-硝基二苯基甲醇(64.2克，0.219摩尔)中分批添加氧化铬(VI)(91.0克，0.919摩尔)的水/乙酸溶液(1∶4)，同时保持反应混合物温度在25℃至35℃。反应混合物于25℃至35℃下搅拌1小时，冷却，加水稀释，真空浓缩，得到残留物。残留物加水稀释，以二氯甲烷萃取。合并有机萃取液，用无水硫酸钠干燥，与硅胶(10克)混合，过滤。滤液真空浓缩，得到油状物，该油状物的甲醇/水溶液经炭脱色，真空浓缩，得到残留物。此残留物用硅胶及二氯甲烷/己烷溶液进行柱层析，产生标题产物的白色固体。
基本上采用相同方法，得到下列化合物：
Figure A9880989802231
W1               W3               W4                  mp℃OCH3             H                 OCH3CH3              H                 OCH3                109-111F                 H                 OCH3                94-95H                 OCH3             H                    79-81
实施例39
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸的制备
Figure A9880989802232
将三氟乙酸(75毫升)加到2-{{2-{5[3，-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸叔丁酯(12.0克，21.4毫摩尔)的二氯甲烷溶液中。反应混合物于室温下搅拌24小时，真空浓缩，产生标题产物的黄色泡沫状物，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802241
W3              W5              W6             mp℃
CH3             CH3             CH3
H                H                H               152-158
H                CH3             H               215-216
CH3             H                H基本上采用相同方法，也得到下列化合物：
实施例40
2-{{2-{5-[3，6-二氢-3-甲基-2，6二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸2-丙炔基酯的制备
Figure A9880989802251
使2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸(0.510克，1.00毫摩尔)与草酰氯(0.380克，3.00毫摩尔)在二氯甲烷中的混合物于室温下搅拌30分钟，真空浓缩，得到黄色泡沫状物。此泡沫状物以二氯甲烷稀释，所得溶液用炔丙醇(0.110克，2.00毫摩尔)的二氯甲烷溶液处理，在室温下搅拌24小时，真空浓缩，得到油状物。此油状物使用硅胶，己烷/二氯甲烷溶液(1∶1)及5％乙醚的二氯甲烷溶液进行快速柱层析，产生标题产物(0.400克)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：W1               W5              W6                  W7CH3              CH3             H               OCH2CH＝CH2CH3              CH3             H               OCH2C≡CCH3CH3              CH3             H               OCH2CH2ClCH3              CH3             H               OCH(CH3)2CH3              H                H               OCH(C2H5)2CH3              H                H               OCH2C(CH3)3CH3              H                H               OCH2CH＝CHCH3CH3              H                H               OCH2CF3CH3              H                H               OC2H5CH3              H                H               OCH(CH3)2CH3              H                H               OCH2C≡CHCH3              H                H               N(C2H5)2CH3              H                H               N[CH(CH3)2]2CH3              H                H               OCH2CH＝CH2CH3              H                H               OCH2CH2N(CH3)2CH3              H                H               OCH2CH2ClCH3              H                H               OCH(CH3)C≡CHW1               W5            W6                W7CH3              H              H              OCH2C≡CCH3CH3              H              H              OCH(CH3)C≡CCH3CH3              H              H              OCH2C(CH3)＝CH2CH3              H              H              OCH2CH＝C(CH3)2CH3              H              H              OCH2CH2OCH2CH3              H              H              O-N＝C(CH3)2CH3              H              H              OCH(CH3)(CH2)4CH3CH3              H              H              O(CH2)11CH3CH3              H              H              OCH2CO2CH3CH3              H              H              OCH2CH2C(CH3)＝CH2CH3              H              H              OCH2CH＝CH-CH＝CHCH3CH3              H              H              OCH(CH3)CH＝CH2CH3              H              H              OCH(CH3)CO2CH3CH3              H              H              OCH(CH3)CH2OCH3CH3              H              H              OCH2CH2CNCH3              H              H              OCH2CF2CF3CH3              H              H              OCH(CH3)(CH2)8CH3CH3              H              H              NHCH2C≡CHCH3              CH3           H              OC(CH3)3CH3              H              H            
Figure A9880989802271
CH3              H              H            
Figure A9880989802272
CH3              CH3           H            
Figure A9880989802273
CH3              H              H            
Figure A9880989802274
CH3              H              H            
Figure A9880989802275
W1               W5              W6               W7CH3              H                H               
Figure A9880989802281
CH3              H                H               
Figure A9880989802282
CH3              H                H               
Figure A9880989802283
CH3              H                H                CH3              H                H               
Figure A9880989802285
CH3              H                H               
Figure A9880989802286
CH3              H                H               
Figure A9880989802287
CH3              H                H               
Figure A9880989802288
CH3              H                H               
Figure A9880989802289
CH3              H                H               
Figure A98809898022810
CH3              CH3             CH3             OCH2CH2ClCH3              CH3             CH3             OCH2CF3CH3              CH3             CH3             OCH2CH2OH3CH3              CH3             CH3             OCH(CH3)2W1               W5             W6             W7H                 H               H               N(CH3)2CH3              H               H               NHCH3H                 H               H               NHCH3H                 H               H               NH2H                 H               H               N(CH3)OHCH3              H               H               N(CH3)OHH                 H               H               N(CH3)OCH3CH3              H               H               NH2CH3              H               H               NHOHCH3              H               H               NHOCH3CH3              H               H              
Figure A9880989802291
CH3              H               H               O(CH2)4SCH3CH3              H               H               O(CH2)8CH3CH3              H               H               OCH(CH＝CH2)(CH2)3CH3CH3              H               H               OCH2C(C2H5)(CH2OCH2CH＝CH2)2CH3              H               H               OCH2CH2C≡(CH2)5CH3CH3              H               H              
Figure A9880989802292
                                             单个非对映异构体CH3              H               H              
                                             单个非对映异构体CH3              H               H              O(CH2)10CH＝CHCH2CH3CH3              H               H              OCH2C(CH3)(CH3)CH2C6H5CH3              H               H              OCH2C(O)CH3CH3              H               H              OCH2CH2C(O)CH3
实施例41
2-氯-4-氟-5-硝基苯甲酰氯的制备
Figure A9880989802301
用草酰氯(30.8毫升，0.353摩尔)滴加处理2-氯-4-氟-5-硝基苯甲酸(50.0克，0.228摩尔)与N，N-二甲基甲酰胺(5滴)在1，2-二氯乙烷中的混合物，回流3小时，冷却，真空浓缩，得到标题产物的澄色固体，以NMR光谱分析法鉴定。
实施例42
2’-氯-4’-氟-5’-硝基乙酰苯的制备
用2-氯-4-氟-5-硝基苯甲酰氯(2.00克，8.40毫摩尔)的四氢呋喃溶液滴加处理2M甲基锌化氯的四氢呋喃(5.00毫升，10.1毫摩尔)溶液，用四(三苯基膦)钯(0)(0.400克，0.350毫摩尔)处理，于室温下搅拌1小时，倒至3N盐酸中。所得水性混合物以乙酸乙酯萃取。合并有机萃取液，依次用水及饱和碳酸氢钠溶液洗涤，用无水硫酸镁干燥，真空浓缩，得到深色液体。此液体使用硅胶及二氯甲烷的己烷溶液(6∶4)进行快速柱层析法，产生标题产物的灰白色固体(mp 66-68℃)，以NMR光谱分析法鉴定。
实施例43
6-氨基-3-甲基-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989802311
将2’-氯-4’-氟-5’-硝基乙酰苯(12.0克，0.0552摩尔)、硫(1.77克，0.0552摩尔)、30％氢氧化铵溶液(100毫升，0.856摩尔)、及甲醇的混合物放入不锈钢圆桶中，于85℃下加热过夜，冷却，再用硫(0.270克)及30％氢氧化铵溶液(50毫升)处理，于85℃下加热过夜，冷却，过滤除去固体，用乙酸乙酯萃取。合并有机萃取液，用水及盐水依次洗涤，用无水硫酸镁干燥，真空浓缩，得到固体。此固体使用硅胶，及0％、1％及2％乙醚的二氯甲烷溶液进行快速柱层析，产生标题产物的橙色固体(4.19克，mp 189-191℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802312
实施例44
6-氯-3-甲基-5-硝基-1，2-苯并异噻唑的制备
将亚硝酸叔丁酯(3.30毫升，0.0278摩尔)及氯化铜(II)(2.98克，0.0222摩尔)在乙腈中的混合物加热至65℃，用6-氨基-3-甲基-5-硝基-1，2-苯并异噻唑(3.88克，0.0185摩尔)分批处理，于65℃下搅拌，冷却至室温，倒至20％盐酸中。所得水性混合物用乙酸乙酯萃取。合并有机萃取液，用20％盐酸洗涤，用无水硫酸镁干燥，真空浓缩，得到固体，此固体使用硅胶及二氯甲烷/己烷溶液(1∶1与3∶1)进行快速柱层析，产生标题产物的浅黄色固体(2.54克，mp 156-158℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802321
实施例45
6-氟-3-甲基-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989802322
在密封的试管里对6-氯-3-甲基-5-硝基-1，2-苯并异噻唑(2.25克，9.80毫摩尔)、氟化钾(2.85克，49.0毫摩尔)及18-冠-6(1.50克，5.70毫摩尔)在乙腈里的混合物加热29天，过滤除去固体，部份真空浓缩，得到液体。以乙酸乙酯稀释此液体，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到深褐色固体。此固体使用硅胶及10％至50％乙酸乙酯的己烷梯度溶液进行快速柱层析，产生含两种成份的黄色固体。此黄色固体使用硅胶及50％至70％二氯甲烷的己烷梯度溶液进行快速柱层析，产生标题产物的浅黄色固体(0.870克，mp 118-119℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802323
实施例46
5-氨基-6-氟-3-甲基-1，2-苯并异噻唑的制备
将6-氟-3-甲基-5-硝基-1，2-苯并异噻唑(0.740克，3.50毫摩尔)，5％乙酸(25.0毫升)及乙酸乙酯的溶液加热至65℃，用铁粉(0.980克，17.5毫摩尔)处理，于65℃下搅拌1小时，冷却至室温，过滤除去固体。分离有机相，依次用水、饱和碳酸氢钠溶液及盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生标题产物的橙色固体(0.610克)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802332
实施例47
2-氯-4-氟-5-硝基苯酮的制备
Figure A9880989802333
使2-氯-4-氟-5-硝基苯甲酰氯(26.7克，0.112摩尔)与苯(12.0毫升，0.134摩尔)的1，1，2，2-四氯乙烷溶液冷却至0℃至5℃，用氯化铝(18.1克，0.136摩尔)处理，于约8℃下搅拌15分钟，加热至50℃并搅拌1小时，冷却至室温，依次用冰-水混合物及浓盐酸稀释。分离有机相，依次用水及饱和碳酸氢钠溶液洗涤，用无水硫酸镁干燥，真空浓缩，得到固体，此固体使用硅胶及二氯甲烷进行快速柱层析，产生标题产物的橙色固体(30.8克)，以NMR光谱分析法鉴定。
实施例48
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯，S，S-二氧化物的制备
Figure A9880989802341
使2-{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸甲酯(2.00克)与3-氯过氧苯甲酸(2.00克)在氯仿(50.0毫升)中的混合物于室温下搅拌过夜，以饱和碳酸氢钠溶液(100毫升)稀释。分离有机相，用无水硫酸钠干燥，真空浓缩，以甲醇(15.0毫升)稀释，加热，冷却至室温，过滤得到固体。用甲醇洗涤此固体，风干，得到标题产物的黄色粉末(1.50克，mp 225-226℃)。
实施例49
3-{3-[5-(溴甲基)-2-甲氧基-苯基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)嘧啶二酮与3-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧苯甲醛的制备
Figure A9880989802351
使3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮(5.00克，11.2毫摩尔)、N-溴琥珀酰亚胺(3.00克，16.9毫摩尔)及苯甲酰过氧化物(0.460克，1.90毫摩尔)在四氯化碳中的混合物回流过夜，冷却至室温，以二氯甲烷稀释，过滤除去固体。滤液依次用5％偏硫酸氢钠溶液及5％碳酸氢钠溶液洗涤，用无水硫酸镁干燥，真空浓缩，得到琥珀色油。此油使用硅胶及己烷/乙酸乙酯溶液(9∶1)进行柱层析，产生3-{3-[5-(溴甲基)-2-甲氧苯基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)嘧啶二酮的浅黄色固体(0.700克，mp 158-160℃)及3-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧苯甲醛的浅黄色固体(1.50克，mp 118-120℃)。
实施例50
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}三甲基溴化铵的制备
将3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(20.0克，0.0480摩尔)与甲苯的混合物加热至90℃，冷却至室温，用液体三乙胺(8.60克，0.145摩尔)处理，于室温下搅拌90分钟，过滤得到固体，用甲苯洗涤此固体，于45-50℃的真空烘箱中干燥，得到标题产物的白色固体，以NMR光谱分析法鉴定。
基本上采用相同方法，但改用合适的仲胺，得到下列化合物：W9                  W10                          mp℃CH3                 CH2CO2C2H5              119-121CH3                 CH3                         200-201
 -CH≡CH-N＝CH-                                206-207H                    SO2CH3                     119-121
实施例51
N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰基}-对-甲苯磺酰胺的制备
使1，1’-羰基二咪唑(0.198克，1.22毫摩尔)及{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸(0.300克，0.610毫摩尔)在四氢呋喃中的混合物于室温下搅拌过夜，回流30分钟，冷却至室温，依次用对-甲苯磺酰胺(0.209克，1.22毫摩尔)的四氢呋喃溶液及1，8-重氮双环[5.4.0]十一碳-7-烯(0.204克，1.34毫摩尔)的四氢呋喃溶液处理，于室温下搅拌3小时，倒至10％盐酸中。所得水性混合物过滤得到固体。此固体用乙腈/水溶液重结晶，产生标题产物的灰白色固体(0.200克，mp 140-144℃)。
基本上采用相同方法，得到下列化合物：W3               W5            W6           W8              W9             mp℃CH3              H              H              CH3             HCH3              H              H                 HCH3              H              H                 HCH3              H              H                 HCH3              H              H             
Figure A9880989802385
    HW3               W5            W6             W8              W9             mp℃CH3              H              H                     HCH3              H              H          
Figure A9880989802392
       HCH3              H              H                     HCH3              H              H             HCH3              H              H          
Figure A9880989802395
     HCH3              H              H          
Figure A9880989802396
   HCH3              H              H          
Figure A9880989802397
      HCH3              H              H          
Figure A9880989802398
          HCH3              H              H           CH＝CH(C6H5)       HCH3              CH3           CH3        H                    CH3W3          W5        W6        W8                     W9        mp℃CH3         H          H                  H          120(dec)H            H          H          CH3                     H          151CH3         H          H        
Figure A9880989802402
    H           235-239CH3         H          H        
Figure A9880989802403
             H           204-207CH3         H          H                H           114-117CH3         H          H        
Figure A9880989802405
  H           156-158CH3         H          H        
Figure A9880989802406
       H          236H            CH3       H         CH3                    H          175-177CH3         H          H         CH2Cl                  H          174-184H            H          H         CH2Cl                  H           220-230CH3         H          H         CH3                    CH3       135-145H            H          H         CH3                    CH3       195-199
W3        W5        W6          W8               W9           mp℃
CH3        H          H         CH2CH2CH3        H
CH3        H          H         CH＝CH2             H
CH3        H          H         CH2CH3             H
H           H          H         CH(CH3)2           H
H           H          H         CH2CH2CH3         H
H           H          H         CH＝CH2              H
H           H          H         CH2CH3             H
CH3        H          H         CH(CH3)2           H
CH3        CH3       H         CH(CH3)2           H
CH3        CH3       H         CH2CH2CH3         H
CH3        CH3       H         CH＝CH2             H
CH3        CH3       H         CH2CH3             H
CH3        CH3       H         CH3                 H
CH3        H          H         (CH2)3CH3         H
H           H          H         (CH2)3CH3         H
CH3        CH3       H         (CH2)3CH3        H
H           H          H         N[CH(CH3)2]2      H
实施例52
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛的制备
用硝酸银(0.340克，0.00200摩尔)处理3-[3-(二溴甲基)-1，2-苯并异噻唑-5基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.500克，0.00100摩尔)在二噁烷/水中的混合物(5∶2)，回流90分钟，冷却至室温并于室温下搅拌过夜，回流3小时，冷却，经硅藻土过滤。所得滤液真空浓缩，得到水性混合物。用二氯甲烷萃取此水性混合物。有机萃取物依次用水及盐水洗涤，用无水硫酸镁干燥及真空浓缩，得到固体。此固体使用硅胶及二氯甲烷进行柱层析，产生标题产物的固体(0.240克，mp 193-194.5℃)。
基本上采用相同方法，由3-[6-氟-3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮制得5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基-6-氟-1，2-苯并异噻唑-3-甲醛。
实施例53
1-甲基-3-{3-[(甲基亚磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802421
用3-氯过氧苯甲酸(0.580克，60％，2.00毫摩尔)处理1-甲基-3-{3-[(甲硫基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.740克，1.90毫摩尔)的二氯甲烷溶液，于室温下搅拌5分钟，再用二氯甲烷稀释，用5％碳酸钠溶液洗涤，用无水硫酸镁干燥，真空浓缩，得到固体。此固体使用硅胶及10％乙酸乙酯的二氯甲烷溶液进行快速柱层析，产生标题产物的白色固体，以NMR光谱分析法鉴定。
基本上采用相同方法，由1-甲基-3-{3-[(苯硫基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮制得1-甲基-3-{3-[(苯亚磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮。
实施例54
1-甲基-3-{3-[(甲基磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802431
在室温下使1-甲基-3-{3-[(甲基亚磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.480克，1.24毫摩尔)及3-氯过氧苯甲酸(0.600克，60％，2.10毫摩尔)的二氯甲烷混合物，于室温下搅拌4小时，以5％碳酸钠溶液洗涤，用无水硫酸镁干燥，真空浓缩，得到固体。此固体使用硅胶及10％乙醚的二氯甲烷溶液进行快速柱层析，产生标题产物的白色固体，以NMR光谱分析法鉴定。
基本上采用相同方法，由1-甲基-3-{3-[(苯亚磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮制得1-甲基-3-{3-[(苯磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮。
实施例55
2-乙氧基-3-[3-(6-羟基-间甲氧基)-1，2-苯并异噻唑-5-基]6-(三氟甲基)-4(3H)-嘧啶酮的制备
Figure A9880989802441
将2-乙氧基-[3-(6-甲氧基-间-甲氧基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-4(3H)-嘧啶酮(0.490克，1.06毫摩尔)的二氯甲烷溶液冷却至-5℃，用1M三溴化硼的二氯甲烷溶液(1.38毫升，1.38毫摩尔)处理，搅拌6小时，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生标题产物的灰白色固体，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
实施例56
{{2-{5-[2-乙氧基-6-氧-4-(三氟甲基)-1(6H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯的制备
使2-乙氧基-3-[3-(6-羟基-间-甲苯基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-4(3H)-嘧啶酮(0.470克，1.05毫摩尔)、碳酸钾(0.190克，1.37毫摩尔)及溴乙酸甲酯(0.210克，1.37毫摩尔)在N，N-二甲基甲酰胺里的混合物，于室温下搅拌过夜，以乙酸乙酯稀释，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到固体。此固体使用硅胶及10％乙醚的二氯甲烷溶液进行快速柱层析，产生标题产物的灰白色固体(0.450克，mp 171-174℃)。
基本上采用相同方法，得到下列化合物：W5              W6                   mp℃H                CH3                  95-99CH3             CH3                  93-100H                CH2C≡CH             187-188
实施例57
2，2’-二硫双[5-硝基苯甲酸]的制备
Figure A9880989802462
用叔丁醇钾(55.5克，0.495摩尔)分批处理2-氯-5-硝基苯甲酸(100克，0.496摩尔)在乙醇中的混合物，再以乙醇稀释，加热至回流，以由硫化钠九水合物(60.0克，0.249摩尔)、硫(8.80克，0.274摩尔)及水形成的溶液分批处理，回流2小时，冷却至室温，用浓盐酸处理。所得酸性混合物搅拌1小时，过滤得到固体。此固体用水洗涤，风干，产生标题产物之黄色粉末，以NMR光谱分析法鉴定。
实施例58
5-硝基-1，2-苯并异噻唑-3(2H)-酮的制备
Figure A9880989802471
用N，N-二甲基甲酰胺(0.800毫升)处理2，2’-二硫双[5-硝基苯甲酸](44.6克，0.113摩尔)及亚硫酰氯(49.0毫升，0.670摩尔)的二氯甲烷溶液，回流过夜，真空浓缩，以1，2-二氯乙烷稀释。所得有机溶液用溴(22.5毫升，0.436摩尔)处理，于室温下搅拌20分钟，回流3.5小时，真空浓缩，得到残留物。使该残留物的1，2-二氯乙烷溶液在冰-水浴中冷却，用浓氨(112毫升)处理15分钟，于室温下搅拌16小时，于冰-水浴中冷却，用浓盐酸处理。所得水性混合物于室温下搅拌1小时，过滤得到固体。用水洗涤此固体，风干，得到标题产物的黄色固体，以NMR光谱分析法鉴定。
实施例59
3-氯-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989802472
使5-硝基-1，2-苯并异噻唑-3(2H)-酮(10.0克，0.0510摩尔)、磷酰氯(40.0毫升，0.429摩尔)与三丁胺(12.0毫升，0.050摩尔)的混合物于103-115℃下加热6小时，于室温下搅拌过夜，倒至冰-水混合物中。所得水性混合物用二氯甲烷萃取。合并的有机萃取液依次用水及饱和碳酸氢钠溶液洗涤，用无水硫酸钠干燥，真空浓缩，得到胶状物。此胶状物使用硅胶及二氯甲烷进行柱层析，产生标题产物的橙黄色固体，以NMR光谱分析法鉴定。
实施例60
α-氰基-5-硝基-1，2-苯并异噻唑-3-乙酸乙酯的制备
用冰浴-丙酮浴冷却乙醇钠溶液(预先由乙醇及钠(1.00克，0.0430摩尔)制备)，分批添加氰基乙酸乙酯(4.51克，0.0398摩尔)，于室温下搅拌30分钟，用3-氯-5-硝基-1，2-苯并异噻唑(4.27克，0.0199摩尔)处理，于室温下搅拌过夜，冷却至0℃，滴加10％盐酸(15.0毫升)处理。所得水性混合物于室温下搅拌1小时，过滤得到固体。以乙醇洗涤此固体，风干，产生标题产物的黄色固体，以NMR光谱分析法鉴定。
实施例61
5-硝基-1，2-苯并异噻唑-3-乙酸乙酯的制备
Figure A9880989802491
将α-氰基-5-硝基-1，2-苯并异噻唑-3-乙酸乙酯(6.67克，0.0229摩尔)加到乙酰氯(67.0毫升)的乙醇溶液中。使反应混合物回流过夜，冷却，过滤除去固体。所得滤液经真空浓缩，得到褐色半固体。使此半固体在乙醚中的混合物搅拌2小时，过滤得到固体。固体以乙醚洗涤，风干，得到标题产物的黄色晶体(1.04克，mp 91-92℃)。
实施例62
5-氨基-1，2-苯并异噻唑-3-乙酸乙酯的制备
Figure A9880989802492
使10％乙酸溶液(31.0毫升)于50℃下搅拌，以铁粉(0.656克)处理，滴加5-硝基-1，2-苯并异噻唑-3-乙酸乙酯(1.03克，3.88毫摩尔)的乙酸乙酯溶液处理，于50℃下搅拌2小时，再以铁粉(0.305克)处理，于50℃下搅拌15分钟，倒至饱和碳酸氢钠溶液中。所得水性混合物以乙酸乙酯萃取。合并的有机萃取液依次用水及盐水洗涤，用无水硫酸钠干燥，真空浓缩，得到油状物。此油状物使用硅胶及二氯甲烷进行柱层析，产生标题产物的黄色油。
实施例63
5-[3，6-二氢-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸乙酯的制备
使5-氨基-1，2-苯并异噻唑-3-乙酸乙酯(0.748克，3.16毫摩尔)与2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(0.660克，3.17毫摩尔)在乙酸中的混合物回流3小时，真空浓缩，以饱和碳酸氢钠溶液稀释。所得混合物以二氯甲烷萃取。合并有机萃取液，以水洗涤，用无水硫酸钠干燥，真空浓缩，产生标题产物的黄褐色固体，以NMR光谱分析法鉴定。
实施例64
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸乙酯的制备
Figure A9880989802502
使5-[3，6-二氢-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸乙酯(0.643克，0.00160摩尔)及碳酸钾(0.243克，0.00170摩尔)在N，N-二甲基甲酰胺中的混合物于室温下搅拌90分钟，以碘甲烷(0.320毫升，0.00500摩尔)处理，于室温下搅拌，加水稀释。所得水性混合物以二氯甲烷萃取。有机萃取液以水洗涤，用无水硫酸镁干燥，真空浓缩，得到褐色油。此油使用硅胶与10％乙酸乙酯的己烷溶液进行柱层析，产生标题产物的黄褐色固体(0.362克，mp 150-152℃)。
实施例65
5-氨基-1，2-苯并异噻唑-3-乙醇的制备
Figure A9880989802511
使5-氨基-1，2-苯并异噻唑-3-乙酸乙酯(3.14克，0.0133摩尔)在四氢呋喃里的混合物冷却至-8℃，滴加2M氢硼化锂的四氢呋喃溶液(5.00毫升，0.0100摩尔)处理，于室温下搅拌3.5小时，冷却至-5℃，再以氢硼化锂溶液(4.20毫升，0.0084摩尔)处理，于室温下搅拌过夜，冷却至0℃，依次添加水(5.00毫升)及10％盐酸(10.0毫升)中止反应，于室温下搅拌1小时，以饱和碳酸氢钠溶液(10.0毫升)中和，真空浓缩，得到残留物。此残留物以5％甲醇的二氯甲烷溶液稀释。所得混合物以水、盐水及二氯甲烷稀释。分离各相。有机相真空浓缩，得到橙色胶状物。此胶状物用甲醇结晶，产生标题产物的黄褐色固体，以NMR光谱分析法鉴定。
实施例66
3-[3-(2-羟乙基)-1，2-苯并异噻唑-5-基-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮乙酸酯的制备
Figure A9880989802521
使5-氨基-1，2-苯并异噻唑-3-乙醇(0.794克，4.09毫摩尔)及2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(0.850克，4.08毫摩尔)在乙酸里的混合物回流5小时，真空浓缩，得到黄褐色固体。以碳酸钾(0.615克，4.45毫摩尔)处理该固体的N，N-二甲基甲酰胺溶液，搅拌1小时，以碘甲烷(0.800毫升，12.8毫摩尔)处理，搅拌过夜，倒至冰-水混合物中。所得水性混合物以二氯甲烷萃取。合并的有机萃取液依次用水、3％盐酸、水、饱和碳酸氢钠溶液及水洗涤，用无水硫酸钠干燥，真空浓缩，得到固体。此固体使用硅胶及二氯甲烷进行柱层析，产生标题产物的白色固体，以NMR光谱分析法鉴定。
实施例67
3-[3-(2-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802531
使3-[3-(2-羟乙基)-1，2-苯并异噻唑-5-基-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮乙酸酯(1.00克，2.42毫摩尔)在10％盐酸(250毫升)里的混合物回流35分钟，经玻璃棉过滤去除固体。所得滤液冷却，以二氯甲烷萃取。合并的有机萃取液以水洗涤，用无水硫酸钠干燥，真空浓缩，产生标题产物的黄色固体，以NMR光谱分析法鉴定。
实施例68
5-硝基-1，2-苯并异噻唑-3-乙腈的制备
Figure A9880989802532
使5-硝基-1，2-苯并异噻唑-3乙酸乙酯(5.00克，17.2毫摩尔)、水(100毫升)及二甲亚砜(35.0毫升)的混合物于107℃下搅拌24小时，于室温下搅拌2天，倒至冰-水混合物中。所得水性混合物搅拌2小时，过滤得到固体。以水洗涤固体，风干，产生标题产物的黄褐色固体。
实施例69
α，α-二甲基-5-硝基-1，2-苯并异噻唑-3-乙腈的制备
Figure A9880989802541
使5-硝基-1，2-苯并异噻唑-3-乙腈(1.29克，5.89毫摩尔)在N，N-二甲基甲酰胺里的混合物冷却至-9℃，以氢化钠(1.00克60％油匀散液)处理，于-3℃下搅拌20分钟，以碘甲烷(5.00毫升)处理，于室温下搅拌4小时，倒至冰上。所得水性混合物以10％盐酸处理，以二氯甲烷萃取。合并的有机萃取液依次用水、饱和碳酸氢钠溶液及水洗涤，用无水硫酸钠干燥，真空浓缩，得到固体。此固体使用硅胶及二氯甲烷进行柱层析，产生标题产物的黄色固体，以NMR光谱分析法鉴定。
实施例70
α，α-二甲基-5-硝基-1，2-苯并异噻唑-3-乙酸乙酯的制备
使α，α-二甲基-5-硝基-1，2-苯并异噻唑-3-乙腈(0.913克，3.69毫摩尔)、水(0.450毫升)、浓硫酸(4.55毫升)及乙醇(9.10毫升)的混合物回流1小时，冷却，倒至冰上。所得水性混合物用饱和碳酸氢钠溶液中和，以二氯甲烷萃取。有机萃取液以水洗涤，用无水硫酸钠干燥，真空浓缩，得到固体。此固体使用硅胶及二氯甲烷进行柱层析，产生标题产物的浅黄色晶体。
实施例71
5-氨基-α，α-二甲基-1，2-苯并异噻唑-3-乙酸乙酯的制备
使α，α-二甲基-5-硝基-1，2-苯并异噻唑-3-乙酸乙酯(0.714克，2.42毫摩尔)、铁粉(0.500克)、10％乙酸(23.0毫升)及乙酸乙酯(23.0毫升)的混合物于54-58℃下搅拌1小时，冷却，倒至饱和碳酸氢钠溶液中。所得水性混合物以乙酸乙酯萃取。合并的有机萃取液依次用水及盐水洗涤，用无水硫酸钠干燥，真空浓缩，得到黄色油。此油使用硅胶及10％乙酸乙酯的二氯甲烷溶液进行柱层析，产生标题产物之浅褐色油，以NMR光谱分析法鉴定。
实施例72
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸乙酯的制备
Figure A9880989802552
5-氨基-α，α-二甲基-1，2-苯并异噻唑-3-乙酸乙酯(0.546克，2.06毫摩尔)和2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(0.430克，2.06毫摩尔)在乙酸中的混合物回流4.5小时，真空浓缩，用饱和碳酸氢钠溶液稀释。所得水性混合物以二氯甲烷萃取。合并的有机萃取液以水洗涤，用无水硫酸钠干燥，真空浓缩，得到褐色泡沫状物。用碳酸钾(0.312克，2.25毫摩尔)处理此泡沫状物的N，N-二甲基甲酰胺溶液，搅拌1小时，用碘甲烷(0.420毫升，6.70毫摩尔)处理，于室温下搅拌过夜，倒至含20毫升浓盐酸的冰-水混合物中。所得水性混合物以二氯甲烷萃取。合并的有机萃取液依次用10％盐酸、水、饱和碳酸氢钠溶液及水洗涤，用无水硫酸钠干燥及真空浓缩，得到褐色油。此油使用硅胶及33％乙酸乙酯的二氯甲烷溶液进行柱层析，产生粉红色泡沫状物，用乙醇重结晶，产生标题产物的粉红色晶体，mp 164-167℃。
实施例73
5-氨基-3-氯-1，2-苯并异噻唑的制备
Figure A9880989802561
用铁粉(8.40克，325筛目)及浓盐酸(8滴)处理3-氯-5-硝基-1，2-苯并异噻唑(2.00克)的甲苯溶液，加热至回流，滴加水(8.00毫升)处理，回流35分钟，冷却至室温，经硅藻土过滤。所得滤液真空浓缩，得到残留物。此残留物使用硅胶及乙酸乙酯/己烷溶液(1∶1)进行快速柱层析，产生标题产物。
实施例74
3-(3-氯-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802571
使5-氨基-3-氯-1，2-苯并异噻唑(1.10克)及2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(1.38克)在乙酸(15.1毫升)中的混合物于90-105℃下搅拌2小时，冷却至室温，过滤得到0.500克标题产物的固体。所得滤液加水稀释，过滤，再得到1.11克标题产物。
实施例75
3-(3-氯-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使3-(3-氯-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.06克)、碳酸钾(0.470克)及碘甲烷(0.500毫升)在N，N-二甲基甲酰胺里的混合物在室温下搅拌90分钟，再用碘甲烷(0.500毫升)处理，于室温下搅拌15分钟，加水稀释。所得水性混合物过滤得到固体。此固体以水洗涤，在室温下的真空烘箱中干燥，产生标题产物的固体，以NMR光谱分析法鉴定。
实施例76
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙二腈腈
Figure A9880989802581
使3-(3-氯-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.500克)、丙二腈(0.270克)及三乙胺(1.50克)在甲基亚砜中的混合物于60℃下搅拌15分钟，冷却至室温，加水稀释。所得水性混合物用乙酸乙酯萃取。有机萃取液以水洗涤，用无水硫酸镁干燥，真空浓缩，得到褐色油。萃取的水相用盐水稀释，用浓盐酸酸化，以乙酸乙酯萃取。有机萃取液用无水硫酸镁干燥，真空浓缩，得到褐色油。合并所得的油，使用硅胶及乙酸乙酯/己烷/甲醇/乙酸溶液(10∶10∶4∶1)进行快速柱层析，产生标题产物的油，用NMR光谱分析法鉴定。
实施例77
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈的制备
Figure A9880989802591
使3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.420克，0.00100摩尔)及氰化钠(0.0750克，0.00150摩尔)在乙腈中的混合物于室温下搅拌过夜，过滤得到固体。此固体溶于二氯甲烷中，所得溶液经无水硫酸钠干燥，真空浓缩，得到灰白色固体。此固体使用硅胶及10％乙酸乙酯的二氯甲烷溶液进行柱层析，产生标题产物的白色固体，以NMR光谱分析法鉴定。
基本上采用相同方法，由3-[3-(溴甲基)-6-氟-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮制得5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-6-氟-3-乙腈。
实施例78
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸乙酯的制备
用浓硫酸(10.0毫升)处理5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈(1.00克)、乙醇(20.0毫升)及水(1.00毫升)的混合物，回流15分钟，倒至冰-水混合物中。所得水性混合物用二氯甲烷萃取。合并的有机萃取液依次用水、饱和碳酸氢钠溶液及水洗涤，用无水硫酸钠干燥，真空浓缩，得到橙色泡沫状物。此泡沫状物使用硅胶及10％乙酸乙酯的二氯甲烷溶液进行柱层析，产生标题产物的固体，以NMR光谱分析法鉴定。
实施例79
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸的制备
Figure A9880989802611
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸乙酯(0.600克)、10％盐酸(20.0毫升)及1，2-二氯乙烷(2.00毫升)的混合物煮沸30分钟，同时使1，2-二氯乙烷蒸发，冷却，倒至冰上。所得水性混合物过滤得到固体。固体以水洗涤，风干，得到标题产物的白色固体(0.550克，mp240-242℃)。
实施例80
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸甲酯的制备
Figure A9880989802621
将乙酰氯(11.0毫升)加到已预先使用冰-丙酮浴冷却的甲醇(110毫升)中。所得混合物于室温下搅拌30分钟，用5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸(0.617克，1.60毫摩尔)处理，回流4小时，倒至饱和碳酸氢钠溶液中。所得水性混合物用二氯甲烷萃取。合并的有机萃取液以水洗涤，真空浓缩，得到残留物。残留物用丙酮/己烷溶液重结晶，产生标题产物的白色固体(0.540克，mp 175-176℃)。
实施例81
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酰胺的制备
Figure A9880989802631
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸(0.960克，0.00250摩尔)与1，1’-羰基二咪唑(0.420克，0.00259摩尔)的四氢呋喃混合物于室温下搅拌4.5小时，用氯化铵(0.230克，0.00430摩尔)处理，于室温下搅拌过夜，以浓氨水(1.00毫升)处理，搅拌5分钟，以10％盐酸酸化，真空浓缩，得到残留物。此残留物以5％甲醇之二氯甲烷溶液稀释，所得混合物搅拌3小时，过滤，得到固体。此固体用5％甲醇的二氯甲烷溶液洗涤，于水中形成浆状物，过滤及干燥，得到标题产物的白色固体，以NMR光谱分析法鉴定。
实施例82
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸钠(DL-型)的制备
使2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸(0.500克)及氢氧化钠(0.0360克)在水中的混合物于室温下搅拌过夜，真空浓缩至一半体积，过滤得到标题产物的固体，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：R                       X+CH3               NH+[CH(CH3)2]2H                  NH+[CH(CH3)2]2CH3                    NH3 +H                       NH3 +H                       Na+
实施例83
2-{{2-{4-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸-2-丙炔酯的制备
Figure A9880989802651
使2-{{2-{4-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸钠叔丁酯(1.00克，0.00172摩尔)、炔丙醇(20.0毫升)及甲磺酸(52.0毫克，0.542毫摩尔)的混合物于75-93℃下搅拌12小时，于室温下搅拌7小时，真空浓缩，得到残留物。残留物以二氯甲烷稀释，所得溶液通过硅胶管柱，真空浓缩，得到黄色胶状物。此胶状物溶于乙醚中，所得溶液以水洗涤，用无水硫酸镁干燥，及真空浓缩，得到黄色胶状物。此胶状物使用硅胶及醚/二氯甲烷/己烷溶液(4∶3∶7)进行柱层析，产生泡沫状物。此泡沫状物用二氯甲烷/己烷溶液重结晶，产生标题产物的白色固体，mp 137-147℃。
基本上采用相同方法，得到下列化合物：W5                             W8CH3                            CH3H                               CH2C≡CH
实施例84
[(5-硝基-1，2-苯并异噻唑-3-基)氧基]乙腈的制备
用碳酸钾(18.5克，134毫摩尔)处理5-硝基-1，2-苯并异噻唑-3(2H)-酮(17.5克，89.2毫摩尔)在N，N-二甲基甲酰胺中的混合物，于室温下搅拌30分钟，以溴乙腈(16.0克，133毫摩尔)处理，于室温下搅拌过夜，倒至冰上。所得水性混合物用盐酸酸化至pH3，用乙酸乙酯萃取。合并的有机萃取液依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到固体。此固体使用硅胶及二氯甲烷进行柱层析，产生标题产物的黄色固体(15.0克，mp 123-124.5℃)。
基本上采用相同方法，得到下列化合物：Y                        mp℃OCH3                    108-109OCH(CH3)2OCH2CH＝CH2OCH2C≡CH               115-117OCH2CO2CH3
实施例85
[(5-氨基-1，2-苯并异噻唑-3-基)氧基]乙腈的制备
Figure A9880989802672
使铁粉(13.0克，0.233摩尔)在5％乙酸溶液(65.0毫升)里的混合物加热至50℃，分批添加[(5-硝基-1，2-苯并异噻唑-3-基)氧基]乙腈(11.0克，0.047摩尔)、乙酸(100毫升)及乙酸乙酯(65.0毫升)的混合物，回流2小时，冷却至40℃，过滤除去固体。分离各相，用乙酸乙酯萃取水相，合并有机相及有机萃取液，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生标题产物的油状物，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989802681
                           Y
                          OCH3
                        OCH(CH3)2
                        OCH2CH＝CH2
                        OCH2C≡CH
                        OCH2CO2CH3
实施例86
{{5-[3，6-二氢-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}氧基}乙腈的制备
Figure A9880989802682
使[(5-氨基-1，2-苯并异噻唑-3-基)氧基]乙腈(4.30克，21.0毫摩尔)与2-二甲氨基-4-(三氟甲基)-6H-1，3-噁嗪-6-酮(4.37克，21.0毫摩尔)在乙酸中的混合物回流3小时，于室温下搅拌过夜，倒至冰-水混合物中。所得水性混合物过滤得到固体。此固体以水洗涤，于55℃的真空烘箱中干燥过夜，产生标题产物的褐色固体(2.63克，mp 254-258℃)。
基本上采用相同方法，得到下列化合物：Y                                          mp℃OCH3OCH(CH3)2                                180-185OCH2CH＝CH2                              210-212OCH2C≡CH                                 212-215OCH2CO2CH3
实施例87
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}氧基}乙腈的制备
Figure A9880989802692
使{{5-[3，6-二氢-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}氧基}乙腈(2.63克，7.15毫摩尔)与碳酸钾(1.97克，14.3毫摩尔)在N，N-二甲基甲酰胺中的混合物搅拌30分钟，用碘甲烷(2.03克，14.3毫摩尔)处理，于室温下搅拌过夜，倒至冰-水混合物中。所得水性混合物过滤得到固体。此固体溶于乙酸乙酯中，所得溶液依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到褐色固体。此固体使用硅胶及二氯甲烷进行柱层析，产生黄色固体。此黄色固体用二氯甲烷/己烷溶液重结晶，产生标题产物的灰白色固体，mp 265-266℃。
基本上采用相同方法，得到下列化合物：Y                          mp℃OCH3                      198-199OCH(CH3)2                125-127OCH2CH＝CH2              184-185OCH2C≡CH                 201-202.5OCH2CO2CH3             181-183
实施例88
3-[3-(二氯甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.750克，0.00150摩尔)与氯化锂(0.950克，0.0225摩尔)的N，N-二甲基甲酰胺溶液于室温下搅拌48小时，用乙酸乙酯稀释。所得混合物依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到泡沫状物。此泡沫状物使用硅胶、二氯甲烷及1％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的白色泡沫状物(0.530克，mp 148-149℃)。
基本上采用相同方法，但改用3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮替代3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，制得3-[3-(氯甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的白色固体，mp201-203℃。
实施例89
3-[3-(氟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802711
使3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.00克，0.00240摩尔)、14.4毫升1M四丁基氟化铵的四氢呋喃溶液(0.0144摩尔)与无水对甲苯磺酸(1.36克，0.00790摩尔)的四氢呋喃溶液于室温下搅拌30分钟，回流3小时，于室温下搅拌3天，回流22小时，部份真空浓缩，以乙酸乙酯稀释。所得混合物依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到橙色固体。此固体使用硅胶及2.5％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的白色固体(0.42克，mp 201-202℃)。
实施例90
3-[3-(二氟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802721
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(0.750克，0.00200摩尔)及二乙氨基三氟化硫(0.260毫升，0.00200摩尔)的二氯甲烷溶液于室温下搅拌1小时，再用二乙氨基三氟化硫(数滴)处理，于室温下搅拌90分钟，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到黄色固体。此固体使用硅胶及1％乙醚的二氯甲烷溶液进行快速柱层析，产生标题产物的白色固体(0.680克，mp 183-184℃)。
实施例91
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}膦酸二乙酯的制备
使3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.00克，0.00240摩尔)的乙醚混合物冷却至10℃，滴加亚磷酸三乙酯(0.580毫升，0.00340摩尔)处理，于10℃下搅拌90分钟，以10毫升四氢呋喃稀释，于室温下搅拌过夜，回流1天，冷却，部分真空浓缩，以二氯甲烷稀释。所得有机溶液以水洗涤，用无水硫酸镁干燥，真空浓缩，得到黄色固体。此固体使用硅胶及乙醚/二氯甲烷溶液(1∶1)进行柱层析，产生标题产物的白色固体(0.930克，mp 142-144℃)。
基本上采用相同方法，采用适当亚磷酸三烷基酯，得到下列化合物：
Figure A9880989802731
X              R23                  mp℃H              CH3                  124-127H              CH(CH3)2            55-65F              CH2CH3              65-75
实施例92
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}膦酸的制备
Figure A9880989802741
使{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}膦酸二乙酯(1.00克，0.00210摩尔)及溴三甲基硅烷(2.20毫升，0.0168摩尔)的二氯甲烷(5.0毫升)溶液于室温下搅拌过夜，真空浓缩，得到残留物。残留物用甲醇(10.0毫升)稀释，于室温下搅拌3.5小时，真空浓缩，得到黄褐色固体。固体于煮沸的二氯甲烷中研磨，过滤及干燥，得到标题产物的米色固体(0.650克，mp＞230℃)。
实施例93
1-甲基-3-(3-丙烯基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(Z)-及1-甲基-3-丙烯基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(E)-与(Z)-，(3∶1)的制备
Figure A9880989802751
使(乙基)三苯基膦化(1.15克，0.00310摩尔)之四氢呋喃混合物，以氢化钠(0.120克，0.00310摩尔)处理，于室温下搅拌1小时，用5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(1.00克，0.00280摩尔)在四氢呋喃中的混合物处理，于室温下搅拌1小时，过滤。所得滤液部份真空浓缩，以二氯甲烷稀释，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到橙色固体。此固体使用硅胶及1％乙醚之二氯甲烷溶液快速柱层析，得到1-甲基-3-(3-丙烯基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(Z)-型的白色固体(0.350克，mp 200-201℃)及1-甲基-3-(3-丙烯基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(E)-型与(Z)-型(3∶1)的白色固体(0.450克，mp 228-230℃)
基本上依相同方法且采用经适当取代之溴化鏻，得到下列化合物：
Figure A9880989802761
W10                   W11                mp℃
CO2CH3               H                   ＞230
C(O)CH3               H                   ＞230
CHO                    H                   ＞230
CH2Br                 H                   235(分解
C(O)C6H5             H
C(O)N(CH3)OCH2       H
CO2CH2＝CH2         H
CHO                     CH2CH3
实施例94
1-甲基-3-(3-吗啉基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802771
使3-(3-氯-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.300克)、吗啉(2.00克)及三乙胺(5.00克)在四氢呋喃中的混合物回流18小时，真空浓缩，得到残留物。残留物使用硅胶及25％与50％乙酸乙酯的庚烷溶液进行柱层析，产生标题产物的黄色固体(0.210克，mp 200-205℃)。
基本上采用相同方法，但改用合适的胺，得到下列化合物：
Figure A9880989802772
                    Y                     mp℃
                 NHSO2CH3              135-145
                 
Figure A9880989802773
             198-203
                 N(C2H5)2
                 
Figure A9880989802774
    ＞280
实施例95
3-[3-(叠氮甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802781
用叠氮化钠(0.325克，5.00毫摩尔)处理3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(2.00克，4.76毫摩尔)的N，N-二甲基甲酰胺溶液，于室温下搅拌过夜，以18-冠-6处理，于室温下搅拌2小时，倒至冰-水混合物中。所得水性混合物过滤得到固体。此固体以水洗涤，风干，得到标题产物的白色固体，以NMR光谱分析法鉴定。
实施例96
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}氨基磷酸二乙酯的制备
Figure A9880989802782
使3-[3-(叠氮甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.61克，4.20毫摩尔)及亚磷酸三乙酯(0.860毫升，5.00毫摩尔)在二噁烷里的混合物回流30分钟，真空浓缩，加水稀释，以二氯甲烷萃取。有机萃取液合并，用无水硫酸镁干燥，真空浓缩，得到黄色油。此油使用硅胶及10％至40％乙腈的二氯甲烷溶液柱层析，产生标题产物的黄色泡沫状物(1.00克，mp 133-134℃)。
实施例97
α-乙酰基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸叔丁酯的制备
使氢化钠(60％油中，0.293克，7.33毫摩尔)在四氢呋喃里的混合物冷却至0℃，滴加乙酰乙酸叔丁酯(1.00毫升，6.03毫摩尔)的四氢呋喃溶液，搅拌数分钟。滴加所得混合物至3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.40克，3.33毫摩尔)的甲基亚砜溶液中。添加完毕后，反应混合物倒至含微量10％盐酸的冰-水混合物中。所得水性混合物以二氯甲烷萃取。有机萃取液合并，用无水硫酸镁干燥，真空浓缩，得到油状物。此油状物使用硅胶及0％、2％、3％与15％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的固体，mp 76-78℃。
基本上采用相同方法，得到下列化合物：
Figure A9880989802801
                  Y                 mp℃
        
Figure A9880989802802
           70-71
        
Figure A9880989802803
           68-69
实施例98
1-甲基-3-[3-(3-氧丁基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与α-乙酰基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸的制备
Figure A9880989802804
使α-乙酰基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸叔丁酯(0.700克)与三氟乙酸(10.0毫升)在二氯甲烷里的混合物于室温下搅拌过夜，真空浓缩，以二氯甲烷及饱和碳酸氢钠溶液稀释。分离各相。有机相用无水硫酸镁干燥，真空浓缩，产生1-甲基-3-[3-(3-氧丁基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮白色固体(0.310克，mp198-199℃)。水相以浓盐酸酸化，搅拌数分钟，过滤得到固体。以水洗涤固体，风干，得到α-乙酰基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸的白色固体，mp 191-193℃。
基本上采用相同方法，得到下列化合物：
Figure A9880989802811
实施例99
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸甲酯的制备
Figure A9880989802812
使{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}丙二酸单甲酯(0.610克)与樟脑磺酸(0.100克)在甲苯里的混合物回流2小时，再以樟脑磺酸(0.400克)处理，回流3小时，真空浓缩，以1，1，2，2-四氯乙烷稀释，回流4小时，冷却至室温，真空浓缩，以二氯甲烷及饱和碳酸氢钠溶液稀释。分离有机相，用无水硫酸镁干燥，真空浓缩，得到固体。固体于己烷中搅拌1小时，过滤及干燥，产生标题产物的白色固体(0.400克，mp176-178℃)。
实施例100
N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}邻苯二甲酰亚胺的制备
使3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.750克)及邻苯二甲酰亚胺化钾(0.350克)之乙腈混合物回流1小时，冷却至室温，倒至冰-水混合物。所得水性混合物过滤得到固体。以水洗涤此固体，风干，产生标题产物(0.720克，mp 204-208℃)。
实施例101
3-[3-(邻-羟苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮三氟甲基磺酸酯的制备
Figure A9880989802822
使3-[3-(邻-羟苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(3.67克，8.75毫摩尔)与三乙胺(0.970克，9.63毫摩尔)在二氯甲烷里的混合物于冰-水浴中冷却，用三氟甲磺酸酐(2.72克，9.63毫摩尔)处理，于室温下搅拌过夜，倒入水中。所得水性混合物以二氯甲烷萃取。合并有机萃取液，以盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到油状物。此油状物使用硅胶及3％乙醚的二氯甲烷溶液进行柱层析，产生标题产物的白色泡沫状物，以NMR光谱分析法鉴定。
实施例102
邻-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}肉桂酸甲酯的制备
Figure A9880989802831
使3-[3-(邻-羟基苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮三氟甲磺酸酯(1.00克，1.81毫摩尔)的N，N-二甲基甲酰胺溶液依次用三乙胺(0.200克，1.99毫摩尔)、丙烯酸甲酯(0.310克，3.62毫摩尔)、二苯基膦基乙烷(DPPE，0.0220克，0.0500毫摩尔)及乙酸钯(II)(0.0100克，0.0450毫摩尔)处理，于100℃搅拌过夜，冷却至室温，倒至水中。所得水性混合物过滤得到固体。以水洗涤固体，溶于二氯甲烷。所得有机溶液依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，得到油状物。此油状物使用硅胶及5％乙醚的二氯甲烷溶液进行柱层析，产生的油与乙醚研磨，产生标题产物的灰白色固体(0.460克，mp 150-152℃)。
实施例103
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，(2∶3)混合物的制备
Figure A9880989802841
使3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(5.00克)、四氟硼酸银(3.50克)、1，4-二噁烷(30.0毫升)、及水(10.0毫升)的溶液回流2小时，冷却，过滤除去固体。所得滤液倒至二氯甲烷与水的混合物中。分离有机相，依次用水及盐水洗涤，用无水硫酸钠干燥，真空浓缩，产生标题产物之2∶3混合物。
实施例104
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸的制备
Figure A9880989802851
使二铬酸钾(10.0克)的1.5M硫酸(200毫升)溶液冷却至0℃，滴加2∶3的3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(12.0克)在乙酸中的混合物，于室温下搅拌2小时，加水稀释。所得水性混合物以二氯甲烷萃取。合并有机萃取液，依次用水及盐水洗涤，用无水硫酸钠干燥，真空浓缩，产生标题产物的白色固体(8.50克，mp 149-152℃)。
实施例105
5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺的制备
Figure A9880989802861
用1，1’-羰基二咪唑(0.260克，1.58毫摩尔)处理5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸(0.400克，1.08毫摩尔)的四氢呋喃溶液，于室温下搅拌30分钟，回流2小时，冷却至室温，滴加甲磺酰胺(0.130克，1.37毫摩尔)与1，8-重氮双环[5.4.0]十一碳-7-烯(0.230克，1.50毫摩尔)的溶液，于室温下搅拌3小时，倒至0.5N盐酸中。所得水性混合物以二氯甲烷萃取。合并有机萃取液，以盐水洗涤，用无水硫酸钠干燥，真空浓缩，得到残留物。残留物使用硅胶及二氯甲烷/乙酸溶液(10∶1)柱层析，产生标题产物的白色固体(0.350克，72％，mp 241-243℃)。
基本上采用相同方法，但改用经适当取代的磺酰胺，得到下列化合物：
Figure A9880989802871
X               R15                    mp℃H               CH2Cl                  190-192H              
Figure A9880989802872
          147-149H                            147-149H              
Figure A9880989802874
      235-237X                      R15                  mp℃H              
Figure A9880989802881
                 177-180H               CH(CH3)CH2CH3           ＞225H              
Figure A9880989802882
            217-219H              
Figure A9880989802883
           172-174H               (CH2)11CH3H               CH(CH3)2                 156-158H               HC2CH3                   197-200H                             ＞225H                 ＞230H              
Figure A9880989802886
      ＞230H              
Figure A9880989802887
        215-220H                     226-228X                       R51                        mp℃H               
Figure A9880989802891
                    155-159H               
Figure A9880989802892
              ＞220F                       CH2C6H5                 120-125H               
Figure A9880989802893
               220-225H                       CH2CH2C6H5             ＞220H               
Figure A9880989802894
                143-148H                       CH＝CHC6H5                198-203
实施例106
2-{{2-[5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}对-甲苯基}氧基-N-(甲磺酰基)乙酰胺的制备
将{{2-[5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}乙酸(1.54克，0.00312摩尔)的四氢呋喃溶液滴加至含1，1’-羰基二咪唑(1.06克，0.00655摩尔)在四氢呋喃里的悬浮液中。所得混合物搅拌1.5小时，冷却至室温。滴加甲磺酰胺(0.594克，0.00624摩尔)、重氮双环十一碳烷(1.09克，0.00702摩尔)与四氢呋喃的混合物。所得混合物于室温下搅拌过夜，倒至10％盐酸中。所得白色固体过滤，干燥，产生标题化合物(1.65克，91.6％，mp 123-125℃)，以NMR光谱分析法鉴定。
实施例107
N-{{2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酰基}甘氨酸甲酯的制备
Figure A9880989802901
在0℃下将1，1’-羰基二咪唑(0.340克，0.00203摩尔)加到{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}乙酸(1.00克，0.00203摩尔)的二甲基甲酰胺溶液中。混合物于0℃下搅拌30分钟，回升至室温。添加甘氨酸甲酯盐酸盐(0.260克，0.00207摩尔)，所得混合物于室温下搅拌3天。加水稀释混合物，过滤产生白色固体，经硅胶使用醚∶二氯甲烷层析，产生标题产物的白色泡沫状物(0.830克，74.8％)，以NMR光谱分析法鉴定
实施例108
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}乙酸的制备
Figure A9880989802911
使{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯(10.9克，0.0190摩尔)，10％盐酸及乙酸的混合物于90℃下搅拌2小时，冷却，倒至水中，以乙酸乙酯萃取。合并有机层，以水及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩，形成泡沫状物。此泡沫状物自乙酸乙酯重结晶，产生标题产物的白色固体(6.20克，66.2％，mp123-126℃)。
实施例109
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}-2-甲基丙酸2-丙炔酯的制备
Figure A9880989802912
使2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基-2-甲基丙酸(0.500克，0.000960摩尔)、对-甲苯磺酸(0.0100克)、炔丙醇(0.0538克，0.000960摩尔)及甲苯的混合物于50℃下搅拌1天，冷却至室温，真空浓缩，得到残留物。此残留物经硅胶以醚∶二氯甲烷层析，产生标题产物(0.360克，67.2％)，以NMR光谱分析法鉴定。
基本上采用相同方法，但改用适当羧酸及醇类，得到下列化合物：
Figure A9880989802921
      W4              W4              W4
      CH3             CH3             CH2C≡CH
      CH3             CH3             CH2C＝CH(CH3)
      CH3             CH3             CH2CH＝CH2
      CH3             CH3             CH(CH3)C≡CH
      CH3             CH3             CH(CH3)CH2OCH3
      H                H                (CH2)3O(CH2)3OCH3
      H                H               
      H                H                (CH2)5Si(CH3)2C(CH3)3
      H                H               
Figure A9880989802923
实施例110
3-[3-(2-羟基-3-碘-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
将N-碘琥珀酰亚胺(0.240克，0.00107摩尔)的丙酮溶液滴加到3-[3-(2-羟基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.430克，0.000992摩尔)的丙酮溶液中，所得混合物于室温下搅拌过夜。再添加N-碘琥珀酰亚胺(0.120克，0.000635摩尔)，混合物于室温下搅拌3小时。混合物真空浓缩，产生红色胶状物，于硅胶上用醚∶二氯甲烷进行色谱层析。用1M硫代硫酸钠及盐水洗涤含标题化合物的组分，用无水硫酸镁干燥，真空浓缩，得到标题化合物的黄色固体(0.280克，46.8％，mp 241-242℃)。
实施例111
3-[3-(5-碘-2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802941
用碘(1.14克，0.00450摩尔)分批处理3-[3-(6-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.34克，0.00300摩尔)、三氟乙酸银及二氯甲烷的混合物，于室温下搅拌过夜，以二氯甲烷稀释，以1M硫代硫酸钠及盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生的褐色油静置时即固化。用醚重结晶，产生标题化合物的浅黄色晶体(1.50克，87.2％，mp 210-212℃)。
实施例112
3-[3-(α，α-二溴-2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989802951
使3-[3-(2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.34克，0.00300摩尔)、N-溴琥珀酰亚胺(1.39克，0.00780摩尔)、苯甲酰过氧化物(0.200克)及四氯化碳的混合物于回流下搅拌3小时，趁热过滤。滤液冷却至室温，真空浓缩。残留物经硅胶使用醚∶二氯甲烷层析，产生标题产物的白色泡沫状物(0.640克，35.3％)，以NMR光谱分析法鉴定。
实施例113
5-硝基-1，2-苯并异噻唑的制备
Figure A9880989802952
将2-氯-5-硝基苯甲醛(300克，1.62摩尔)与硫(54.4克，1.70摩尔)加到氢氧化铵(1000毫升)与N，N-二甲基甲酰胺的混合物中。混合物缓缓加热至90℃并搅拌1小时，冷却至室温，倒至冰上，加水稀释。过滤，产生标题化合物的黄色固体(277.1克，94.9％)。
实施例114
3-氯-5-硝基-1，2-苯并异噻唑的制备
将5-硝基-1，2-苯并异噻唑(271克，1.50摩尔)在乙酸中的悬浮液加热至80℃形成溶液。离开加热源，于70-80℃下，连续通入氯气6小时直到混合物饱和为止。混合物冷却至室温，搅拌过夜。过滤，产生标题化合物的黄色晶体(237克，73.6％)，以NMR光谱分析法鉴定。
实施例115
2’-氯-2-甲基-2-乙酯基丙酰苯的制备
Figure A9880989802962
将2-氯苯甲酰氯(52.2克，0.298摩尔)、2-溴异丁酸乙酯(58.2克，0.298摩尔)及醚的混合物分批加至锌箔(19.5克，0.298摩尔)中，所得混合物于回流下搅拌3小时，于室温下过夜。混合物倒至冷的稀硫酸中，有机层以饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，真空浓缩成黄色油。此油经硅胶使用己烷∶乙酸乙酯层析，产生标题化合物的无色油(41.8克，55.1％)。
实施例116
2’-氯-5’-硝基-2-甲基-2-乙酯基丙酰苯的制备
将’-氯-2-甲基-2-乙酯基丙酰苯(4.00克，0.01570摩尔)加到5℃的浓硫酸(15.0毫升)中，然后滴加浓硝酸(90％，0.740毫升，0.0204摩尔)。搅拌5分钟后，混合物倒至冰上，以乙酸乙酯萃取。有机层以饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩，产生标题化合物的黄色油(3.90克，83.0％)，以NMR光谱分析法鉴定。
实施例117
α，α-二甲基-5-硝基-1，2-苯并异噻唑-3-乙酸乙酯的制备
用氢氧化铵(9毫升)滴加处理2’-氯-5’-硝基-2-甲基-2-乙酯基丙酰苯(3.24克，0.00108摩尔)、N，N-二甲基甲酰胺及硫(0.350克，0.00109摩尔)的混合物，加热至70-80℃并搅拌2小时，冷却至室温，加水稀释。过滤产生标题化合物的固体(2.49克，78.3％，mp 75-77℃)，以NMR光谱分析法鉴定。
实施例118
1-苯并噻吩-2，3-二酮的制备
Figure A9880989802972
将草酰氯(175克，1.38摩尔)的醚溶液滴加到硫酚(100克，0.907摩尔)的醚溶液中。混合物回流搅拌2小时，真空浓缩。残留物溶于二氯甲烷中，冷却至0℃。分批添加氯化铝(145克，1.09摩尔)，保持温度不超过25℃。所得混合物回流搅拌30分钟，冷却至室温，搅拌倒至冰水中。有机层以饱和碳酸氢钠、水及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩成橙色固体，用二氯甲烷∶己烷重结晶，产生标题化合物(102克，69.0％)，以NMR光谱分析法鉴定。
实施例119
1，2-苯并异噻唑-3-甲酰胺的制备
Figure A9880989802981
在5-10℃下将1-苯并噻吩-2，3-二酮(87.0克，0.530摩尔)加到氢氧化铵(1.78升)中后，再加过氧化氢(30％水溶液，178毫升)。所得混合物过滤，得到黄色固体，干燥(77.0克，81.7％)，以NMR及IR光谱分析法鉴定标题化合物。
实施例120
3-氰基-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989802982
在0-5℃下用硝酸(90％，4.12毫升)滴加处理1，2-苯并异噻唑-3-甲酰胺(12.0克，0.0674摩尔)的浓硫酸溶液，并保持温度不超过10℃，于5℃下搅拌1小时，于激烈搅拌下倒至冰水中。所得悬浮液过滤，得到固体。干燥此固体，用乙腈重结晶，产生白色固体(10.0克)，以磷酸氯(60.0毫升)处理。所得混合物于90-100℃下搅拌90分钟，冷却至室温，于搅拌下缓缓倒至冰水中，过滤得到固体。此固体用二氯甲烷∶己烷重结晶，产生标题化合物的橙色固体(8.00克，87.9％，mp 168-170℃)，NMR及IR光谱分析法鉴定。
实施例121
2，4-二氟-5-硝基苯甲酰氯的制备
Figure A9880989802991
将草酰氯(94.0克，0.739摩尔)滴加到2，4-二氟-5-硝基苯甲酸(100.0克，0.492摩尔)、二氯甲烷及N，N-二甲基甲酰胺(0.600毫升)的混合物中。所得混合物于回流下搅拌3.25小时，冷却至室温，真空浓缩，产生标题化合物的褐色油(111克，95.2％)。
实施例122
2’，4’-二氟-2-甲氧基-5-甲基-5’-硝基苯酮的制备
Figure A9880989802992
使氯化铝(62.3克，0.467摩尔)与二氯甲烷的混合物冷却至-20℃至-10℃，用4-甲基苯甲醚(60.1克，0.492摩尔)处理，在10分钟里滴加2，4-二氟-5-硝基苯甲酰氯(111克，0.468摩尔)与二氯甲烷的混合物处理，温热至0℃，在室温下搅拌过夜，于搅拌下缓缓倒至冰上，以二氯甲烷稀释。有机层以水及盐水洗涤，用无水硫酸镁干燥及真空浓缩成固体。此固体用乙腈重结晶，产生标题化合物的黄色固体(82.1克，54.0％)，以NMR光谱分析法鉴定。
实施例123
3-(6-甲氧基-间-甲苯基)-6-氨基-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989803001
在冰浴上将氢氧化铵(330毫升)加到2’，4’-二氟-2-甲氧基-5-甲基-5’-硝基苯酮(60.0克，0.186摩尔)、硫(6.25克，0.195摩尔)及N，N-二甲基甲酰胺悬浮液中。所得混合物回升至35℃，以2小时时间逐渐加温至81℃，冷却至室温，倒至水中。所得固体溶于乙酸乙酯与N，N-二甲基甲酰胺中，以水洗涤。有机层真空浓缩，产生标题化合物，以NMR光谱分析法鉴定。
实施例124
3-(6-甲氧基-间-甲苯基)-6-氯-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989803002
将亚硝酸叔丁酯(5.90克，0.0571摩尔)、氯化铜(6.20克，0.0457摩尔)及乙腈的混合物加热至65-75℃，用3-(6-甲氧基-间-甲苯基)-6-氨基-5-硝基-1，2-苯并异噻唑(12.0克，0.0381摩尔)处理10分钟，于67-75℃下搅拌2小时，以亚硝酸叔丁酯(1.50毫升)及氯化铜(1.00克)处理，于67-75℃下搅拌40分钟，冷却至室温，以乙酸乙酯稀释。有机层以10％盐酸洗涤及过滤。滤液以水洗涤，真空浓缩，产生标题化合物的固体(10.6克，83.1％)，以NMR光谱分析法鉴定。
实施例125
3-(6-甲氧基-间-甲苯基)-6-氟-5-硝基-1，2-苯并异噻唑的制备
Figure A9880989803011
使3-(6-甲氧基-间-甲苯基)-6-氯-5-硝基-1，2-苯并异噻唑(7.30克，0.0218摩尔)、氟化钾(6.33克，0.109摩尔)、18-冠-6(2.31克，0.0872摩尔)及环丁砜的混合物于154℃下搅拌19小时，冷却至室温，倒至冰水中。所得固体过滤，经硅胶使用二氯甲烷层析，产生的固体用乙腈重结晶，产生黄褐色粉末。此粉末用乙酸乙酯重结晶，产生标题化合物的黄褐色固体(2.09克，29.9％)，以NMR光谱分析法鉴定。
实施例126
5-氨基-4-溴-6-氟-3-甲基-1，2-苯并异噻唑的制备
向5-氨基-6-氟-3-甲基-1，2-苯并异噻唑(0.600克，0.00329摩尔)的1，2-二氯乙烷溶液中加入N-溴琥珀酰亚胺(0.586克，0.00329摩尔)，然后加入1，1’-偶氮双(环己腈)(0.0200克)。混合物于70℃下搅拌2小时，再加入N-溴琥珀酰亚胺(0.240克，0.00135摩尔)，混合物于70℃下搅拌40分钟。混合物再冷却至室温，过滤及真空浓缩，得到残留物。此残留物经硅胶层析，得到标题化合物(0.870克，100％)，以NMR光谱分析法鉴定。
实施例127
5-氯-1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备使1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.00克，0.00293摩尔)、硫酰氯(2.00克，0.0148摩尔)与1，2-二氯乙烷的混合物于回流下搅拌5小时，冷却至室温，以二氯甲烷稀释。所得混合物以饱和碳酸氢钠及盐水洗涤，用无水硫酸钠干燥，过滤及真空浓缩，得到残留物。此残留物经硅胶使用乙酸乙酯/己烷层析，产生标题产物的白色固体(0.350克，31.8％，mp252-254℃)，以NMR光谱分析法鉴定。
实施例128
3-[3-(1-溴乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与3-[3-(1，1-二溴乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803031
使1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.44克，0.00405摩尔)、N-溴琥珀酰亚胺(0.790克，0.00446摩尔)及1，2-二氯乙烷的混合物在150瓦灯泡下，于60℃下搅拌1小时，冷却至室温，真空浓缩，产生黄色固体。此黄色固体经硅胶使用80％至70％己烷∶乙酸乙酯进行快速层析，产生1，1-二溴乙基苯并异噻唑的白色泡沫状物(0.0600克，2.88％)。及1-溴乙基苯并异噻唑的白色晶体(1.73克，98.9％，mp 163℃)。这二种产物以NMR光谱分析法鉴定。
用相似的方法，以N-氯琥珀酰亚胺处理上述反应物，产生3-[3-(1-氯乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的白色固体，mp 169-171℃。
实施例129
3-[3-(溴氯甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使3-[3-(氯甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.00克，0.00266摩尔)、偶氮-双-异丁腈(0.100克)、N-溴琥珀酰亚胺(0.712克，0.00400摩尔)与1，2-二氯乙烷的混合物于回流下搅拌1小时。再添加偶氮-双-异丁腈(0.0500克)及N-溴琥珀酰亚胺(0.100克)，混合物于回流下搅拌2小时，冷却至室温，以二氯甲烷稀释，以水洗涤，用无水硫酸镁干燥，真空浓缩成橙色胶状物。此胶状物经硅胶使用二氯甲烷∶醚层析，产生标题化合物的白色泡沫物(0.950克，80.2％， mp 93-96℃)，以NMR光谱分析法鉴定。
实施例130
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-溴-1，2-苯并异噻唑-3-乙酸甲酯的制备
Figure A9880989803051
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸甲酯(0.400克，0.00100摩尔)、N-溴琥珀酰亚胺(0.370克，0.00210摩尔)、苯甲酰过氧化物(0.0100克)与四氯乙烷的混合物于回流下搅拌2.5小时，冷却至室温，经硅胶使用二氯甲烷层析，产生标题化合物的灰白色固体(0.430克，90.0％，mp 84-87℃)，以NMR光谱分析法鉴定。
实施例131
3-[3-(2-溴乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
向3-[3-(2-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.690克，0.00185摩尔)的二氯甲烷溶液中加入四溴化碳(0.655克，0.00197摩尔)，然后加入三苯基膦(0.517克，0.00197摩尔)。使混合物在氛围温度下搅拌3小时，再以四溴化碳(0.328克，0.000988摩尔)及三苯基膦(0.259克，0.000987摩尔)处理。所得混合物搅拌85分钟，以甲醇稀释，真空浓缩。所得固体溶于二氯甲烷中，以饱和碳酸氢钠及水洗涤，用无水硫酸钠干燥，过滤及真空浓缩成黄色固体。此黄色固体经硅胶使用二氯甲烷层析，产生标题产物的灰白色固体(0.530克，66.0％)，以NMR及元素分析法鉴定。
实施例132
3-[3-(2，2-二溴乙烯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803071
将三苯基膦(0.354克，0.00138摩尔)加到四溴化碳(0.223克，0.000676摩尔)的二氯甲烷溶液中。所得混合物于室温下搅拌10分钟，滴加5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(0.200克，0.000563摩尔)的二氯甲烷溶液处理。所得混合物搅拌20分钟，并真空浓缩。所得残留物经硅胶使用10∶1二氯甲烷/乙酸乙酯进行快速柱层析法纯化，产生标题产物的白色固体(0.240克，83.6％，mp 260-262℃)，以NMR及IR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989803072
      W10             W11             mp℃
      Br               F
      Cl               Cl               254-256
实施例133
(1R，2S)-3-[3-(1，2-二溴丙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与(1R，2R)-3-[3-(1，2-二溴丙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803081
向1-甲基-(3-丙烯基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.500克，0.00136摩尔)与四氯化碳的混合物中加入溴(0.220克，0.00138摩尔)。所得混合物于室温下搅拌2.5小时，真空浓缩成黄色泡沫状物，经硅胶使用二氯甲烷∶醚层析。首先洗脱出(1R，2S)-异构物，分离得到灰白色固体(0.310克，41.9％，mp 214℃)，以NMR光谱分析法鉴定。其次洗脱出(1R，2R)-异构物，为灰白色泡沫状物(0.290克，39.2％，mp 188-189℃)，以NMR光谱分析法鉴定。
实施例134
3-[3-(2(和1)-溴-1(和2)-羟丙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(4∶1)非对映异构物的混合物
Figure A9880989803091
向1-甲基-(3-丙烯基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.00克，0.00272摩尔)、二噁烷与水的混合物中加入N-溴琥珀酰亚胺(0.570克，0.00321摩尔)。所得混合物于室温下搅拌23小时，倒至水中，以醚萃取。有机层以水洗涤，用无水硫酸镁干燥，过滤及真空浓缩，产生黄色泡沫状物。此泡沫状物经硅胶使用二氯甲烷∶醚层析，产生标题之异构物混合物之白色泡沫状物(1.03克，82.4％，mp 100-103℃)，以NMR光谱分析法鉴定。
实施例135
5-[3，6-二氢-5-溴-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二溴-1，2-苯并异噻唑-3-乙酸甲酯与5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二溴-1，2-苯并异噻唑-3-乙酸甲酯的制备
Figure A9880989803101
使5-[3，6-二氢-5-溴-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸甲酯(1.20克，0.00300摩尔)、二甲基-N，N-二溴乙内酰(4.20克，0.0150摩尔)与1，2-二氯乙烷的混合物于回流下搅拌3天，冷却至室温，以二氯甲烷稀释，以10％硫代硫酸钠、水及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩。所得残留物经硅胶使用二氯甲烷层析。首先洗脱出溴尿嘧啶取代的α，α-二溴-1，2-苯并异噻唑-3-乙酸酯，并分离出白色固体(0.400克，30.0％，mp 241℃)，以NMR光谱分析法鉴定。然后洗脱出α，α-二溴-1，2-苯并异噻唑-3-乙酸酯，并分离出白色固体(0.520克，31.1％，mp 194-196℃)。以NMR光谱分析法鉴定。
实施例136
α-溴-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈的制备
Figure A9880989803111
将N-溴琥珀酰亚胺(0.250克，0.00140摩尔)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈(0.500克，0.00140摩尔)的1，2-二氯乙烷溶液中。所得混合物经UV灯照射，于回流下搅拌6小时。再加N-溴琥珀酰亚胺(0.250克，0.00140摩尔)，所得混合物于UV灯下，回流搅拌1.5小时。混合物冷却至室温，真空浓缩。所得残留物溶于二氯甲烷中，以水洗涤，以木炭处理，用无水硫酸镁干燥，过滤，及真空浓缩，产生标题产物的红色玻璃状物(0.350克，56.2％，mp 185-187℃)，以IR及NMP光谱分析法鉴定。
实施例137
{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}异硫氰酸甲酯的制备
Figure A9880989803121
将3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.500克，0.00119摩尔)加到硫氰酸钾(0.300克，0.00309摩尔)的二甲亚砜溶液中。所得混合物于室温下搅拌2小时，以乙酸乙酯稀释，以水洗涤，用无水硫酸镁干燥，过滤，真空浓缩，产生标题化合物的白色固体(0.475克，100％，mp 239-241℃)，以NMR及IR光谱分析法鉴定。
实施例138
3-[3-羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮硝酸酯的制备
使3-[3-(二溴-(33％)及-溴甲基(67％))-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(2.00克，0.00434摩尔)、硝酸银(1.50克，0.00887摩尔)、二噁烷及水的混合物于回流下搅拌1小时，冷却至室温，过滤。滤液真空浓缩。残留物分布在二氯甲烷与水之间。有机层以盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩。残留物经硅胶使用二氯甲烷∶甲醇层析，产生标题化合物的白色固体(0.450克，25.9％，mp 188-190℃)，以NMR光谱分析法鉴定。
实施例139
3-[3-(1-甲氧乙基)-1，2苯并异噻唑5基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
将三氟甲磺酸银(0.510克，0.00199摩尔)加到3-[3-(1-溴乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.720克，0.00166摩尔)、甲醇与1，2二氯乙烷的混合物中。所得混合物于室温下搅拌23小时，经硅藻土使用乙酸乙酯过滤。向滤液中加入饱和碳酸氢钠，所得混合物激烈搅拌1小时。保留有机层，同时以乙酸乙酯萃取水层。合并的有机层以硫酸镁干燥，过滤及真空浓缩成浆状物，经硅胶使用己烷∶乙酸乙酯层析，产生标题化合物的白色固体(0.660克，100％，mp 133-135℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，但改用适当醇替代甲醇，制备下列化合物：
Figure A9880989803142
实施例140
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-甲氧基-1，2-苯并异噻唑-3-乙酸甲酯的制备使5-[3，6-二氧-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-溴-1，2-苯并异噻唑-3-乙酸甲酯(0.600克，0.00125摩尔)、三氟甲磺酸银(0.400克，0.00156摩尔)及甲醇的混合物于回流下搅拌36小时，冷却及真空浓缩。残留物分布在二氯甲烷及饱和碳酸氢钠之间。保留有机层，以二氯甲烷萃取水层。合并的有机层以盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩。残留物经硅胶使用二氯甲烷层析，产生标题化合物的白色固体(0.220克，41.0％，mp 166-168℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，由5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二溴-1，2-苯并异噻唑-3-乙酸甲酯制备5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲氧基-1，2-苯并异噻唑-3-乙酸甲酯。
实施例141
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲醛，3-(二甲基缩醛)的制备将三氟甲磺酸银(0.620克，0.00241摩尔)加到3-[6-氟-3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.500克，0.000967摩尔)、1，2-二氯乙烷及甲醇(1.00毫升)的混合物中。所得混合物于室温及遮光下搅拌过夜。混合物使用二氯甲烷洗涤过滤。滤液以饱和碳酸氢钠、水及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩成油状物。此油经硅胶使用乙酸乙酯∶己烷层析，产生标题化合物的白色固体(0.330克，81.4％，mp 63-65℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
实施例142
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}(甲磺酰基)氨基甲酸叔丁酯的制备
Figure A9880989803171
在0℃下将(甲磺酰基)氨基甲酸叔丁酯(1.52克，0.00780摩尔)加到氢化钠(60％，0.312克，0.00780摩尔)与四氢呋喃的混合物中。使混合物回升到室温，滴加3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(3.00克，0.00714摩尔)的二甲亚砜溶液。所得混合物于室温下搅拌过夜，倒至稀盐酸中，以二氯甲烷萃取。合并的有机层以水洗涤，用无水硫酸镁干燥，过滤及真空浓缩。所得残留物经硅胶使用醚∶二氯甲烷层析，产生标题化合物的白色固体(3.00克，78.7％，mp 109-111℃)，以NMR光谱分析法鉴定。
实施例143
3[3-(羟甲基)1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮苯甲酸酯的制备
在0℃下向3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.650克，0.00182摩尔)与二氯甲烷的混合物中加入三乙胺(0.330毫升，0.00236摩尔)，然后加入苯甲酰氯(0.210毫升，0.00182摩尔)。混合物于0℃下搅拌1小时，在15分钟里搅拌添加饱和碳酸氢钠以中止反应。所得混合物以醚稀释，有机层以饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，过滤，真空浓缩成橙色浆状物。此浆状物经硅胶使用己烷∶乙酸乙酯层析，产生固体。此固体用乙酸乙酯及己烷重结晶，产生标题化合物的白色固体(0.340克，40.5％，mp140-142℃)。
基本上采用相同方法，但改用合适的酰氯及羟烷基苯并异噻唑，得到下列化合物：
Figure A9880989803191
W12          R13                           mp℃H             CH2Cl                         166-168H             CH2C6H5                    125-127H           
Figure A9880989803192
       144-146H           
Figure A9880989803193
                139-142H                     164-167H           
Figure A9880989803195
         124-126W12             R12                  mp℃H        
Figure A9880989803201
              81-83H              CH(CH2CH3)C6H5H        
Figure A9880989803202
          245-247H                      148-150H        
Figure A9880989803204
         195-198H        
Figure A9880989803205
               178-180H        
Figure A9880989803206
              201-204H              CH2OCH3           165-166H        
Figure A9880989803207
                 134-136H                       178-180H              C(CH3)3           50-52H            160-162W12               R12                 mp℃H         
Figure A9880989803211
            148-150H                CH(Cl)C6H5         159-161H                 195-197H         
Figure A9880989803213
            160-162CH3            CH2Cl                45-147CH3            CH2OCH3            11-114CH3       
Figure A9880989803214
CH3      
Figure A9880989803215
             102-104CH3            CH(Cl)C6H5         66-68CH3       
Figure A9880989803216
              79-81CH3            CH3                 76
实施例144
3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803221
在-78℃下，以15分钟将甲基氯化镁(14.1毫升，0.0422摩尔)滴加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(6.00克，0.00170摩尔)的四氢呋喃溶液中。所得混合物于-70℃下搅拌30分钟，用饱和氯化铵中止反应，使之回升至室温。以乙酸乙酯稀释后，以饱和氯化铵、水及盐水洗涤混合物，用无水硫酸镁干燥，过滤，真空浓缩成固体。此固体经硅胶使用己烷/乙酸乙酯层析，产生标题化合物的白色晶体(4.49克，71.1％)，以NMR光谱分析法鉴定。
实施例145
3-(3-乙酰基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803231
在氮气大气压下向3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(3.99克，0.0107摩尔)的无水二氯甲烷溶液中加入4分子筛，然后加入二铬酸吡啶鎓(4.85克，0.0129摩尔)。所得混合物于室温下搅拌22小时，以醚稀释，经硅胶及硅藻土过滤，真空浓缩成固体。此固体用乙酸乙酯∶己烷重结晶，产生标题化合物的白色固体(2.34克，59.2％，mp 149℃)，以NMR光谱分析法鉴定。
实施例146
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮甲基氨基甲酸酯的制备
Figure A9880989803241
在0℃下向3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.00克，0.00280摩尔)及二氯甲烷的混合物中加入三乙胺(0.590毫升，0.00420摩尔)，然后加入异氰酸甲酯(0.190毫升，0.00320摩尔)。所得混合物在氛围温度下搅拌27小时，以乙酸乙酯及饱和碳酸氢钠溶液稀释，并搅拌15分钟。以饱和碳酸氢钠及盐水洗涤有机层，用无水硫酸镁干燥，过滤及真空浓缩成黄色固体。此固体用乙酸乙酯重结晶，产生标题化合物的黄褐色晶体(0.440克，37.9％，mp＞230℃)。
基本上采用相同方法，但改用合适的异氰酸酯，得到下列化合物：
Figure A9880989803242
                R26                 mp℃
                C6H5               209
                CH2C6H5           174-177
实施例147
3-[3-(1-羟乙基)-1，2苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮甲磺酸酯的制备
Figure A9880989803251
在0℃下，向3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.650克，0.00175摩尔)的二氯甲烷溶液中加入甲磺酰氯(0.150毫升，0.00193摩尔)，然后加入三乙胺(0.320毫升，0.00228摩尔)。所得混合物于0℃下搅拌80分钟，以pH7缓冲液中止反应。以乙酸乙酯及醚稀释有机层后，以pH7缓冲液及盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩成无色浆状物。此浆状物溶于乙酸乙酯中，添加己烷使之结晶，产生标题化合物的白色晶体(0.640克，81.4％，mp157℃)。以NMR光谱分析法鉴定。
基本上采用相同方法，但改用合适的磺酰氯，制备下列化合物：
Figure A9880989803252
                R47                    mp℃
                CH(CH3)2             113-115
                (CH2)3CH3           124-125
                C6H5                 92-94
用基本上相同的方法，但改用合适的磺酰氯与3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮反应，得到下列化合物：
Figure A9880989803261
                R47                   mp℃
                CH3                   178-180
                CH(CH3)2             141-143
                (CH2)3CH3           142-145
                C6H5                 150-152
实施例148
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛3-(二乙基缩醛)的制备
Figure A9880989803262
将正甲酸三乙酯(0.560毫升，0.00338摩尔)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(0.800克，0.00225摩尔)的乙醇悬浮液中后，再添加硝酸铵(0.0100克)。所得混合物于室温下搅拌19小时，回流下搅拌3小时。冷却至室温后，混合物真空浓缩成黄色油。此油经硅胶使用己烷∶乙酸乙酯层析，产生标题化合物的黄色泡沫状物(0.690克，71.4％，mp 49℃)，以NMR光谱分析法鉴定。
实施例149
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-[双(3-羟丙基)二硫缩醛]的制备
向5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(2.86克，0.00805摩尔)与乙腈的混合物中加入3-巯基-1-丙醇(0.600毫升，0.00684摩尔)，然后加入氯化铋(III)(0.0900克)。所得混合物于室温下搅拌过夜。再加入3-巯基-1-丙醇(0.200毫升，0.00228摩尔)，混合物真空浓缩。残留物经硅胶使用丙酮∶乙酸乙酯层析，分离出第二个成份的黄色油，溶于醚中，以水及盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩，产生标题化合物的黄色固体(1.00克，23.8％)，以NMR光谱分析法鉴定。
实施例150
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-[双(2-羟乙基)二硫缩醛]，二乙酸酯(二酯)的制备
Figure A9880989803281
向5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-[双(2-羟乙基)二硫缩醛](0.500克，0.00101摩尔)的二氯甲烷溶液中加入三乙胺(0.400毫升，0.00300摩尔)，然后加入乙酰氯(0.160毫升，0.00220摩尔)。所得混合物于室温下搅拌1小时，倒至水中，以二氯甲烷稀释。保留有机层，以二氯甲烷萃取水层。合并的有机层以水及盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩成黄色油。此油经硅胶使用己烷∶乙酸乙酯层析，产生标题化合物的黄色油(0.340克，58.3％)，以NMR光谱分析法鉴定。
基本上采用相同方法，由5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-[双(3-羟丙基)二硫缩醛]制得5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-[双(3-羟丙基)二硫缩醛]，二乙酸酯(二酯)。
实施例151
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-[双(2-羟乙基)二硫缩醛]的制备
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(3.00克，0.00844摩尔)、2-巯基乙醇(1.80毫升，0.0252摩尔)、对-甲苯磺酸(0.0800克，0.000420摩尔)及甲苯的混合物于回流下搅拌2小时，共沸除去水。冷却至室温后，混合物搅拌过夜，以乙酸乙酯稀释，以水及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩，得到褐色油。此油经硅胶层析，产生标题化合物的白色固体(1.10克，31.3％)，以NMR光谱分析法鉴定。
实施例152
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-肟，(E)-异构物的制备
Figure A9880989803301
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛(0.200克，0.000563摩尔)、羟胺盐酸盐(0.0700克，0.00100摩尔)、乙酸钠(0.150克，0.00183摩尔)及乙醇的混合物于50-60℃下搅拌1小时，真空浓缩。残留物分布在二氯甲烷与水之间。分离有机相，以盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩。残留物经硅胶使用二氯甲烷∶乙酸乙酯层析，产生标题化合物的白色固体(0.140克，67.3％，mp 234-236℃)，以NMR光谱分析法鉴定。
基本上依相同方法，但改用适当醛与各种羟胺或肼，得到下列肟及腙：
Figure A9880989803302
                n              W12              mp℃
                1              OH                186-188
                0              OCH3             235-237
                0              NHC6H5          ＞220
                0              N(CH3)2         192-192.5
                0              N(CH3)C6H5     198.5
实施例153
3-[3-(氯乙酰基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803311
将硫酰氯(0.350毫升，0.00433摩尔)加到3-(3-乙酰基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧嘧二酮(0.570克，0.00154摩尔)的氯仿溶液中。所得混合物于回流下搅拌1小时。加入浓盐酸(1滴)，然后加入硫酰氯(1.05毫升，0.0130摩尔)，所得混合物于回流下搅拌3天。混合物冷却至室温，以乙酸乙酯及醚稀释，以饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，及真空浓缩成固体。所得固体经硅胶使用己烷∶乙酸乙酯层析，产生白色固体。此固体经硅胶使用氯仿层析，产生白色固体，用乙酸乙酯及己烷重结晶，产生标题化合物的白色晶体(mp 215-215℃)，以NMR光谱分析法鉴定。
实施例154
3-[3-(溴乙酰基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
在室温下，向3-(3-乙酰基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.800克，0.00217摩尔)的乙酸乙酯溶液中加入氢溴酸(48％，3滴)，然后加入溴在乙酸乙酯里的物质(0.522 M，4.35毫升，0.00277摩尔)。所得混合物于回流下搅拌2小时，冷却至室温，以乙酸乙酯稀释，依次用硫代硫酸钠、饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩成白色固体。此固体用己烷∶乙酸乙酯重结晶，产生标题化合物的白色晶体(mp 191-193℃)，以NMR光谱分析法鉴定。
实施例155
(E)-与(Z)-α-(环丙基亚甲基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈的制备
Figure A9880989803331
                    (E)-和(Z)-
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈(0.730克，0.00199摩尔)、环丙醛(0.300克，0.00428摩尔)、吗啉(0.100毫升)、乙酸(0.0500毫升)及乙醇的混合物于回流下搅拌45分钟，冷却并倒至10％盐酸水溶液中。所得沉淀物过滤，以水洗涤，真空干燥，产生标题化合物(0.780克，93.8％，mp 201-205℃)，以IR及NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989803341
W14                 mp℃
Figure A9880989803342
               231-232CH(CH3)2
        W14                    mp℃
Figure A9880989803351
基本上采用相同方法，以5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸甲酯为反应物，并使用适当醛，得到下列化合物：
    W14
实施例156
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-乙腈的制备
Figure A9880989803363
向5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈(0.730克，0.00199摩尔)的二甲亚砜溶液中加入碘乙烷(0.170毫升，0.00210摩尔)，然后加入碳酸钾(0.750克，0.00543摩尔)。所得混合物于室温下搅拌过夜，倒至冰与5％盐酸水溶液的混合物上。所得固体过滤，干燥，溶于最少量二氯甲烷中，使用硅胶及100％至99∶1二氯甲烷/乙醚进行快速柱层析，产生标题化合物的白色固体(0.220克，28.0％，mp 107-109℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，使用碘甲烷为烷化剂，得到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-甲基-1，2-苯并异噻唑-3-乙腈。
基本上采用相同方法，由适当烷化剂及5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸甲酯为反应物，得到下列化合物：
               W15
               CH3
            CH2CH(CH3)2
实施例157
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二乙基-1，2-苯并异噻唑-3-乙腈的制备
向5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈(0.730克，0.00199摩尔)的二甲亚砜溶液中加入碘乙烷(0.326毫升，0.00408摩尔)，然后加入碳酸钾(0.750克，0.00543摩尔)。所得混合物于室温下搅拌过夜，倒至水中，以二氯甲烷萃取。合并的有机层用无水硫酸镁干燥，真空浓缩成黄色油。此油经硅胶使用100％至99∶1二氯甲烷/乙醚快速层析，得到标题化合物的白色固体(0.430克，51.2％，mp76-78℃)，以NMR光谱分析法鉴定。
采用相同起始物，不同烷化剂及基本上相同的方法，得到下列化合物：
W15                 W16
CH3                 CH3
       -CH2CH2-CH2CH＝CH2         CH2CH＝CH2CH2C≡CH            CH2C≡CHCH2C6H5          CH2C6H5
实施例158
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸2-丁炔酯的制备
Figure A9880989803392
将N， N-二甲基甲酰胺(8滴)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸(2.00克，0.00538摩尔)、二氯甲烷及四氢呋喃的混合物中。所得混合物于冰浴上冷却，以草酰氯(6.70毫升，0.0135摩尔)处理，于冰浴上搅拌1小时，真空浓缩。将12.5％残留物的四氢呋喃溶液加到2-丁炔-1-醇(0.200毫升)、三乙胺及四氢呋喃混合物中。所得混合物于氛围温度下搅拌过夜，倒至冷的10％盐酸中。以二氯甲烷萃取混合物，合并的有机层用无水硫酸镁干燥，过滤及真空浓缩，产生标题化合物的灰白色固体(0.140克，49.1％，mp 138-139℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，使用适当醇或硫醇，得到下列化合物：
Figure A9880989803401
X                    W17                          mp℃H                OCH2CH2SCH2CH3              118-119H                OCH2C(Cl)＝CH2                147H                OCH2CH2NHCOCH3               188H                O(CH2)6CH3                   79H                OCH2CH2OCH2CH2OCH3        68H                OCH2CH2CH3OH                 72-75H                OCH2CH2OCH3                  148-149H                SCH2C6H5                     185-187H                SCH2CH3                       165-167F                OCH2CH3                       145-148.5F                OCH3                           186.5-189.5H                SCH3                           184H                SCH(CH3)2                     94H                S(CH2)3CH3                   174.5F                SCH3CH3H                SC(CH3)3                      114F               
Figure A9880989803402
实施例159
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯的制备
在室温下，将硫酸(98％，5滴)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸(0.300克，0.000809摩尔)的甲醇溶液中。所得混合物于室温下搅拌过夜，真空浓缩。残留物溶于二氯甲烷中，以饱和碳酸氢钠及盐水洗涤，用无水硫酸钠干燥，过滤及真空浓缩。残留物经硅胶使用二氯甲烷∶乙酸乙酯进行柱层析，产生标题化合物的白色固体(0.235克，75.3％，mp153-156℃)。
实施例160
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸异丙酯的制备
Figure A9880989803412
在室温下，将1-(3-二甲胺丙基)-3-乙基碳化二亚胺盐酸盐(0.200克，0.00105摩尔)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基-1，2-苯并异噻唑-3-羧酸(0.200克，0.000539摩尔)、二甲氨基吡啶(0.0100毫克)、异丙醇(0.200克，0.00330摩尔)与二氯甲烷的混合物中。所得混合物于室温下搅拌过夜，在水与二氯甲烷之间分配。分离有机层，以水及盐水洗涤，用无水硫酸钠干燥，过滤，及真空浓缩。所得残留物经硅胶使用二氯甲烷∶乙酸乙酯层析，产生标题化合物的白色固体(0.180克，80.7％，mp 94-97℃)。
基本上采用相同方法，但改用适当醇，得到下列化合物：
Figure A9880989803421
                W47               mp℃
                C6H5            103-106
                
Figure A9880989803422
   99-102
实施例161
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺的制备
使5-[3，6-二氢-3-甲基-2，6-二氧4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸(1.00克，0.00270摩尔)及羰基二咪唑(0.480克，0.00296摩尔)的四氢呋喃溶液于回流下搅拌。30分钟后，反应混合物冷却至室温，以N，N-二异丙基磺酰胺处理，搅拌15分钟，以1，8-重氮双环[5.4.0]十一碳-7-烯(0.400毫升，0.00270摩尔)处理。于室温下搅拌过夜，反应混合物真空浓缩，在水与乙酸乙酯之间分配。水层以乙酸乙酯萃取，合并的有机层以盐水洗涤，用无水硫酸镁干燥，真空浓缩。所得残留物经硅胶使用1∶2乙酸乙酯/己烷快速层析，产生标题化合物的白色固体(0.200克，mp 241℃)。
基本上采用相同方法，得到下列化合物：
Figure A9880989803431
X              R46                  R44                    mp℃H              CH3                  CH3                   213H              H                     CH(CH3)2             236H              CH3                   174-175F              CH(CH3)2            CH(CH3)2            206-207基本上采用相同方法，但改用适当C-3苯基酸为起始物，得到下列化合物：
Figure A9880989803433
X              W3                   mp℃H              H                     121-123H              CH3                  193-195F              CH3                  192
实施例162
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-氨磺酰基-1，2-苯并异噻唑-3-甲酰胺的制备
Figure A9880989803441
在10℃下，用草酰氯(1.68毫升，0.00337摩尔)及N，N-二甲基甲酰胺(1滴)处理5-(3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基-1，2-苯并异噻唑-3-羧酸(0.500克，0.00135摩尔)在9∶1二氯甲烷/四氢呋喃中的溶液。1小时后，反应混合物真空浓缩，溶于1，4-二噁烷中，在0℃下滴加到磺酰胺(1.29克，0.0135摩尔)的1，4-二噁烷溶液中。于室温下搅拌过夜后，反应混合物真空浓缩，溶于乙酸乙酯中，依次用盐水及10％HCl水溶液洗涤，用无水硫酸镁干燥，真空浓缩，产生粗制品。粗制品经硅胶使用6∶4乙酸乙酯/己烷过滤，产生标题产物的灰白色固体，mp 221℃。
实施例163
5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-N-异丙基-1，2-苯并异噻唑-3-甲酰胺的制备
在室温下，将1-(3-二甲氨丙基)-3-乙基碳化二亚胺盐酸盐(0.300克，0.00157摩尔)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸(0.400克，0.00108摩尔)、异丙胺(0.140克，0.00237摩尔)、二甲胺吡啶(0.000100克)与二氯甲烷的混合物中。所得混合物于室温下搅拌过夜，在二氯甲烷及水之间分配。以0.5M盐酸及盐水洗涤有机层，用无水硫酸钠干燥，过滤，真空浓缩。所得残留物经硅胶使用二氯甲烷∶乙酸乙酯层析，产生标题化合物的白色固体(0.250克，56.2％，mp 110-113℃)。
基本上采用相同方法，但改用适当取代的胺，得到下列化合物：
Figure A9880989803461
R11             R12                           mp℃H                       93-96CH3        
Figure A9880989803463
            117-119H                H                             227-229CH3             CH3                         95-98H              
Figure A9880989803464
             275H                CH2CO2H
实施例164
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-甲氧基-1，2-苯并异噻唑-3-甲酰胺的制备
在冰浴上依次将N，N-二甲基甲酰胺(5滴)及草酰氯(13.5毫升，0.0269摩尔)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸(4.00克，0.0108摩尔)、二氯甲烷与四氢呋喃的混合物中。所得混合物于氛围温度下搅拌90分钟，真空浓缩。残留物溶于四氢呋喃中，取25％此溶液加至含O-甲基羟胺盐酸盐(0.900克，0.0108摩尔)、四氢呋喃与三乙胺(2.25毫升，0.0162摩尔)的混合物中。所得混合物于室温下搅拌过夜，倒至冰水中，以二氯甲烷萃取。有机层用无水硫酸镁干燥，过滤，及真空浓缩。残留物经硅胶使用二氯甲烷层析，产生标题化合物的浅黄色固体(0.240克，22.3％，mp125-127℃)。
基本上采用相同方法，使用适当羟胺，得到下列化合物：
Figure A9880989803481
R12              R21                     mp℃H                 CH2CH＝CH2            91-92CH3              H                       118-120H                 CH2C6H5             96-97H                 SO2OH                  221H                 H                       234
实施例165
1-甲基-6-(三氟甲基)-3-(3-戊烯基-1，2-苯并异噻唑-5-基)-2，4(1H，3H)-嘧啶二酮的制备
向5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸(0.200克，0.000540摩尔)的二氯甲烷溶液中加入N，N-二甲基甲酰胺(1滴)，然后加入草酰氯的二氯甲烷溶液(2.0M，0.540毫升，0.00108摩尔)。所得混合物于室温下搅拌90分钟，真空浓缩成白色固体，保留备用。于-78℃下，在含氰化铜(0.061克，0.000675摩尔)的四氢呋喃溶液中滴加正丁基锂(2.5M己烷溶液，0.540毫升，0.00135摩尔)。使反应混合物回温5分钟，然后再降回-78℃。用第一个步骤所得白色固体的四氢呋喃溶液处理混合物，所得混合物于-78℃下搅拌1小时。以饱和氯化铵中止反应混合物的反应，以乙酸乙酯稀释。有机层依次饱和氯化铵、水及盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩成黄色浆状物。此浆状物经硅胶使用己烷∶乙酸乙酯层析，产生标题化合物的无色浆状物(0.142克，64.0％)，以NMR光谱分析法鉴定。
基本上采用相同方法，得到下列化合物：
Figure A9880989803491
                    R12                    mp℃
                    C(CH3)2              83-85
                    C6H5                 93-95
                CH(CH3)CH2CH3           75-77
实施例166
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N甲基-N-(甲磺酰基)1，2-苯并异噻唑-3-甲酰胺的制备
Figure A9880989803501
向5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-羧酸胺(0.300克，0.000670摩尔)的丙酮溶液中添加硫酸二甲酯(0.180克，0.00140摩尔)，然后加入碳酸钾(0.250克，0.00180摩尔)至含。所得混合物于回流下搅拌1小时，真空浓缩。残留物分布在二氯甲烷与水之间。保留有机层，以二氯甲烷萃取水层。合并的有机层以水洗涤，用无水硫酸钠干燥，过滤，及真空浓缩。残留物经硅胶使用乙酸乙酯∶己烷层析，产生标题化合物的白色固体(0.232克，74.9％，mp 120-122℃)。
基本上采用相同方法，得到下列化合物：
          R42                  R42                 mp℃
      CH2OCH2CH3           CH3                  91-93
      CH2OCH2CH3           CH2C6H5           185-186
      CH2CO2CH3            CH2C6H5           158-160
         CH3                 CH2C6H5           ＞225
实施例167
3-(3-异丙基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
使5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸(2.00克，0.00484摩尔)及喹啉(20.0毫升)的混合物搅拌加热至140℃。15分钟后，混合物冷却至室温，以乙酸乙酯稀释，依次用2N盐酸，饱和碳酸氢钠溶液及盐水洗涤，用无水硫酸镁干燥，及真空浓缩成黄色固体。此固体用己烷∶二氯甲烷重结晶，产生标题化合物的灰白色固体(0.640克，35.8％，mp 139-140℃)，以NMR及IR光谱分析法鉴定。
实施例168
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸，烯丙酯的制备
Figure A9880989803512
将N，N-二甲基甲酰胺(8滴)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸(2.00克，0.00484摩尔)与二氯甲烷的混合物中。混合物于冰浴上冷却，添加草酰氯(2.0M二氯甲烷溶液，6.05毫摩尔，0.0121摩尔)。所得混合物于冰浴上搅拌1小时，真空浓缩。残留物溶于四氢呋喃中，在此溶液中添加烯丙醇(0.420克，0.0185摩尔)及三乙胺(1.50毫升，0.0108摩尔)。混合物于室温下搅拌3天。添加二甲氨基吡啶(0.0100克)，混合物于室温下搅拌24小时，过滤，滤液真空浓缩。残留物溶于醚中，以饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩。残留物经硅胶使用己烷∶乙酸乙酯层析，产生标题化合物的白色固体(mp 115-116℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，但改用适当醇或硫醇，得到下列化合物：
W14                     mp℃
OCH3
OCH(CH3)2             207-209
Figure A9880989803532
        164-165
OCH2C6H5
Figure A9880989803533
SCH2CH3
实施例169
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸的制备
在0℃下将三溴化硼的二氯甲烷溶液(1.0M，100毫升，0.100摩尔)加到5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸乙酯(6.30克，0.0143摩尔)的二氯甲烷溶液中，保持温度不超过15℃。所得混合物于氛围温度下搅拌1小时，以3N盐酸中止反应，以二氯甲烷稀释。分离有机层，依次用水及盐水洗涤，用无水硫酸镁干燥，真空浓缩，产生标题化合物的灰白色固体(mp155-156℃)，以NMR及IR光谱分析法鉴定。
基本上采用相同方法，由其乙酯制得5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-羧酸。
实施例170
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-α，α-二甲基-1，2-苯并异噻唑-3-乙酰胺的制备
Figure A9880989803541
将N，N-二甲基甲酰胺(8滴)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸(0.800克，0.00194摩尔)及二氯甲烷的混合物中。混合物于冰浴上冷却，添加草酰氯(2.0M二氯甲烷溶液，2.42毫升，0.00485摩尔)。所得混合物于冰浴上搅拌一小时，真空浓缩。残留物溶于四氢呋喃中。添加N，N-二异丙氨基磺酰胺(0.410克，0.00278摩尔)、乙基二异丙胺(0.310克，0.00240摩尔)及二甲胺吡啶(0.0100克)，所得混合物于室温下搅拌过夜。混合物过滤，滤液真空浓缩，产生黄色树脂。树脂经硅胶过滤，产生标题化合物的黄褐色树脂(0.500克，44.8％)。
实施例171
3-[3-(1，1-二甲基-2-氧丙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
将N，N-二甲基甲酰胺(8滴)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸(0.800克，0.00194摩尔)及二氯甲烷的混合物中。混合物于冰浴上冷却，添加草酰氯(2.0M二氯甲烷溶液，2.42毫升，0.00484摩尔)。所得混合物于冰浴上搅拌一小时，真空浓缩。残留物溶于四氢呋喃中。所得溶液滴加至甲基锌化氯(2.0M，0.970毫升，0.00194摩尔)的四氢呋喃混合物中，然后添加四-三苯基膦钯(0.220克，0.000190摩尔)。所得混合物于室温下搅拌过夜，添加10％盐酸中止反应，以乙酸乙酯萃取。有机层以饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，过滤及真空浓缩成橙色固体。此固体经硅胶层析，产生标题化合物的灰白色固体(0.270克，65.7％，mp 195-196℃)。
实施例172
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酰胺的制备
Figure A9880989803561
将N，N-二甲基甲酰胺(8滴)加到5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸(2.00克，0.00484摩尔)及二氯甲烷的混合物中。混合物于冰浴上冷却，添加草酰氯(2.0M二氯甲烷溶液，6.05毫升，0.0121摩尔)。所得混合物于冰浴上搅拌一小时，真空浓缩。残留物溶于四氢呋喃中。所得溶液经氨气饱和后，添加三乙胺。混合物过滤，滤液真空浓缩成固体。此固体用二氯甲烷∶己烷重结晶，产生标题化合物的黄褐色固体(1.65克，82.7％，mp 192-196℃)，以NMR及IR光谱分析法鉴定。
实施例173
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-N-(甲磺酰基)-1，2-苯并异噻唑-3-乙酰胺的制备
将N，N-二甲基甲酰胺(8滴)加到5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸(2.00克，0.00484摩尔)及二氯甲烷的混合物中。混合物于冰浴上冷却，添加草酰氯(2.0M二氯甲烷溶液，6.05毫升，0.0121摩尔)。所得混合物于冰浴上搅拌一小时，真空浓缩。残留物溶于四氢呋喃中。添加甲磺酰胺(0.690克，0.00726摩尔)后，添加乙基二异丙胺(0.940克，0.00727摩尔)及二甲氨基吡啶(0.100克)。所得混合物于室温下搅拌并过滤。滤液真空浓缩，残留物经硅胶使用己烷∶乙酸乙酯过滤。滤液真空浓缩成黄褐色固体。此固体悬浮于二氯甲烷中，搅拌，再过滤一次，产生标题化合物的白色固体(0.320克，13.5％，mp264-265℃)。
基本上采用相同方法，得到下列化合物：
Figure A9880989803581
                    R41
                  CH2CH3
                  CH(CH3)2
                C(CH3)CH2CH3
                    R61
                
Figure A9880989803582
实施例174
{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}磺酰基}乙酸的制备
使{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}磺酰基}乙酸甲酯(1.00克，0.00210摩尔)、乙酸及10％盐酸(2.00毫升)的混合物于60℃下搅拌过夜。再添加盐酸(37％，1.20毫升)，混合物于80℃下搅拌5小时。混合物冷却至室温，于搅拌下倒至冰水中，过滤，产生标题化合物的白色固体(0.760克，78.4％，mp 215℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，由其甲酯制得{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫代}乙酸。
实施例175
{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}磺酰基}乙酸甲酯的制备
Figure A9880989803591
在0℃下将间-氯过苯甲酸(纯度70％，1.91克，0.00774摩尔)的二氯甲烷溶液加到{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫代}乙酸甲酯(1.00克，0.00225摩尔)的二氯甲烷溶液中。当由薄层层析法判断反应完成时，混合物依次用5％碳酸钠及盐水洗涤，及真空浓缩成白色泡沫状物。此泡沫状物于醚中研磨，产生标题化合物的白色固体(0.500克，46.7％，mp 209-210℃)，以NMR光谱分析法鉴定。
实施例176
N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}-N-(甲磺酰基)甘氨酸甲酯的制备
Figure A9880989803601
向2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}-N-(甲磺酰基)-乙酰胺(0.500克，0.00115摩尔)的混合物中加入溴乙酸甲酯(0.130毫升，0.00138摩尔)后加入氢化钠(60％，00690克，0.00173摩尔)。所得混合物倒至水中，以二氯甲烷萃取。合并的有机层用无水硫酸镁干燥，过滤，及真空浓缩成油。此油状物于醚中研磨，产生标题化合物的白色固体(0.270克，46.4％，mp 135-136℃)，以NMR光谱分析法鉴定。
实施例177
3[3-[(乙氧甲氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
向3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.800克，0.00224摩尔)与二氯甲烷的混合物中加入乙基二异丙胺(0.780毫升，0.00448摩尔)及氯甲基乙基醚(0.310毫升，0.00336摩尔)。所得混合物于室温下搅拌42.5小时，加醚稀释，依次用1M盐酸水溶液、饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩成黄色浆物。此浆物经硅胶使用己烷∶乙酸乙酯层析，产生产物的白色固体，以NMR光谱分析法鉴定。
基本上采用相同方法，但改用适当烷化剂，得到下列化合物：
Figure A9880989803612
                   R22                     mp℃
                
Figure A9880989803613
                CH2OCH2C6H5           114
                CH2OCH3                  138-141
                
Figure A9880989803614
R22                     mp℃
Figure A9880989803621
CH2SCH3              145-147
Figure A9880989803622
实施例178
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸的制备
将37％盐酸(5.00毫升)加到{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸甲酯(4.19克，0.00977摩尔)与乙酸的混合物中。所得混合物于65℃下搅拌过夜，冷却至室温。混合物真空浓缩。残留物悬浮于水中，缓缓添加碳酸氢钠固体至中性pH，以中止反应。所得混合物分布在醚与饱和碳酸氢钠之间，过滤。滤液以二氯甲烷洗涤，以盐酸酸化，过滤，得到标题产物的白色固体(2.87克，70.7％，mp 191-192℃)，以NMR光谱分析法鉴定。
实施例179
2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}-N-(甲磺酰基)乙酰胺二甲胺盐的制备
Figure A9880989803631
将二甲胺(2.0M四氢呋喃溶液，1.04毫升，0.00208摩尔)加到2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}-N-(甲磺酰基)乙酰胺(0.510克，0.00104摩尔)的四氢呋喃溶液中。所得混合物搅拌5分钟，真空浓缩。残留物溶于四氢呋喃中，添加醚使之结晶。所得灰白色固体(0.420克，75.1％，mp 102-107℃)，以NMR光谱分析法鉴定为标题化合物。
基本上采用相同方法，由2-{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫代}-N-(甲磺酰基)乙酰胺制得2-{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫代}-N-(甲磺酰基)乙酰胺二甲胺盐。
实施例180
{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸二甲胺盐的制备
将二甲胺的四氢呋喃溶液(2.0M，1.23毫升，0.00246摩尔)加到{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸(0.510克，0.00123摩尔)的四氢呋喃溶液中。混合物搅拌15分钟，以醚稀释，分离所得的灰白色固体(0.420克，74.2％，mp 175-176℃)，以NMR光谱分析法鉴定为标题化合物。
基本上采用相同方法，由{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫代}乙酸得到{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫代}乙酸二甲胺盐。
实施例181
2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基-N-(甲磺酰基)-乙酰胺的制备
将1，1’-羰基二咪唑(1.17克，0.00722摩尔)加到{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸(1.50克，0.00361摩尔)的四氢呋喃溶液中。混合物于回流下搅拌1小时，冷却至室温。添加甲磺酰胺(0.755克，0.00794摩尔)后，添加1，8-重氮双环[5.4.0]十一碳-7-烯(1.19毫升，0.00794摩尔)。所得混合物于室温下搅拌过夜，倒至10％盐酸中，过滤。所得白色固体于四氢呋喃中研磨，过滤，产生标题化合物的灰白色固体(1.00克，56.2％，mp＞240℃)，以NMR光谱分析法鉴定。
基本上采用相同方法，由{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}磺酰基}乙酸制得2-{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫}-N-(甲磺酰基)乙酰胺。
实施例182
3-{3-[溴(苯磺酰基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803661
向3-[3-(苯磺酰基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(0.400克，0.000831摩尔)的乙酸乙酯溶液中加入48％氢溴酸(4滴)后再加入溴之乙酸乙酯溶液(0.522M，1.67毫升，0.000872摩尔)。所得混合物于回流下搅拌1.5小时。再添加溴在乙酸乙酯里的物质(1.67毫升)，所得混合物于回流下搅拌1小时。混合物冷却至室温，以乙酸乙酯稀释，依次用0.1M亚硫酸钠、饱和碳酸氢钠及盐水洗涤，用无水硫酸镁干燥，过滤，真空浓缩。残留物经硅胶使用己烷∶乙酸乙酯层析，产生标题化合物的白色晶体(0.420克，90.1％，mp 182-183℃)，以NMR光谱分析法鉴定。
实施例183
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-乙酸甲酯的制备
Figure A9880989803662
将氢化钠(60％，0.0900克，0.00225摩尔)分批加入5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸甲酯(0.400克，0.00100摩尔)、N，N-二甲基甲酰胺与乙基碘(0.980克，0.00628摩尔)的混合物中。混合物于室温下搅拌5天，以二氯甲烷稀释，依次用8％盐酸、水及盐水洗涤，用无水硫酸镁干燥，过滤，及真空浓缩。残留物经硅胶使用醚∶己烷∶二氯甲烷层析，产生标题化合物(0.260克，60.9％)，以NMR光谱分析法鉴定。
基本上采用相同方法，但改用适当烷化剂，得到下列化合物：
Figure A9880989803671
W15                  W16
H                     CH2CH＝CH2CH2CH＝CH2             CH2CH＝CH2
H                     CH7C≡CHCH7C≡CH                CH7C≡CH
H                     CH2C6H5CH2C6H5               CH2C6H5
          -CH2CH2-
实施例184
1-甲基-3-{3-[1-(甲磺酰基)乙基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮的制备
Figure A9880989803672
将氢化钠(60％，0.120克，0.00300摩尔)加到1-甲基-3-{3-[1-(甲磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(1.00克，0.00238摩尔)的四氢呋喃悬浮液中。所得混合物于室温下搅拌1小时，以碘甲烷(0.220毫升，0.00360摩尔)处理。混合物于室温下搅拌2小时，部份真空浓缩，加水稀释，以乙酸乙酯萃取。以水洗涤有机层，用无水硫酸镁干燥，真空浓缩成褐色泡沫状物。此泡沫状物经硅胶使用二氯甲烷/醚层析，产生标题化合物的灰白色固体(0.420克，40.4％)，以NMR光谱分析法鉴定。
基本上采用相同方法，但使用适当烷化剂，得到下列化合物：
                           W19
                        CH2CH＝CH2
                        CH2C≡CH
                        CH2C6H5
实施例185
对试验化合物的芽后除草性评估
由下列试验证明本发明化合物芽后除草活性，其中以试验化合物处理各种双子叶及单子叶植物。试验中，使幼苗于专用盘中生长约2周。试验化合物分散在含0.5％TWEEN20(一种来自亚特拉斯化学工业(Atlas Chemical Industries)的聚氧乙烯山梨糖醇酐单月桂酸酯表面活性剂)的50/50丙酮/水混合物中。当利用40psi喷嘴施用至植物一段固定时间时，其用量足以提供相当于每公顷约0.0157公斤至0.500公斤活性化合物。喷洒后，植物置于温室平台上，根据常规温室方法照料。处理后4至5周，检查幼苗，根据如下的分级系统分级。数据示于下表I。若某指定化合物涉及一个以上的试验时，则数据取平均值。
这些评估法中采用的植物品种用字母缩写、俗名及学名表示。
该芽后除草评估法中采用的化合物用化合物编号表示，并说明其名称。表I中的数据按化合物编号表示。
除草性分级表
除草性评估结果以分级表示(0至9)。此等级系根据肉眼观察植物直立性、活力、变形、大小、变色及整体植物的外观，与对照组比较来评定。
分级              定义                       相对于对照组的控制％
9                 完全消灭                   100
8                 几乎完全消灭               91-99
7                 良好除草效果               80-90
6                 有除草效果                 65-79
5                 严重受损                   45-64
4                 受损                       30-44
3                 中度影响                   16-29
2                 轻度影响                   6-15
1                 微量影响                   1-5
0                 无影响                     0
"空白"表示没有进行评估。
除草性评估中采用的植物品种字母缩写              俗名             学名ABUTH                 茼麻             Abutilon theophrasti，Medic.AMBEL                 猪草             Ambrosia artemisifolia，L.CASOB                 山扁豆           Cassia obtusifolia，L.CHEAL                 藜               Chenopodium album，L.GALAP                 猪殃殃           Galium aparineIPOHE                 藤牵牛           Ipomoea hederacea，(L.)Jacq.IPOSS                 牵牛属           Ipomoea Spp.ECHCG                 野稗             Echinochloa crus-galli，(L.)BeauSETVI                 莠草             Setaria viridis，(L.)Beau字母缩写              俗名             学名GLXMAW                威廉种大         Glycine max，(L.)Merr.cv WilliamsGLXMA                 大豆             Glycine max，(L.)Merr.ORYSAT    狄波耐种稻     Oryza sativa，(L.)TebonnetTRZAWR    冬小麦理班种   Triticum aestivum，cv RibandZEAMX     玉米           Zea mays，L.
                经评估为除草剂的化合物化合物编号
1. 3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)2，4(1H，3H)-嘧啶二酮
2.{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯
3. 2-{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯
4. 1-甲基-3-(3-苯基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
5. 3-[3-(对-乙苯基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
6. 1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
7. 3-[3-(2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
8.{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯
9. 2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}丙酸甲酯
10. 2-[3-(6-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
11. 3-[3-(6-羟基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
12.{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}乙酸甲酯
13. 2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯
14. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯，(R)-
15. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯，(S)-
16. 3-[3-(溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
17. 3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
18. 3-[3-(2-甲氧基-3，5-二甲苯基)-1，2-苯并异噻唑-5-基]1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
19. 3-(3-异丙氧基-1，2-苯并异噁唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
20. 3-(3-氯-1，2-苯并异噁唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
21. 1-甲基-3-(3-氯-1，2-苯并异噁唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
22.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}氧基}乙酸甲酯
23. 3-(6-氟-3-甲基-1，2-苯并异噁唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
24. 3-[3-(6-甲基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1，6-二甲基-2，4(1H，3H)-嘧啶二酮
25. 1-甲基-3-(3-苯基-1，2-苯并异噁唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
26.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，4-二甲苯基}氧基}乙酸甲酯
27. 2-{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，4-二甲苯基}氧基}丙酸甲酯
28. 2-{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-乙基苯氧基}丙酸甲酯
29. 1-乙基-3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
30. 2-{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-异丙基苯氧基}丙酸甲酯
31. 3-[3-(甲氧甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
32. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，乙酸酯
33. 2-{{2-{5-[3，6-二氢-3-甲基-2-氧-6硫代-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯
34. 3-[3-(6-甲氧基-2，3，4-三甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
35. 3-(1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
36. 3-(3-溴-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
37. 3-(3-氯-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
38.{{2-{5-[3，6-二氢-3，4-二甲基-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯
39. 2-{{2-{5-[3，6-二氢-3，4-二甲基-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯
40. 3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
41. 3-(4-氯-3-(6-羟基-间-甲苯基)-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
42. 3-(3-甲氧基-1，2-苯并异噁唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
43. 3-[3-(邻-甲氧苯氧基)-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
44. 1-甲基-3-(2-甲基-3-氧-1，2-苯并异噁唑啉-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
45. 3-[3-(5-乙基-2-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
46. 3-[3-(5-异丙基-2-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
47. 2-{邻-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}氧基}苯氧基}丙酸甲酯
48.{邻-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}氧基}苯氧基}乙酸甲酯
49.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸乙酯
50.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸异丙酯
51.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-丙炔酯
52. 1-甲基-3-{3-{6-[(吗啉羰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
53.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-吗啉乙酯
54. 1-甲基-3-{3-{6-{[(4-苯基-1-哌嗪基)羰基]-甲氧基}间-甲苯基}-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
55. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丁酸甲酯
56. 1-甲基-3-{3-[6-(2-丙炔氧基)-间-甲苯基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
57. 3-{3-[6-(氰甲氧基)-间-甲苯基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
58. 3-{3-[6-(1-氰乙氧基)-间-甲苯基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
59. 3-[3-(6-异丙氧基-间-甲苯基)-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
60. 3-{3-{6-[(二乙基氨基甲酰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
61. 3-{3-{6-[(二异丙基氨基甲酰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
62. 3-{3-{6-[(1-苯并咪唑基羰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
63. 3-{3-{6-{[(间-氰苯基)氨基甲酰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
64.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸
65. 3-{3-[6-(烯丙氧基)-间-甲苯基}-1，2-苯并异噁唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
66. 3-[3-(6-乙氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
67. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丁酸乙酯
68.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸叔丁酯
69.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸烯丙酯
70.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-(二甲氨基)乙酯
71.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-氯乙酯
72.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-吡啶甲酯
73.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸3-苯基-2-丙炔酯
74.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-甲基-2-丙炔酯
75.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-丁炔酯
76.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-甲基-2-丁炔酯
77. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸2-丙炔酯
78. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸烯丙酯
79. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸糠酯
80. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸2-丁炔酯
81. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸2-氯乙酯
82. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸异丙酯
83.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-乙酸丙酯
84.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸环戊酯
85.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1，2，2-三甲基丙酯
86.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1，2-二甲基丙酯
87.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2，2-二甲基丙酯
88.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-丁烯酯，(E)-或(Z)-
89.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸肉桂酯，(E)-或(Z)-
90.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2，2，2-三氟乙酯
91. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸叔丁酯
92. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸
93.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸甲酯
94. 1-烯丙基-3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
95. 1-异丙基-3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
96.{{2-{5-[3-乙基-3，6-二氢-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸甲酯
97. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸甲酯
98. 1-甲基-3-{3-[(甲硫基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
99.{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫}乙酸甲酯
100. 1-甲基-3-{3-[(甲磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
101. 3-{3-[(二甲氨基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
102.N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}-N-甲基甘氨酸乙酯
103.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}乙酸2-丙炔酯
104. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸乙酯
105. 3-[3-(邻-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)嘧啶二酮
106. 3-[3-(咪唑-1-基甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
107. 1-甲基-3-[3-(2-丙炔氧基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
108.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}氧基}乙腈
109. 3-[3-(烯丙氧基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
110. 3-(3-异丙氧基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
111. 3-(3-甲氧基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
112.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}氧基}乙酸甲酯
113. 5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛
114. 3-[3-(二氯甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
115.{{2-{5-[3-烯丙基-3，6-二氢-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-丙炔酯
116. 1-甲基-3-(3-吗啉基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
117.N-{5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲磺酰胺
118. 3-[3-(二乙氨基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
119. 3-(3-乙基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
120. 3-[3-(邻-羟苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲)-2，4(1H，3H)-嘧啶二酮
121.N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰基}甲磺酰胺
122.N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}对-甲苯磺酰胺
123.对-氯-N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰基}苯磺酰胺
124.N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰基}-α-甲苯磺酰胺
125. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-丙炔酯
126. 3-{3-[5-(溴甲基)-2-甲氧苯基]-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
127. 3-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧基苯甲醛
128. 3-[3-(氯甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
129.α-乙酰基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸叔丁酯
130.α-乙酰基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸
131. 1-甲基-3-[3-(3-氯丁基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
132.{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酸甲酯
133. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}丙酸甲酯
134.{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酸2-丙炔酯
135.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}乙酸2-丙炔酯
136.{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲酰苯氧基}乙酸甲酯
137. 3-[3-(氟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
138.{{2-{4-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯
139. 3-[3-(对-氯苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
140. 3-[3-(二氟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
141. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈
142.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸2-丙炔酯
143. 3-[3-(2-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，乙酸酯
144. 2-{{2-{4-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}丙酸2-丙炔酯
145.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}丙二酸二-叔丁酯
146.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}丙二酸叔丁基甲酯
147.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}丙二酸单甲酯
148. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙酸甲酯
149. 3-{3-[(2-氯-5-硝基苯氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
150. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸
151. 1-甲基-3-[3-(1-哌嗪基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
152. 3-{3-{[5-氯-4-(三氟甲基)-2-噻唑基]氨基}-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
153. 2-{{2-{4-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}丙酸甲酯
154. 3-[3-(2-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
155.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}膦酸二乙酯
156.{{5-[3，6-二氢-3-甲基-2，6-二氧4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}三甲基铵化溴
157. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酸甲酯
158.N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}邻苯二甲酰亚胺
159.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}氨基磷酸二乙酯
160.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}膦酸
161. 3-(4-氯-6-氟-3-甲基-1，2-苯并异噁唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
162.{{2-{5-[2-(甲硫基)-6-氧-4-(三氟甲基)-1(6H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸甲酯
163.{{2-{5-[2-(甲硫基)-6-氧-4-(三氟甲基)-1(6H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-丙炔酯
164.邻-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}肉桂酸甲酯
165. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙二腈
166. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸甲酯，S，S-二氧化物
167. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙酰胺
168. 1-甲基-3-{3-[(甲亚磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
169. 3-[3-(对-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
170. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基-丙酸甲酯
171. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}戊酸乙酯，DL-
172.{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰氧基}乙酸甲酯
173. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸钠，DL-
174. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸，DL-，与二异丙胺化合
175.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸，与二异丙胺化合
176. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸，铵盐，DL-
177.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸，铵盐
178.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸钠
179. 3-{3-[(异丙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
180. 3-{3-[(2-氟乙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
181. 3-{3-[(苄氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
182.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸3-甲基-3-丁烯酯
183.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-甲基烯丙酯
184.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2，4-己二烯酯
185.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-环己烯-1-基酯
186.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-甲烯丙酯
187.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸3-甲基-2-丁烯酯
188. 4-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}2-丁烯酸甲酯，(E)-与(Z)-
189. 1-甲基-3-{3-{6-[(四氢-5-甲基-2-氧-3-呋喃基)氧]-间-甲苯基}-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，DL-
190. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰氧基}丙酸，DL-
191.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-甲氧乙酯
192.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-甲基-2-甲氧乙酯，DL-
193. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}-N-(2-丙炔基)乙酰胺
194.邻-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰氧基}肟丙酮
195. 3-[3-(乙氧甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
196. 3-{3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
197. 1-甲基-3-{3-[(间-甲苄基)硫代]甲基}-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
198. 3-{3-[(2-氯乙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
199. 3-{3-[2-氯-1-(氯甲基)乙基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
200. 3-{3-[(2-乙氧乙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
201. 1-甲基-3-{3-[(2，2，2-三氟乙氧基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
202. 3-{3-[(异丙硫基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
203. 3-{3-[(2，2-二氟乙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
204. 3-[3-(丁氧甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
205. 3-{3-[(2-丁烯氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
206. 1-甲基-3-{3-[(1-甲基烯丙氧基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
207. 3-{3-{[2-氟-1-(氟甲基)乙氧基]甲基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
208. 1-甲基-6-(三氟甲基)-3-[(2，2，2-三氟-1-甲基乙氧基)甲基]-1，2-苯并异噻唑5-基]-2，4(1H，3H)-嘧啶二酮
209. 3-{3-[(2-环己烯-1-基氧)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
210. 1-甲基-3-{3-[(3-甲基-2-丁烯氧基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
211. 1-甲基-3-{3-{{[4-(1-甲基乙烯基)-1-环己烯-1-基]甲氧基}甲基}-1，2-苯并异噻唑-5-基}-2，4(1H，3H)-嘧啶二酮
212. 3-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}-2-亚甲基丁酸甲酯
213. 3，4-二氢-3-(3-甲基-1，2-苯并异噻唑-5-基)-2，4-二氧-6-(三氟甲基)-1(2H)-嘧啶乙腈
214. 1-乙基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与2-乙氧基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-4(3H)-嘧啶二酮(1∶1)
215. 1-异丁基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与2-异丁氧基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6(三氟甲基)-4(3H)-嘧啶二酮(55∶45)
216. 1-烯丙基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮与2-(烯丙氧基)-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-4(3H)-嘧啶二酮(85∶15)
217. 3-(3-甲基-1，2-苯并异噻唑-5-基)-1-(2-丙炔基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
218. 1-苄基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
219. 1-甲基-3-{3-[(4-戊烯氧基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
220. 3-{3-[(3-己烯氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(E)-
221. 1-甲基-3-{3-{[(对-甲基苯乙基)氧]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
222. 3-{[(2，4-二甲基苯乙基)氧]甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
223. 3-{3-[(3-丁烯氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
224. 3-{3-[(3-氯丙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
225. 3-[3-(羟甲基)-1，2-苯并异噻唑-5基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
226. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(邻-甲苯磺酰基)乙酰胺
227. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3基}对-甲苯基}氧基}-N-(苯乙烯基磺酰基)乙酰胺
228. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(间-硝基苯基)磺酰基]乙酰胺
229. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(对-硝基苯基)磺酰基]乙酰胺
230. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(对-氟苯基)磺酰基]乙酰胺
231. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(对-甲氧苯基)磺酰基]乙酰胺
232. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(苯磺酰基)乙酰胺
233. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(α，α，α-三氟-间-甲苯基)磺酰基]乙酰胺
234. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(邻-氟苯基)磺酰基]乙酰胺
235. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(间氯苯基)磺酰基]乙酰胺
236.邻-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}苄腈
237. 1-甲基-3-{3-[(邻-硝基苯氧基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
238. 1-甲基-6-(三氟甲基)-3-{3-{[(α，α，α-三氟邻甲苯基)氧]甲基}-1，2-苯并异噻唑-5-基}-2，4(1H，3H)-嘧啶二酮
239.{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基水杨酸酯
240. 1-甲基-3-{3-{[间-(甲氨基)苯氧基]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
241. 3-{3-[(间-乙酰苯氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
242.间-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}苄腈
243. 1-甲基-6(三氟甲基)-3-{3-{[(α，α，α-三氟间-甲苯基)氧]甲基}-1，2-苯并异噻唑-5-基}-2，4(1H，3H)-嘧啶二酮
244. 1-甲基-3-{3-{[间-(三氟甲氧基)苯氧基]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
245. 2-(烯丙氧基)-3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-4(3H)-嘧啶二酮
246.{{2-{5-[2-乙氧基-6-氧-4-(三氟甲基)-1(6H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸甲酯
247. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲苯基-1，2-苯并异噻唑-3-乙酸乙酯
248. 3-{3-[(间-氟苯氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
249.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-氰基乙酯
250.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-甲基己酯，DL-
251.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2，2，3，3，3-五氟丙酯
252.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸十二烷基酯
253.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸3-呋喃基甲酯
254.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸四氢糠基酯，DL-
255.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-甲基癸基酯，DL-
256.5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙腈
257.{对-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酸甲酯
258. 2-{对-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}丙酸甲酯
259.{对-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酸2-丙炔酯
260. 3-[3-(2-溴乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
261.{{2-{4-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}对甲基}氧基}乙酸甲酯
262. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲烷膦酸二甲酯
263.5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲烷膦酸二异丙酯
264.α-溴-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈
265.{{2-{4-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}乙酸叔丁酯
266. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙醛-3-肟，(E)-与(Z)-
267. 3-[3-(2-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
268. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-(甲磺酰基)乙酰胺
269.N-[(5-乙酰氨基-1，3，4-噻二唑-2-基)磺酰基]-2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰胺
270. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(3，5-二甲基异噁唑-4-)磺酰基]-乙酰胺
271. 5-氯-1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
272.{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}磺酰基}乙酸甲酯
273.{对-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酸叔丁酯
274.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，3-二甲苯基}氧基}乙酸甲酯
275. 2-{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，3-二甲苯基}氧基}丙酸甲酯
276. 1-甲基-6-(三氟甲基)-3-(3-乙烯基-1，2-苯并异噻唑-5-基)-2，4(1H，3H)-嘧啶二酮
277. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛-3-(O-甲基肟)，(E)-
278. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛-3-肟，(E)-
279. 5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙烯酸甲酯，(E)-
280.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，3-二甲苯基}氧基}乙酸2-丙炔酯
281.{对-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酸
282.{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}磺酰基}乙酸
283.{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫}乙酸
284. 3-[3-(2，2-二溴乙烯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
285. 1-甲基-3-[3-(3-氧-1-丁烯基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(E)-
286. 3-[3-(2-溴-2-氟乙烯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
287. 3-[3-(2，2-二氯乙烯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
288. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(2，4-二甲基噻唑-5-基)磺酰基]-乙酰胺
289. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-[(5-乙氧苯并噻唑-2-基)磺酰基]-乙酰胺
290.N-[(5-氯-3-甲基苯并[b}噻吩-2-基)磺酰基]-2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰胺
291. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙烯醛，(E)-
292.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸甲酯
293.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸
294. 2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}-N-(甲磺酰基)乙酰胺
295. 2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}-N-(甲磺酰基)乙酰胺二甲胺盐
296.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲氧基}乙酸二甲胺盐
297. 2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫}-N-(甲磺酰基)乙酰胺
298. 2-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫}-N-(甲磺酰基)乙酰胺二甲胺盐
299.{{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}硫}乙酸二甲胺盐
300. 3-[3-(溴氯甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
301. 3-[3-(间-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
302. 3-[3-(1，2-二溴丙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(1R，2S)-
303. 3-[3-(1，2-二溴丙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(1R，2R)-
304.{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}(甲磺酰基)氨甲酸叔丁酯
305.N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}甲磺酰胺
306.N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}甲基}-N-(甲磺酰基)甘氨酸甲酯
307. 3-(3-乙酰基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
308. 3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
309. 3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮甲磺酸酯
310. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮硝酸酯
311.{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}异硫氰酸甲酯
312.{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基基}乙酸
313. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰基异羟肟酸
314. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}丙酸
315. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸
316. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-甲氧基乙酰胺
317. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯
318. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯
319. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸苯酯
320. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸对氟苯酯
321. 3-[3-(2(和1)-溴1(和2)-羟丙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，非对映异构体的(4∶1)混合物
322. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
323. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺
324.N-[(氯甲基)磺酰基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
325. 2-{间-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}丙酸甲酯
326.{间-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2苯并异噻唑-3-基}苯氧基}乙酸2-丙炔酯
327. 3-[3-(间-乙氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
328. 3-[3-(间-异丙氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
329. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N，N-二甲基-1，2-苯并异噻唑-3-甲酰胺
330. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-异丙基-1，2-苯并异噻唑-3-甲酰胺
331.N-(5-叔丁基异噁唑-3-基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
332.{间-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酸甲酯
333. 3-[3-(2，5-二甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
334.N-[(氯甲基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
335. 2-{邻{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-(甲磺酰基)丙酰胺
336. 2-{邻{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-甲基乙酰基异羟肟酸
337. 3-[3-(溴乙酰基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
338. 3-[3-(氯乙酰基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
339. 3-[3-(1-溴乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
340. 3-[3-(1，1-二溴乙基)-1，2-苯并异噻唑5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
341.N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
342. 1-甲基-3-[3-[6-(甲硫基)间-甲苯基]-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
343.N-[(氯甲基)磺酰基]-2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基氧基}乙酰胺
344.N-[(氯甲基)磺酰基]-2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酰胺
345. 3-[6-氟-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
346. 3-[6-氟-3-(6-羟基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
347.{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧苯氧基}乙酸甲酯
348. 2-{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧苯氧基}丙酸甲酯
349.{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧苯氧基}乙酸2-丙炔酯
350. 3-[3-(1-甲氧乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
351. 3-{3-[1-(烯丙氧基)乙基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
352. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(苯磺酰基)-1，2-苯并异噻唑-3-甲酰胺
353. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(对-甲苯磺酰基)-1，2-苯并异噻唑-3-甲酰胺
354. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-甲氧基-N-甲基乙酰胺
355. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-甲基乙酰基异羟肟酸
356.N-[(对-氯苯基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
357. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(2-萘基磺酰基)-1，2-苯并异噻唑-3-甲酰胺
358. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(十二烷磺酰基)-1，2-苯并异噻唑-3-甲酰胺
359.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}乙酸甲酯
360. 3-[3-(3-溴丙烯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(E)-
361. 3-[3-(2-羟基-5-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
362. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺
363. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮甲磺酸酯
364. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮苯甲酸酯
365. 4’-氟-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-甲基-1，2-苯并异噻唑-3-羧基酰苯胺(carboxanilide)
366. 3-(6-氟-3-甲基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
367. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-甲基-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺
368. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮氯乙酸酯
369. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮苯乙酸酯
370. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙氧甲基)-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺
371. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮1-甲基乙磺酸酯
372. 3-[3-(二溴甲基)-6-氟-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
373. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-腈
374. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮甲基氨基甲酸酯
375. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮苯基氨基甲酸酯
376. 3-[3-(溴甲基)-6-氟-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
377. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲膦酸二乙酯
378. 3-[6-氟-3-(甲氧甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
379. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-乙腈
380. 3-[3-(6-甲氧基-5-茚满基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
381. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮丁磺酸酯
382. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮苯磺酸酯
383. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺
384. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸2-丁炔酯
385. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸2-(乙硫基)乙酯
386. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸2-氯烯丙酯
387. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸2-乙酰氨基乙酯
388. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸庚酯
389. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸2-(2-甲氧乙氧基)乙酯
390. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮苄基氨基甲酸酯
391. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(2-噻吩磺酰基)-1，2-苯并异噻唑-3-甲酰胺
392. 1-甲基-3-{3-[(苯硫基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
393. 1-甲基-3-{3-[(苯磺酰基)甲基]-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
394. 1-甲基-3-{3-[(苯亚磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
395. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(1-甲基丙基)磺酰基]-1，2-苯并异噻唑-3-甲酰胺
396. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸苄酯
397. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸对甲氧苄酯
398. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-甲基-1，2-苯并异噻唑-3-羧基异羟肟酸
399.N-(烯丙氧基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
400. N-(苄氧基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
401. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(2，4-二氯苯基)乙酸酯
402. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(邻-氯苯基)乙酸酯
403. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-甲氧基-1，2-苯并异噻唑-3-甲酰胺
404. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(邻-硝基苄基)磺酰基]-1，2-苯并异噻唑-3-甲酰胺
405. N-[(对-叔丁基苄基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
406. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-{[对-(三氟甲氧基)苄基]磺酰基}-1，2-苯并异噻唑-3-甲酰胺
407. 3-{3-[溴(苯磺酰基)甲基]-1，2-苯并异噻唑-5基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
408. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛3-(苯基腙)，(E)
409. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛3-(二甲基腙)，(E)-
410. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸3-羟丙酯
411. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸2-甲氧乙酯
412. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛3-(甲苯基腙)，(E)-
413. 3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮1-甲基乙磺酸酯
414. 3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮丁磺酸酯
415. 3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮苯磺酸酯
416. 3-[3-(1-氯乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
417. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧基异羟肟酸硫酸氢酯
418. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛-3-[双(2-羟乙基)二硫缩醛]二乙酸酯
419. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛-3-[双(2-羟乙基)二硫缩醛]
420.N-[(对-氯苄基)甲基氨磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
421. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-硫羧酸S-苄酯
422. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-硫羧酸S-乙酯
423. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-羧酸乙酯
424. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛-3-[双(3-羟丙基)二硫缩醛]
425.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}乙酸
426. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-硫基醛-3-[双(2-羟丙基)二硫缩醛]二乙酸酯
427. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(α-甲基苄基)磺酰基)-1，2-苯并异噻唑-3-甲酰胺
428. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1-(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}对-甲苯基}氧基}-N-(甲磺酰基)乙酰胺
429. 3-[3-(5-碘-2-甲氧基对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
430. 4’-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-N-甲基-N-甲磺酰苯胺
431. 1-甲基-6-(三氟甲基)-3-(3-戊酰基-1，2-苯并异噻唑-5-基)-2，4(1H，3H)-嘧啶二酮
432. 1-甲基-3-(3-新戊酰基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
433. 1-甲基-3-[(2-甲基丁酰基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
434.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-5-茚满基}氧基}乙酸甲酯
435. 2-{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-5-茚满基}氧基}丙酸甲酯
436.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-5-茚满基}氧基}乙酸2-丙炔酯
437. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-甲基-N-(甲磺酰基)乙酰胺
438. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-甲基-N-(甲磺酰基)乙酰胺
439.N-[5-氯-4-(三氟甲基)噻唑-2-基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
440.N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙氧甲基)-1，2-苯并异噻唑-3-甲酰胺
441.N-(苄磺酰基)-N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}羰基}甘氨酸甲酯
442. 3-[6-氯-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
443.{{2-{6-氯-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸甲酯
444. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-乙腈
445. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二乙基-1，2-苯并异噻唑-3-乙腈
446. 1-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}环丙腈
447. 3-[3-(α，α-二溴-2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
448. 3-[3-(5-碘-2-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
449. 3-(3-苯甲酰基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
450. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(对-甲氧苯基)乙酸酯
451. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮噻吩基乙酸酯
452. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(对-氯苯基)乙酸酯
453. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛-3-(二甲基缩醛)
454. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(间-甲氧苯基)乙酸酯
455. 3-{3-[(乙氧甲氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
456. 1-甲基-3-{3-{[(四氢-2H-吡喃-2-基)氧]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
457. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(3-甲基-2-亚噻吩基)-1，2-苯并异噻唑-3-乙腈
458.α-(环丙基亚甲基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈，(E)-与(Z)-
459.{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-碘苯氧基}乙酸甲酯
460.{2-{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-碘苯氧基}丙酸甲酯
461. 3-{3-[(苄氧基)甲氧基)甲基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
462. 3-[6-氟-3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
463. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮异烟酸酯
464. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(对-甲基苄基)磺酰基]-1，2-苯并异噻唑-3-甲酰胺
465. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(邻-甲基苄基)磺酰基]-1，2-苯并异噻唑-3-甲酰胺
466. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸
467. 3-{{2-[5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙醛1-(二甲基缩醛)
468.N-[(对-氯苄基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
469.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-碘-间-甲苯基}氧基}乙酸甲酯
470. 2-{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-碘-间-甲苯基}氧基}丙酸甲酯
471. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧基异羟肟酸
472. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-氨磺酰基-1，2-苯并异噻唑-3-甲酰胺
473. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮2-苯基丁酸酯
474. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮2，6-二氯异烟酸酯
475. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮5-异噁唑羧酸酯
476. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮5-硝基-2-呋喃甲酸酯
477. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮2-噻吩羧酸酯
478. 3-{3-[(甲氧甲氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
479.{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯
480. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮2-氯烟酸酯
481. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮6-氯烟酸酯
482.N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲酰胺
483. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(间-甲苄基)磺酰基]-1，2-苯并异噻唑-3-甲酰胺
484. 1-甲基-3-{3-{[(甲硫基)甲氧基]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
485. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(苯乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺
486.N-[(间-氯苄基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺
487. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸糠酯
488. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-N-(甲磺酰基)-1，2-苯并异噻唑-3-乙酰胺
489. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸异丙酯
490. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸甲酯
491. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸烯丙酯
492. 2-{{5-氯-2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酸甲酯
493.{{5-氯-2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸甲酯
494.N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-甲基-1，2-苯并异噻唑-3-甲酰胺
495. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮甲氧乙酸酯
496. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮环丙烷羧酸酯
497. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮2-呋喃甲酸酯
498. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮新戊酸酯
499. 3-(3-异丙基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
500. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺
501. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(苯乙烯基磺酰基)-1，2-苯并异噻唑-3-甲酰胺，(E)-
502. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(3，4-二甲氧苯基)乙酸酯
503. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮(2，5-二甲氧苯基)乙酸酯
504. 3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮氯苯基乙酸酯
505. 3-{3-[6-(烯丙氧基)-5-碘-间-甲苯基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
506. 3-[3-[4-氯-6-甲氧基-间-甲苯基]-1，2-苯并异噻唑5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
507. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3甲酰胺
508. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺
509. 5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酰胺
510. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸2-吡啶基甲酯
511. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-α，α-二甲基-1，2-苯并异噻唑-3-乙酰胺
512. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-(二异丙基氨磺酰基)-乙酰胺
513. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-羧酸甲酯
514. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸叔丁酯
515. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸
516. 1-(2氟乙基)-3-(3-甲基-1，2-苯并异噻唑-5-基)-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
517.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸(1-苯基-环丙基)甲酯
518.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸4-(甲硫基)丁酯
519.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸壬酯
520.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸1-乙烯基戊酯
521.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2，2-双[(烯丙氧基)甲基]丁酯
522.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸3-癸炔酯
523.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸3-(3-甲氧丙氧基)丙酯
524.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸，带有4-羟基环己烷羧酸乙酯的酯，异构物A
525.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸，带有4-羟基环己烷羧酸乙酯的酯，异构物B
526.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸11-十四烯酯，(E)-
527.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2，2-二甲基-3-苯基丙酯
528. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸2-丙炔酯
529. 2-{{2-{5-[3，6-二氢3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸2-丁烯酯
530. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸烯丙酯
531. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸1-甲基-2-丙炔酯
532. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸2-甲氧基-1-甲基乙酯
533.{{2-{5[3，6二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-(5，5-二甲基-间-二噁烷-2-基)乙酯
534.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸5-(叔丁基二甲硅烷氧基)戊酯
535.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸(四氢-3-呋喃基)甲酯，DL-
536.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸3-(3-甲氧丙氧基)丙酯
537. 1-甲基-3-{3-[6-(苯甲酰甲基氧基)-间-甲苯基]-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
538. 3-{3-{6-[(对-氯苯甲酰甲基)氧]间-甲苯基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
539. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰胺
540. 3-{3-[6-(3，3-二甲基-2-氧丁氧基)间-甲苯基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
541.对-{2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-丙酰氨基}苯甲酸乙酯
542. 3-{3-[6-[1-(3，4-二甲基苯甲酰基)乙氧基]间-甲苯基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
543. 3-{3-[6-{[对-(二氟甲氧基)苯甲酰甲基]氧基}间-甲苯基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
544. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸2-氯乙酯
545. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸2，2，2-三氟乙酯
546. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸2-甲氧基乙酯
547. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基丙酸异丙酯
548. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酰胺
549. 3-{3-[邻-(3，3-二甲基-2-氧丁氧基)苯基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
550. 3-{3-[邻-(1-(3，4-二甲基苯甲酰基)乙氧基]苯基}-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
551. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N，N-二甲基丙酰胺
552. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(丙磺酰基)乙酰胺
553. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(乙烯基磺酰基)乙酰胺
554. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(乙磺酰基)乙酰胺
555. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-(异丙磺酰基)乙酰胺
556. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-(丙磺酰基)乙酰胺
557. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-(乙烯基磺酰基)乙酰胺
558. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-(乙磺酰基)乙酰胺
559. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}二氟乙酸乙酯
560. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(异丙基磺酰基)乙酰胺
561. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-甲基乙酰胺
562. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-N-甲基乙酰胺
563. 2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}-乙酰胺
564. 1-甲基-3-[3-(3-氧-3-苯丙烯基)-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，(E)-
565. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-甲氧基-N-甲基-1，2-苯并异噻唑-3-丙烯酰胺，(E)-
566. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-丙烯酸烯丙酯，(E)-
567. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-丙烯醛，(E)-
568. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(异丙磺酰基)丙酰胺
569. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(丙磺酰基)丙酰胺
570. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(乙烯基磺酰基)丙酰胺
571. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(乙磺酰基)丙酰胺
572. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-N-(甲磺酰基)丙酰胺
573.N-(丁磺酰基)-2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酰胺
574.N-(丁磺酰基)-2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}苯氧基}乙酰胺
575.N-(丁磺酰基)-2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}丙酰胺
576. 2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}-2-甲基-N-(甲磺酰基)丙酰胺
577.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-氧丁酯
578.{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}对-甲苯基}氧基}乙酸2-羟基乙酯，乙酸酯
579.N-{{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}羰基}甘氨酸
580.α，α-二烯丙基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈
581. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二-2-丙炔基-1，2-苯并异噻唑-3-乙腈
582.α，α-二苄基-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈
583. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-甲基-1，2-苯并异噻唑-3-乙腈
584. 3-{3-{[(对-氯苄基)氧]甲基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
585. 3-{3-{[(2，4-二氯苄基)氧]甲基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
586. 3-{3-{[(3，4-二氯苄基)氧]甲基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
587. 1-甲基-3-{3-{[(间-甲基苄基)氧]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
588. 1-甲基-3-{3-{[(间-硝基苄基)氧]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
589. 1-甲基-3-{3-{[(对-硝基苄基)氧]甲基}-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
590. 1-甲基-3-{3-[1-(甲磺酰基)乙基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
591. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(2-甲基亚丙基)-1，2-苯并异噻唑-3-乙腈
592. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(2-吡啶亚甲基)-1，2-苯并异噻唑-3-乙腈
593. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(3-呋喃亚甲基)-1，2-苯并异噻唑-3-乙腈
594. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-亚糠基-1，2-苯并异噻唑-3-乙腈
595. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(咪唑-5-基亚甲基)-1，2-苯并异噻唑-3-乙腈
596. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(4-吡啶亚甲基)-1，2-苯并异噻唑-3-乙腈
597. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(对-甲基亚苄基)-1，2-苯并异噻唑-3-乙腈
598. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(吡咯-2-基亚甲基)-1，2-苯并异噻唑-3-乙腈
599. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(邻-甲氧亚苄基)-1，2-苯并异噻唑-3-乙腈
600. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(对-羟基亚苄基)-1，2-苯并异噻唑-3-乙腈
601. 5-[3，6-二氢-3-甲基-2，6二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(吲哚-2-基亚甲基)-1，2-苯并异噻唑-3-乙腈
602. 1-甲基-3-{3-[1-(甲磺酰基)-3-丁烯基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
603. 1-甲基-3-{3-[1-(甲磺酰基)-3-丁炔基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
604. 1-甲基-3-{3-[α-(甲磺酰基)苯乙基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮
605. 5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-(邻-氟亚苄基)-1，2-苯并异噻唑-3-乙腈
606.α-(邻氰基亚苄基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈，(E)-与(Z)-
607.α-(环戊基亚甲基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈，(E)-与(Z)-
                                                   表1
                                         对试验化合物的芽后除草评估
                                                                                         G               O       T
                 A       A       C       C       G       I       I       E       S       L       G       R       R       Z
                 B       M       A       H       A       P       P       C       E       X       L       Y       Z       E
                 U       B       S       E       L       O       O       H       T       M       X       S       A       A化合物   施用率      T       E       O       A       A       H       S       C       V       A       M       A       W       M编号  (公斤/公顷)   H       L       B       L       P       E       S       G       I       W       A       T       R       X1       0.5000     9.0     9.0     9.0     9.0     9.0             9.0     9.0     9.0     9.0     8.0     7.0     7.0     8.0
      0.2500     9.0     9.0     8.0     9.0     9.0             9.0     9.0     9.0     7.0     9.0     5.0     5.5     7.0
      0.1250     9.0     9.0     9.0     9.0     9.0             9.0     9.0     9.0     7.0     9.0     5.0     5.0     5.0
      0.0630     9.0     9.0     9.0     9.0     9.0     9.0             7.0     9.0     6.0             4.3     5.3     6.0
      0.0625     9.0     9.0     9.0     9.0     9.0             9.0     7.0     9.0     4.0     8.0     4.5     3.5     5.0
      0.0315     9.0     9.0     9.0     9.0     9.0     9.0             5.0     9.0     6.3             5.0     7.0     5.7
      0.0313     9.0     9.0     9.0     9.0     9.0             9.0     6.0     9.0     3.0     8.0     3.0     3.5     4.0
      0.0158     9.0     9.0     9.0     9.0     5.0     9.0             4.0     9.0     5.3             3.0     4.0     5.7
      0.0157     9.0     9.0     9.0     9.0     9.0             9.0     4.0     9.0     3.0     6.0     3.0     3.0     3.52        0.5000     9.0     9.0     9.0     9.0                     9.0     9.0     9.0             9.0     9.0     7.0     8.0
      0.2500     9.0     9.0     9.0     9.0     9.0             9.0     9.0     9.0             9.0     9.0     9.0     7.5
      0.1250     9.0     9.0     9.0     9.0     9.0             9.0     9.0     9.0             9.0     8.5     6.5     7.5
      0.0630     9.0     9.0     6.5     9.0     9.0     9.0             9.0     9.0     8.8             7.8     7.2     8.0
      0.0625     9.0     9.0     9.0     9.0     9.0             9.0     9.0     9.0             8.5     8.5     6.5     6.5
      0.0320     9.0     9.0     5.0     9.0     9.0     9.0             9.0     9.0     8.3             6.3     5.3     6.3
      0.0315     9.0     9.0     6.5     9.0     9.0     9.0             9.0     9.0     8.0             7.6     6.6     7.8
      0.0313     7.0     9.0     9.0     9.0                     9.0     9.0     9.0             7.5     8.0     5.5     6.0
      0.0160     9.0     9.0     7.2     9.0     5.8     9.0     9.0     9.0     9.0     7.4             6.0     5.5     6.8
      0.0158     9.0     9.0     6.5     8.0     7.0     9.0             9.0     8.0     7.8             7.2     6.4     7.4
      0.0157     9.0     9.0     4.0     9.0     9.0             9.0     9.0     9.0             6.5     7.0     5.5     6.0
                                                         表1(续)
                                                                                               G                 O        T
                  A        A        C        C        G        I        I        E        S        L        G        R        R   Z
                  B        M        A        H        A        P        P        C        E        X        L        Y        Z   E
                  U        B        S        E        L        O        O        H        T        M        X        S        A   A化合物 施用率     T        E        O        A        A        H        S        C        V        A        M        A        W   M编号 (公斤/公顷) H        L        B        L        P        E        S        G        I        W        A        T        R   X
       0.5000    9.0      9.0      9.0      9.0      9.0               9.0      9.0      9.0               8.0      9.0      9.0  9.03      0.2500    9.0      9.0      9.0      9.0                        9.0      9.0      9.0               7.5      9.0      8.0  9.0
       0.1250    9.0      9.0      9.0      9.0      9.0               9.0      9.0      9.0               7.5      8.5      8.0  8.5
       0.0630    9.0      9.0      9.0      9.0      9.0      9.0               9.0      9.0      7.0               7.2      8.8  8.3
       0.0625    9.0      9.0      9.0      9.0      9.0               9.0      9.0      9.0               6.5      9.0      8.5  8.0
       0.0315    9.0      9.0      6.7      9.0      7.5      9.0               9.0      9.0      6.8               6.8      8.7  8.2
       0.0313    9.0      9.0      4.0      9.0      9.0               9.0      9.0      9.0               4.5      8.5      5.5  6.5
       0.0160    9.0      9.0      3.0      9.0      9.0      9.0               9.0      9.0      5.5               6.3      7.5  7.3
       0.0158    9.0      9.0      5.3      8.3      7.5      9.0               9.0      9.0      5.8               6.0      8.3  7.7
       0.0157    9.0      9.0      2.0      9.0      9.0               9.0      7.0      9.0               4.0      7.0      5.5  6.54      0.5000    9.0      9.0      9.0      9.0      9.0               9.0      9.0      9.0               9.0      4.0      4.0  3.0
       0.2500    9.0      9.0      9.0      9.0      9.0               9.0      8.0      9.0               9.0      3.0      3.0  3.0
       0.1250    9.0      9.0      9.0      9.0      9.0               9.0      8.0      9.0               7.0      3.0      3.0  3.0
       0.0625    9.0      9.0      9.0      9.0      9.0               9.0      7.0      9.0               4.0      2.0      3.0  3.0
       0.0313    9.0      7.0      7.0      9.0      9.0               7.0      5.0      9.0               5.0      2.0      2.0  2.0
       0.0157    9.0      9.0      7.0      9.0      4.0                        2.0      8.0               6.0      2.0      2.0  2.05      0.5000    9.0      9.0      9.0      9.0      8.0               9.0      9.0      9.0               7.0      3.0      3.0  3.0
       0.2500    9.0      9.0      9.0      9.0      9.0               9.0      7.0      9.0               7.0      3.0      2.0  3.0
       0.1250    9.0      9.0      9.0      9.0      9.0               9.0      7.0      9.0               7.0      3.0      2.0  3.0
       0.0625    9.0      9.0      7.0      9.0      9.0               9.0      7.0      9.0               7.0      2.0      2.0  2.0
       0.0313    9.0      9.0      9.0      9.0      9.0               9.0      6.0      9.0               6.0      2.0      2.0  2.0
       0.0157    7.0      9.0      7.0      9.0      7.0               4.0      6.0      8.0               4.0      1.0      2.0  1.0
                                                            表1(续)
                                                                                                       G                  O        T
                    A        A        C         C         G        I        I        E        S        L        G         R        R        Z
                    B        M        A         H         A        P        P        C        E        X        L         Y        Z        E
                    U        B        S         E         L        O        O        H        T        M        X         S        A        A化合物  施用率      T        E        O         A         A        H        S        C        V        A        M         A        W        M编号 (公斤/公顷)   H        L        B         L         P        E        S        G        I        W        A         T        R        X6       0.5000     9.0      9.0      7.0       9.0       9.0               9.0      7.0      9.0               7.0       5.0      6.0      3.0
         0.2500     9.0      9.0      8.0       9.0       9.0               9.0      6.0      9.0      7.0      6.0       5.0      5.0      3.5
         0.1250     9.0      9.0      7.0       9.0       9.0               9.0      7.0      9.0      7.0      6.0       4.5      2.5      3.5
         0.0640     9.0      9.0                9.0       9.0      9.0               3.0      7.0      6.0                1.0      3.0      5.0
         0.0630     9.0      6.5      2.5       7.0       5.0      5.0               1.5      2.0      4.8                1.8      1.5      4.5
         0.0625     9.0      9.0      4.0       9.0       9.0               9.0      2.0      9.0      7.0      4.0       1.5      2.0      3.5
         0.0320     9.0      9.0      2.3       6.5       3.0      9.0      9.0      1.0      6.0      5.5      5.0       1.5      2.5      3.8
         0.0315     9.0      6.0      1.5       5.0       3.0      4.0               1.0      2.5      3.8                1.0      0.8      4.3
         0.0313     9.0      8.0      0.0       9.0       9.0               8.0      2.0      7.0      7.0      4.0       1.5      1.5      3.5
         0.0160     5.7      7.7      0.0       3.0       2.7      6.0      7.5      0.7      3.7      5.5      2.5       1.5      2.0      3.5
         0.0158     5.0      3.0      0.0       0.0       0.0      2.5               0.0      0.0      3.0                0.5      0.0      4.0
         0.0157     8.0      7.0      0.0       9.0       4.0               7.0      2.0      7.0               4.0       2.0      2.0      2.07       0.2500     9.0      9.0      9.0       9.0       8.0               9.0      8.0      9.0      9.0                6.5      7.0      7.0
         0.1250     9.0      9.0      9.0       9.0       7.0               9.0      7.0      9.0      7.5                5.5      5.5      6.0
         0.0625     9.0      9.0      9.0       9.0       5.0               8.0      3.0      9.0      9.0                4.5      5.0      5.5
         0.0313     9.0      9.0      9.0       9.0       5.0               9.0      3.0      9.0      8.5                3.5      5.5      6.0
         0.0157     9.0      9.0      8.0       9.0       3.0               9.0      3.0      9.0      8.0                4.0      5.0      6.0
                                               表1(续)
                                                                              G             O      T
               A      A      C      C      G      I      I      E      S      L      G      R      R      Z
               B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
               U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷) H      L      B      L      P      E      S      G      I      W      A      T      R      X8      0.2500    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0    9.0           8.5    9.0    9.0
     0.1250    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0    9.0           8.5    9.0    9.0
     0.0625    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0    9.0           8.5    9.0    9.0
     0.0320    9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           5.0    9.0    7.0
     0.0313    9.0    9.0    9.0           7.0           9.0    9.0    9.0    9.0           8.5    8.5    8.0
     0.0160    9.0           9.0           5.0    9.0           5.0    5.0    8.5           4.5    7.5    7.0
     0.0157    9.0    9.0    9.0           7.0           9.0    9.0    9.0    8.5           7.5    8.5    8.09      0.2500    9.0    9.0    9.0           8.0           9.0    9.0    9.0    9.0           9.0    9.0    9.0
     0.1250    9.0    9.0    9.0           9.0           9.0    9.0    9.0    9.0           8.5    9.0    9.0
     0.0625    9.0    9.0    9.0    9.0    7.0           7.0    9.0    9.0    9.0           8.5    9.0    9.0
     0.0320    9.0           9.0    9.0    4.0    9.0           9.0    9.0    8.0           7.0    9.0    8.5
     0.0313    9.0    6.0    9.0           6.0           9.0    9.0    9.0    9.0           7.0    8.0    8.5
     0.0160    9.0           9.0           2.0    9.0           9.0    9.0    7.0           6.5    9.0    7.0
     0.0157    9.0    9.0    9.0    9.0    5.0           9.0    9.0    9.0    7.5           6.5    7.5    9.010      0.2500    9.0    9.0    9.0    9.0    7.0           9.0    5.0    9.0    7.5           3.5    5.5    6.0
     0.1250    9.0    9.0    9.0    9.0    8.0           9.0    3.0    9.0    8.0           2.5    5.0    6.0
     0.0625    9.0    9.0    9.0    9.0    4.0           9.0    2.0    9.0    7.5           2.5    5.0    6.0
     0.0313    9.0    9.0    9.0    9.0    3.0           9.0    2.0    9.0    6.0           2.5    3.5    6.0
     0.0157    9.0    8.0    5.0    8.0    2.0           5.0    2.0    8.0    6.0           2.0    3.5    5.5
                                                表1(续)
                                                                               G             O      T
                A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X11      0.2500    9.0    9.0    7.0    9.0    6.0           9.0    7.0    8.0    6.0           2.0    5.0    5.5
      0.1250    9.0    9.0    6.0    6.0    4.0           8.0    7.0    9.0    6.0           2.0    4.0    5.5
      0.0625    8.0    9.0    4.0    9.0    2.0           5.0    4.0    9.0    5.5           1.5    3.0    6.0
      0.0313    9.0    9.0    4.0    8.0    2.0           2.0    4.0    7.0    5.5           1.5    4.0    5.5
      0.0157    7.0    6.0    3.0    5.0    5.0           1.0    2.0    6.0    4.0           1.5    3.0    5.512      0.2500    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0    9.0           9.0    9.0    9.0
      0.1250    9.0    9.0    9.0    9.0    7.0           9.0    9.0    9.0    9.0           8.0    7.5    9.0
      0.0625    9.0    9.0    9.0    9.0    7.0           9.0    9.0    9.0    9.0           7.5    9.0    9.0
      0.0313    9.0    9.0    9.0    9.0    5.0           9.0    9.0    9.0    8.5           7.0    9.0    8.0
      0.0160    9.0    9.0    5.0           3.0    9.0           4.0    7.0    7.5           4.5    6.5    7.0
      0.0157    9.0    9.0    7.0    9.0    4.0           9.0    8.0    8.0    7.5           7.5    8.0    7.513      0.2500    9.0    9.0    9.0    9.0    8.0           9.0    9.0    9.0    8.5           8.0    8.5    9.0
      0.1250    9.0    9.0    9.0    9.0    7.0           9.0    9.0    9.0    8.0           8.0    7.5    9.0
      0.0625    9.0    9.0    7.0    9.0    5.0           8.0    9.0    7.0    7.5           7.5    8.0    9.0
      0.0320    9.0           8.0    9.0    3.0    9.0           7.0    7.0    4.0           3.0    3.5    7.0
      0.0313    9.0    9.0    9.0    9.0    4.0           9.0    9.0    9.0    8.0           6.0    6.0    8.5
      0.0160    9.0    9.0    5.0    9.0    2.0    9.0           5.0    6.0    4.0           3.0    3.0    5.0
      0.0157    9.0    9.0    7.0    9.0    3.0           9.0    9.0    9.0    6.5           5.5    6.0    8.5
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R     Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z     E
                 U      B      S      E      L      O      O      H      T      M      X      S      A     A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W     M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R     X14       0.1250     9.0    9.0    7.0    9.0    6.0    9.0           9.0    9.0    7.0           7.0    7.5   8.5
      0.0640     9.0    9.0    3.0    9.0    6.0    5.0           9.0    9.0    5.0           5.5    5.5   7.5
      0.0625     9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    6.5           3.0    7.5   6.0
      0.0320     9.0    7.0    3.0    6.0    4.0    6.0           8.0    9.0    4.5           3.5    7.0   7.5
      0.0313     9.0    9.0    6.0    9.0    5.0    8.0           9.0    9.0    5.5           3.0    7.5   8.0
      0.0160     9.0           2.0    5.0    3.0    5.0           5.0    5.0    4.0           3.0    5.0   6.0
      0.0156     9.0    9.0    4.0    9.0    4.0    9.0           7.0    9.0    4.5           1.5    4.5   7.015       0.0640     9.0    9.0    4.0    9.0    6.0    9.0           8.0    9.0    7.5           9.0    8.5   7.5
      0.0630     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.5           7.5    8.5   8.5
      0.0320     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    6.5           6.0    8.5   7.5
      0.0315     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.0           7.0    9.0   8.5
      0.0160     9.0    9.0    6.0    9.0    4.0    4.0           9.0    9.0    5.5           4.5    8.0   6.5
      0.0158     9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    6.5           5.0    8.5   8.516       0.0840     8.0    3.0           0.0    3.0    2.0           2.0    4.0    4.0           0.5    0.5   1.5
      0.0320     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.5           0.0    0.0   0.0
      0.0160     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.5           0.0    0.0   0.017       0.0640     9.0    9.0    7.0    9.0    5.0    5.0           3.0    7.0    6.0           4.0    3.5   6.0
      0.0320     9.0    5.0    5.0    5.0    4.0    5.0           2.0    5.0    4.5           2.0    2.5   5.5
      0.0160     9.0    6.0    4.0    7.0    3.0    3.0           2.0    3.0    4.5           2.5    2.5   5.5
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X18      0.0630     9.0    6.0           9.0    5.0    9.0           4.0    5.0    4.0           2.0    2.5    5.0
      0.0315     6.0    9.0    9.0    9.0    4.0    4.0           3.0    7.0    3.5           2.0    2.0    5.5
      0.0158     5.0    9.0    2.0    9.0    0.0    2.0           0.0    0.0    3.5           1.5    1.5    5.019      0.0640     5.0    4.0    2.0    0.0    3.0    2.0           0.0    1.0    5.5           1.0    1.5    5.5
      0.0320     4.0    3.0    0.0    0.0    3.0    2.0           0.0    0.0    5.0           1.0    1.0    5.0
      0.0160     1.0    2.0    0.0    0.0    0.0    0.0           0.0    0.0    4.5           0.0    0.0    4.520      0.0640     5.0    2.0    0.0    0.0    3.0    3.0           2.0    0.0    4.5           1.0    1.0    5.0
      0.0320     4.0    0.0    0.0    0.0    0.0    0.0           0.0    3.0    3.5           0.5    0.5    4.5
      0.0160     1.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.5           0.0    0.0    4.021      0.2500                                                                    7.0           2.0    2.0    5.0
      0.1250                                                                    7.0           2.0    1.0    5.0
      0.0640     9.0    7.0    6.0    9.0    6.0    5.0           0.0    6.0    5.5           1.0    1.0    4.5
      0.0625                                                                    7.0           2.0    1.0    5.0
      0.0320     9.0    5.0    4.0    8.0    4.0    3.0           0.0    1.0    5.5           1.0    1.0    5.0
      0.0313                                                                    6.0           1.0    1.0    5.0
      0.0160     6.0    0.0    0.0    0.0   0.0     2.0           0.0    1.0    4.5           0.5    0.0    3.5
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X22       0.0640     0.0    0.0    0.0    0.0    0.0    1.0           3.0    0.0    5.0           2.0    2.0    5.0
      0.0320     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.5           2.0    2.0    4.5
      0.0160     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.5           1.0    1.0    3.023       0.0640     9.0    9.0    7.0    9.0    9.0    9.0           2.0    8.0    7.5           2.0    3.0    6.0
      0.0320     9.0    9.0    5.0    9.0    9.0    9.0           0.0    4.0    6.5           2.0    2.0    5.5
      0.0160     9.0    6.0    5.0    6.0    4.0    7.0           0.0    6.0    6.5           1.0    1.0    5.524       0.0630     7.0    3.0           0.0    0.0    4.0           0.0    0.0    3.0           0.5    3.0    5.0
      0.0315     4.0    3.0           0.0    0.0    3.0           0.0    0.0    3.0           3.5    2.0    5.0
      0.0158     0.0    0.0    0.0    0.0    0.0    3.0           0.0    0.0    2.0           0.0    0.0    4.025       0.0630     9.0    5.0           9.0    5.0    8.0           2.0    7.0    7.0           3.5    3.5    4.5
      0.0315     9.0    5.0    9.0    9.0    2.0    5.0           2.0    6.0    4.0           2.0    3.5    4.5
      0.0158     7.0    5.0           9.0    2.0    5.0           2.0    9.0    4.0           0.0    3.0    5.026       0.0630     9.0    9.0    6.0    9.0    9.0    9.0           9.0    9.0    7.5           2.0    8.0    7.0
      0.0315     9.0    9.0    5.0    9.0    6.0    9.0           7.0    7.0    7.0           2.5    8.0    7.0
      0.0158     9.0    9.0    5.0    9.0    4.0    9.0           5.0    5.0    7.5           1.0    8.5    7.0
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X27       0.0630     9.0    9.0    4.0    9.0    9.0    9.0           7.0    7.0    7.0           4.5    8.5    7.0
      0.0315     9.0    9.0    3.0    9.0    6.0    9.0           7.0    9.0    7.0           3.0    6.5    7.0
      0.0158     9.0    6.0    2.0    9.0    3.0    6.0           7.0    9.0    6.0           1.5    4.5    7.0
28       0.0630     9.0    9.0    6.0    9.0    9.0    9.0           9.0    9.0    4.0           9.0    9.0    8.0
      0.0315     9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    3.5           4.0    8.0    8.0
      0.0158     9.0    9.0    4.0    9.0    4.0    9.0           8.0    5.0    4.0           1.0    4.5    7.029       0.0630     5.0    4.0    3.0    5.0    2.0    5.0           3.0    6.0    4.5           2.0    3.5    5.5
      0.0315     4.0    3.0    2.0    4.0    2.0    4.0           0.0    9.0    2.5           1.0    1.0    5.0
      0.0158     0.0    0.0    0.0    0.0    0.0    1.0           0.0    9.0    2.5           1.0    1.0    5.030       0.0630     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    7.0           7.5    7.5    9.0
      0.0315     9.0    9.0    8.0    9.0    4.0    9.0           7.0    7.0    6.0           5.5    6.5    9.0
      0.0158     9.0    8.0    9.0    9.0    3.0    9.0           4.0    7.0    5.5           2.5    5.5    9.031       0.0630     9.0    9.0    9.0    9.0    8.0    9.0           4.0    9.0    9.0           3.0    3.0    6.0
      0.0315     9.0    9.0    7.0    9.0    5.0    9.0           1.0    9.0    7.5           2.5    2.5    6.0
      0.0158     9.0    9.0    5.0    9.0    3.0    9.0           1.0    4.0    6.5           1.5    1.5    5.5
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X32       0.0630     9.0    9.0    4.0    9.0    7.0    9.0           2.0    5.0    5.5           1.0    2.0    5.5
      0.0315     9.0    7.0    4.0    9.0    3.0    9.0           2.0    5.0    4.5           1.0    1.0    5.0
      0.0158     9.0    5.0    2.0    9.0    2.0    7.0           0.0    1.0    4.0           0.0    0.0    4.033       0.0630     9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    6.0           7.5    8.5    8.5
      0.0315     9.0    9.0    4.0    9.0    5.0    9.0           9.0    9.0    5.5           4.5    8.5    9.0
      0.0158     9.0    9.0    6.0    9.0    4.0    9.0           5.0           5.0           3.0    7.5    7.034       0.0630     0.0    1.0    0.0    4.0    0.0    0.0           1.0    7.0    3.0           0.0    0.0    4.0
      0.0315     0.0    0.0    0.0    0.0    0.0    0.0           0.0    6.0    3.0           0.0    0.5    3.0
      0.0158     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.0           0.0    0.0    2.535       0.0315     9.0    9.0    5.0    9.0           4.0           2.0    2.0    4.0           1.0    1.5    5.0
      0.0158     9.0    5.0    2.0    9.0    2.0    3.0           1.0    2.0    3.5           0.5    1.0    4.536       0.0630     0.0    0.0    0.0    0.0    0.0    1.0           1.0    9.0    0.0           0.5    0.5    1.5
      0.0315     0.0    0.0    0.0    0.0    0.0    0.0           0.0    9.0    0.0           0.5    0.5    1.0
      0.0158     0.0    0.0    0.0    0.0    0.0    0.0           0.0    9.0    0.0           0.5    0.5    0.5
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X37       0.0630     1.0    0.0    0.0    0.0    0.0    1.0           0.0    0.0    1.5           0.5    0.5    2.0
      0.0315     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.5           0.5    0.5    2.0
      0.158      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.5    0.5    0.038       0.1250     1.0    1.0    1.0    1.0    1.0    2.0           5.0    6.0    2.5           3.0    3.5    5.5
      0.0625     1.0    1.0    1.0    1.0    0.0    1.0           5.0    6.0    2.0           2.5    3.5    4.5
      0.0313     1.0    1.0    1.0    1.0    0.0    1.0           1.0    2.0    2.0           1.5    3.5    4.5
      0.0156     0.0    0.0    1.0    0.0    0.0    1.0           1.0    1.0    2.0           1.5    3.0    4.539       0.1250     8.0    3.0    0.0    1.0    1.0    2.0           3.0    5.0    2.5           1.5    4.0    5.0
      0.0625     4.0    1.0    0.0    1.0    1.0    2.0           2.0    1.0    2.5           1.0    3.5    4.5
      0.0313     1.0    1.0    0.0    0.0    0.0    1.0           1.0    1.0    1.0           1.0    2.5    4.5
      0.0156     1.0    0.0    0.0    0.0    0.0    1.0           1.0    1.0    1.0           1.0    2.0    4.540       0.1250     9.0    9.0    6.0    6.0    5.0    9.0           2.0    8.0    6.0           3.5    5.5    5.0
      0.0625     9.0    9.0    6.0    6.0    1.0    9.0           2.0    7.0    6.0           3.5    5.0    4.5
      0.0313     9.0    4.0    4.0    5.0    1.0    9.0           2.0    7.0    5.0           2.0    4.0    4.5
      0.0156     9.0    3.0    3.0    4.0    0.0    9.0           2.0           5.0           2.0    4.5    4.5
                                                表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X41       0.1250     9.0    1.0    2.0    1.0    1.0    4.0           0.0    0.0    5.5           2.0    4.0    4.5
      0.0625     9.0    1.0    0.0    1.0    1.0    4.0           0.0    0.0    4.5           2.0    3.0    4.0
      0.0313     5.0    1.0    0.0    1.0    1.0    2.0           0.0    0.0    3.0           1.5    2.0    4.0
      0.0156     2.0    0.0    0.0    0.0    0.0    1.0           0.0    0.0    2.5           1.5    2.0    4.042       0.1250     8.0    3.0    3.0    2.0    2.0    6.0           2.0    3.0    4.5           3.0    3.0    4.5
      0.0625     8.0    2.0    3.0    1.0    1.0    4.0           1.0    3.0    4.5           2.5    2.0    4.5
      0.0313     8.0    2.0    0.0    1.0    0.0    3.0           1.0    3.0    4.5           0.5    1.5    4.0
      0.0156     1.0    1.0    0.0    0.0    0.0    3.0           0.0    3.0    3.5           0.5    1.5    3.543       0.1250     9.0    9.0    3.0    5.0    4.0    9.0           3.0    9.0    7.0           3.5    4.0    5.5
      0.0625     9.0    7.0    2.0    4.0    2.0    9.0           3.0    1.0    6.0           2.5    3.5    5.5
      0.0313     9.0    6.0    1.0    3.0    2.0    3.0           3.0           5.5           2.5    3.5    5.0
      0.0156     7.0    4.0    1.0    1.0    1.0    3.0           0.0    1.0    5.0           1.0    1.5    4.544       0.1250     6.0    3.0    2.0    2.0    1.0    4.0           0.0    3.0    5.0           0.5    2.0    4.5
      0.0625     5.0    2.0    0.0    1.0    1.0    4.0           0.0    0.0    4.0           0.5    1.5    4.5
      0.0313     5.0    2.0    0.0    1.0    1.0    4.0           0.0    0.0    4.0           1.0    1.0    4.0
      0.0156     3.0    2.0    0.0    0.0    0.0    1.0           0.0    0.0    3.0           0.5    1.0    4.5
                                                   表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X45       0.1250      9.0    9.0    9.0    7.0    5.0    9.0           7.0    8.0    6.5           4.0    6.0    5.5
      0.0625      9.0    9.0    7.0    7.0    9.0    9.0           7.0    9.0    6.5           4.0    5.5    5.5
      0.0313      9.0    9.0    6.0    7.0    3.0    9.0           5.0    8.0    6.5           4.0    4.5    5.5
      0.0156      9.0    5.0    0.0    7.0    2.0    9.0           5.0    5.0    5.5           3.5    4.5    5.546       0.1250      9.0    9.0    7.0    9.0    4.0    9.0           7.0    7.0    7.0           4.0    5.0    6.0
      0.0625      9.0    9.0    7.0    7.0    4.0    9.0           7.0    7.0    7.0           3.5    5.0    6.0
      0.0313      9.0    9.0    6.0    7.0    3.0    8.0           4.0    5.0    6.0           3.5    5.0    5.5
      0.0156      9.0    8.0    3.0    5.0    1.0    9.0           4.0           6.0           3.0    3.5    5.047       0.1250      9.0    9.0    6.0    6.0    4.0    9.0           5.0    9.0    8.0           8.0    8.5    9.0
      0.0625      9.0    7.0    6.0    4.0    4.0    9.0           7.0    7.0    7.5           9.0    8.0    7.5
      0.0313      9.0    9.0    5.0    4.0    2.0    9.0           7.0    7.0    6.5           7.5    8.0    7.048       0.1250      9.0    9.0    7.0    6.0    6.0    9.0           7.0    9.0    8.0           7.0    8.5    8.5
      0.0625      9.0    9.0    3.0    5.0    6.0    9.0           7.0    9.0    7.5           8.5    8.5    8.5
      0.0313      9.0    9.0    3.0    2.0    2.0    9.0           6.0    9.0    7.5           6.5    7.0    8.0
      0.0156      9.0    6.0    0.0    1.0    1.0    9.0           5.0    6.0    6.0           5.0    8.5    7.049       0.0320      9.0    9.0    5.0    9.0    4.0    9.0           9.0    9.0    7.5           5.5    4.0    6.5
      0.0160      9.0    9.0    3.0    9.0    5.0    9.0           9.0    9.0    6.0           5.0    4.0    6.0
                                                   表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X50       0.0320      9.0    9.0    4.0    9.0    4.0    9.0           9.0    9.0    7.0           4.5    4.5    6.5
      0.0160      9.0    9.0    4.0    9.0    3.0    9.0           9.0    9.0    6.0           2.0    2.0    6.051       0.0640      9.0    9.0    4.0           9.0    9.0           9.0    9.0    7.5           6.0    6.0    7.5
      0.0320      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.5           6.0    6.0    7.0
      0.0160      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    6.5           5.0    4.0    6.052       0.0640      8.0    7.0    6.0    8.0    4.0    2.0           2.0    4.0    4.0           2.0    2.0    5.0
      0.0320      9.0    5.0    5.0    5.0    0.0    2.0           0.0    2.0    4.0           1.5    1.5    4.553       0.0640      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.5           6.5    6.5    7.5
      0.0320      9.0    9.0    4.0    9.0    5.0    9.0           9.0    9.0    6.0           5.5    5.0    6.5
      0.0160      9.0    9.0    9.0    9.0    9.0    9.0           9.0    4.0    6.0           3.0    3.5    5.554       0.0630      9.0    9.0    2.0    9.0    1.0    9.0           9.0    7.0    6.5           1.0    2.0    5.5
      0.0315      9.0           2.0    9.0    0.0    7.0           5.0    9.0    4.0           0.5    3.0    5.0
      0.0158      9.0    3.0    1.0    9.0    0.0    7.0           5.0    6.0    3.5           0.0    1.0    4.555       0.0640      9.0    9.0    7.0    9.0    4.0    7.0           8.0    8.0    5.5           1.5    7.0    7.5
      0.0320      9.0    9.0    9.0    9.0    4.0    5.0           7.0    7.0    5.0           1.5    7.5    7.0
      0.0160      9.0    7.0    5.0    7.0    1.0    4.0           5.0    3.0    4.0           1.5    4.5    5.5
                                                    表1(续)
                                                                                 G              O      T
                  A      A      C      C      G      I      I      E      S      L       G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X       L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M       X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A       M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W       A      T      R      X56       0.1600      9.0    8.0    8.0    7.0    0.0    1.0           0.0    0.0    4.0            1.5    1.5    4.5
      0.0640      9.0    9.0           9.0    6.0    6.0           2.0    4.0    4.5            1.5    2.0    5.5
      0.0320      9.0    9.0           9.0    4.0    1.0           0.0    2.0    3.5            1.5    2.0    4.557       0.0640      9.0    9.0    9.0           9.0    9.0           4.0    7.0    7.5            4.5    5.0    6.5
      0.0320      9.0    9.0    9.0           9.0    9.0           2.0    6.0    5.0            2.5    3.5    5.5
      0.0160      9.0    9.0    9.0    9.0    6.0    5.0           2.0    2.0    4.5            2.5    3.0    5.058       0.0640      9.0           4.0    9.0    6.0    9.0           4.0    5.0    4.5            3.5    4.0    6.5
      0.0320      9.0    9.0    9.0    9.0    3.0    8.0           2.0    5.0    5.0            3.0    3.5    5.5
      0.0160             8.0           9.0    2.0    8.0           2.0    5.0    4.5            2.0    3.0    5.059       0.0640      9.0    7.0    9.0           3.0    6.0           3.0    7.0    5.0            2.5    3.5    5.5
      0.0320      9.0    6.0           9.0    3.0    4.0           2.0    5.0    4.5            2.5    2.5    5.5
      0.0160      9.0    5.0    0.0    5.0    1.0    4.0           2.0    2.0    3.0            1.5    1.5    4.560       0.0640      9.0    7.0           8.0    2.0    4.0           2.0    4.0    6.0            2.0    2.5    6.5
      0.0320      9.0    4.0    5.0    7.0    1.0    3.0           2.0    2.0    5.0            1.5    1.5    6.0
      0.0160      4.0    0.0    0.0    5.0    0.0    0.0           0.0    2.0    4.5            1.0    1.0    5.0
                                                    表1(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X61       0.0640       5.0    9.0           9.0    4.0    4.0           5.0    5.0    4.5           0.5    2.5    5.0
      0.0320       6.0    4.0           4.0    0.0    3.0           3.0    4.0    4.0           0.5    2.0    5.0
      0.0160       6.0    4.0    0.0    4.0    0.0    0.0           2.0    2.0    1.0           0.0    0.0    1.062       0.0630       9.0    9.0    7.0    9.0    6.0    9.0           9.0    9.0    9.0           5.5    5.5    7.0
      0.0315       9.0    9.0    4.0    9.0    7.0    9.0           9.0    9.0    7.0           2.0    4.0    4.0
      0.0158       9.0    9.0    5.0    9.0    6.0    9.0           9.0    7.0    7.0           3.0    3.0    5.563       0.06330      9.0    9.0    3.0    9.0    2.0    5.0           9.0    7.0    5.0           2.0    3.5    4.5
      0.0315       9.0    9.0    3.0    9.0    0.0    5.0           9.0    9.0    5.0           2.0    3.0    4.5
      0.0158       9.0    9.0    2.0    9.0    0.0    3.0           9.0    6.0    4.0           1.0    1.0    4.064       0.0640       9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.0           5.5    5.5    7.0
      0.0320       9.0    9.0    9.0    9.0    9.0    9.0           9.0    8.0    5.5           5.0    5.0    5.5
      0.0160       9.0    9.0           9.0           9.0           8.0    7.0    5.5           4.5    4.5    5.565       0.0630       9.0    9.0    9.0    9.0    4.0    9.0           1.0    9.0    5.5           1.5    3.5    5.5
      0.0315       9.0    9.0    2.0    9.0    2.0    4.0           3.0    3.0    5.5           0.0    3.0    5.5
      0.0158       9.0    5.0    2.0    9.0    1.0    9.0           3.0    9.0    5.0           0.0    2.0    5.5
                                                    表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X66       0.0630      9.0    9.0    9.0    9.0    4.0    9.0           3.0    9.0    6.0           1.0    3.0    6.0
      0.0315      9.0    9.0    7.0    9.0    3.0    9.0           3.0    9.0    6.0           0.5    2.0    5.5
      0.0158      9.0    9.0    5.0    9.0    2.0    4.0           2.0    9.0    5.0           0.5    2.0    5.067       0.0630      9.0    9.0    5.0    9.0    1.0    9.0           6.0    9.0    4.5           1.5    6.5    4.5
      0.0315      9.0    5.0    2.0    5.0    1.0    5.0           5.0    9.0    4.5           1.0    3.5    4.5
      0.0158      9.0    2.0    0.0    0.0    1.0    9.0           2.0    6.0    4.0           0.0    2.5    4.0
      0.0630      6.0    5.0    9.0    9.0    2.0    9.0           5.0    9.0    5.5           2.0    3.5    5.068
      0.0315      9.0    5.0    5.0    9.0    1.0    9.0           4.0    8.0    5.0           2.0    3.0    5.5
      0.0158      9.0    4.0    5.0    5.0    0.0    7.0           1.0    4.0    4.5           0.5    2.0    5.069       0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    8.0    8.5
      0.0315      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.5    8.0
      0.0158      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    7.5           4.5    4.5    7.070       0.0630      9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    8.0           3.0    5.0    6.0
      0.0315      9.0    9.0    5.0    9.0    4.0    9.0           9.0    9.0    8.0           2.0    4.0    8.0
      0.0158      9.0    9.0    2.0    9.0    2.0    9.0           9.0    8.0    7.0           2.0    3.0    6.0
                                                    表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X71       0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    9.0    8.5
      0.0315      9.0    9.0    7.0    9.0    5.0    9.0           9.0    9.0    9.0           6.5    6.5    7.5
      0.0158      9.0    9.0    8.0    9.0    8.0    9.0           9.0    9.0    7.0           5.0    7.0    5.572       0.0630      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    9.0           7.5    7.5    8.0
      0.0315      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    9.0           5.0    5.0    7.0
      0.0158      9.0    9.0    7.0    9.0    5.0    9.0           9.0    9.0    7.0           3.0    4.0    6.073       0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           5.5    4.5    6.0
      0.0315      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.5           3.0    4.5    5.5
      0.0158      9.0    9.0    7.0    9.0    8.0    9.0           9.0    9.0    8.5           2.5    3.0    5.574       0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.5    8.5
      0.3115      9.0    9.0    5.0    9.0    9.0    9.0           9.0    9.0    9.0           6.5    7.5    7.5
      0.0158      9.0    9.0    7.0    9.0    7.0    9.0           9.0    9.0    7.5           2.5    4.5    6.575       0.0630      9.0    9.0    7.0    9.0    7.0    9.0           9.0    9.0    9.0           6.5    9.0    7.5
      0.0315      9.0    9.0    8.0    9.0    8.0    9.0           9.0    9.0    9.0           6.5    6.0    8.0
      0.0158      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           5.5    6.0    6.0
                                                    表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X76       0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    9.0    8.0
      0.0315      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    8.5           5.0    5.5    5.5
      0.0158      9.0    9.0    4.0    9.0    5.0    9.0           9.0    9.0    7.0           2.0    4.0    5.577       0.0830      9.0    9.0    4.0    9.0    9.0    9.0           9.0    9.0    7.0           9.0    9.0    8.0
      0.0315      9.0    9.0    3.0    9.0    7.0    9.0           9.0    9.0    6.5           7.0    8.5    7.0
      0.0158      9.0    9.0    1.0    7.0    7.0    9.0           9.0    9.0    6.5           7.0    7.5    7.078       0.0630      9.0    9.0    3.0    9.0    7.0    9.0           9.0    9.0    6.5           7.0    9.0    7.5
      0.0315      9.0    9.0    2.0    9.0    7.0    9.0           9.0    9.0    6.5           6.5    8.5    7.5
      0.0158      9.0    9.0    2.0    6.0    3.0    9.0           9.0    9.0    6.0           6.5    8.0    7.579       0.0630      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    7.5           7.5    8.5    7.5
      0.0315      9.0    9.0    2.0    9.0    6.0    9.0           9.0    9.0    6.5           6.5    8.0    7.5
      0.0158      9.0    9.0    2.0    4.0    3.0    9.0           9.0    9.0    6.5           5.5    8.0    7.080       0.0630      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    7.5           7.5    8.0    7.5
      0.0315      9.0    9.0    1.0    7.0    9.0    9.0           9.0    9.0    7.5           7.5    8.5    7.5
      0.0158      9.0    9.0    1.0    6.0    7.0    9.0           9.0    9.0    6.5           6.0    7.5    7.0
                                                    表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X81       0.0630      9.0    9.0    3.0    9.0    9.0    9.0           9.0    9.0    7.0           8.0    8.5    8.0
      0.0315      9.0    9.0    2.0    9.0    9.0    9.0           9.0    9.0    6.5           7.5    8.5    7.5
      0.0158      9.0    9.0    1.0    6.0    6.0    9.0           9.0    8.0    6.0           6.0    8.5    6.582       0.0630      9.0    6.0    1.0    9.0    4.0    9.0           7.0    9.0    5.5           5.5    6.0    5.5
      0.31315     9.0    9.0    0.0    7.0    2.0    9.0           7.0    9.0    5.0           3.5    5.0    5.5
      0.0158      9.0    2.0    0.0    4.0    1.0    9.0           5.0    9.0    4.0           2.0    3.5    4.083       0.0630      9.0    9.0    3.0    9.0    7.0    9.0           9.0    9.0    8.0           7.5    6.5    6.0
      0.0315      9.0    9.0    1.0    9.0    7.0    9.0           9.0    9.0    7.0           6.5    6.0    6.0
      0.0158      9.0    9.0    1.0    8.0    7.0    9.0           9.0    9.0    7.0           5.0    5.0    6.084       0.0630      9.0    9.0    4.0    9.0    9.0    9.0           9.0    9.0    8.0           8.0    8.0    7.5
      0.0315      9.0    9.0    3.0    9.0    7.0    9.0           9.0    9.0    7.5           7.0    7.0    6.5
      0.0158      9.0    9.0    1.0    9.0    6.0    9.0           9.0    9.0    7.0           6.5    6.5    6.085       0.0630      5.0    2.0    2.0    5.0    5.0    9.0           7.0    8.0    7.0           5.0    5.5    6.5
      0.0315      3.0    1.0    1.0    4.0    4.0    5.0           3.0    7.0    5.0           4.0    5.5    6.0
      0.0158      1.0    1.0    1.0    1.0    1.0    5.0           1.0    3.0    5.0           3.5    4.0    5.5
                                                   表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X86        0.0630     9.0    9.0    7.0    9.0    7.0    9.0           9.0    9.0    7.5           7.0    6.5    6.0
       0.0315     9.0    9.0    1.0    8.0    8.0    9.0           7.0    7.0    7.0           6.5    6.5    6.0
       0.0158     9.0    9.0    1.0    5.0    6.0    9.0           7.0    7.0    6.5           4.5    5.0    5.587        0.0630     9.0    9.0    6.0    9.0    9.0    9.0           9.0    9.0    7.5           7.5    7.0    7.0
       0.0315     9.0    9.0    2.0    7.0    7.0    9.0           9.0    7.0    6.5           5.5    6.0    6.0
       0.0158     9.0    9.0    1.0    6.0    5.0    9.0           6.0    3.0    6.5           5.5    5.5    5.588        0.0630     9.0    9.0    4.0    9.0    7.0    9.0           9.0    9.0    8.5           6.5    6.5    7.5
       0.0315     9.0    9.0    4.0    9.0    7.0    9.0           9.0    9.0    8.0           6.5    6.5    7.5
       0.0158     9.0    9.0    2.0    8.0    7.0    9.0           9.0    8.0    7.5           6.0    5.5    6.089        0.0630     9.0    9.0    3.0    8.0    7.0    9.0           9.0    9.0    7.5           7.5    7.5    6.5
       0.0315     9.0    9.0    3.0    7.0    7.0    9.0           9.0    9.0    7.0           6.5    6.5    6.5
       0.0158     9.0    9.0    2.0    6.0    5.0    9.0           9.0    9.0    6.5           4.0    5.0    5.5
90        0.0630     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.5           8.0    7.5    7.5
       0.0315     9.0    9.0    3.0    7.0    7.0    9.0           9.0    9.0    7.5           7.0    7.0    7.5
       0.0158     9.0    7.0    1.0    7.0    5.0    9.0           9.0    9.0    7.0           5.5    6.0    6.5
                                                表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X91       0.0630     9.0    4.0    1.0    5.0    0.0    5.0           6.0    9.0    3.5           3.5    4.5    5.0
      0.0315     3.0    1.0    4.0    0.0    4.0    2.0           6.0    3.5    2.0           4.0    5.0
      0.0158     7.0    1.0    1.0    3.0    0.0    2.0           1.0    3.0    2.0           2.0    3.5    4.592       0.0630     9.0    9.0    3.0    8.0    7.0    9.0           9.0    9.0    7.5           8.0    9.0    8.0
      0.0315     9.0    9.0    3.0    7.0    3.0    9.0           9.0    9.0    7.5           7.5    9.0    7.5
      0.0158     9.0    9.0    1.0    5.0    1.0    9.0           9.0    9.0    7.0           6.5    8.5    7.093       0.0630     9.0    9.0    3.0    7.0    5.0    9.0           9.0    9.0    7.5           6.5    8.0    7.5
      0.0315     9.0    9.0    3.0    7.0    3.0    9.0           9.0    9.0    6.5           5.5    8.0    7.5
      0.0158     9.0    9.0    1.0    6.0    1.0    9.0           9.0    9.0    6.0           5.5    8.0    7.594       0.0630     0.0    0.0    0.0    0.0    0.0    1.0           1.0    1.0    3.0           2.5    3.0    4.5
      0.0315     0.0    0.0    0.0    0.0    0.0    0.0           0.0    1.0    3.0           1.5    1.5    4.0
      0.0158     0.0    0.0    0.0    0.0    0.0    0.0           0.0    1.0    1.5           1.5    1.5    3.095       0.0630     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    1.5
      0.0315     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0158     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X96       0.0630      9.0    9.0    0.0    6.0    1.0    9.0           8.0    9.0    6.5           5.5    7.0    7.5
      0.0315      9.0    5.0    0.0    4.0    0.0    9.0           7.0    6.0    6.5           4.0    6.0    7.5
      0.0158      5.0    4.0    0.0    2.0    0.0    9.0           7.0    2.0    4.5           2.0    4.5    6.097       0.0830      9.0    9.0    0.0    9.0    6.0    9.0           9.0    9.0    7.5           7.5    9.0    8.0
      0.0315      9.0    9.0    0.0    4.0    2.0    9.0           8.0    9.0    7.5           7.5    8.0    8.0
      0.0158      9.0    3.0    0.0    4.0    2.0    9.0           6.0    9.0    6.0           6.0    8.0    7.598       0.1250      9.0    9.0    4.0    6.0    7.0    9.0           0.0    2.0    8.5           2.0    5.0    5.5
      0.0630      9.0    9.0    3.0    7.0    7.0    9.0           0.0    8.0    8.5           4.5    5.5    6.0
      0.0625      9.0    9.0    4.0    4.0    4.0    9.0           0.0    0.0    8.0           2.0    3.5    5.0
      0.0315      9.0    9.0    0.0    7.0    7.0    9.0           0.0    3.0    7.5           3.5    5.0    6.0
      0.0313      9.0    7.0    4.0    4.0    4.0    9.0           0.0    0.0    6.0           1.5    2.5    4.5
      0.0158      9.0    9.0    0.0    5.0    4.0    6.0           0.0    3.0    5.5           2.5    4.5    5.0
      0.0156      9.0    4.0    0.0    2.0    3.0    9.0           0.0    0.0    6.0           1.0    2.5    4.599       0.0630      9.0    4.0    3.0    7.0    1.0    9.0           7.0    7.0    7.5           6.0    6.0    7.5
      0.0315      9.0    2.0    1.0    5.0    1.0    7.0           4.0    4.0    5.5           4.5    4.5    7.0
      0.0158      9.0    2.0    0.0    3.0    0.0    6.0           2.0    8.0    5.5           4.0    4.0    6.5
                                                表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X100      0.1250                                                                    9.0           4.0    4.0    6.0
      0.0630     9.0    9.0    0.0    8.0    8.0    9.0           3.0    2.0    7.5           2.5    2.0    6.5
      0.0625                                                                    8.0           3.0    3.0    6.0
      0.0315     9.0    9.0    0.0    6.0    5.0    9.0           0.0    0.0    7.0           2.5    2.0    6.0
      0.0313                                                                    7.0           2.0    3.0    5.0
      0.0158     9.0    9.0    0.0    5.0    4.0    9.0           0.0    0.0    6.0           1.0    1.5    5.5
      0.0156                                                                    7.0           2.0    3.0    5.0101      0.0630     9.0    3.0    0.0    2.0    1.0    5.0           0.0    0.0    4.0           1.0    2.0    4.5
      0.0315     4.0    1.0    0.0    2.0    0.0    4.0           0.0    0.0    3.0           1.0    1.5    3.5
      0.0158     3.0    1.0    0.0    0.0    0.0    4.0           0.0    0.0    1.5           0.5    1.0    3.5102      0.0630     9.0    7.0    0.0    4.0    2.0    9.0           1.0    3.0    8.0           3.5    4.0    6.0
      0.0315     7.0    7.0    0.0    3.0    2.0    9.0           0.0    0.0    8.0           2.5    3.0    6.0
      0.0158     7.0    5.0    0.0    3.0    2.0    9.0           0.0    0.0    7.0           2.0    2.5    5.5103      0.0630     9.0    9.0    5.0    9.0    6.5    9.0           9.0    9.0    7.3           8.0    8.8    7.8
      0.0315     9.0    9.0    2.0    7.5    4.5    9.0           9.0    9.0    7.3           6.8    7.0    7.8
      0.0158     9.0    9.0    0.5    8.0    2.0    9.0           9.0    9.0    7.0           5.8    6.8    7.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X104      0.0630      9.0    9.0    1.5    5.0    7.5    9.0           6.0    8.5    7.3           6.5    5.8    7.3
      0.0315      9.0    9.0    1.0    3.5    5.5    9.0           3.5    9.0    6.0           6.0    5.5    7.3
      0.0158      9.0    6.0    0.0    3.5    5.0    9.0           1.0    5.5    5.8           4.3    5.5    7.0105      0.1250                                                                     8.0           6.0    6.0    7.0
      0.0630      9.0    9.0    8.5    7.5    7.0    9.0           6.5    9.0    8.5           5.0    5.0    6.5
      0.0625                                                                     8.0           5.0    6.0    7.0
      0.0315      9.0    9.0    8.0    7.0    5.5    9.0           4.5    6.5    7.8           3.8    4.0    5.8
      0.0313                                                                     7.0           5.0    5.0    6.0
      0.0158      9.0    9.0    6.0    6.0    5.0    9.0           2.0    6.0    7.5           3.3    3.3    5.8
      0.0156                                                                     7.0           4.0    4.0    6.0106      0.0630      4.0    2.0    0.0    0.0    1.0    4.0           0.0    0.0    3.5           1.5    2.5    5.0
      0.0315      4.0    0.0    0.0    0.0    1.0    2.0           0.0    0.0    3.0           1.0    1.5    5.0
      0.0158      1.0    0.0    0.0    0.0    0.0    1.0           0.0    0.0    2.5           0.5    1.0    4.5107      0.0630      9.0    6.0    2.0    4.0    1.0    9.0           0.0    5.0    5.5           3.0    4.5    4.0
      0.0315      9.0    4.0    1.0    4.0    1.0    9.0           0.0    3.0    5.5           2.5    3.5    3.5
      0.0158      5.0    1.0    0.0    2.0    1.0    0.0           0.0    0.0    4.0           2.5    2.0    3.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R     Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z     E
                  U      B      S      E      L      O      O      H      T      M      X      S      A     A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W     M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R     X108      0.0630      5.0    5.0    1.0    5.0    2.0    6.0           0.0    0.0    4.5           2.5    3.5   4.0
      0.0315      5.0    4.0    1.0    4.0    1.0    3.0           0.0    0.0    3.5           2.0    2.0   3.0
      0.0158      3.0    0.0    0.0    0.0    0.0    4.0           0.0    0.0    4.0           2.0    2.0   4.0109      0.0630      9.0    5.0    4.0    4.0    5.0    9.0           1.0    4.0    5.0           2.5    4.5   4.0
      0.0315      9.0    6.0    3.0    4.0    2.0    9.0           2.0    2.0    6.0           2.5    3.5   4.0
      0.0158      9.0    4.0    0.0    1.0    1.0    9.0           0.0    0.0    4.0           2.5    3.0   4.5110      0.1250      9.0    9.0    5.0    5.0    6.0    9.0           2.0    9.0    8.5           4.0    4.0   6.0
      0.0630      9.0    9.0    2.0    5.0    2.0    9.0           1.0    5.0    7.0           3.0    3.0   5.0
      0.0625      9.0    7.0    2.0    2.0    1.0    9.0           0.0    3.0    6.0           2.0    2.5   5.0
      0.0315      9.0    9.0    2.0    4.0    1.0    9.0           0.0    5.0    5.5           2.5    2.5   5.0
      0.0313      9.0    2.0    0.0    2.0    0.0    9.0           0.0    0.0    5.0           1.5    2.5   5.0
      0.0158      9.0    2.0    0.0    2.0    0.0    4.0           0.0    0.0    5.5           2.5    2.5   4.0
      0.0156      9.0    1.0    0.0    1.0    0.0    9.0           0.0    0.0    4.0           1.0    1.5   4.5111      0.0630      9.0    6.0    1.0    2.0    0.0    9.0           0.0    0.0    5.0           3.0    3.0   5.0
      0.0315      9.0    4.0    1.0    1.0    0.0    9.0           0.0    0.0    4.5           2.0    2.0   4.0
      0.0158      4.0    2.0    0.0    1.0    0.0    2.0           0.0    0.0    3.5           2.0    2.0   3.5
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X112      0.0630      9.0    3.0    1.0    3.0    2.0    9.0           2.0    5.0    7.0           3.0    2.5    7.0
      0.0315      8.0    3.0    1.0    1.0    2.0    8.0           2.0    2.0    5.5           2.5    2.5    7.0
      0.0158      6.0    0.0    0.0    1.0    1.0    4.0           0.0    2.0    4.0           2.5    2.5    6.0113      0.0630      9.0    9.0    4.0    5.0    6.0    9.0           4.0    6.0    6.0           5.0    5.0    7.0
      0.0315      9.0    7.0    2.0    5.0    2.0    9.0           1.0    4.0    4.5           3.5    3.5    6.0
      0.0158      9.0    9.0    0.0    2.0    1.0    9.0           0.0    0.0    4.0           3.5    3.5    5.0114      0.0630      9.0    9.0    4.5    5.0    6.5    9.0           2.0    5.0    6.8           3.8    4.5    5.8
      0.0315      9.0    8.0    1.5    2.5    3.5    9.0           0.5    6.5    5.5           2.8    3.3    5.5
      0.0158      8.0    7.5    1.0    3.0    1.5    9.0           0.0    0.5    5.8           2.5    3.0    5.0115      0.1250      7.0    3.0    0.0    2.0    1.0    9.0           5.0    8.0    5.5           3.0    4.5    7.5
      0.0625      7.0    3.0    0.0    2.0    1.0    9.0           5.0    8.0    5.5           2.5    3.5    7.5
      0.0313      7.0    2.0    0.0    1.0    0.0    7.0           4.0    3.0    5.0           1.5    3.0    7.0
      0.0156      7.0    1.0    0.0    0.0    0.0    9.0           4.0    0.0    4.0           1.5    2.5    6.5116      0.1250      0.0    0.0    0.0    0.0    0.0    1.0           0.0    0.0    1.5           0.0    0.0    1.5
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.5           0.0    0.0    0.5
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                     表1(续)
                                                                                          G               O       T
                  A       A       C       C       G       I       I       E       S       L       G       R       R       Z
                  B       M       A       H       A       P       P       C       E       X       L       Y       Z       E
                  U       B       S       E       L       O       O       H       T       M       X       S       A       A化合物    施用率      T       E       O       A       A       H       S       C       V       A       M       A       W       M编号   (公斤/公顷)   H       L       B       L       P       E       S       G       I       W       A       T       R       X117      0.1250      0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     1.0             0.0     0.0     1.0
      0.0625      0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.0             0.0     0.0     0.0
      0.0313      0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.0             0.0     0.0     0.0
      0.0156      0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.0             0.0     0.0     0.0118      0.1250      1.0     0.0     0.0     0.0     0.0     1.0             0.0     0.0     1.0             0.5     0.5     2.0
      0.0625      0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     1.0             0.0     0.0     1.0
      0.0313      0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.5             0.0     0.0     0.0
      0.0156      0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.0             0.0     0.0     0.0119      0.1250      9.0     9.0     5.0     8.0     9.0     9.0             5.0     8.0     8.0             4.5     4.0     6.0
      0.0630      9.0     9.0     2.0     9.0     9.0     9.0             1.0     9.0     6.5             2.5     3.0     6.0
      0.0625      9.0     9.0     2.0     6.0     8.0     9.0             2.0     7.0     7.5             3.0     4.0     6.0
      0.0315      9.0     9.0     2.0     9.0     7.0     9.0             0.0     0.0     6.0             1.5     2.5     4.5
      0.0313      9.0     8.0     1.0     3.0     5.0     9.0.            0.0     2.0     7.5             2.0     3.5     6.0
      0.0158      9.0     7.0     1.0     9.0     4.0     9.0             0.0     0.0     4.0             0.5     1.5     4.5
      0.0156      9.0     7.0     0.0     3.0     2.0     9.0             0.0     0.0     6.5             1.5     3.0     5.0120      0.0630      9.0     9.0     9.0     6.0     5.0     9.0             9.0     8.0     7.5             5.0     5.0     6.5
      0.0315      9.0     9.0     9.0     5.0     4.0     9.0             6.0     4.0     7.5             3.5     4.5     6.5
      0.0158      9.0     9.0     9.0     5.0     4.0     9.0             6.0     3.0     6.0             2.5     4.5     5.0
                                                表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X121      0.0630     9.0    9.0    7.0    6.0    6.0    9.0           7.0    9.0    9.0           6.5    6.5    8.0
      0.0315     9.0    9.0    6.0    5.0    6.0    9.0           7.0    9.0    8.5           6.0    6.5    7.5
      0.0158     9.0    9.0    5.0    6.0    4.0    9.0           7.0    9.0    6.5           4.0    5.0    8.0122      0.0630     9.0    9.0    6.0    8.0    6.0    9.0           6.5    9.0    6.5           3.5    4.8    7.0
      0.0315     9.0    9.0    5.0    7.0    5.0    9.0           6.5    8.0    6.5           3.3    4.5    6.3
      0.0158     9.0    9.0    4.5    6.0    2.0    9.0           5.5    8.5    5.3           3.3    4.5    5.5123      0.0830     9.0    9.0    5.0    8.0    2.0    9.0           4.0    7.5    6.3           3.0    4.3    5.5
      0.0315     9.0    9.0    4.5    6.5    0.5    9.0           2.0    2.0    5.8           2.3    3.8    5.3
      0.0158     9.0    8.0    3.5    6.5    0.5    9.0           0.0    0.5    5.5           1.5    3.8    5.0124      0.0630     9.0    9.0    5.5    7.0    5.0    9.0           6.5    7.5    7.0           2.8    4.8    6.5
      0.0315     9.0    9.0    4.5    6.5    2.5    9.0           3.5    6.5    5.8           2.0    4.3    5.8
      0.0158     9.0    6.5    2.0    5.5    0.5    7.0           1.5    5.0    5.3           2.0    3.5    5.8125      0.1250     9.0    9.0    7.0    7.0    3.0    9.0           9.0    9.0    7.5           7.5    9.0    9.0
      0.0625     9.0    9.0    2.0    4.0    1.0    9.0           9.0    9.0    7.5           7.5    8.5    7.5
      0.0313     9.0    8.0    2.0    2.0    0.0    9.0           9.0    9.0    7.0           3.0    7.5    8.0
      0.0156     9.0    3.0    2.0    1.0    0.0    8.0           9.0    9.0    7.0           3.0    7.5    7.5
                                             表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X126      0.0630      9.0    6.0    5.0    4.0    6.0    9.0           1.0    4.0    6.5           2.5    4.0    7.0
      0.0315      7.0    4.0    5.0    4.0    4.0    9.0           0.0    1.0    5.5           2.5    3.5    6.0
      0.0158      7.0    1.0    3.0    0.0    0.0    9.0           0.0    1.0    5.5           2.5    3.0    5.5127      0.0830      9.0    5.0    6.0    3.0    6.0    9.0           1.0    9.0    7.0           4.5    7.0    7.5
      0.0315      9.0    4.0    5.0    1.0    6.0    9.0           1.0    1.0    7.0           2.5    5.5    7.0
      0.0158      9.0    1.0    4.0    1.0    6.0    9.0           1.0    2.0    5.5           2.5    4.5    5.5128      0.0630      9.0    6.0    3.0    5.0    4.0    8.0           1.5    3.0    5.3           2.5    3.8    4.0
      0.0315      8.0    4.5    1.0    1.0    2.5    5.5           0.5    1.5    4.5           1.5    1.8    2.8
      0.0158      8.5    4.0    1.0    1.5    1.5    3.0           0.5    1.5    4.3           1.3    1.3    1.8129      0.0630      9.0    6.0    2.0    7.0    4.0    9.0           2.0    3.0    7.0           3.0    5.5    6.0
      0.0315      9.0    4.0    2.0    4.0    2.0    9.0           1.0    1.0    6.5           3.5    4.5    5.5
      0.0158      9.0    2.0    3.0    4.0    2.0    9.0           1.0    1.0    6.0           2.5    2.5    5.0130      0.0630      9.0    6.0    2.0    7.0    5.0    9.0           2.0    4.0    7.5           3.0    4.5    6.0
      0.0315      9.0    5.0    2.0    6.0    3.0    9.0           4.0    6.0    8.0           3.0    4.5    5.5
      0.0158      9.0    2.0    2.0    3.0    1.0    8.0           1.0    1.0    7.0           2.5    4.5    5.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X131      0.0630      9.0    6.0    3.0    6.0    6.0    9.0           2.0    4.0    7.0           2.5    4.5    6.0
      0.0315      9.0    4.0    2.0    3.0    4.0    9.0           2.0    1.0    5.0           2.5    3.0    4.0
      0.0158      9.0    4.0    1.0    2.0    3.0    9.0           2.0    1.0    4.5           2.5    3.0    3.5
132      0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    7.0    8.0
      0.0315      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    6.0    8.0
      0.0158      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           6.5    6.5    8.0133      0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    9.0    8.0
      0.0315      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    8.5    7.5
      0.0158      9.0    9.0    8.0    9.0    8.0    9.0           9.0    9.0    7.5           7.5    8.5    7.5134      0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    7.0    7.5
      0.0315      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    7.0    8.0
      0.0158      9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    7.5           7.5    7.0    7.0135      0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.5           7.5    9.0    8.5
      0.0315      9.0    9.0    7.0    9.0    8.0    9.0           9.0    9.0    7.5           7.5    9.0    8.5
      0.0158      9.0    9.0    6.0    9.0    6.0    9.0           9.0    6.0    8.0           7.0    8.5    8.5
                                                 表1(续)
                                                                                  G             O      T
                  A      A       C      C      G      I      I      E      S      L      G      R      R       Z
                  B      M       A      H      A      P      P      C      E      X      L      Y      Z       E
                  U      B       S      E      L      O      O      H      T      M      X      S      A       A化合物    施用率      T      E       O      A      A      H      S      C      V      A      M      A      W       M编号   (公斤/公顷)   H      L       B      L      P      E      S      G      I      W      A      T      R       X136      0.0630      9.0    6.0     0.0    3.0    1.0    9.0           0.0    6.0    3.0           2.5    2.0     4.5
      0.0315      9.0    2.0     1.0    3.0    1.0    9.0           0.0    4.0    3.5           2.0    3.5     5.0
      0.0158      7.0    1.0     0.0    0.0    1.0    4.0           0.0    0.0    3.5           1.5    2.5     5.5137      0.0630      9.0    9.0     5.0    7.0    7.0    9.0           3.0    7.0    6.5           4.5    4.5     6.0
      0.0315      9.0    9.0     2.0    5.0    6.0    9.0           2.0    4.0    6.0           4.0    4.5     6.0
      0.0158      9.0    8.0     1.0    3.0    3.0    9.0           0.0    0.0    6.0           2.5    4.0     5.5138      0.0630      9.0    9.0     8.0    7.0    7.0    9.0           7.5    9.0    9.0           6.3    5.8     8.3
      0.0315      9.0    9.0     5.0    5.0    7.0    9.0           4.5    9.0    8.0           5.5    5.3     8.0
      0.0158      9.0    6.5     1.5    1.0    2.5    9.0           4.5    9.0    6.8           4.8    4.8     7.5139      0.2500                                                                      7.0           3.0    4.0     6.0
      0.1250                                                                      7.0           3.0    3.0     6.0
      0.0630      9.0    7.0     1.0    5.0    3.0    9.0           0.0    2.0    5.5           3.5    4.0     6.5
      0.0625                                                                      7.0           3.0    3.0     6.0
      0.0315      9.0    9.0     1.0    4.0    5.0    7.0           0.0    0.0    6.0           2.5    3.0     5.5
      0.0313                                                                      7.0           3.0    3.0     6.0
      0.0158      9.0    6.0     0.0    1.0    2.0    6.0           0.0    0.0    5.5           2.5    3.0     5.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X140      0.0630      9.0    9.0    2.0    8.0    7.0    9.0           2.0    4.0    7.5           4.0    5.0    6.5
      0.0315      8.0    8.0    2.0    6.0    7.0    9.0           1.0    4.0    6.0           3.0    3.0    5.5
      0.0158      9.0    7.0    0.0    4.0    3.0    9.0           0.0    2.0    5.5           2.5    2.5    5.5141      0.1250                                                                     8.0           3.0    3.0    7.0
      0.0630      9.0    7.0    1.0    7.5    8.0    9.0           0.5    0.5    7.0           2.5    3.0    6.0
      0.0625                                                                     7.0           1.0    3.0    7.0
      0.0315      9.0    7.0    1.0    8.5    5.0    9.0           0.0    0.0    5.5           2.0    3.0    5.5
      0.0313                                                                     7.0           1.0    3.0    6.0
      0.0158      9.0    6.5    0.5    7.0    3.0    8.0           0.0    0.0    5.5           1.8    2.3    5.3
      0.0156                                                                     6.0           1.0    2.0    5.0142      0.0630      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           7.5    8.5    8.5
      0.0315      9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    9.0           7.0    9.0    8.0
      0.0158      9.0    9.0    9.0    9.0    7.0    9.0           8.0    9.0    9.0           6.5    8.0    7.0
                                              表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X143      0.2500                                                                     8.0           5.0    5.0    5.0
      0.1250                                                                     8.0           4.0    5.0    6.0
      0.0630      9.0    6.0    0.0    7.0    7.0    9.0           0.0    0.0    6.0           1.5    3.0    4.0
      0.0625                                                                     7.0           4.0    5.0    5.0
      0.0315      9.0    6.0    0.0    6.0    4.0    9.0           0.0    0.0    6.0           1.5    3.0    4.0
      0.0313                                                                     7.0           4.0    4.0    5.0
      0.0158      8.0    2.0    0.0    2.0    2.0    2.0           0.0    0.0    5.0           1.5    2.5    3.5
      0.0156                                                                     7.0           4.0    3.0    5.0144      0.0630      9.0    9.0    1.0    5.0    9.0    9.0           7.0    8.0    7.5           8.0    8.5    8.5
      0.0315      9.0    9.0    1.0    7.0    9.0    5.0           7.0    7.0    6.5           5.5    7.0    7.5
      0.0158      9.0    9.0    1.0    2.0    5.0    3.0           4.0    7.0    6.5           2.0    6.5    7.5145      0.2500                                                                     7.0           5.0    6.0    7.0
      0.1250      9.0    6.0    4.0    6.0    3.0    7.0           2.0    3.0    6.0           4.3    4.7    6.0
      0.0625      9.0    3.0    3.0    3.0    2.0    9.0           2.0    2.0    5.3           3.7    4.0    5.7
      0.0313      4.0    3.0    1.0    3.0    1.0    9.0           0.0    1.0    5.0           3.3    3.3    5.3
      0.0156      3.0    1.0    1.0    4.0    1.0    1.0           1.0    2.0    5.0           2.7    3.0    5.3
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X146      0.2500                                                                     8.0           7.0    7.0    8.0
      0.1250      9.0    9.0    1.0    9.0    6.0    9.0           9.0    9.0    6.0           6.3    6.3    7.7
      0.0625      9.0    9.0    2.0    9.0    4.0    9.0           9.0    9.0    6.3           5.7    5.3    7.3
      0.0313      9.0    7.0    2.0    9.0    2.0    9.0           4.0    9.0    6.0           5.0    5.3    7.3
      0.0156      9.0    4.0    1.0    6.0    2.0    9.0           2.0    7.0    5.3           3.7    4.0    6.7147      0.2500                                                                     8.0           6.0    6.0    7.0
      0.1250      9.0    4.0    2.0    4.0    4.0    9.0           3.0    7.0    6.0           3.7    4.3    6.3
      0.0625      9.0    2.0    1.0    4.0    1.0    9.0           2.0    9.0    5.3           3.0    3.7    4.7
      0.0313      5.0    2.0    1.0    4.0    1.0    3.0           0.0    2.0    5.3           2.7    3.0    3.7
      0.0156      3.0    1.0    1.0    4.0    1.0    1.0           0.0    1.0    4.7           2.0    2.7    3.0148      0.1250      9.0    9.0    4.0    9.0    7.0    9.0           2.0    9.0    6.5           6.0    6.0    7.5
      0.0625      9.0    9.0    3.0    9.0    6.0    9.0           2.0    2.0    6.5           5.5    5.0    7.0
      0.0313      9.0    7.0    1.0    3.0    4.0    9.0           1.0    2.0    6.0           4.0    4.5    6.5
      0.0156      9.0    4.0    1.0    5.0    2.0    9.0           1.0    5.0    5.5           3.5    4.0    6.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X149      0.1250      9.0    1.0    1.0    2.0    2.0    9.0           1.0    1.0    5.0           4.5    4.5    5.5
      0.0630                                                                     7.0           4.0    5.0    6.0
      0.0625      9.0    1.0    1.0    1.0    2.0    9.0           0.0    0.0    4.0           3.5    4.0    4.5
      0.0315                                                                     6.0           4.0    4.0    6.0
      0.0313      9.0    2.0    1.0    1.0    2.0    9.0           0.0    0.0    4.0           3.0    3.5    5.0
      0.0158                                                                     6.0           4.0    4.0    5.0
      0.0156      7.0    1.0    0.0    0.0    1.0    4.0           0.0    0.0    3.5           2.0    3.0    5.0150      0.1250      9.0    9.0    3.0    9.0    9.0    9.0           9.0    9.0    8.0           7.3    6.7    7.7
      0.0625      9.0    9.0    2.0    7.0    7.0    9.0           4.0    5.0    7.0           6.3    6.3    7.3
      0.0313      9.0    6.0    2.0    7.0    4.0    9.0           2.0    6.0    6.3           4.3    5.0    7.0
      0.0156      9.0    7.0    1.0    3.0    2.0    5.0           0.0    0.0    6.3           4.7    4.7    6.7151      0.5000      1.0    0.0    0.0    1.0    1.0    0.0           0.0    0.0    1.5           1.0    1.0    2.0
      0.2500      1.0    0.0    0.0    1.0    1.0    0.0           0.0    0.0    1.5           0.0    1.0    1.0
      0.1250      1.0    0.0    0.0    1.0    0.0    0.0           0.0    0.0    1.5           0.0    1.0    1.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.5           0.0    0.0    1.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.5           0.0    0.0    0.0152      0.0630      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.5           1.5    2.0    2.5
      0.0315      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.5           0.5    1.0    2.0
      0.0158      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.5           0.0    1.0    1.0
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X153      0.0630      9.0    9.0    3.0    7.0    9.0    9.0           8.0    7.0    8.5           6.0    6.0    8.0
      0.0315      9.0    4.0    0.0    2.0    3.0    9.0           3.0    9.0    7.5           6.0    6.0    8.0
      0.0158      9.0    3.0    0.0    1.0    3.0    4.0           2.0    9.0    6.5           5.5    6.0    7.5154      0.0630      9.0    9.0    0.0    7.0    9.0    9.0           0.0    0.0    6.0           1.5    2.5    5.5
      0.0315      9.0    7.0    0.0    4.0    5.0    9.0           0.0    0.0    5.5           1.0    1.5    4.5
      0.0158      9.0    2.0    0.0    2.0    3.0    9.0           0.0    0.0    5.5           1.0    1.5    4.0155      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           0.0    8.0    9.0           2.0    5.5    6.5
      0.1250      9.0    9.0    3.0    9.0    7.0    9.0           0.0    4.0    8.0           2.0    4.5    5.0
      0.0625      9.0    9.0    0.0    9.0    5.0    9.0           0.0    4.0    7.0           2.0    4.0    5.0
      0.0313      9.0    9.0    0.0    9.0    0.0    9.0           0.0    3.0    6.5           1.5    4.0    4.5
      0.0156      9.0    4.0    0.0    3.0    0.0    9.0           0.0    3.0    5.5           1.0    4.0    4.5156      0.1250      9.0    5.0    2.0    9.0    3.0    4.0           1.0    1.0    4.5           2.5    3.0    3.5
      0.0625      4.0    3.0    1.0    1.0    2.0    1.0           1.0    0.0    4.0           2.5    2.0    3.5
      0.0313      3.0    1.0    1.0    1.0    1.0    1.0           0.0    0.0    3.0           1.5    1.5    1.5
      0.0156      1.0    1.0    0.0    2.0    1.0    0.0           0.0    0.0    3.0           0.5    0.5    1.0
                                               表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X157      0.1250      9.0    9.0    5.0    9.0    9.0    9.0           7.0    9.0    7.5           6.5    6.0    7.5
      0.0625      9.0    9.0    4.0    7.0    7.0    9.0           6.0    7.0    7.0           6.5    5.5    7.0
      0.0313      9.0    7.0    3.0    6.0    7.0    9.0           4.0    4.0    7.0           5.5    5.0    7.0
      0.0156      9.0    5.0    2.0    6.0    5.0    6.0           1.0    1.0    6.0           4.0    3.5    7.0158      0.1250      9.0    9.0    5.0    9.0    9.0    9.0           2.0    7.0    6.0           4.5    4.5    7.0
      0.0625      9.0    6.0    6.0    9.0    6.0    9.0           2.0    5.0    6.0           5.0    5.0    7.0
      0.0313      9.0    6.0    3.0    7.0    4.0    9.0           2.0    2.0    5.0           3.5    4.0    5.5
      0.0156      9.0    3.0    3.0    4.0    3.0    4.0           1.0    2.0    5.0           3.0    3.0    5.0159      0.1250      9.0    9.0    6.0    9.0    5.0    9.0           3.0    4.0    7.5           5.0    5.0    6.5
      0.0625      9.0    9.0    6.0    9.0    6.0    9.0           3.0    2.0    6.5           4.0    4.5    6.0
      0.0313      9.0    6.0    2.0    7.0    3.0    9.0           1.0    1.0    5.0           3.5    4.0    5.0
      0.0156      7.0    6.0    2.0    6.0    1.0    3.0           0.0    1.0    5.0           2.5    4.0    5.0160      0.1250      1.0    2.0    1.0    1.0    2.0    1.0           0.0    0.0    3.0           0.5    1.0    1.0
      0.0625      0.0    0.0    1.0    1.0    0.0    1.0           0.0    0.0    3.0           0.5    0.5    0.5
      0.0313      0.0    0.0    1.0    0.0    0.0    1.0           0.0    0.0    2.5           0.0    0.5    0.5
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.0           0.0    0.5    0.5
                                              表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X161     0.1250      9.0    7.0    5.0    9.0    9.0    9.0           5.0    6.0    8.0           3.5    4.0    6.0
     0.0625      9.0    6.0    4.0    6.0    4.0    9.0           4.0    5.0    5.5           2.5    3.0    5.0
     0.0313      6.0    4.0    1.0    6.0    1.0    6.0           2.0    5.0    6.5           3.0    2.0    5.0
     0.0156      3.0    1.0    1.0    3.0    1.0    3.0           1.0    1.0    4.5           1.5    2.0    4.0162     0.1250                                                                     5.0           3.0    4.0    7.0
     0.0625                                                                     4.0           3.0    3.0    6.0
     0.0313                                                                     4.0           3.0    3.0    6.0
     0.0156                                                                     4.0           2.0    3.0    5.0163     0.1250                                                                     5.0           4.0    5.0    7.0
     0.0625                                                                     4.0           3.0    4.0    6.0
     0.0313                                                                     4.0           2.0    4.0    6.0
     0.0156                                                                     3.0           2.0    3.0    5.0164     0.0630                                                                     7.0           5.0    8.0    8.0
     0.0315                                                                     7.0           5.0    7.0    7.0
     0.0158                                                                     7.0           4.0    5.0    7.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X165      0.1250                                                                     7.0           3.0    4.0    6.0
      0.0625                                                                     7.0           2.0    3.0    6.0
      0.0313                                                                     7.0           1.0    3.0    5.0
      0.0156                                                                     7.0           1.0    3.0    5.0166      0.0630                                                                     4.0           2.0    4.0    6.0
      0.0315                                                                     4.0           2.0    4.0    6.0
      0.0158                                                                     2.0           2.0    4.0    5.0167      0.1250                                                                     6.0           2.0    3.0    5.0
      0.0625                                                                     6.0           2.0    3.0    5.0
      0.0313                                                                     5.0           2.0    2.0    4.0
      0.0156                                                                     5.0           1.0    2.0    4.0168      0.1250                                                                     8.0           4.0    4.0    6.0
      0.0625                                                                     7.0           3.0    3.0    6.0
      0.0313                                                                     7.0           2.0    3.0    5.0
      0.0156                                                                     7.0           1.0    3.0    5.0
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X169      0.1250                                                                     3.0           4.0    4.0    3.0
      0.0625                                                                     2.0           2.0    2.0    2.0
      0.0313                                                                     1.0           1.0    1.0    1.0
      0.0156                                                                     1.0           1.0    1.0    1.0170      0.1250      9.0    7.0    9.0    8.0    9.0    9.0           9.0    9.0    7.5           8.0    8.0    9.0
      0.0630      9.0    9.0    6.0    9.0    6.0    9.0           9.0    9.0    7.0           7.0    7.0    9.0
      0.0625      9.0    9.0    7.0    7.0    9.0    9.0           8.0    9.0    7.5           8.0    8.5    9.0
      0.0315      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    6.0           7.0    7.0    9.0
      0.0313      9.0    9.0    5.0    5.0    9.0    9.0           8.0    9.0    6.5           7.5    9.0    8.5
      0.0158      9.0    9.0    6.0    7.0    6.0    9.0           7.0    7.0    5.0           7.0    7.0    8.0
      0.0156      9.0    5.0    0.0    4.0    3.0    9.0           3.0    8.0    6.0           6.5    7.5    8.5171      0.0630      9.0    1.0    1.0    7.0    1.0    5.0           2.0    1.0    4.0           4.0    4.0    5.0
      0.0315      3.0    1.0    1.0    1.0    1.0    7.0           2.0    0.0    3.0           4.0    4.0    5.0
      0.0158      4.0    1.0    0.0    0.0    0.0    5.0           0.0    0.0    3.0           3.0    3.0    5.0172      0.0630      9.0    9.0    7.0    9.0    7.0    9.0           9.0    9.0    9.0           8.0    6.0    7.0
      0.0315      9.0    9.0    5.0    9.0    6.0    9.0           9.0    9.0    7.0           6.0    5.0    7.0
      0.0158      9.0    9.0    5.0    5.0    5.0    9.0           9.0    9.0    7.0           6.0    8.0    4.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物      施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      F      S      G      I      W      A      T      R      X173       0.1250     9.0    9.0    9.0    6.0    5.0    9.0           9.0    9.0    7.0           7.5    8.5    8.0
       0.0630     9.0    9.0    6.0    8.0    4.0    9.0           9.0    9.0    7.0           5.0    9.0    7.0
       0.0625     9.0    9.0    3.0    8.0    5.0    9.0           3.0    9.0    7.0           4.5    8.5    8.0
       0.0315     9.0    9.0    4.0    5.0    2.0    9.0           9.0    7.0    6.0           4.0    7.0    7.0
       0.0313     9.0    8.0    3.0    2.0    1.0    9.0           3.0    9.0    6.5           4.0    6.0    8.0
       0.0158     9.0    9.0    3.0    2.0    1.0    9.0           9.0    7.0    3.0           4.0    5.0    4.0
       0.0156     9.0    7.0    0.0    2.0    0.0    7.0           2.0    7.0    6.5           3.0    5.5    6.0174       0.0630     9.0    9.0    6.0    8.0    6.0    9.0           9.0    9.0    9.0           5.0    8.0    7.0
       0.0625     9.0    9.0    3.0    6.0    4.0    9.0           9.0    9.0    7.5           6.0    7.0    8.0
       0.0315     9.0    9.0    3.0    8.0    2.0    9.0           9.0    9.0    7.0           3.0    5.0    7.0
       0.0313     9.0    9.0    1.0    4.0    1.0    9.0           9.0    9.0    7.0           5.0    7.0    8.0
       0.0158     9.0    9.0    2.0    7.0    2.0    9.0           8.0    7.0    6.0           3.0    4.0    5.0
       0.0156     9.0    9.0    0.0    3.0    0.0    9.0           5.0    4.0    7.0           4.5    5.0    6.5
                                                 表1(续)
                                                                                  G             O      T
                  A       A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T       E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H       L      B      L      P      E      S      G      I      W      A      T      R      X175      0.0630      9.0     9.0    6.0    9.0    5.0    9.0           9.0    9.0    9.0           5.0    5.0    6.0
      0.0315      9.0     9.0    2.0    5.0    4.0    9.0           8.0    9.0    7.0           4.0    4.0    5.0
      0.0158      9.0     9.0    2.0    5.0    1.0    9.0           9.0    7.0    7.0           4.0    4.0    5.0176      0.1250      9.0     9.0    9.0    7.0    7.0    9.0           9.0    9.0    8.0           7.5    9.0    8.5
      0.0630      9.0     8.0    5.0    8.0    5.0    9.0           9.0    9.0    7.0           5.0    9.0    7.0
      0.0625      9.0     9.0    8.0    7.0    7.0    9.0           8.0    9.0    8.0           7.5    9.0    8.0
      0.0315      9.0     9.0    4.0    7.0    4.0    9.0           8.0    9.0    6.0           6.0    9.0    7.0
      0.0313      9.0     9.0    7.0    7.0    2.0    9.0           7.0    9.0    7.5           6.5    9.0    8.5
      0.0158      9.0     9.0    4.0    6.0    2.0    9.0           8.0    8.0    5.0           5.0    8.0    6.0
      0.0156      9.0     6.0    2.0    5.0    0.0    9.0           3.0    3.0    7.0           4.0    7.5    7.0177      0.0630      9.0     9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           6.0    5.0    7.0
      0.0315      9.0     9.0    5.0    8.0    5.0    9.0           9.0    9.0    7.0           6.0    7.0    5.0
      0.0158      9.0     9.0    3.0    8.0    6.0    9.0           8.0    9.0    7.0           4.0    4.0    5.0178      0.0630      9.0     9.0    5.0    8.0    8.0    9.0           9.0    9.0    9.0           4.0    4.0    7.0
      0.0315      9.0     9.0    2.0    7.0    7.0    9.0           9.0    9.0    7.0           4.0    3.0    5.0
      0.0158      9.0     9.0    2.0    4.0    5.0    9.0           7.0    9.0    5.0           4.0    3.0    5.0
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X179      0.1250      9.0    9.0    3.0    8.0    7.0    9.0           8.0    8.0    8.0           7.5    6.5    7.0
      0.0630      9.0    9.0    3.0    8.0    5.0    9.0           2.0    7.0    7.0           4.0    4.0    5.0
      0.0625      9.0    9.0    2.0    4.0    6.0    9.0           5.0    5.0    7.5           3.0    4.0    5.5
      0.0315      9.0    9.0    2.0    6.0    4.0    9.0           2.0    9.0    5.0           3.0    3.0    4.0
      0.0313      9.0    5.0    1.0    3.0    1.0    9.0           1.0    2.0    7.5           2.0    3.5    5.0
      0.0158      9.0    8.0    2.0    4.0    3.0    9.0           3.0    7.0    5.0           2.0    2.0    4.0
      0.0156      9.0    3.0    0.0    1.0    1.0    9.0           0.0           5.5           1.5    2.0    4.5180      0.0630      9.0    9.0    7.0    8.0    7.0    9.0           1.0    6.0    7.0           2.0    2.0    5.0
      0.0315      9.0    8.0    2.0    7.0    6.0    9.0           0.0    1.0    7.0           2.0    2.0    5.0
      0.0158      9.0    9.0    2.0    4.0    3.0    9.0           0.0    0.0    7.0           2.0    2.0    4.0181      0.0630      9.0    8.0    7.0    8.0    6.0    9.0           4.0    9.0    6.0           4.0    6.0    4.0
      0.0315      9.0    7.0    4.0    7.0    6.0    9.0           4.0    9.0    5.0           4.0    4.0    5.0
      0.0156      9.0    6.0    4.0    5.0    4.0    9.0           4.0    8.0    5.0           3.0    3.0    4.0182      0.0780      9.0    9.0    5.0    9.0    9.0    9.0           9.0    9.0    7.5           4.5    4.5    7.0
      0.0390      9.0    9.0    5.0    9.0    9.0    9.0           9.0    9.0    8.5           4.5    4.5    6.5
      0.0195      9.0    9.0    3.0    7.0    5.0    9.0           9.0    9.0    7.5           4.5    4.5    5.5
                                                   表1(续)
                                                                                    G             O      T
                  A       A       C       C      G      I      I      E      S      L      G      R      R      Z
                  B       M       A       H      A      P      P      C      E      X      L      Y      Z      E
                  U       B       S       E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T       E       O       A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H       L       B       L      P      E      S      G      I      W      A      T      R      X183      0.0780      9.0     9.0     9.0     9.0    9.0    9.0           9.0    9.0    8.5           9.0    7.5    8.0
      0.0390      9.0     9.0     7.0     9.0    9.0    9.0           9.0    9.0    8.0           6.5    7.5    7.5
      0.0195      9.0     9.0     4.0     8.0    5.0    9.0           9.0    9.0    7.5           4.0    6.0    6.5184      0.0780      9.0     9.0     3.0     9.0    9.0    9.0           9.0    9.0    7.0           8.0    9.0    7.5
      0.0390      9.0     9.0     3.0     7.0    7.0    9.0           9.0    9.0    7.0           5.5    7.5    6.5
      0.0195      9.0     9.0     0.0     5.0    3.0    9.0           9.0    9.0    6.5           3.5    5.5    6.0185      0.0640      9.0     9.0     3.0     9.0    9.0    9.0           9.0    9.0    8.5           7.0    7.0    7.5
      0.0320      9.0     9.0     3.0     9.0    9.0    9.0           9.0    9.0    8.0           5.5    5.5    6.0
      0.0160      9.0     9.0     1.0     3.0    5.0    9.0           7.0    8.0    8.5           4.5    5.5    5.0186      0.0630      9.0     9.0     7.0     9.0    9.0    9.0           9.0    9.0    8.0           7.0    6.5    8.0
      0.0315      9.0     9.0     5.0     9.0    6.0    9.0           9.0    9.0    7.5           7.0    6.0    7.0
      0.0158      9.0     9.0     0.0     5.0    5.0    9.0           9.0    9.0    7.5           4.5    5.0    6.0187      0.0630      9.0     9.0     3.0     9.0    7.0    9.0           9.0    9.0    7.5           5.0    6.5    7.5
      0.0315      9.0     9.0     3.0     9.0    6.0    9.0           9.0    7.0    7.0           5.0    5.5    5.5
      0.0158      9.0     8.0     0.0     8.0    4.0    9.0           7.0    3.0    6.5           3.0    5.0    5.5
                                                 表1(续)
                                                                                 G      O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X188      0.0630      9.0    9.0    2.0    1.0    1.0    9.0           2.0    5.0    5.5           4.0    4.0    7.0
      0.0315      9.0    7.0    2.0    0.0    0.0    9.0           5.0    9.0    5.5           4.0    4.5    6.0
      0.0158      9.0    9.0    1.0    1.0    1.0    6.0           1.0    8.0    5.5           3.0    3.5    5.0189      0.0630      9.0    6.0    4.0    6.0    1.0    7.0           4.0    9.0    4.5           3.0    3.5    4.5
      0.0315      9.0    5.0    4.0    5.0    1.0    9.0           4.0    3.0    4.0           2.5    3.0    5.0
      0.0158      9.0    2.0    1.0    4.0    1.0    7.0           1.0    1.0    4.0           1.5    3.5    3.5190      0.0630      9.0    9.0    6.0    7.5    9.0    9.0           9.0    9.0    8.5           7.0    6.3    7.5
      0.0315      9.0    9.0    6.0    8.0    7.0    9.0           9.0    9.0    8.0           6.3    6.0    7.3
      0.0158      9.0    9.0    5.5    4.5    5.5    9.0           8.0    7.0    7.0           5.3    5.3    6.0191      0.0630      9.0    9.0    8.0    8.0    8.5    9.0           9.0    9.0    8.0           7.5    6.8    8.0
      0.0315      9.0    9.0    7.0    9.0    7.0    9.0           9.0    9.0    7.3           6.5    6.5    7.5
      0.0158      8.0    9.0    4.0    7.5    7.0    9.0           9.0    9.0    7.3           5.3    5.8    6.8192      0.0630      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.5           7.0    7.0    7.5
      0.0315      9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    8.5           6.5    6.5    7.0
      0.0158      9.0    9.0    6.0    9.0    6.0    9.0           9.0    9.0    7.0           5.5    6.0    5.5193      0.0630      9.0    9.0    3.0    6.0    1.5    9.0           0.5    2.0    5.0           3.5    4.0    5.5
      0.0315      9.0    7.0    3.5    6.5    1.5    9.0           0.5    1.0    5.5           3.3    3.3    5.3
      0.0158      9.0    6.5    1.5    4.5    1.5    7.0           0.5    0.5    5.3           3.3    3.5    5.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X194      0.0630      9.0    9.0    8.0    9.0    7.0    9.0           9.0    9.0    8.5           7.5    6.0    8.0
      0.0315      9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    8.0           7.0    5.5    7.5
      0.0158      9.0    9.0    3.0    9.0    4.0    9.0           9.0    9.0    7.5           5.0    5.0    5.5195      0.0630      9.0    9.0    5.0    9.0    9.0    9.0           5.0    9.0    8.5           5.5    5.0    5.5
      0.0315      9.0    9.0    5.0    9.0    5.0    9.0           2.0    9.0    8.5           5.0    4.0    5.5
      0.0158      9.0    7.0    4.0    7.0    2.0    9.0           1.0    4.0    7.5           3.0    3.5    5.0196      0.0630      9.0    9.0    5.0    9.0    7.0    9.0           6.0    8.0    7.3           4.3    4.3    5.7
      0.0315      9.0    9.0    5.0    9.0    4.0    9.0           4.0    4.0    6.7           3.3    3.3    5.3
      0.0158      9.0    7.0    2.0    7.0    1.0    9.0           2.0    2.0    6.3           3.0    3.0    5.3197      0.2500      9.0    9.0    2.0    9.0    9.0    9.0           0.0    3.0    5.5           1.5    4.5    5.5
      0.1250      9.0    6.5    4.0    8.0    4.5    9.0           0.0    4.5    6.0           2.3    4.0    5.5
      0.0625      9.0    4.0    2.5    5.5    3.5    7.0           0.0    3.0    5.5           1.5    3.8    5.5
      0.0313      9.0    2.5    1.5    3.5    1.0    9.0           0.0    1.5    5.0           1.5    3.3    5.0
      0.0156      8.5    1.0    0.0    2.0    0.5    6.0           0.0    0.0    4.5           0.8    2.8    5.0198      0.1250      9.0    9.0    2.0    5.0    7.0    9.0           2.0    5.0    7.0           4.5    4.5    6.5
      0.0625      9.0    9.0    2.0    3.0    5.0    9.0           0.0    3.0    6.0           2.5    3.0    5.0
      0.0313      9.0    5.0    0.0    1.0    1.0    9.0           0.0    0.0    6.0           1.5    3.0    4.5
      0.0156      9.0    5.0    0.0    1.0    1.0    9.0           0.0    0.0    4.5           1.5    2.5    4.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X199       0.1250     9.0    4.0    2.0    1.0    4.0    9.0           0.0    1.0    5.5           2.0    2.5    6.0
       0.0625     9.0    2.0    2.0    1.0    2.0    9.0           0.0    1.0    5.5           1.5    2.5    5.0
       0.0313     9.0    1.0    2.0    1.0    1.0    9.0           0.0    1.0    4.5           1.0    2.0    5.0
       0.0156     7.0    1.0    0.0    1.0    1.0    6.0           0.0    0.0    4.5           1.0    2.0    5.0200       0.1250     9.0    9.0    4.0    7.0    7.0    9.0           7.0    7.0    8.5           4.5    4.5    6.5
       0.0625     9.0    7.0    3.0    6.0    7.0    9.0           0.0    2.0    7.0           4.5    4.0    6.0
       0.0313     9.0    7.0    0.0    2.0    2.0    9.0           0.0    0.0    6.5           2.5    3.0    5.0
       0.0156     9.0    2.0    0.0    1.0    2.0    9.0           0.0    0.0    5.5           2.0    2.5    5.0201       0.1250     9.0    6.0    4.0    6.0    6.0    9.0           0.0    3.0    7.5           3.5    4.0    5.5
       0.0625     9.0    6.0    2.0    3.0    2.0    9.0           0.0    2.0    6.0           3.0    3.5    5.5
       0.0313     9.0    3.0    0.0    1.0    1.0    9.0           0.0    2.0    5.0           2.5    3.0    5.5
       0.0156     7.0    2.0    0.0    1.0    0.0    6.0           0.0    0.0    5.0           2.0    2.5    5.0
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X202       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           0.0    9.0    8.0           2.5    5.5    6.0
       0.1250     9.0    9.0    1.0    9.0    9.0    9.0           0.0    9.0    8.0           2.0    4.0    5.5
       0.0630     9.0    7.0    6.0    7.0    6.0    9.0           3.0    4.0    7.5           4.0    4.5    5.5
       0.0625     9.0    6.0    1.0    9.0    6.0    9.0           0.0    0.0    6.5           1.5    2.5    5.0
       0.0315     9.0    6.0    6.0    6.0    4.0    9.0           2.0    1.0    6.5           4.0    4.5    5.5
       0.0313     9.0    4.0    0.0    9.0    4.0    9.0           0.0    0.0    5.5           0.5    2.0    4.5
       0.0158     9.0    6.0    4.0    6.0    4.0    7.0           2.0    1.0    6.0           3.0    3.5    5.0
       0.0156     9.0    3.0    0.0    9.0    2.0    3.0           0.0    0.0    5.5           0.5    2.0    4.5203       0.0630     9.0    8.0    6.0    9.0    6.0    9.0           5.0    5.0    7.5           5.0    5.0    6.0
       0.0315     9.0    9.0    5.0    6.0    6.0    9.0           2.0    5.0    7.0           4.0    4.0    5.5
       0.0158     9.0    7.0    4.0    4.0    4.0    9.0           2.0    3.0    7.0           3.0    3.5    5.5204       0.0630     9.0    9.0    6.0    7.0    6.0    9.0           4.0    5.0    7.5           5.5    5.5    6.0
       0.0315     9.0    7.0    6.0    6.0    5.0    9.0           3.0    2.0    6.0           3.5    4.5    5.5
       0.0158     9.0    4.0    3.0    3.0    3.0    9.0           2.0    2.0    6.0           4.0    4.5    5.5205       0.0630     9.0    9.0    6.0    9.0    6.0    9.0           4.0    7.0    8.5           4.5    5.5    6.0
       0.0315     9.0    8.0    5.0    8.0    5.0    9.0           3.0    4.0    7.0           4.5    4.5    5.5
       0.0158     9.0    6.0    4.0    6.0    3.0    9.0           2.0    2.0    7.5           3.0    3.5    4.5
                                               表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X206       0.0630     9.0    8.0    7.0    8.0    6.0    9.0           5.0    6.0    7.5           4.0    5.0    6.5
       0.0315     9.0    8.0    5.0    8.0    3.0    7.0           3.0    4.0    7.0           3.0    4.0    5.5
       0.0158     9.0    4.0    4.0    4.0    1.0    9.0           3.0    2.0    6.5           3.5    4.0    5.5207       0.0630     9.0    9.0    6.0    9.0    8.0    9.0           4.0    5.0    7.5           4.0    4.0    6.0
       0.0315     9.0    7.0    5.0    8.0    6.0    9.0           3.0    4.0    7.5           4.0    4.0    6.0
       0.0158     9.0    6.0    3.0    8.0    5.0    9.0           2.0    2.0    6.5           3.0    3.5    5.5208       0.0630     9.0    6.0    4.0    5.0    4.0    9.0           2.0    3.0    6.0           3.5    4.0    5.5
       0.0315     9.0    7.0    3.0    7.0    4.0    9.0           2.0    2.0    6.5           3.0    4.0    5.5
       0.0158     8.0    4.0    3.0    5.0    3.0    8.0           2.0    2.0    6.5           2.5    3.0    5.0209       0.0630     9.0    9.0    6.0    5.0    6.0    9.0           1.0    9.0    7.5           4.5    4.5    6.0
       0.0315     9.0    6.0    0.0    3.0    3.0    9.0           0.0    7.0    6.5           3.5    4.0    5.0
       0.0158     9.0    4.0    1.0    4.0    2.0    9.0           0.0    2.0    5.5           1.5    2.5    5.5210       0.0630     9.0    9.0    1.0    8.0    9.0    9.0           1.0    4.0    6.0           3.0    5.0    5.5
       0.0315     9.0    6.0    0.0    6.0    7.0    9.0           0.0    4.0    6.0           1.5    3.5    5.0
       0.0158     9.0    4.0    0.0    3.0    7.0    3.0           0.0    4.0    6.0           1.5    3.5    5.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X211      0.0630      9.0    9.0    2.0    7.0    9.0    9.0           0.0    2.0    6.0           1.5    4.0    5.5
      0.0315      9.0    4.0    1.0    4.0    5.0    9.0           0.0    0.0    5.0           1.5    3.5    5.0
      0.0158      9.0    0.0    0.0    0.0    0.0    2.0           0.0    0.0    4.5           1.0    3.5    5.0212      0.0630      9.0    6.0    0.0    6.0    6.0    9.0           0.0    0.0    5.5           1.5    3.5    5.5
      0.0315      9.0    3.0    0.0    0.0    5.0    3.0           0.0    0.0    5.0           1.5    3.0    5.0
      0.0158      9.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.0           1.5    2.0    4.5213      0.2500      9.0    3.0    2.0    5.0    3.0    6.0           2.0    7.0    4.5           4.5    4.5    5.5
      0.1250      9.0    2.0    1.0    4.0    1.0    9.0           0.0    0.0    4.0           3.5    3.5    5.5
      0.0630                                                                     8.0           6.0    6.0    7.0
      0.0625      9.0    2.0    1.0    4.0    1.0    7.0           0.0    0.0    4.5           3.5    3.5    5.0
      0.0315                                                                     8.0           5.0    5.0    7.0
      0.0313      7.0    1.0    1.0    1.0    1.0    4.0           1.0    1.0    4.5           3.5    4.0    5.0
      0.0158                                                                     8.0           5.0    5.0    6.0
      0.0156      2.0    0.0    0.0    0.0    1.0    2.0           0.0    0.0    4.0           3.0    3.5    3.5214      0.2500      6.0    2.0    2.0    7.0    2.0    4.0           1.0    3.0    5.5           3.0    4.0    5.0
      0.1250      4.0    0.0    1.0    2.0    2.0    2.0           1.0    3.0    3.5           2.0    2.5    5.0
      0.0625      4.0    1.0    0.0    2.0    1.0    1.0           0.0    0.0    3.5           2.5    2.0    4.5
      0.0313      3.0    0.0    0.0    1.0    0.0    0.0           0.0    0.0    3.5           2.0    2.5    3.5
      0.0156      3.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.5           2.5    2.0   3.5
                                                 表1(续)
                                                                                  G             O      T
                  A       A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T       E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H       L      B      L      P      E      S      G      I      W      A      T      R      X215      0.2500      1.0     1.0    0.0    4.0    1.0    1.0           1.0    5.0    3.5           1.0    1.0    2.5
      0.1250      0.0     0.0    0.0    2.0    0.0    1.0           0.0    5.0    4.0           0.5    0.5    2.0
      0.0625      0.0     0.0    0.0    3.0    0.0    0.0           0.0    1.0    3.0           0.5    1.0    0.5
      0.0313      0.0     0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.5           0.5    0.5    0.5
      0.0156      0.0     0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.0           0.5    0.5    0.5216      0.2500      5.0     3.0    1.0    4.0    1.0    1.0           0.0    0.0    3.5           1.0    1.0    1.5
      0.1250      4.0     3.0    0.0    4.0    0.0    0.0           0.0    0.0    4.0           1.0    0.5    1.0
      0.0625      2.0     1.0    0.0    1.0    0.0    0.0           0.0    0.0    4.0           0.5    0.5    1.0
      0.0313      1.0     0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.0           0.5    0.5    1.0
      0.0156      0.0     0.0    0.0    0.0    0.0    1.0           0.0    0.0    3.5           0.0    0.0    2.0217      0.2500      9.0     1.0    1.0    4.0    3.0    3.0           0.0    9.0    3.5           2.5    3.5    4.0
      0.1250      9.0     1.0    0.0    2.0    1.0    2.0           0.0    0.0    4.0           1.0    2.0    3.5
      0.0625      9.0     0.0    0.0    0.0    1.0    3.0           0.0    0.0    4.5           2.5    3.0    4.5
      0.0313      4.0     1.0    0.0    1.0    0.0    3.0           0.0    0.0    3.5           2.0    3.0    3.0
      0.0156      0.0     0.0    0.0    0.0    0.0    3.0           0.0    3.0    4.5           2.0    2.0    4.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X218      0.2500      5.0    1.0    1.0    2.0    2.0    0.0           0.0    0.0    4.0           1.0    1.0    2.0
      0.1250      2.0    0.0    0.0    3.0    1.0    0.0           0.0    0.0    3.5           0.5    0.5    1.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.5           0.5    0.5    1.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.5           0.5    0.5    1.5
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.5           0.5    1.0    1.5219      0.2500      9.0    9.0    4.0    9.0    9.0    9.0           2.0    9.0    9.0           6.0    6.5    7.0
      0.1250      9.0    9.0    2.0    9.0    9.0    9.0           0.0    9.0    9.0           4.5    6.0    6.0
      0.0625      9.0    7.0    0.0    9.0    7.0    9.0           0.0    3.0    8.5           3.5    5.0    5.0
      0.0313      9.0    4.0    0.0    9.0    5.0    9.0           0.0    0.0    7.0           2.0    4.5    4.5
      0.0156      9.0    1.0    0.0    3.0    0.0    4.0           0.0    0.0    5.5           2.0    3.0    4.5220      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    8.5           6.4    7.0    8.0
      0.1250      9.0    9.0    3.0    9.0    7.0    9.0           3.0    9.0    7.5           6.0    6.0    8.0
      0.0625      9.0    7.0    1.0    9.0    4.0    9.0           0.0    9.0    7.5           6.0    6.0    7.0
      0.0313      9.0    5.0    1.0    9.0    4.0    9.0           0.0    5.0    5.5           3.0    5.5    6.0
      0.0156      9.0    1.0    0.0    4.0    4.0    9.0           0.0           5.0           2.0    4.5    4.5
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X221       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           2.0    9.0    8.5           4.0    5.0    6.5
       0.1250     9.0    9.0    7.0    9.0    8.0    9.0           2.0    9.0    7.5           3.5    5.0    6.5
       0.0625     9.0    4.0    9.0    9.0    9.0    9.0           2.0    7.0    7.0           3.0    4.5    6.0
       0.0313     9.0    3.0    3.0    9.0    6.0    9.0           0.0           6.0           2.0    3.5    5.0
       0.0156     9.0    3.0    0.0    8.0    3.0    9.0           0.0    0.0    5.5           2.0    3.0    5.0222       0.2500     9.0    9.0    9.0    9.0    7.0    9.0           1.0    9.0    6.5           2.5    4.0    6.0
       0.1250     9.0    7.0    7.0    9.0    7.0    9.0           0.0    9.0    6.5           2.0    4.0    6.0
       0.0625     9.0    9.0    3.0    9.0    5.0    9.0           0.0    6.0    6.0           1.0    4.0    5.0
       0.0313     9.0    4.0    2.0    7.0    5.0    7.0           0.0           5.5           0.5    3.5    5.0
       0.0156     9.0    3.0    0.0    4.0    5.0    3.0           0.0    6.0    4.5           0.5    3.0    5.0223       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.0    7.0
       0.1250     9.0    9.0    7.0    9.0    7.0    9.0           4.0    9.0    9.0           5.0    6.0    7.0
       0.0625     9.0    9.0    6.0    8.0    7.0    9.0           3.0    9.0    7.5           5.0    5.5    6.5
       0.0313     9.0    5.0    4.0    7.0    3.0    9.0           3.0    4.0    6.0           4.5    5.0    5.5
       0.0156     9.0    5.0    4.0    9.0    3.0    9.0           2.0    4.0    6.0           3.0    4.5    5.5224       0.1250     9.0    9.0    4.0    9.0    9.0    9.0           2.0    3.0    6.5           5.0    5.5    6.5
       0.0625     9.0    6.0    4.0    6.0    7.0    9.0           2.0    3.0    7.5           5.0    5.0    6.5
       0.0313     9.0    6.0    1.0    6.0    4.0    9.0           2.0    1.0    5.5           4.5    5.0    6.0
       0.0156     9.0    3.0    1.0    5.0    3.0    7.0           0.0    1.0    5.0           3.0    4.0    5.0
                                              表1(续)
                                                                               G             O      T
                A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X225     0.2500     9.0    9.0    7.0    9.0    9.0    9.0           4.0    7.0    9.0           5.0    6.0    6.5
     0.1250     9.0    9.0    6.0    9.0    7.0    9.0           3.0    4.0    6.0           5.0    5.0    6.0
     0.0825     9.0    9.0    3.0    7.0    6.0    9.0           3.0    5.0    6.0           3.5    4.0    6.0
     0.0313     9.0    6.0    1.0    4.0    3.0    9.0           1.0    2.0    5.5           3.0    3.0    5.0
     0.0156     9.0    4.0    1.0    4.0    2.0    9.0           1.0    2.0    4.5           3.0    2.5    5.0226     0.0630     9.0    9.0    3.0    9.0    2.0    9.0           3.0    9.0    5.0           3.0    5.0    6.5
     0.0315     9.0    9.0    6.0    9.0    2.0    8.0           2.0    8.0    5.0           2.5    4.0    6.0
     0.0158     9.0    4.0    0.0    4.0    0.0    9.0           2.0    7.0    4.5           2.0    3.5    5.5227     0.0630     9.0    9.0    0.0    9.0    6.0    9.0           7.0    9.0    8.0           1.5    4.5    8.5
     0.0315     9.0    9.0    0.0    9.0    2.0    9.0           3.0    8.0    5.5           1.5    4.0    6.0
     0.0158     9.0    9.0    0.0    9.0    0.0    9.0           0.0    3.0    5.0           1.5    4.0    5.5228     0.0630     9.0    9.0    4.0    5.0    3.0    9.0           2.0    9.0    6.0           2.0    5.5    6.0
     0.0315     9.0    6.0    3.0    5.0    0.0    9.0           2.0    7.0    4.5           2.0    4.0    5.5
     0.0158     9.0    4.0    0.0    5.0    0.0    9.0           2.0    6.0    4.5           1.5    3.5    5.5229     0.0630     3.0    0.0    0.0    4.0    1.0    6.0           0.0    4.0    5.5           2.0    3.5    4.5
     0.0315     3.0    0.0    0.0    4.0    0.0    2.0           0.0    0.0    4.0           1.0    3.5    4.5
     0.0158     2.0    0.0    0.0    0.0    0.0    1.0           0.0           3.5           1.0    3.5    4.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X230       0.0630     9.0    9.0    2.0    9.0    3.0    9.0           2.0    0.0    6.0           2.5    6.5    6.5
       0.0315     9.0    9.0    0.0    9.0    0.0    9.0           0.0    0.0    6.0           2.5    5.0    5.5
       0.0158     9.0    9.0    0.0    6.0    0.0    9.0           0.0           5.5           1.5    3.0    5.5231       0.0630     9.0    9.0    4.0    9.0    4.0    9.0           9.0    9.0    6.5           2.5    5.0    7.0
       0.0315     9.0    9.0    2.0    9.0    2.0    9.0           4.0    9.0    6.0           2.0    4.5    5.5
       0.0158     9.0    4.0    2.0    5.0    2.0    9.0           4.0    7.0    6.0           2.0    4.5    5.5232       0.0630     9.0    9.0    6.0    9.0    2.0    9.0           6.0    9.0    7.5           3.0    7.5    8.5
       0.0315     9.0    9.0    6.0    9.0    0.0    9.0           6.0    8.0    7.0           2.5    6.5    7.0
       0.0158     9.0    7.0    3.0    9.0    0.0    9.0           5.0    5.0    6.5           2.5    7.0    6.0233       0.0630     9.0    9.0    3.0    9.0    0.0    9.0           0.0    7.0    5.5           1.5    4.0    5.5
       0.0315     9.0    8.0    0.0    7.0    0.0    9.0           0.0    7.0    5.5           1.5    4.0    5.5
       0.0158     4.0    3.0    0.0    4.0    0.0    9.0           0.0    4.0    5.0           1.0    4.0    5.5234       0.0630     9.0    9.0    7.0    9.0    4.0    9.0           5.0    9.0    5.5           2.5    4.5    7.0
       0.0315     9.0    9.0    0.0    9.0    0.0    9.0           0.0    6.0    5.0           2.0    3.5    5.5
       0.0158     9.0    9.0    0.0    4.0    0.0    7.0           0.0    7.0    5.0           1.0    2.5    4.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X235      0.0630      9.0    9.0    4.0    9.0    3.0    9.0           4.0    9.0    6.0           2.5    5.5    6.5
      0.0315      7.0    7.0    4.0    5.0    0.0    9.0           0.0    9.0    6.0           2.5    4.0    6.5
      0.0158      9.0    9.0    4.0    5.0    0.0    9.0           0.0    3.0    5.5           1.5    3.5    5.0236      0.1250      9.0    4.0    1.0    6.0    2.0    2.0           1.0    1.0    4.5           2.5    3.0    5.0
      0.0625      8.0    3.0    1.0    5.0    2.0    2.0           1.0    1.0    4.0           2.0    2.0    5.0
      0.0313      6.0    1.0    1.0    4.0    7.0    3.0           1.0    1.0    4.0           2.0    2.0    4.5
      0.0156      4.0    2.0    1.0    3.0    1.0    1.0           0.0    0.0    2.5           1.5    1.5    3.5237      0.1250      9.0    6.0    4.0    7.0    7.0    9.0           2.0    7.0    6.0           3.0    3.5    5.0
      0.0625      9.0    6.0    3.0    9.0    5.0    9.0           3.0    9.0    5.5           2.0    3.0    5.0
      0.0313      9.0    5.0    2.0    6.0    3.0    4.0           2.0    4.0    4.0           1.5    2.0    5.0
      0.0156      2.0    3.0    0.0    2.0    1.0    2.0           0.0    0.0    3.0           1.0    2.0    4.0238      0.1250      9.0    9.0    4.0    9.0    6.0    9.0.          2.0    4.0    5.5           2.5    3.0    5.0
      0.0625      9.0    9.0    4.0    7.0    5.0    9.0           1.0    2.0    5.0           2.5    3.0    4.5
      0.0313      9.0    7.0    2.0    6.0    3.0    9.0           1.0    2.0    4.5           2.0    2.0    4.5
      0.0156      5.0    4.0    1.0    3.0    2.0    3.0           1.0    1.0    3.5           0.5    1.0    3.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X239      0.1250      9.0    9.0    6.0    9.0    7.0    9.0           5.0    9.0    7.0           4.0    5.0    5.5
      0.0825      9.0    9.0    4.0    7.0    5.0    9.0           3.0    3.0    6.0           3.0    3.0    5.5
      0.0313      9.0    9.0    3.0    6.0    4.0    9.0           2.0    2.0    5.5           2.0    2.5    5.0
      0.0156      9.0    5.0    2.0    4.0    2.0    9.0           1.0    2.0    4.0           2.0    2.5    4.0240      0.1250                                                                     7.0           5.0    6.0    6.0
      0.0625                                                                     7.0           4.0    5.0    6.0
      0.0313                                                                     7.0           3.0    4.0    6.0
      0.0156                                                                     6.0           3.0    3.0    5.0241      0.1250                                                                     6.0           4.0    5.0    5.0
      0.0625                                                                     6.0           3.0    4.0    5.0
      0.0313                                                                     6.0           3.0    5.0    5.0
      0.0156                                                                     5.0           3.0    4.0    4.0242      0.1250                                                                     7.0           5.0    5.0    6.0
      0.0625                                                                     7.0           4.0    5.0    6.0
      0.0313                                                                     7.0           4.0    4.0    6.0
      0.0156                                                                     6.0           4.0    5.0    6.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X243      0.1250                                                                     7.0           4.0    4.0    6.0
      0.0625                                                                     7.0           4.0    5.0    6.0
      0.0313                                                                     7.0           4.0    4.0    6.0
      0.0156                                                                     6.0           4.0    4.0    5.0244      0.1250                                                                     7.0           4.0    4.0    6.0
      0.0625                                                                     7.0           4.0    4.0    6.0
      0.0313                                                                     6.0           4.0    4.0    6.0
      0.0156                                                                     6.0           3.0    4.0    5.0245      0.0630      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           0.5    0.0    0.5
      0.0315      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0158      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0246      0.0630      9.0    2.0    0.0    2.0    1.0    6.0           5.0    8.0    4.5           3.0    4.5    7.5
      0.0315      9.0    0.0    0.0    2.0    0.0    9.0           6.0    3.0    4.0           2.5    3.0    6.0
      0.0158      0.0    0.0    0.0    0.0    0.0    1.0           1.0    1.0    4.0           2.0    2.5    5.0
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X247      0.1250                                                                     8.0           6.0    6.0    7.0
      0.0625                                                                     8.0           5.0    6.0    6.0
      0.0313                                                                     8.0           3.0    5.0    6.0
      0.0156                                                                     7.0           3.0    5.0    6.0248      0.5000                                                                     7.0           5.0    6.0    7.0
      0.2500                                                                     7.0           4.0    6.0    7.0
      0.1250                                                                     6.0           2.0    4.0    6.0
      0.0625                                                                     6.0           1.0    4.0    5.0
      0.0313                                                                     5.0           1.0    4.0    5.0
      0.0156                                                                     5.0           1.0    3.0    4.0249      0.1250                                                                     9.0           9.0    9.0    8.0
      0.0625                                                                     9.0           9.0    8.0    8.0
      0.0313                                                                     8.0           8.0    7.0    8.0
      0.0156                                                                     8.0           5.0    6.0    8.0250      0.1250                                                                     8.0           7.0    5.0    5.0
      0.0625                                                                     8.0           7.0    4.0    5.0
      0.0313                                                                     7.0           3.0    4.0    5.0
      0.0156                                                                     6.0           2.0    4.0    5.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X251      0.1250                                                                     9.0           9.0    8.0    8.0
      0.0625                                                                     8.0           8.0    8.0    8.0
      0.0313                                                                     8.0           5.0    7.0    6.0
      0.0156                                                                     8.0           4.0    4.0    6.0252      0.1250                                                                     7.0           3.0    4.0    6.0
      0.0625                                                                     7.0           2.0    4.0    6.0
      0.0313                                                                     5.0           0.0    2.0    4.0
      0.0156                                                                     5.0           0.0    2.0    4.0253      0.1250                                                                     9.0           9.0    8.0    8.0
      0.0625                                                                     9.0           8.0    8.0    8.0
      0.0313                                                                     8.0           8.0    8.0    8.0
      0.0156                                                                     8.0           7.0    6.0    7.0254      0.1250                                                                     9.0           9.0    9.0    8.0
      0.0625                                                                     9.0           9.0    9.0    8.0
      0.0313                                                                     9.0           8.0    8.0    8.0
      0.0156                                                                     8.0           6.0    7.0    7.0
                                                 表1(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X255       0.1250                                                                     6.0           2.0    4.0    6.0
       0.0625                                                                     5.0           2.0    3.0    6.0
       0.0313                                                                     4.0           1.0    2.0    4.0
       0.0156                                                                     1.0           0.0    1.0    1.0256       0.0620      9.0    9.0    4.0    9.0    9.0    9.0           2.0    9.0    9.0           7.0    6.5    7.0
       0.0320      9.0    9.0    2.0    9.0    9.0    9.0           0.0    7.0    9.0           5.5    5.0    6.5
       0.0160      9.0    9.0    0.0    9.0    7.0    9.0           0.0    0.0    9.0           4.0    3.5    5.0257       0.0620      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    9.0    8.0
       0.0320      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           5.5    8.5    8.0
       0.0160      9.0    9.0    2.0    9.0    9.0    9.0           7.0    7.0    9.0           2.0    6.5    7.0258       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    9.0
       0.0620      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.0320      8.9    9.0    4.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.0160      8.6    9.0    9.0    9.0    7.0    9.0           8.0    9.0    8.5           7.0    9.0    8.5259       0.0620      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           5.0    8.0    8.0
       0.0320      9.0    9.0    9.0    9.0    8.0    9.0           9.0    7.0    9.0           3.5    6.5    8.0
       0.0160      9.0    9.0    3.0    9.0    9.0    9.0           6.0    9.0    8.0           2.5    5.5    8.0
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X260      0.1250      3.0    0.0    0.0    0.0    0.0    1.0           0.0    0.0    2.5           3.0    2.0    1.0
      0.0620      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.5           2.0    2.0    1.0261      0.0620      9.0    9.0    0.0    9.0    4.0    9.0           9.0    9.0    9.0           8.0    7.0    8.0
      0.0320      9.0    8.0    0.0    5.0    3.0    9.0           7.0    9.0    7.5           8.0    6.0    7.5
      0.0160      9.0    3.0    0.0    3.0    2.0    9.0           2.0    3.0    6.5           6.5    5.0    7.0262      0.1250      9.0    9.0    0.0    9.0    8.0    9.0           0.0    0.0    6.5           3.5    4.5    5.0
      0.0620      9.0    9.0    0.0    0.0    5.0    9.0           0.0    0.0    6.0           3.0    4.0    4.5
      0.0320      9.0    3.0    0.0    0.0    0.0    1.0           0.0    0.0    4.0           1.5    3.5    4.0
      0.0160      9.0    3.0    0.0    0.0    0.0    0.0           0.0    0.0    4.0           1.0    3.0    4.0263      0.1250      9.0    9.0    0.0    3.0    4.0    9.0           0.0    0.0    7.0           2.5    5.0    5.0
      0.0620      9.0    3.0    0.0    3.0    3.0    4.0           0.0    0.0    4.5           1.5    4.0    4.5
      0.0320      9.0    1.0    0.0    0.0    3.0    4.0           0.0    0.0    4.0           1.0    4.0    3.0
      0.0160      9.0    0.0    0.0    0.0    0.0    4.0           0.0    0.0    3.0           0.5    3.0    3.0264      0.1250      9.0    9.0    0.0    5.0    9.0    9.0           0.0    0.0    6.5           1.5    2.5    5.0
      0.0620      9.0    5.0    0.0    3.0    8.0    9.0           0.0    0.0    5.0           0.5    2.0    4.0
      0.0320      9.0    5.0    0.0    0.0    5.0    9.0           0.0    0.0    5.0           0.5    1.5    3.5
      0.0160      9.0    2.0    0.0    0.0    0.0    4.0           0.0    0.0    3.0           0.5    1.5    3.0
                                                 表1(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X265       0.1250      2.0    0.0    0.0    9.0    7.0    0.0           0.0    0.0    4.5           5.5    3.0    7.0
       0.0620      2.0    0.0    0.0    5.0    7.0    0.0           0.0    0.0    3.5           3.5    3.0    4.5
       0.0320      0.0    0.0    0.0    5.0    5.0    0.0           0.0    0.0    3.0           1.5    1.0    3.5
       0.0160      0.0    0.0    0.0    3.0    0.0    0.0           0.0    0.0    2.0           0.5    0.5    2.5266       0.1250      9.0    5.0    0.0    7.0    4.0    9.0           0.0    0.0    5.0           3.0    5.5    5.5
       0.0620      9.0    3.0    0.0    7.0    4.0    9.0           0.0    0.0    4.5           2.0    4.0    3.5
       0.3220      0.0    0.0    0.0    0.0    2.0    0.0           0.0    0.0    3.0           1.0    2.5    1.5
       0.0160      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.5           0.5    1.5    1.0267       0.0620      9.0    9.0    0.0    9.0    9.0    9.0           0.0    0.0    5.0           3.5    5.0    5.0
       0.0320      9.0    4.0    0.0    8.0    7.0    5.0           0.0    0.0    4.5           2.5    4.5    5.0
       0.0160      9.0    2.0    0.0    4.0    3.0    1.0           0.0    0.0    3.5           2.0    3.0    4.5268       0.0320      9.0    9.0    9.0    9.0    7.0    9.0           9.0    8.0    9.0           7.3    6.3    8.5
       0.0160      9.0    9.0    6.0    9.0           9.0           9.0    9.0    9.0           8.0    7.0    9.0269       0.0620      1.0    2.0    0.0    5.0    0.0    9.0           0.0    0.0    3.5           3.0    2.5    4.5
       0.0320      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.0           2.5    2.5    4.0
                                                 表1(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X270       0.0620      9.0    9.0    9.0    9.0    4.0    9.0           4.0    4.0    7.5           7.0    7.0    7.5
       0.3320      9.0    9.0    2.0    6.0    2.0    9.0           4.0    6.0    6.0           5.0    4.5    6.5
       0.0160      9.0    5.0    0.0    5.0    1.0    9.0           0.0    4.0    5.0           4.0    4.5    4.5271       0.0620      9.0    6.0    2.0    9.0    6.0    9.0           1.0    3.0    5.5           2.5    3.0    4.5
       0.0320      9.0    4.0    0.0    7.0    7.0    9.0           1.0    1.0    4.5           2.5    3.0    3.5
       0.0160      2.0    2.0    0.0    5.0    9.0    0.0           0.0    0.0    4.0           2.5    2.0    3.5272       0.1250      9.0    8.0    0.0    2.0    3.0    9.0           0.0    0.0    6.0           1.0    2.0    4.5
       0.0620      9.0    4.0    0.0    0.0    1.0    9.0           0.0    0.0    5.5           0.0    1.0    4.0
       0.0320      3.0    0.0    0.0    0.0    0.0    9.0           0.0    0.0    4.5           0.0    1.0    3.5
       0.0160      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.5           0.0    1.0    2.0273       0.0620      9.0    9.0    9.0    9.0    5.0    9.0           3.0    6.0    9.0           3.5    4.5    5.5
       0.3220      9.0    7.0    9.0    9.0    5.0    9.0           2.0    2.0    7.5           3.5    4.5    6.0
       0.0160      9.0    6.0    2.0    7.0           9.0           1.0    1.0    5.0           3.0    3.0    5.5274       0.0620      9.0    9.0    6.0    6.0    5.0    9.0           9.0    9.0    9.0           9.0    7.5    9.0
       0.0320      9.0    7.0    2.0    7.0    3.0    7.0           9.0    9.0    9.0           7.5    7.5    7.5
       0.0160      9.0    6.0    2.0    4.0    2.0    9.0           9.0    9.0    8.5           7.5    5.5    7.5
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X275       0.0620     9.0    9.0    6.0    9.0    5.0    9.0           9.0    9.0    6.5           8.5    8.5    9.0
       0.0320     9.0    6.0    2.0    9.0    9.0    9.0           7.0    5.0    6.0           7.5    7.5    9.0
       0.0160     9.0    9.0    4.0    4.0    6.0    9.0           6.0    7.0    4.5           5.5    8.5    8.5276       0.0620     9.0    7.0    4.0    6.0    6.0    9.0           2.0    4.0    5.5           3.5    4.5    5.0
       0.0320     9.0    9.0    2.0    3.0    3.0    9.0           1.0    3.0    4.5           2.5    2.5    3.5
       0.0160     9.0    3.0    1.0    1.0    4.0    4.0           2.0    1.0    3.0           1.5    1.5    3.0277       0.0620     9.0    9.0    2.0    7.0    7.0    9.0           2.0    5.0    8.0           6.0    5.0    6.0
       0.0320     9.0    9.0    2.0    5.0    9.0    7.0           2.0    4.0    8.0           5.5    4.0    5.5
       0.0160     9.0    6.0    1.0    4.0    7.0    6.0           1.0    2.0    5.0           3.5    3.5    3.5278       0.0620     9.0    7.0    1.0    6.0    9.0    6.0           2.0    7.0    5.5           4.5    4.5    5.0
       0.0320     9.0    4.0    1.0    3.0    7.0    5.0           1.0    5.0    5.5           4.5    2.5    4.5
       0.0160     9.0    2.0    0.0    1.0    1.0    2.0           1.0    1.0    4.5           2.0    1.5    2.0279       0.0620     6.0    7.0    2.0    3.0    7.0    9.0           3.0    3.0    6.5           2.5    3.5    5.5
       0.0320     9.0    6.0    2.0    3.0    6.0    7.0           2.0    3.0    6.0           2.0    3.5    5.0
       0.0160     4.0    4.0    0.0    1.0    9.0    0.0           2.0    1.0    4.0           1.5    2.5    3.5
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X280       0.0620     9.0    9.0    9.0    8.0    9.0.   9.0           9.0    9.0    9.0           9.0    7.5    9.0
       0.0320     9.0    9.0    4.0    9.0    6.0    9.0           9.0    9.0    9.0           7.0    7.0    8.0
       0.0160     9.0    9.0    4.0    9.0    6.0    9.0           6.0    9.0    9.0           8.0    6.0    8.0281       0.0620     9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    9.0           7.0    6.5    8.0
       0.0320     9.0    7.0    9.0    9.0    7.0    9.0           7.0    7.0    9.0           5.5    6.5    7.5
       0.0160     9.0    9.0    6.0    9.0    9.0    9.0           6.0    9.0    7.5           5.5    6.5    7.5282       0.0620     5.0    4.0    1.0    3.0    2.0    1.0           1.0    2.0    5.0           1.5    3.0    2.0
       0.0320     1.0    3.0    1.0    2.0    2.0    1.0           1.0    0.0    3.5           1.0    1.5    2.0
       0.0160     0.0    1.0    1.0    0.0    1.0    1.0           1.0    0.0    2.0           1.0    1.5    1.5283       0.0620     9.0    5.0    1.0    9.0    6.0    5.0           3.0    6.0    7.5           5.5    6.0    7.0
       0.0320     9.0    4.0    1.0    7.0    5.0    9.0           3.0    4.0    7.0           5.0    6.0    7.0
       0.0160     9.0    2.0    0.0    3.0    4.0    9.0           0.0    5.0    6.5           4.0    3.5    7.0284       0.0620     9.0    4.0    1.0    2.0    7.0    9.0           2.0    2.0    5.5           4.0    3.5    7.0
       0.0320     6.0    4.0    1.0    1.0    2.0    7.0           1.0    2.0    4.0           2.5    2.5    6.0
       0.0160     3.0    2.0    1.0    0.0    1.0    4.0           0.0    2.0    3.5           2.0    3.0    3.0285       0.0620     9.0    9.0    1.0    6.0    9.0    9.0           2.0    4.0    7.0           5.0    5.0    5.0
       0.0320     9.0    9.0    1.0    6.0    7.0    9.0           2.0    2.0    6.5           3.5    4.0    4.5
       0.0160     9.0    7.0    0.0    0.0    6.0    7.0           1.0    4.0    6.5           3.5    3.0    3.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X286       0.0620     9.0    7.0    0.0    1.0    2.0    5.0           1.0    2.0    5.5           3.5    4.0    7.0
       0.0320     2.0    3.0    0.0    2.0    3.0    9.0           1.0    4.0    5.0           3.0    3.5    4.5
       0.0160     4.0    2.0    0.0    1.0    2.0    1.0           0.0    1.0    3.5           1.5    2.0    1.5287       0.0620     9.0    7.0    1.0    6.0    3.0    9.0           2.0    2.0    5.5           3.5    3.5    5.0
       0.0320     9.0    5.0    0.0    2.0    1.0    9.0           2.0    2.0    6.5           3.0    3.0    5.0
       0.0160     6.0    2.0    0.0    0.0    0.0    7.0           0.0    1.0    4.5           2.0    2.5    4.5288       0.0620     9.0    9.0    6.0    9.0    6.0    9.0           9.0    7.0    9.0           3.0    6.5    9.0
       0.0320     7.0    9.0    5.0    9.0    6.0    9.0           9.0    9.0    9.0           3.5    7.0    9.0
       0.0160     9.0    9.0    2.0    9.0    3.0    9.0           5.0    3.0    6.0           2.0    4.0    7.0289       0.0620     9.0    7.0    1.0    9.0    2.0    9.0           3.0    4.0    5.5           2.5    3.5    5.0
       0.0320     9.0    9.0    2.0    5.0    1.0    9.0           2.0    6.0    5.5           1.5    3.0    4.5
       0.0160     9.0    7.0    0.0    2.0    1.0    9.0           0.0    1.0    5.5           0.5    2.0    3.5290       0.0620     9.0    9.0    1.0    9.0    1.0    9.0           1.0    2.0    4.5           1.5    3.0    5.0
       0.0320     6.0    7.0    1.0    9.0    1.0    6.0           1.0    1.0    4.5           1.0    2.5    4.5
       0.0160     9.0    9.0    0.0    2.0    1.0    9.0           0.0    0.0    4.0           0.5    2.0    4.5
                                                   表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X291       0.0620     9.0    4.0    0.0    2.0    4.0    7.0           0.0    0.0    7.0           2.5    3.0    5.5
       0.0320     6.0    1.0    0.0    1.0    2.0    2.0           0.0    0.0    6.5           2.0    2.0    5.0
       0.0180     3.0    0.0    0.0    0.0    1.0    2.0           0.0    0.0    6.5           2.0    2.0    4.5292       0.1250     9.0    9.0    0.0    7.0    9.0    9.0           5.0    7.0    8.0           5.0    6.5    7.5
       0.0620     9.0    4.0    0.0    4.0    9.0    9.0           0.0    0.0    8.5           4.0    5.5    7.5
       0.0320     9.0    4.0    0.0    4.0    6.0    9.0           0.0    0.0    5.5           4.0    5.5    7.0
       0.0160     9.0    4.0    0.0    0.0    6.0    2.0           0.0    0.0    5.0           3.0    4.5    6.5293       0.1250     9.0    9.0    0.0    5.0    8.0    7.0           6.0    8.0    6.5           4.5    6.5    8.0
       0.0620     9.0    9.0    0.0    3.0    4.0    5.0           2.0    5.0    6.0           5.0    6.0    7.5
       0.0320     9.0    1.0    0.0    2.0    4.0    5.0           0.0    0.0    6.0           3.5    5.0    7.5
       0.0160     9.0    0.0    0.0    0.0    2.0    1.0           0.0    0.0    4.5           3.0    4.5    6.5294       0.1250     9.0    4.0    0.0    3.0    9.0    8.0           0.0    0.0    7.0           5.0    5.5    7.0
       0.0620     9.0    4.0    0.0    3.0    3.0    8.0           0.0    0.0    7.0           3.5    5.0    6.5
       0.0320     4.0    4.0    0.0    1.0    3.0    8.0           0.0    0.0    6.0           3.5    4.5    6.0
       0.0160     0.0    0.0    0.0    0.0    0.0    2.0           0.0    0.0    5.0           3.0    4.0    5.5295       0.1250     9.0    9.0    0.0    4.0    9.0    7.0           0.0    3.0    7.0           3.5    4.5    5.5
       0.0620     7.0    9.0    0.0    0.0    6.0    4.0           0.0    0.0    5.5           3.0    4.0    5.5
       0.0320     4.0    5.0    0.0    0.0    2.0    2.0           0.0    0.0    5.5           2.5    4.5    6.0
       0.0160     2.0    3.0    0.0    0.0    2.0    2.0           0.0    0.0    4.5           2.5    3.0    5.0
                                                   表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X296       0.1250     9.0    9.0    0.0    4.0    7.0    9.0           2.0    7.0    7.5           5.5    6.0    7.5
       0.0620     9.0    4.0    0.0    0.0    4.0    7.0           1.0           6.0           4.0    5.5    7.0
       0.0320     9.0    1.0    0.0    0.0    4.0    4.0           0.0    0.0    5.0           3.0    5.0    6.5
       0.0160     7.0    0.0    0.0    0.0    3.0    1.0           0.0    0.0    5.0           3.0    5.0    6.5297       0.1250     9.0    4.0    0.0    4.0    4.0    9.0           0.0    0.0    7.5           4.0    5.0    7.5
       0.0620     9.0    4.0    0.0    3.0    4.0    3.0           0.0    2.0    7.5           3.0    5.0    7.0
       0.0320            3.0    0.0    2.0    2.0    2.0           0.0           7.0           3.0    4.5    7.0
       0.0160     9.0    0.0    0.0    0.0    0.0    1.0           0.0    0.0    5.0           3.0    4.0    6.0298       0.1250     9.0    9.0    0.0    4.0    7.0    8.0           1.0    3.0    6.5           3.0    4.5    6.5
       0.0620     9.0    9.0    0.0    4.0    5.0    3.0           0.0    0.0    6.5           3.0    4.0    6.0
       0.0320     9.0    2.0    0.0    0.0    1.0    1.0           0.0    0.0    6.5           3.0    4.0    6.0
       0.0160     3.0           0.0    0.0    0.0    0.0           0.0    0.0    6.0           3.0    4.0    6.0299       0.1250     9.0    6.0    0.0    7.0    3.0    9.0           0.0    0.0    7.5           4.5    5.5    7.0
       0.0620     9.0    3.0    0.0    3.0    1.0    7.0           0.0    0.0    7.0           3.0    5.0    7.0
       0.0320     9.0    1.0    0.0    0.0    0.0    3.0           0.0    0.0    6.5           3.0    4.5    6.5
       0.0160     9.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.5           2.5    4.0    6.5
                                                表1(续)
                                                                                  G             O      T
                  A       A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T       E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H       L      B      L      P      E      S      G      I      W      A      T      R      X300       0.2500     9.0     9.0    7.0    9.0    7.0    9.0           6.0    9.0    7.5           7.5    6.5    7.0
       0.1250     9.0     8.5    5.0    9.0    8.5    9.0           2.0    9.0    7.0           5.0    4.8    7.0
       0.0620     9.0     7.0    3.0    5.5    7.0    9.0           1.0    8.5    6.3           4.3    4.3    6.5
       0.0320     9.0     6.0    1.5    4.0    4.5    7.0           1.0    2.0    6.0           2.8    3.5    5.5
       0.0160     9.0     6.0    1.5    4.0    3.0    6.0           0.5    2.0    5.0           1.8    2.8    6.0301       0.0620     9.0     4.0    9.0    9.0    9.0    9.0           0.0    1.0    5.5           1.0    3.5    5.0
       0.0320     9.0     3.0    4.0    4.0    4.0    9.0           0.0    1.0    5.5           0.5    3.5    4.5
       0.0160     9.0     2.0    0.0           2.0    9.0           0.0    0.0    5.0           0.5    3.5    3.5302       0.0620     9.0     9.0    1.0    9.0    3.0    9.0           0.0    9.0    7.5           2.0    4.5    4.5
       0.0320     9.0     9.0    0.0    9.0    4.0    9.0           0.0    3.0    7.0           1.5    4.0    4.5
       0.0160     9.0     5.0    0.0    6.0    1.0    9.0           0.0    0.0    5.0           1.0    3.0    4.0303       0.0620     9.0     9.0    3.0    9.0    7.0    9.0           0.0    8.0    7.5           2.0    3.5    5.0
       0.0320     9.0     3.0    1.0    4.0    3.0    9.0           0.0    4.0    7.5           1.5    3.5    4.5
       0.0160     9.0     3.0    0.0    4.0    0.0    9.0           0.0    0.0    7.0           1.0    3.0    4.5304       0.0620     9.0     7.0    1.0    9.0    2.0    9.0           1.0    4.0    6.0           2.0    3.0    5.0
       0.0320     9.0     6.0    0.0    6.0    2.0    6.0           0.0    1.0    5.5           1.5    2.5    5.0
       0.0160     9.0     4.0    0.0    4.0    1.0    3.0           1.0    0.0    5.0           1.0    2.0    4.5
                                                    表1(续)
                                                                                 G             O      T
                 A       A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率    T       E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)  H       L      B      L      P      E      S      G      I      W      A      T      R      X305      0.0620     9.0     7.0    2.0    7.0    7.0    9.0           1.0    5.0    6.5           2.5    4.5    5.0
      0.0320     9.0     7.0    1.0    9.0    4.0    6.0           1.0    1.0    6.0           1.5    2.5    5.0
      0.0160     9.0     6.0    0.0    4.0    2.0    1.0           0.0    0.0    4.0           0.0    2.0    3.5306      0.0620     9.0     5.0    1.0    5.0    3.0    9.0           2.0    3.0    6.5           2.5    5.0    6.5
      0.0320     9.0     2.0    0.0    2.0    1.0    4.0           1.0    1.0    5.5           2.5    4.0    5.5
      0.0160     9.0     1.0    0.0    1.0    1.0    3.0           1.0    0.0    5.0           1.5    2.5    5.0307      0.0620     9.0     9.0    7.0    9.0    9.0    9.0           3.0    6.0    9.0           3.0    4.0    6.0
      0.0320     6.2     9.0    6.0    5.0    9.0    9.0           3.0    4.0    9.0           3.0    4.0    5.5
      0.0160     6.4     9.0    3.0    3.0    5.0    9.0           3.0    3.0    6.5           1.5    3.0    5.5308      0.0620     9.0     9.0    9.0    9.0    9.0    9.0           7.0    7.0    9.0           4.5    4.5    6.5
      0.0320     6.4     9.0    6.0    9.0    9.0    9.0           3.0    5.0    8.0           3.5    3.5    6.0
      0.0160     5.6     9.0    2.0    4.0    7.0    9.0           1.0    1.0    6.0           2.5    3.0    5.0309      0.0620     9.0     9.0    7.0    9.0    9.0    9.0           2.0    9.0    9.0           4.0    4.0    6.0
      0.0320     9.0     9.0    5.0    9.0    9.0    9.0           3.0    3.0    8.0           2.5    3.5    6.0
      0.0160     9.0     9.0    1.0    3.0    6.0    9.0           1.0    3.0    8.5           2.0    3.0    5.0
                                                表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X310       0.0620     9.0    9.0    3.0    7.0    4.0    9.0           4.0    5.0    4.0           2.5    5.0    5.0
       0.0320     9.0    2.0    0.0    3.0    2.0    9.0           1.0    1.0    4.0           1.0    3.0    4.5
       0.0160     9.0    4.0    0.0    3.0    0.0    9.0           0.0    0.0    3.0           0.5    2.5    4.0311       0.0620     9.0    4.0    1.0    3.0    3.0    3.0           1.0    1.0    4.5           0.5    1.5    3.5
       0.0320     9.0    3.0    0.0    2.0    0.0    3.0           0.0    3.0    3.5           0.0    1.0    3.5
       0.0160     0.0    1.0    0.0    0.0    0.0    0.0           0.0    0.0    4.0           0.0    1.0    1.5312       0.0620     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.5    7.0    7.5
       0.0320     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           5.5    5.5    7.5
       0.0160     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           4.5    5.0    6.5313       0.0620     9.0    9.0    4.0    9.0    7.0    9.0           9.0    9.0    7.0           4.5    4.0    7.5
       0.0320     9.0    9.0    1.0    7.0    7.0    9.0           6.0    9.0    6.0           4.0    3.5    5.5
       0.0160     9.0    4.0    1.0    9.0    1.0    6.0           3.0    5.0    6.0           2.0    2.5    5.5314       0.0620     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.5    9.0    9.0
       0.0320     9.0    7.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           5.5    9.0    9.0
       0.0160     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           4.0    5.5    7.5
                                             表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X315       0.0620     9.0    9.0    1.0    9.0    8.0    9.0           7.0    9.0    9.0           6.0    5.5    7.5
       0.0320     9.0    7.0    0.0    9.0    5.0    7.0           3.0    6.0    7.0           4.5    5.0    7.0
       0.0160     4.0    5.0    0.0    5.0    5.0    4.0           0.0    4.0    6.0           1.5    4.0    6.5316       0.0620     9.0    9.0    3.0    9.0    9.0    9.0           9.0    9.0    8.5           6.0    5.5    5.5
       0.0320     9.0    9.0    1.0    9.0    9.0    9.0           9.0    9.0    8.5           6.0    5.0    5.5
       0.0160     9.0    9.0    0.0    9.0    5.0    9.0           9.0    9.0    8.0           6.5    4.5    6.0317       0.0620     9.0    9.0    2.0    9.0    9.0    9.0           2.0    9.0    9.0           5.0    5.0    7.0
       0.0320     9.0    9.0    0.0    4.0    9.0    9.0           0.0    9.0    8.5           4.0    4.5    7.0
       0.0160     9.0    9.0    0.0    3.0    9.0    9.0           0.0    9.0    7.5           3.0    3.5    6.0318       0.0620     9.0    9.0    3.0    8.0    9.0    9.0           0.0    9.0    8.5           5.0    5.0    6.0
       0.0320     9.0    9.0    2.0    9.0    4.0    9.0           0.0    6.0    8.5           4.0    3.5    5.0
       0.0160     9.0    5.0    0.0    3.0    4.0    9.0           0.0    5.0    8.0           2.5    3.0    4.0319       0.0620     9.0    9.0    5.0    6.0    8.0    9.0           7.0    9.0    8.5           6.5    6.5    7.0
       0.0320     9.0    9.0    1.0    6.0    8.0    9.0           6.0    9.0    8.5           5.5    5.5    7.0
       0.0160     9.0    2.0    1.0    5.0    6.0    9.0           4.0    7.0    7.5           6.0    5.0    6.5
                                                   表1(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X320       0.0620      9.0    9.0    1.0    9.0    9.0    9.0           7.0    9.0    7.5           7.0    6.5    7.0
       0.0320      9.0    7.0    1.0    6.0    7.0    9.0           4.0    9.0    8.5           5.5    5.5    7.0
       0.0160      9.0    4.0    1.0    7.0    6.0    9.0           3.0    4.0    7.5           5.5    5.0    6.5321       0.0620      9.0    9.0    6.0    9.0    8.0    9.0           0.0    6.0    7.5           4.0    4.5    4.5
       0.0320      9.0    9.0    4.0    9.0    7.0    9.0           0.0    5.0    7.0           4.0    4.5    4.5
       0.0160      9.0    9.0    2.0    9.0    5.0    9.0           0.0    3.0    7.0           3.5    4.5    4.5322       0.0620      9.0    3.0    0.0    1.0    1.0    9.0           0.0    0.0    6.5           2.0    3.0    4.5
       0.0320      7.0    1.0    0.0    0.0    0.0    8.0           0.0    0.0    5.0           1.5    1.5    3.5
       0.0160      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.0           1.0    1.0    3.5323       0.2500      9.0    9.0    5.0    9.0    9.0    9.0           9.0    9.0    8.5           8.5    5.5    8.0
       0.1250      9.0    9.0    4.0    9.0    8.0    9.0           9.0    9.0    7.3           6.8    5.5    7.5
       0.0620      9.0    9.0    1.0    8.0    8.0    9.0           9.0    9.0    7.0           6.5    6.5    7.5
       0.0320      7.3    9.0    1.0    5.0    7.0    9.0           7.0    9.0    7.0           6.0    5.0    7.0
       0.0160      6.6    9.0    1.0    3.0    5.0    9.0           6.0    5.0    6.5           5.0    5.0    7.0324       0.0620      9.0    9.0    7.0    9.0    7.0    9.0           3.0    9.0    9.0           7.0    6.0    8.0
       0.0320      9.0    9.0    6.0    9.0    6.0    9.0           0.0    8.0    8.5           5.5    5.0    7.5
       0.0160      9.0    9.0    6.0    9.0    3.0    9.0           0.0    4.0    7.0           2.5    4.0    5.0
                                                    表1(续)
                                                                                   G             O      T
                  A      A       C       C      G      I      I      E      S      L      G      R      R      Z
                  B      M       A       H      A      P      P      C      E      X      L      Y      Z      E
                  U      B       S       E      L      O      O      H      T      M      X      S      A      A化合物      施用率    T      E       O       A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L       B       L      P      E      S      G      I      W      A      T      R      X325       0.0620     9.0    9.0     9.0     9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.0320     9.0    5.0     9.0     9.0    9.0    9.0           9.0    9.0    9.0           8.0    8.0    9.0
       0.0160     9.0    4.0     2.0     9.0    6.0    9.0           9.0    9.0    8.0           8.0    7.5    9.0326       0.0620     9.0    9.0     4.0     9.0    6.0    9.0           9.0    9.0    9.0           6.5    7.5    8.0
       0.0320     9.0    9.0     3.0     9.0    6.0    9.0           9.0    9.0    9.0           6.0    7.5    8.0
       0.0160     9.0    4.0     0.0     9.0    6.0    9.0           8.0    9.0    8.0           3.5    6.0    8.0327       0.0620     9.0    9.0     3.0     9.0    5.0    9.0           0.0    8.0    8.0           3.0    4.0    5.0
       0.0320     9.0    9.0     1.0     9.0    4.0    9.0           0.0    6.0    8.0           3.0    4.0    4.5
       0.0160     9.0    6.0     1.0     5.0    2.0    7.0           0.0    3.0    6.5           1.5    3.0    4.5328       0.0620     9.0    7.0     1.0     9.0    7.0    9.0           0.0    3.0    7.0           3.5    4.0    5.0
       0.0320     9.0    3.0     0.0     9.0    4.0    9.0           0.0    3.0    7.0           3.5    4.0    5.0
       0.0160     9.0    3.0     0.0     9.0    2.0    4.0           0.0    0.0    4.5           3.5    3.5    4.5329       0.0620     9.0    7.0     4.0     6.0    6.0    9.0           2.0    5.0    7.0           5.0    5.0    5.0
       0.0320     9.0    6.0     1.0     6.0    5.0    9.0           1.0    1.0    6.5           3.0    3.0    4.5
       0.0160     9.0    6.0     1.0     3.0    1.0    3.0           1.0    1.0    6.0           2.0    2.0    4.5
                                                   表1(续)
                                                                                  G             O      T
                  A       A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T       E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H       L      B      L      P      E      S      G      I      W      A      T      R      X330      0.0620      9.0     6.0    1.0    4.0    2.0    9.0           1.0    1.0    6.5           3.0    3.0    4.5
      0.0320      9.0     4.0    1.0    2.0    1.0    9.0           2.0    1.0    5.5           2.0    2.5    2.5
      0.0160      1.0     2.0    0.0    1.0    1.0    1.0           1.0    0.0    4.5           2.0    2.0    2.5331      0.0620      8.0     2.0    0.0    4.0    2.0    9.0           0.0    0.0    5.0           1.5    3.0    4.5
      0.0320      4.0     0.0    0.0    2.0    1.0    9.0           0.0    0.0    4.0           0.5    3.0    4.0
      0.0160      3.0     0.0    0.0    0.0    0.0    6.0           0.0    0.0    3.5           0.0    2.0    3.5332      0.0620      9.0     9.0    4.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    8.0    8.5
      0.0320      9.0     9.0    4.0    9.0    9.0    9.0           9.0    9.0    9.0           6.5    7.5    8.5
      0.0160      9.0     9.0    3.0    9.0    9.0    9.0           9.0    9.0    9.0           3.5    6.0    7.5333      0.0620      9.0     9.0    9.0    9.0    5.0    9.0           0.0    7.0    7.0           2.5    4.5    5.0
      0.0320      9.0     9.0    2.0    5.0    4.0    9.0           0.0    7.0    7.0           2.5    4.0    4.5
      0.0160      9.0     9.0    2.0    3.0    2.0    9.0           0.0    3.0    6.5           2.0    3.5    4.5334      0.0620      9.0     7.0    2.0           2.0    9.0           3.0    7.0    6.5           3.5    4.0    5.5
      0.0320      9.0     6.0    1.0    4.0    1.0    9.0           1.0    2.0    5.0           2.5    3.5    4.5
      0.0160      9.0     2.0    1.0    4.0    1.0    7.0           0.0    1.0    4.0           2.5    3.5    3.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X335       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.1250     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.5    9.0
       0.0620     9.0    9.0    9.0           7.0    9.0           9.0    9.0    9.0           7.5    8.0    9.0
       0.0320     8.7    9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           7.5    8.0    9.0
       0.0160     8.4    9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           6.5    6.5    9.0336       0.0620     9.0    9.0    6.0           7.0    9.0           9.0    9.0    9.0           6.0    5.5    7.5
       0.0320     9.0    9.0    1.0    9.0    6.0    9.0           5.0    7.0    7.5           5.5    5.5    5.5
       0.0160     9.0    7.0    1.0           1.0    9.0           5.0    7.0    7.0           5.5    5.5    5.5337       0.0620     9.0    9.0    9.0           9.0    9.0           2.0    9.0    9.0           3.5    3.5    4.5
       0.0320     9.0    9.0    4.0    7.0    3.0    9.0           2.0    9.0    6.5           3.5    3.5    5.0
       0.0160     9.0    7.0    3.0    7.0    2.0    9.0           2.0    4.0    6.5           2.0    2.5    4.5338       0.0620     9.0    9.0    7.0    9.0    7.0    9.0           6.0    6.0    8.0           4.0    5.0    6.0
       0.0320     9.0    9.0    7.0    9.0    9.0    9.0           2.0    4.0    7.5           3.5    4.0    5.5
       0.0160     9.0    7.0    3.0    7.0    9.0    9.0           1.0    1.0    7.5           2.5    4.0    5.5339       0.0620     9.0    9.0    1.0           7.0    9.0           2.0    7.0    6.5           4.0    4.5    5.5
       0.0320     9.0    7.0    1.0    7.0    4.0    9.0           2.0    4.0    5.5           3.5    5.0    4.5
       0.0160     9.0    9.0    1.0    9.0    2.0    9.0           1.0    2.0    5.5           3.0    3.0    4.0
                                                   表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X340       0.0620     9.0    9.0    9.0           9.0    9.0           3.0    9.0    8.0           5.0    5.0    6.5
       0.0320     9.0    9.0    4.0    9.0    9.0    9.0           2.0    6.0    7.0           5.0    5.0    5.0
       0.0160     9.0    9.0    1.0    9.0    8.0    9.0           2.0    3.0    6.5           3.5    4.0    5.0341       0.0620     9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           6.0    6.5    8.0
       0.0320     7.9    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    6.5    8.0
       0.0160     7.4    9.0    2.0    7.0    4.0    9.0           9.0    9.0    8.5           5.0    5.0    7.5342       0.0620     9.0    7.0    2.0           2.0    9.0           1.0    1.0    5.5           4.5    5.0    5.5
       0.0320     9.0    5.0    1.0    7.0    2.0    9.0           1.0    1.0    5.0           3.5    3.5    5.0
       0.0160     9.0    4.0    1.0    4.0    1.0    6.0           1.0    1.0    4.5           3.0    3.5    4.5343       0.0620     9.0    9.0    4.0           1.0    9.0           9.0    9.0    7.5           5.5    5.5    7.0
       0.0320     9.0    9.0    1.0    9.0    1.0    9.0           9.0    9.0    5.5           4.5    4.5    5.0
       0.0160     9.0    9.0    1.0    9.0    1.0    9.0           9.0    1.0    5.5           3.5    4.5    5.0344       0.0620     9.0    9.0    9.0           9.0    9.0           9.0    9.0    9.0           6.5    6.0    7.5
       0.0320     9.0    9.0    7.0    9.0    7.0    9.0           9.0    9.0    7.0           6.0    6.0    5.0
       0.0160     9.0    9.0    2.0    9.0    3.0    9.0           7.0    9.0    6.5           4.5    5.0    5.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X345       0.0620     9.0    9.0    9.0    9.0    4.0    9.0           3.0    9.0    8.5           5.0    6.0    6.0
       0.0320     9.0    7.0    9.0    9.0    4.0    9.0           0.0    9.0    7.5           3.0    4.0    4.5
       0.0160     9.0    4.0    4.0    9.0    3.0    9.0           0.0    4.0    6.0           3.5    3.5    2.0346       0.0620     7.0    7.0                  7.0           7.0    9.0    9.0    6.0           3.0    4.0    2.0347       0.0620     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.0320     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    9.0    9.0
       0.0160     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    9.0           8.0    9.0    9.0348       0.0620     9.0    9.0           9.0    9.0    9.0           9.0    9.0    8.0           9.0    9.0    9.0
       0.0320     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.0           5.0    9.0    9.0
       0.0160     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.0           4.0    8.0    9.0349       0.0620     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.5    9.0
       0.0320     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    9.0           8.5    8.5    6.5
       0.0160     9.0    9.0    0.0    7.0    4.0    9.0           9.0    9.0    7.5           8.5    8.5    8.0350       0.0620     9.0    9.0    9.0    9.0    9.0    9.0           3.0    9.0    9.0           4.5    4.0    6.0
       0.0320     9.0    9.0    4.0    9.0    9.0    9.0           0.0    9.0    9.0           3.0    3.5    5.0
       0.0160     9.0    9.0    3.0    8.0    9.0    9.0           0.0    6.0    7.0           1.5    2.5    3.0
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物      施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X351       0.0620     9.0    9.0    9.0    9.0    7.0    9.0           2.0    9.0    9.0           4.0    4.0    5.0
       0.0320     9.0    9.0    4.0    7.0    6.0    9.0           0.0    4.0    8.0           3.5    3.5    4.5
       0.0160     9.0    9.0    2.0    4.0    6.0    9.0           0.0           7.0           0.5    1.5    3.5352       0.0620     9.0    9.0    2.0    9.0    2.0    9.0           2.0    2.0    9.0           6.0    3.5    7.5
       0.0320     9.0    9.0    0.0    9.0    2.0    9.0           0.0    0.0    9.0           2.0    2.5    7.5
       0.0160     9.0    9.0    0.0    9.0    0.0    9.0           0.0    0.0    8.0           1.5    2.5    7.5353       0.1250     9.0    7.0    5.0    7.0    7.0    9.0           3.0    7.0    8.0           4.5    4.5    7.5
       0.0620     9.0    9.0    3.0    7.0    2.0    9.0           2.0    6.0    7.0           4.0    4.0    7.0
       0.0320     9.0    7.0    1.0    7.0    2.0    9.0           2.0    1.0    6.5           3.5    3.5    6.0
       0.0160     6.0    4.0    1.0    3.0    1.0    7.0           1.0    1.0    5.5           3.5    3.5    5.0354       0.1250     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    9.0    8.0
       0.0620     9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    9.0           8.0    8.0    8.0
       0.0320     9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           7.0    7.0    6.5
       0.0160     9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           6.0    6.0    6.0355       0.1250     9.0    7.0    4.0    9.0    6.0    9.0           9.0    9.0    6.0           6.5    5.5    5.5
       0.0620     9.0    9.0    2.0    9.0    3.0    9.0           9.0    7.0    6.5           6.0    5.5    5.0
       0.0320     9.0    9.0    3.0    2.0    1.0    7.0           7.0    7.0    5.5           4.5    5.5    4.5
       0.0160     9.0    9.0    1.0    4.0    1.0    9.0           4.0    1.0    4.0           4.5    5.0    5.0
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X356       0.1250     9.0    9.0    7.0    9.0    1.0    9.0           4.0    3.0    9.0           4.5    4.5    8.0
       0.0620     9.0    9.0    9.0    9.0    1.0    9.0           3.0    3.0    8.0           4.0    4.0    7.5
       0.0320     9.0    9.0    1.0    7.0    2.0    9.0           2.0    3.0    9.0           3.0    3.5    7.5
       0.0160     9.0    9.0    1.0    9.0    1.0    9.0           1.0    1.0    7.5           2.5    3.0    7.5357       0.1250     9.0    9.0    4.0    9.0    4.0    9.0           5.0    7.0    9.0           5.0    5.0    7.5
       0.0620     9.0    9.0    1.0    9.0    1.0    9.0           1.0    2.0    9.0           3.0    4.5    7.5
       0.0320     9.0    9.0    1.0    7.0    1.0    9.0           2.0    3.0    7.5           3.0    4.0    7.5
       0.0160     9.0    9.0    1.0    9.0    0.0    9.0           1.0    1.0    6.0           2.5    2.5    6.5358       0.1250     9.0    9.0    3.0    4.0    3.0    9.0           0.0    0.0    5.5           1.5    3.5    5.0
       0.0620     9.0    9.0    0.0    3.0    0.0    9.0           0.0    0.0    4.0           1.0    3.5    4.5
       0.0320     9.0    4.0    0.0    1.0    0.0    9.0           0.0    0.0    3.5           1.0    3.0    3.5
       0.0160     9.0    4.0    0.0    0.0    0.0    5.0           0.0    0.0    3.5           0.5    2.5    3.5359       0.1250     9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           8.5    9.0    9.0
       0.0620     9.0    9.0    9.0    9.0    7.7    9.0           9.0    9.0    8.1           8.7    9.0    9.0
       0.0320     9.0    9.0    8.3    9.0    6.3    9.0           8.3    9.0    8.0           8.0    8.9    9.0
       0.0160     9.0    9.0    6.7    9.0    6.0    9.0           9.0    9.0    7.0           6.9    7.9    8.1
                                                   表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X360       0.1250     9.0    9.0    3.0    9.0    3.0    9.0           0.0    3.0    9.0           3.5    4.5    6.5
       0.0620     9.0    9.0    0.0    3.0    3.0    9.0           0.0    0.0    6.5           2.5    4.5    5.5
       0.0320     9.0    4.0    0.0    2.0    1.0    9.0           0.0    0.0    5.0           2.0    4.0    4.5
       0.0160     9.0    0.0    0.0    0.0    0.0    3.0           0.0    0.0    4.0           1.5    3.5    4.0361       0.1250     9.0    3.0    3.0    9.0    4.0    9.0           0.0    0.0    6.5           3.0    4.0    5.0
       0.0620     9.0    2.0    3.0    7.0    3.0    9.0           0.0    0.0    5.0           1.5    3.0    4.0
       0.0320     9.0    2.0    0.0    3.0    0.0    7.0           0.0    0.0    3.5           2.0    3.0    4.0
       0.0160     9.0    2.0    0.0    2.0    0.0    1.0           0.0    0.0    3.5           1.5    3.0    4.0362       0.2500     9.0    9.0    3.0    9.0    9.0    9.0           9.0    9.0    9.0           7.5    6.5    8.0
       0.1250     9.0    9.0    1.0    9.0    5.0    9.0           9.0    9.0    8.0           7.5    5.5    8.0
       0.0620     9.0    9.0    1.0    9.0    3.0    9.0           9.0    8.0    8.0           7.0    5.0    7.5
       0.0320     9.0    9.0    6.0    9.0    3.0    9.0           8.0    8.0    8.0           5.5    4.0    7.5
       0.0160     9.0    9.0    0.0    9.0    1.0    9.0           5.0    4.0    7.5           5.0    4.0    7.5363       0.1250     9.0    9.0    0.0    2.0    5.0    9.0           0.0    0.0    4.5           1.0    3.5    3.0
       0.0620     9.0    7.0    0.0    0.0    5.0    3.0           0.0    0.0    4.5           0.0    2.0    3.0
       0.0320     5.0    3.0    0.0    0.0    0.0    2.0           0.0    0.0    4.0           0.0    1.0    2.0
       0.0160     4.0    0.0    0.0    0.0    0.0    1.0           0.0    0.0    3.0           0.0    0.5    2.0
                                                     表1(续)
                                                                                     G             O       T
                  A       A       C       C      G       I      I      E      S      L      G      R       R       Z
                  B       M       A       H      A       P      P      C      E      X      L      Y       Z       E
                  U       B       S       E      L       O      O      H      T      M      X      S       A       A化合物    施用率      T       E       O       A      A       H      S      C      V      A      M      A       W       M编号   (公斤/公顷)   H       L       B       L      P       E      S      G      I      W      A      T       R       X364      0.2500      9.0     9.0     2.0     9.0    9.0     9.0           2.0    3.0    7.0           4.0     4.5     5.0
      0.1250      9.0     9.0     2.0     9.0    8.0     9.0           0.0    1.0    7.0           3.0     4.5     5.0
      0.0620      9.0     9.0     0.0     8.0    7.0     9.0           0.0    0.0    6.0           2.0     3.5     5.0
      0.0320      9.0     9.0     0.0     6.0    4.0     9.0           0.0    0.0    5.5           2.0     3.0     4.5
      0.0160      9.0     4.0     0.0     4.0    2.0     9.0           0.0    0.0    5.5           2.0     2.5     4.5365      0.2500      9.0     9.0     6.0     9.0    9.0     9.0           5.0    9.0    8.5           5.5     6.0     7.0
      0.1250      9.0     9.0     2.0     7.0    6.0     9.0           0.0    5.0    8.0           5.0     5.0     5.5
      0.0620      9.0     9.0     1.0     7.0    4.0     9.0           0.0    0.0    8.0           3.0     4.0     5.0
      0.0320      9.0     2.0     0.0     7.0    2.0     9.0           0.0    0.0    6.0           2.0     3.0     5.0
      0.0160      9.0     1.0     0.0     4.0    1.0     9.0           0.0    0.0    5.5           1.5     3.0     5.0366      0.2500      9.0     9.0     9.0     9.0    9.0     9.0           8.0    9.0    9.0           7.5     7.0     7.5
      0.1250      9.0     9.0     8.5     9.0    9.0     9.0           8.0    9.0    9.0           7.0     6.8     7.3
      0.0620      9.0     9.0     5.5     9.0    8.5     9.0           7.0    9.0    9.0           5.8     5.3     6.5
      0.0320      9.0     9.0     5.0     9.0    6.0     9.0           3.5    9.0    8.5           4.5     4.0     5.3
      0.0160      9.0     9.0     3.5     9.0    7.5     9.0           2.5    6.0    7.8           3.0     3.0     4.8
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X367      0.0620      9.0    9.0    1.0    9.0    2.0    9.0           4.0    9.0    8.5           5.0    5.0    7.0
      0.0320      9.0    7.0    1.0    5.0    2.0    9.0           3.0    9.0    7.5           5.0    4.5    7.0
      0.0160      9.0    4.0    1.0    5.0    2.0    9.0           2.0    4.0    7.0           5.0    4.5    6.5368      0.0620      9.0    9.0    2.0    7.0    4.0    9.0           2.0    2.0    7.5           4.0    4.0    5.5
      0.0320      7.0    7.0    2.0    4.0    4.0    9.0           2.0    1.0    5.5           3.0    4.0    5.0
      0.0160      7.0    4.0    1.0    3.0    4.0    9.0           1.0    0.0    4.5           2.5    3.0    4.0369      0.1250                                                                     8.0           4.0    4.0    6.0
      0.0620      9.0    9.0    4.0    9.0    5.0    9.0           2.0    3.0    6.5           4.0    4.0    5.0
      0.0320      6.2    7.0    1.0    9.0    3.0    9.0           2.0    1.0    6.0           3.0    4.0    4.5
      0.0160      5.2    6.0    0.0    1.0    2.0    9.0           2.0    0.0    5.5           3.0    3.5    4.0370      0.0620      9.0    9.0    1.0    9.0    2.0    9.0           9.0    9.0    9.0           5.0    4.5    7.5
      0.0320      9.0    9.0    1.0    9.0    1.0    9.0           4.0    7.0    9.0           4.5    4.0    7.5
      0.0160      7.0    1.0    0.0    2.0    1.0    9.0           1.0    1.0    8.0           4.0    4.0    7.0371      0.0620      9.0    7.0    1.0    2.0    2.0    9.0           1.0    1.0    4.5           2.5    3.5    4.0
      0.0320      4.0    4.0    0.0    0.0    1.0    3.0           0.0    0.0    3.0           1.5    2.5    2.5
      0.0160      1.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.5           1.0    1.5    1.0
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X372       0.1250     9.0    9.0    9.0    9.0    6.0    9.0           3.0    9.0    8.5           6.5    6.0    7.0
       0.0620     9.0    9.0    5.0    9.0    3.0    9.0           3.0    7.0    8.5           5.5    5.0    5.5
       0.0320     9.0    9.0    3.0    9.0    3.0    9.0           2.0    7.0    8.5           4.5    4.5    4.5
       0.0160     9.0    6.0    2.0    9.0    1.0    9.0           1.0    4.0    7.0           4.0    4.0    4.5373       0.0620     9.0    9.0    0.0    4.0    8.0    9.0           3.0    6.0    7.0           0.5    3.0    7.0
       0.0320     9.0    7.0    0.0    3.0    3.0    9.0           3.0    6.0    7.0           0.5    3.0    7.0
       0.0160     7.0    4.0    0.0    3.0    1.0    9.0           0.0    2.0    7.0           0.5    2.0    5.0374       0.0620     9.0    9.0    3.0    5.0    7.0    9.0           0.0    3.0    9.0           2.0    3.0    5.0
       0.0320     9.0    4.0    0.0    3.0    4.0    9.0           0.0    0.0    9.0           1.0    3.0    5.0
       0.0160     9.0    3.0    0.0    2.0    4.0    9.0           0.0    0.0    5.5           0.5    2.5    5.0375       0.0620     9.0    9.0    5.0    9.0    3.0    9.0           2.0    9.0    8.5           2.5    4.5    5.0
       0.0320     9.0    7.0    5.0    5.0    3.0    9.0           0.0    7.0    8.5           1.5    4.5    5.0
       0.0160     9.0    3.0    0.0    4.0    3.0                  0.0    2.0    5.0           1.0    3.0    5.0376       0.0620     9.0    9.0    0.0    1.0    4.0    9.0           0.0    0.0    7.5           1.0    3.5    3.0
       0.0320     9.0    3.0    0.0    0.0    2.0    9.0           0.0    0.0    5.0           0.5    3.0    2.0
       0.0160     4.0    0.0    0.0    0.0    0.0    3.0           0.0    0.0    3.5           0.0    2.0    1.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X377      0.0620      9.0    9.0    7.0    9.0    5.0    9.0           2.0    6.0    8.5           1.5    4.0    5.0
      0.0320      9.0    9.0    3.0    9.0    5.0    9.0           0.0    3.0    7.5           1.0    4.0    5.0
      0.0160      9.0    9.0    1.0    9.0    2.0    9.0           0.0    2.0    7.5           1.0    3.5    5.0378      0.0620      9.0    9.0    7.0    9.0    9.0    9.0           8.0    8.0    9.0           6.0    6.0    7.5
      0.0320      9.0    9.0    6.5    9.0    9.0    9.0           7.5    9.0    9.0           7.5    6.0    6.5
      0.0160      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    9.0           7.5    6.0    6.0379      0.0320      9.0    9.0    4.0    9.0    7.0    9.0           0.0    4.0    9.0           2.0    3.5    5.0
      0.0160      9.0    9.0    1.0    4.0    4.0    9.0           0.0    2.0    7.5           0.5    3.0    4.5380      0.1250      9.0    9.0    9.0    9.0    7.0    9.0           6.0    9.0    8.5           4.5    4.5    5.0
      0.0620      9.0    9.0    7.0    9.0    4.0    9.0           1.0    6.0    6.0           4.0    4.5    5.0
      0.0320      9.0    9.0    6.0    7.0    4.0    9.0           3.0    9.0    5.5           3.5    4.5    4.5
      0.0160      9.0    9.0    4.0    5.0    1.0    9.0           1.0    1.0    5.5           3.5    4.0    4.5381      0.0620      9.0    9.0    3.0    0.0    3.0    9.0           0.0    0.0    5.0           2.0    2.5    5.0
      0.0320      9.0    8.0    0.0    0.0    3.0    9.0           0.0    0.0    5.0           1.0    2.0    4.0
      0.0160      4.0    3.0    0.0    0.0    0.0    3.0           0.0    0.0    4.0           0.0    1.5    4.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X382       0.0620     9.0    9.0    2.0    2.0    3.0    9.0           0.0   0.0     7.0           1.5    2.5    4.5
       0.0320     9.0    4.0    0.0    1.0    1.0    9.0           0.0   0.0     5.0           0.5    2.5    3.5
       0.0160     4.0    0.0    0.0    0.0    0.0    3.0           0.0   0.0     4.0           0.0    1.5    2.5383       0.0620     9.0    9.0    2.0    9.0    9.0    9.0           9.0   9.0     8.0           6.5    5.5    8.5
       0.0320     9.0    9.0    2.0    9.0    4.0    9.0           9.0   9.0     7.5           5.0    5.0    8.0
       0.0160     9.0    9.0    0.0    9.0    3.0    9.0           9.0   9.0     7.5           3.5    4.0    7.5384       0.0620     9.0    9.0    3.0    9.0    9.0    9.0           9.0   9.0     8.5           6.5    5.5    8.0
       0.0320     9.0    9.0    3.0    5.0    7.0    9.0           5.0   7.0     8.5           5.5    5.0    8.0
       0.0160     9.0    9.0    1.0    4.0    4.0    9.0           5.0   4.0     8.0           4.5    4.5    7.5385       0.0620     9.0    9.0    3.0    7.0    7.0    9.0           9.0   9.0     9.0           4.0    5.5    8.0
       0.0320     9.0    9.0    0.0    7.0    5.0    9.0           5.0   9.0     9.0           3.5    5.5    8.0
       0.0160     9.0    4.0    0.0    3.0    3.0    9.0           2.0   3.0     8.0           2.0    4.0    8.0386       0.0620     9.0    9.0    3.0    7.0    7.0    9.0           7.0   9.0     9.0           5.0    6.0    8.0
       0.0320     9.0    9.0    0.0    5.0    9.0    9.0           7.0   9.0     9.0           4.0    5.5    8.0
       0.0160     9.0    6.0    0.0    1.0    9.0    9.0           3.0   9.0     7.5           2.5    4.0    7.5
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物      施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X387        0.0620    9.0    9.0    2.0    5.0    9.0    9.0           5.0    9.0    9.0           4.5    5.5    8.0
        0.0320    9.0    9.0    1.0    4.0    3.0    9.0           4.0    5.0    8.5           3.5    5.0    7.5
        0.0160    9.0    7.0    0.0    2.0    3.0    9.0           4.0    5.0    7.5           2.0    4.5    7.5388        0.0620    9.0    9.0    5.0    9.0    6.0    9.0           9.0    9.0    9.0           4.5    6.5    6.0
        0.0320    9.0    7.0    2.0    9.0    4.0    9.0           5.0    5.0    7.5           3.0    5.5    5.5
        0.0160    8.0    3.0    1.0    3.0    3.0    9.0           1.0    5.0    7.5           1.5    4.0    5.0389        0.0620    9.0    9.0    3.0    9.0    9.0    9.0           5.0    9.0    8.5           5.0    5.5    8.0
        0.0320    9.0    9.0    2.0    4.0    6.0    9.0           2.0    8.0    8.5           4.5    5.0    8.5
        0.0160    9.0    9.0    0.0    2.0    4.0    9.0           0.0    2.0    8.0           3.0    4.5    6.0390        0.1250    9.0    9.0    9.0    9.0    8.0    9.0           4.0    9.0    9.0           4.5    5.0    5.5
        0.0620    9.0    9.0    6.0    9.0    7.0    9.0           3.0    7.0    9.0           4.5    4.5    5.5
        0.0320    9.0    9.0    5.0    9.0    4.0    9.0           2.0    6.0    8.5           3.5    4.0    4.5
        0.0160    9.0    9.0    6.0    9.0    7.0    9.0           2.0    4.0    8.0           3.5    3.5    4.5391        0.1250    9.0    9.0    3.0    9.0    1.0    9.0           7.0    9.0    6.5           3.5    4.5    7.0
        0.0620    9.0    9.0    1.0    9.0    1.0    9.0           7.0    7.0    6.5           2.5    3.5    7.0
        0.0320    9.0    9.0    1.0    9.0    1.0    9.0           4.0    6.0    6.5           2.5    3.0    7.0
        0.0160    9.0    9.0    1.0    9.0    1.0    9.0           4.0    2.0    6.0           2.5    2.5    6.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X392      0.0620      9.0    9.0    3.0    9.0    4.0    9.0           1.0    3.0    7.5           2.5    4.5    6.0
      0.0320      9.0    9.0    2.0    9.0    3.0    9.0           0.0    3.0    6.5           2.0    3.5    5.5
      0.0160      9.0    3.0    0.0    7.0    3.0    9.0           0.0    0.0    5.5           2.0    3.5    5.0393      0.0620      9.0    9.0    3.0    9.0    4.0    9.0           2.0    3.0    8.0           2.5    5.0    6.0
      0.0320      9.0    9.0    1.0    9.0    3.0    9.0           1.0    1.0    7.0           2.0    4.5    5.5
      0.0160      9.0    9.0    0.0    9.0    1.0    5.0           0.0    0.0    7.0           1.5    4.0    4.5394      0.0620      9.0    9.0    1.0    9.0    5.0    9.0           0.0    1.0    8.0           2.5    5.0    6.0
      0.0320      9.0    8.0    0.0    9.0    3.0    9.0           0.0    0.0    7.5           2.0    4.5    5.0
      0.0160      9.0    4.0    0.0    5.0    0.0    7.0           0.0    0.0    7.0           1.5    4.0    5.0395      0.0620      9.0    9.0    3.0    9.0    5.0    9.0           7.0    5.0    6.5           6.0    5.0    8.0
      0.0320      9.0    9.0    3.0    9.0    2.0    9.0           4.0    3.0    7.0           5.5    5.0    8.0
      0.0160      9.0    9.0    0.0    9.0    0.0    9.0           2.0    3.0    6.0           2.0    3.5    7.5396      0.0620      9.0    9.0    2.0    9.0    4.0    9.0           3.0    5.0    8.5           6.5    7.0    6.0
      0.0320      9.0    9.0    2.0    9.0    4.0    9.0           2.0    5.0    7.5           6.5    7.0    5.5
      0.0160      9.0    9.0    0.0    9.0    3.0    9.0           0.0    0.0    6.5           3.5    6.5    5.5
                                                 表1(续)
                                                                                 G             O      T
                 A      A      C      C      G      I      I       E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P       C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O       H      T      M      X      S      A      A化合物     施用率    T      E      O      A      A      H      S       C      V      A      M      A      W      M编号    (公斤/公顷) H      L      B      L      P      E      S       G      I      W      A      T      R      X397       0.0620    9.0    9.0    9.0    9.0    5.0    9.0            1.0    3.0    9.0           8.0    7.5    6.0
       0.0320    9.0    9.0    9.0    9.0    4.0    9.0            1.0    2.0    9.0           6.0    6.5    6.0
       0.0160    9.0    9.0    0.0    9.0    1.0    9.0            0.0    0.0    7.5           4.5    5.5    5.5398       0.0620    9.0    9.0    1.0    9.0    6.0    9.0            1.0    3.0    7.5           1.5    4.0    5.5
       0.0320    9.0    4.0    0.0    9.0    3.0    9.0            1.0    2.0    7.5           1.5    4.0    5.0
       0.0160    9.0    4.0    0.0    9.0    0.0    5.0            1.0    2.0    5.5           1.5    3.5    4.5399       0.0620    9.0    8.0    1.0    9.0    3.0    9.0            0.0    2.0    7.0           2.0    4.0    5.5
       0.3220    9.0    4.0    0.0    8.0    0.0    9.0            0.0    2.0    7.0           1.0    3.5    5.0
       0.0160    8.0    2.0    0.0    5.0    0.0    7.0            0.0    0.0    5.0           1.0    3.5    4.5400       0.0620    9.0    9.0    1.0    9.0    4.0    9.0            1.0    3.0    7.0           2.5    4.0    5.5
       0.0320    9.0    4.0    0.0    4.0    2.0    9.0            0.0    0.0    6.5           1.0    3.5    5.0
       0.0160    8.0    3.0    0.0    0.0    0.0    5.0            0.0    0.0    5.5           1.0    3.5    5.0401       0.0620    9.0    7.0    1.0    9.0    3.0    9.0            2.0    2.0    5.0           3.0    4.0    5.0
       0.0320    9.0    7.0    1.0    6.0    3.0    9.0            3.0    2.0    5.0           2.5    3.0    5.0
       0.0160    7.0    7.0    0.0    3.0    1.0    7.0            2.0    2.0    5.0           3.0    3.0    4.5
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X402       0.0620    9.0    9.0    1.0    7.0    6.0    9.0           2.0    1.0    5.0           3.5    3.5    5.0
       0.0320    9.0    7.0    0.0    3.0    1.0    6.0           3.0    0.0    5.0           3.0    3.0    4.5
       0.0160    9.0    2.0    0.0    2.0    0.0    9.0           2.0    0.0    4.0           2.5    3.0    4.0403       0.0620    9.0    5.0    0.0    9.0    3.0    9.0           2.0    4.0    8.0           2.0    4.5    4.0
       0.3220    9.0    2.0    0.0    4.0    2.0    9.0           0.0    0.0    7.0           1.0    3.5    4.0
       0.0160    5.0    0.0    0.0    3.0    0.0    4.0           0.0    0.0    5.0           0.0    3.0    2.5404       0.0620    9.0    9.0    2.0    9.0    3.0    9.0           7.0    6.0    7.0           4.0    4.5    5.0
       0.0320    9.0    7.0    2.0    9.0    2.0    9.0           5.0    2.0    7.0           3.0    3.5    4.5
       0.0160    9.0    6.0    1.0    9.0    1.0    9.0           3.0    2.0    7.0           2.5    3.0    4.0405       0.0620    9.0    9.0    4.0    6.0    2.0    9.0           5.0    6.0    8.0           5.0    5.5    8.0
       0.0320    9.0    9.0    1.0    6.0    1.0    9.0           4.0    3.0    7.5           5.0    5.5    7.5
       0.0160    9.0    9.0    1.0    3.0    1.0    7.0           2.0    2.0    6.5           3.5    4.5    7.0406       0.0620    9.0    9.0    6.0    9.0    3.0    9.0           7.0    7.0    9.0           5.0    5.5    8.0
       0.0320    9.0    9.0    6.0    9.0    2.0    9.0           9.0    7.0    7.0           3.5    4.5    8.0
       0.0160    9.0    7.0    4.0    9.0    1.0    9.0           7.0    9.0    7.0           3.0    3.5    7.0
                                                 表1(续)
                                                                                G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X407       0.0620     9.0    9.0    0.0    4.0    4.0    9.0           1.0    2.0    6.0           3.5    5.5    5.0
       0.0320     9.0    9.0    0.0    3.0    2.0    9.0           0.0    0.0    5.5           3.0    5.0    4.5
       0.0160     7.0    3.0    0.0    2.0    2.0    5.0           0.0    0.0    5.5           2.5    4.5    4.5408       0.0620     9.0    7.0    2.0    7.0    3.0    9.0           3.0    9.0    8.0           5.5    5.5    7.5
       0.0320     7.0           0.0    4.0    1.0    9.0           2.0    5.0    7.5           3.0    5.0    5.5
       0.0160     7.0    1.0    0.0    3.0    0.0    7.0           2.0    2.0    6.5           2.5    4.5    3.5409       0.0620     9.0    9.0    2.0    9.0    7.0    9.0           3.0    7.0    8.0           6.0    6.0    7.5
       0.0320     9.0    9.0    0.0    4.0    3.0    9.0           1.0    4.0    7.5           3.5    5.0    7.0
       0.0160     9.0    4.0    0.0    4.0    0.0    9.0           0.0    0.0    5.5           3.5    4.0    4.5410       0.0620     9.0    4.0    0.0    9.0    4.0    9.0           3.0    6.0    7.5           5.5    5.5    7.5
       0.0320     9.0    3.0    0.0    4.0    4.0    9.0           2.0    4.0    7.5           4.5    5.0    5.5
       0.0160     9.0    2.0    0.0    3.0    3.0    9.0           1.0    3.0    7.0           4.0    4.5    4.5411       0.0620     9.0    9.0    7.0    7.0    6.0    9.0           7.0    9.0    8.5           5.5    5.5    7.5
       0.0320     9.0    9.0    4.0    7.0    4.0    9.0           8.0    9.0    8.5           5.0    5.0    7.0
       0.0160     9.0    4.0    3.0    4.0    3.0    9.0           2.0    3.0    8.5           4.0    3.5    6.5
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X412       0.0620     9.0    9.0    4.0    7.0   6.0     9.0           6.0    7.0    7.0           6.0    5.5    7.0
       0.0320     9.0    9.0    3.0    7.0   4.0     9.0           5.0    5.0    6.5           4.0    4.0    7.0
       0.0160     4.0    9.0    1.0    2.0   1.0     9.0           4.0    2.0    5.0           3.0    3.0    5.0413       0.0620     9.0    9.0    5.0    9.0   5.0     9.0           4.0    4.0    7.5           4.0    4.0    5.5
       0.0320     9.0    9.0    3.0    9.0   4.0     9.0           3.0    4.0    7.0           3.5    3.5    5.0
       0.0160     9.0    9.0    1.0    7.0   4.0     9.0           2.0    2.0    5.5           3.5    3.5    5.0414       0.0620     9.0    9.0    7.0    7.0   7.0     9.0           2.0    2.0    7.0           3.5    3.5    5.5
       0.0320     9.0    9.0    2.0    7.0   6.0     9.0           2.0    2.0    6.0           3.0    3.0    5.5
       0.0160     9.0    7.0    1.0    4.0   2.0     7.0           2.0    1.0    6.0           3.0    3.5    5.5415       0.0620     9.0    9.0    6.0    9.0   6.0     9.0           4.0    5.0    6.5           3.5    4.0    5.5
       0.0320     9.0    9.0    2.0    4.0   4.0     9.0           3.0    4.0    7.0           3.5    3.5    5.5
       0.0160     9.0    9.0    1.0    7.0   3.0     9.0           2.0    1.0    6.0           2.5    2.5    5.5416       0.0620     9.0    9.0    4.0    9.0   5.0     9.0           3.0    9.0    7.5           4.5    5.0    5.5
       0.0320     9.0    9.0    3.0    9.0   4.0     9.0           3.0    7.0    7.0           4.0    4.0    5.0
       0.0160     9.0    9.0    2.0    7.0   3.0     9.0           2.0    2.0    7.0           3.5    3.5    5.0417       0.0620     9.0    7.0    4.0    7.0   4.0     9.0           7.0    7.0    7.5           4.5    4.5    6.0
       0.0320     6.0    5.0    1.0    4.0   3.0     9.0           4.0    4.0    7.0           3.5    3.5    6.0
       0.0160     4.0    4.0    1.0    2.0   1.0     3.0           1.0    1.0    7.0           2.5    2.0    5.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X418       0.0620     9.0    9.0    1.0    7.0    1.0    9.0           3.0    9.0    7.5           4.5    4.5    6.0
       0.0320     9.0    9.0    0.0    4.0    0.0    9.0           2.0    3.0    6.0           3.5    3.5    5.0
       0.0160     9.0    3.0    0.0    2.0    0.0    9.0           1.0    1.0    4.5           3.0    3.0    5.0419       0.0620     9.0    9.0    1.0    7.0    3.0    9.0           3.0    4.0    5.5           5.0    5.0    5.5
       0.0320     9.0    4.0    0.0    3.0    0.0    7.0           1.0    1.0    5.0           4.0    4.0    5.0
       0.0160     2.0    1.0    0.0    1.0    0.0    9.0           0.0    0.0    4.5           3.0    3.5    5.0420       0.0620     9.0    9.0    9.0    9.0    4.0    9.0           9.0    8.0    7.5           5.0    4.5    7.5
       0.0320     9.0    9.0    3.0    9.0    3.0    9.0           3.0    2.0    6.5           4.0    4.0    7.5
       0.0160     9.0    9.0    3.0    9.0    2.0    9.0           1.0    1.0    5.0           3.5    3.5    6.5421       0.0620     9.0    9.0    1.0    9.0    9.0    9.0           5.0    4.0    9.0           3.5    3.5    6.5
       0.0320     9.0    9.0    0.0    4.0    1.0    9.0           4.0    2.0    8.5           4.0    3.5    6.0
       0.0160     2.0    1.0    0.0    1.0    1.0    9.0           1.0    2.0    4.5           3.0    3.0    5.5422       0.0620     9.0    9.0    3.0    9.0    9.0    9.0           5.0    9.0    9.0           5.5    5.5    7.0
       0.0320     9.0    9.0    3.0    8.0    6.0    9.0           4.0    9.0    8.0           5.5    5.5    6.0
       0.0160     9.0    9.0    1.0    4.0    5.0    9.0           1.0    6.0    7.5           4.5    4.5    6.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X423       0.0620     9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    9.0           7.5    9.0    7.5
       0.0320     9.0    9.0    6.0    9.0    8.0    9.0           3.0    7.0    9.0           7.5    8.5    6.5
       0.0160     9.0    9.0    9.0    9.0    4.0    9.0           2.0    6.0    8.0           5.0    6.0    5.5424       0.0620     9.0    6.0    1.0    5.0    2.0    9.0           4.0    5.0    5.5           2.5    3.0    4.5
       0.0320     9.0    6.0    1.0    4.0    2.0    9.0           2.0    1.0    4.0           2.5    3.0    3.5
       0.0160     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.0           1.5    1.5    3.5425       0.0620     9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    7.0           8.0    8.5    9.0
       0.0320     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    6.5           7.0    7.5    7.5
       0.0160     9.0    9.0    2.0    3.0    4.0    9.0           0.0    2.0    6.0           7.0    7.5    7.0426       0.0620     9.0    7.0    1.0    2.0    0.0    8.0           1.0    0.0    4.0           3.5    4.0    5.0
       0.0320     9.0    3.0    0.0    0.0    0.0    9.0           0.0    0.0    2.5           2.5    3.5    4.5
       0.0160     7.0    0.0    0.0    0.0    0.0    5.0           0.0    0.0    2.5           2.5    3.0    3.5427       0.0620     9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    9.0           7.0    7.0    8.5
       0.0320     9.0    9.0    9.0    5.0    0.0    9.0           9.0    9.0    9.0           5.5    6.0    8.5
       0.0160     9.0    9.0    9.0    3.0    0.0    9.0           9.0    9.0    9.0           5.0    6.0    7.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物      施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X428        0.0620    9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    8.5           7.0    9.0    8.5
        0.0320    9.0    9.0    3.0    9.0    2.0    9.0           9.0    7.0    9.0           7.0    9.0    9.0
        0.0160    9.0    9.0    1.0    9.0    1.0    9.0           7.0    1.0    9.0           5.5    7.0    8.0429        0.0620    9.0    9.0    9.0    7.0    0.0    9.0           1.0    7.0    5.5           2.5    3.0    5.0
        0.0320    9.0    9.0    3.0    4.0    0.0    9.0           0.0    2.0    5.5           2.5    2.5    4.5
        0.0160    9.0    7.0    1.0    5.0    0.0    9.0           1.0    2.0    4.5           2.0    2.5    4.0430        0.0620    9.0    9.0    9.0    9.0    5.0    9.0           1.0    7.0    9.0           3.0    4.5    5.0
        0.0320    9.0    9.0    6.0    9.0    2.0    9.0           0.0    7.0    8.0           2.5    4.0    5.0
        0.0160    9.0    9.0    2.0    9.0    0.0    9.0           0.0    3.0    8.0           2.0    3.5    5.0431        0.0620    9.0    7.0    1.0    9.0    1.0    9.0           1.0    3.0    5.5           2.5    2.5    5.0
        0.0320    9.0    7.0    1.0    9.0    0.0    9.0           1.0    9.0    8.0           2.0    2.0    5.0
        0.0160    9.0    7.0    1.0    7.0    0.0    9.0           1.0    9.0    5.0           2.0    1.5    5.0432        0.0620    9.0    9.0    3.0    9.0    1.0    9.0           2.0    9.0    8.0           2.5    2.5    5.5
        0.0320    9.0    7.0    1.0    9.0    1.0    9.0           1.0    9.0    5.5           1.5    2.5    5.0
        0.0160    9.0    7.0    0.0    4.0    0.0    9.0           0.0    9.0    5.0           2.0    2.5.   4.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X433       0.0620     9.0    9.0    1.0    4.0    2.0    9.0           1.0    9.0    9.0           2.0    3.5    5.0
       0.0320     9.0    9.0    0.0    4.0    2.0    9.0           0.0    9.0    6.0           1.5    3.5    4.5
       0.0160     9.0    9.0    0.0    4.0    0.0                  0.0    5.0    5.5           1.0    2.5    4.0434       0.0620     9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    9.0           5.5    7.5    9.0
       0.0320     9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    9.0           5.5    7.5    9.0
       0.0160     9.0    9.0    9.0    9.0    1.0    9.0           9.0    9.0    9.0           5.0    7.5    9.0435       0.0620     9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    8.5           5.5    6.5    9.0
       0.0320     9.0    9.0    4.0    9.0    1.0    9.0           8.0    9.0    7.0           5.0    6.0    9.0
       0.0160     9.0    9.0    3.0    9.0    0.0    9.0           5.0    9.0    6.5           3.5    5.0    9.0436       0.0620     9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    9.0           3.5    7.5    9.0
       0.0320     9.0    9.0    9.0    9.0    2.0    9.0           9.0    9.0    9.0           3.5    7.5    9.0
       0.0160     9.0    9.0    9.0    9.0    2.0    9.0           9.0    9.0    9.0           3.5    8.5    9.0437       0.0620     9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    9.0           8.5    8.0    9.0
       0.0320     9.0    9.0    7.0    9.0    2.0    9.0           9.0    9.0    9.0           7.5    8.0    7.5
       0.0160     9.0    9.0    4.0    9.0    0.0    9.0           9.0    9.0    9.0           7.5    5.5    6.0
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X438       0.0620     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    9.0           9.0    8.0    9.0
       0.0320     9.0    9.0    9.0    9.0    2.0    9.0           9.0    9.0    9.0           9.0    8.0    9.0
       0.0160     9.0    9.0    9.0    9.0    0.0    9.0           9.0    9.0    9.0           9.0    7.0    5.5439       0.1250     9.0    9.0    5.0    9.0    5.0    9.0           4.0    6.0    6.5           3.5    3.5    5.0
       0.0620     9.0    9.0    4.0    9.0    4.0    9.0           3.0    6.0    6.5           3.0    2.5    4.5
       0.0320     9.0    9.0    1.0    9.0    3.0    9.0           3.0    3.0    6.0           1.5    1.5    4.5
       0.0160     9.0    9.0    1.0    9.0    2.0    9.0           2.0    3.0    5.5           2.0    2.0    4.5440       0.1250     9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           6.0    6.5    8.0
       0.0620     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    9.0           6.5    5.5    8.0
       0.0320     9.0    9.0    8.0    9.0    5.0    9.0           9.0    9.0    9.0           5.5    5.5    8.0
       0.0160     9.0    9.0    8.0    9.0    4.0    9.0           9.0    9.0    7.5           4.5    4.0    7.5441       0.1250     9.0    9.0    1.0    6.0    1.0    7.0           4.0    5.0    4.5           2.0    3.0    5.0
       0.0620     4.0    4.0    1.0    5.0    1.0    4.0           2.0    2.0    4.5           1.5    2.5    4.5
       0.0320     4.0    2.0    0.0    0.0    0.0    9.0           1.0    0.0    4.5           1.5    2.0    4.5
       0.0160     0.0    0.0    0.0    0.0    0.0    9.0           1.0    1.0    4.0           1.5    2.0    4.5
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X442       0.1250     9.0    9.0    2.0    9.0    3.0    9.0           1.0    9.0    8.0           2.5    4.0    5.5
       0.0620     9.0    9.0    2.0    9.0    0.0    9.0           1.0    9.0    5.5           1.5    4.0    5.0
       0.0320     9.0    5.0    0.0    9.0    0.0    9.0           0.0    3.0    5.5           1.0    4.0    5.0
       0.0160     9.0    4.0    0.0    9.0    0.0    9.0           0.0    3.0    5.0           0.5    3.5    5.0443       0.1250     9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    8.5           5.0    8.0    8.5
       0.0620     9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    8.5           3.5    8.0    8.5
       0.0320     9.0    9.0    5.0    9.0    3.0    9.0           9.0    9.0    6.5           3.0    6.5    8.5
       0.0160     9.0    9.0    4.0    9.0    1.0    9.0           7.0    9.0    5.5           2.5    5.0    8.0444       0.0620     9.0    9.0    5.0    9.0    5.0    9.0           0.0    9.0    9.0           1.0    3.5    4.5
       0.0320     9.0    9.0    2.0    9.0    4.0    9.0           0.0    9.0    9.0           1.0    3.5    4.5
       0.0160     9.0    9.0    0.0    9.0    2.0    9.0           0.0    4.0    9.0           0.5    3.5    4.0445       0.0620     9.0    9.0    7.0    9.0    5.0    9.0           0.0    9.0    9.0           2.0    4.0    6.0
       0.0320     9.0    9.0    1.0    9.0    4.0    9.0           0.0    9.0    8.5           1.5    3.5    5.5
       0.0160     9.0    9.0    0.0    9.0    3.0    9.0           0.0    9.0    8.0           1.5    3.5    5.0446       0.0620     9.0    9.0    2.0    9.0    5.0    9.0           1.0    9.0    9.0           2.0    4.0    5.0
       0.0320     9.0    9.0    1.0    9.0    4.0    9.0           0.0    4.0    8.0           1.5    3.5    4.5
       0.0160     9.0    9.0    0.0    9.0    4.0    9.0           0.0           7.5           0.5    3.5    4.0
                                                 表1(续)
                                                                               G             O      T
                  A     A     C      C      G      I      I      E      S      L      G      R      R      Z
                  B     M     A      H      A      P      P      C      E      X      L      Y      Z      E
                  U     B     S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T     E     O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H     L     B      L      P      E      S      G      I      W      A      T      R      X447       0.1250     9.0   9.0   4.0    9.0    4.0    9.0           9.0    9.0    8.5           7.5    6.5    8.0
       0.0620     9.0   9.0   2.0    9.0    2.0    9.0           2.0    9.0    8.0           5.5    6.0    8.0
       0.0320     9.0   9.0   0.0    9.0    2.0    9.0           2.0    9.0    7.0           4.0    5.0    7.5
       0.0160     9.0   9.0   0.0    7.0    2.0    9.0           1.0    4.0    6.5           2.0    3.5    5.0448       0.1250     9.0   9.0   5.0    9.0    3.0    9.0           3.0    9.0    7.5           2.0    4.5    5.5
       0.0620     9.0   9.0   5.0    9.0    2.0    9.0           1.0    7.0    5.5           2.0    4.0    5.5
       0.0320     9.0   9.0   4.0    9.0    1.0    9.0           0.0    4.0    5.5           1.5    4.0    5.5
       0.0160     9.0   9.0   4.0    9.0    1.0    9.0           0.0           5.0           1.0    3.0    5.5449       0.2500                                                                  8.0           5.0    6.0    8.0
       0.1250                                                                  8.0           4.0    5.0    7.0
       0.0620                                                                  8.0           4.0    5.0    6.0
       0.0320                                                                  9.0           4.0    5.0    6.0
       0.0160                                                                  9.0           4.0    4.0    6.0450       0.1250                                                                  9.0           4.0    5.0    6.0
       0.0620     9.0   8.0   5.0    9.0    9.0    9.0           1.0    9.0    8.0           2.0    4.0    4.3
       0.0320     9.0   7.0   5.0    9.0    5.0    9.0           1.0    9.0    7.3           2.3    4.0    4.3
       0.0160     9.0   3.0   1.0    9.0    5.0    9.0           1.0    9.0    6.7           1.7    3.7    3.7
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X451       0.1250                                                                    8.0           4.0    4.0    6.0
       0.0620     9.0    9.0    3.0    8.0    7.0    9.0           1.0    1.0    8.0           2.0    4.0    4.3
       0.0320     9.0    9.0    1.0    7.0    2.0    9.0           0.0    1.0    7.7           2.0    3.7    3.7
       0.0160     9.0    5.0    1.0    7.0    1.0    9.0           0.0           7.3           2.7    3.0    3.7452       0.1250                                                                    6.0           3.0    4.0    6.0
       0.0620     9.0    9.0    1.0    9.0    8.0    9.0           1.0    9.0    7.0           3.3    3.0    4.3
       0.0320     9.0    5.0    1.0    9.0    3.0    9.0           0.0    2.0    6.7           2.3    2.7    4.0
       0.0160     9.0    3.0    0.0    5.0    2.0    8.0           0.0    1.0    6.7           1.7    2.0    3.7453       0.2500                                                                    9.0           7.0    7.0    8.0
       0.1250                                                                    8.0           5.0    5.0    7.0
       0.0620     9.0     9.0   9.0    9.0    9.0    9.0           7.0    9.0    8.7           6.0    6.3    6.3
       0.0320     9.0     9.0   3.0    9.0    9.0    9.0           3.0    9.0    8.3           5.7    5.7    6.0
       0.0160     9.0     9.0   2.0    8.0    4.0    9.0           1.0    4.0    7.2           4.6    5.0    4.8454       0.1250     9.0     9.0   6.0    9.0    7.0    9.0           4.0    9.0    9.0           2.5    5.0    8.0
       0.0620     9.0     9.0   3.0    9.0    7.0    9.0           0.0    7.0    8.5           0.5    4.0    7.5
       0.0320     9.0     9.0   1.0    9.0    3.0    9.0           0.0    4.0    7.5           0.5    3.0    5.0
       0.0160     9.0     9.0   1.0    9.0    3.0    9.0           0.0    3.0    6.5           0.5    2.5    4.5
                                                   表1(续)
                                                                                  G             O      T
                  A       A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T       E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H       L      B      L      P      E      S      G      I      W      A      T      R      X455       0.2500     9.0     9.0    5.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    8.0    8.0
       0.1250     9.0     9.0    9.0    9.0    9.0    9.0           3.0    9.0    9.0           4.5    7.0    7.5
       0.0620     9.0     9.0    5.0    9.0    9.0    9.0           3.0    9.0    9.0           3.5    5.0    6.0
       0.0320     9.0     9.0    5.0    9.0    5.0    9.0           3.0    9.0    8.5           1.5    4.0    5.0
       0.0160     9.0     9.0    1.0    6.0    3.0    9.0           1.0    4.0    7.5           1.0    4.0    5.0456       0.2500     9.0     9.0    7.0    9.0    9.0    9.0           6.0    9.0    9.0           5.5    7.0    8.0
       0.1250     9.0     9.0    3.0    9.0    8.0    9.0           2.0    9.0    8.0           3.5    6.0    7.5
       0.0620     9.0     9.0    3.0    9.0    7.0    9.0           0.0    9.0    8.5           2.5    4.5    6.0
       0.0320     9.0     9.0    2.0    4.0    5.0    9.0           0.0    7.0    8.5           1.5    4.0    5.5
       0.0160     9.0     9.0    1.0           3.0    9.0           0.0    7.0    6.0           1.0    3.5    4.5457       0.2500     9.0     9.0    0.0    9.0    3.0    9.0           0.0    9.0    7.5           1.5    3.5    4.5
       0.1250     9.0     9.0    2.0    9.0    3.0    9.0           0.0    7.0    7.5           1.5    3.5    4.5
       0.0620     9.0     9.0    2.0    9.0    2.0    9.0           0.0    4.0    7.5           1.0    3.0    4.0
       0.0320     9.0     9.0    0.0    4.0    0.0    9.0           0.0    0.0    6.0           0.5    2.5    3.0
       0.0160     9.0     9.0    0.0    0.0    0.0    9.0           0.0    0.0    4.5           0.5    2.5    3.0
                                                 表1(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X458       0.2500    9.0    9.0    9.0    9.0    9.0    9.0           3.0    8.0    7.5           2.0    3.5    5.0
       0.1250    9.0    9.0    7.0    9.0    5.0    9.0           2.0    8.0    7.5           1.5    3.5    5.0
       0.0620    9.0    9.0    3.0    9.0    4.0    9.0           1.0    7.0    8.5           1.0    2.5    5.0
       0.0320    9.0    9.0    2.0    3.0    3.0    9.0           0.0    4.0    6.0           1.0    2.5    4.5
       0.0160    9.0    9.0    1.0    3.0    1.0    9.0           0.0    3.0    6.0           0.5    2.0    4.5459       0.1250    9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    9.0           3.5    9.0    9.0
       0.0620    9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    8.5           3.5    8.5    9.0
       0.0320    9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    8.5           2.5    8.5    8.5
       0.0160    9.0    9.0    3.0    9.0    3.0    9.0           9.0    9.0    8.0           2.5    8.5    7.5460       0.1250    9.0    9.0    5.0    9.0    4.0    9.0           9.0    9.0    9.0           3.5    9.0    9.0
       0.0620    9.0    9.0    2.0    9.0    3.0    9.0           9.0    9.0    8.0           2.5    8.0    9.0
       0.0320    9.0    9.0    2.0    9.0    1.0    9.0           9.0    9.0    6.5           2.5    7.5    9.0
       0.0160    9.0    9.0    1.0    9.0    0.0    9.0           7.0    9.0    5.5           2.0    6.0    6.5461       0.0620    9.0    9.0    2.0    9.0    3.0    9.0           1.0    4.0    9.0           2.0    5.0    5.0
       0.0320    9.0    9.0    2.0    9.0    1.0    9.0           0.0           8.5           1.5    4.5    5.0
       0.0160    9.0    9.0    0.0    7.0    1.0    9.0           0.0    3.0    6.5           1.0    4.0    4.0
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X462       0.0620     9.0    9.0    9.0    9.0    3.0    9.0           4.0    9.0    8.5           3.0    5.5    5.5
       0.0320     9.0    9.0    9.0    9.0    3.0    9.0           2.0    9.0    9.0           3.0    5.5    5.0
       0.0160     9.0    9.0    7.0    9.0    2.0    9.0           1.0    4.0    7.5           2.0    5.5    5.0463       0.0620     9.0    9.0    0.0    9.0    5.0    9.0           0.0    3.0    7.5           1.0    3.5    5.0
       0.0320     9.0    9.0    0.0    3.0    2.0    9.0           0.0    0.0    7.5           1.0    3.0    5.0
       0.0160     9.0    4.0    0.0    0.0    0.0    9.0           0.0    0.0    5.0           0.5    2.5    3.5464       0.0620     9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           5.5    5.0    8.0
       0.0320     9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    9.0           5.5    5.0    8.0
       0.0160     9.0    9.0    7.0    9.0    4.0    9.0           9.0    9.0    9.0           5.0    5.0    7.5465       0.0620     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    8.5           3.5    4.0    8.0
       0.0320     9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    8.5           3.5    3.5    8.0
       0.0160     9.0    9.0    8.0    9.0    4.0    9.0           9.0    9.0    8.5           3.5    3.5    8.0466       0.0620     9.0    9.0    3.0    9.0    7.0    9.0           5.0    9.0    8.0           6.5    6.5    7.5
       0.0320     9.0    9.0    2.0    9.0    5.0    9.0           4.0    9.0    7.5           5.5    5.5    7.0
       0.0160     9.0    9.0    2.0    9.0    4.0    9.0           5.0    6.0    6.5           5.0    4.5    6.0
                                             表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X467       0.0620     9.0    9.0    4.0    9.0    4.0    9.0           4.0    9.0    6.0           2.5    3.0    4.5
       0.0320     9.0    9.0    3.0    9.0    3.0    9.0           4.0    6.0    5.5           2.0    4.0    4.5
       0.0160     9.0    3.0    1.0    4.0    3.0    9.0           2.0    4.0    5.5           1.5    4.0    4.5468       0.0620     9.0    9.0    5.0    9.0    7.0    9.0           9.0    9.0    9.0           3.5    7.0    8.0
       0.0320     9.0    9.0    5.0    9.0    2.0    9.0           9.0    9.0    8.5           2.0    6.5    8.0
       0.0160     9.0    9.0    5.0    9.0    2.0    9.0           8.0    8.0    8.5           1.0    6.5    8.0
       0.0320     9.0    9.0    4.0    9.0    3.0    9.0           9.0    7.0    6.5           3.5    5.0    8.0
       0.0160     9.0    7.0    3.0    9.0    2.0    9.0           4.0    4.0    5.5           3.5    4.0    7.5470       0.0620     9.0    9.0    5.0    9.0    4.0    9.0           5.0    9.0    5.5           4.0    4.0    8.0
       0.0320     9.0    9.0    2.0    9.0    4.0    9.0           2.0    4.0    5.0           4.0    4.0    7.5
       0.0160     5.0    7.0    2.0    7.0    3.0    9.0           2.0    2.0    5.0           3.0    3.0    5.0471       0.0620     9.0    4.0    0.0    4.0    4.0    9.0           2.0    3.0    8.5           1.5    4.0    4.5
       0.0320     3.0    2.0    0.0    0.0    0.0    4.0           0.0    2.0    7.5           1.5    3.5    4.5
       0.0160     3.0    0.0    0.0    0.0    0.0    3.0           0.0    0.0    6.0           0.5    3.5    3.5
                                                 表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X472       0.0620     7.0    9.0    0.0    2.0    2.0    9.0           6.0    9.0    8.5           3.5    5.5    8.0
       0.0320     4.0    9.0    0.0    2.0    0.0    9.0           3.0    5.0    8.0           3.0    5.0    7.5
       0.0160     4.0    3.0    0.0    2.0    0.0    9.0           3.0           8.0           0.5    4.5    7.5473       0.0620     9.0    7.0    2.0    9.0    4.0    9.0           0.0    2.0    6.5           2.0    7.0    5.0
       0.0320     9.0    7.0    0.0    3.0    4.0    9.0           0.0    0.0    6.0           1.0    4.5    4.0
       0.0160     9.0    3.0    0.0    3.0    2.0    9.0           0.0    0.0    5.5           0.5    4.0    4.0474       0.0620     9.0    5.0    0.0    1.0    1.0    9.0           0.0    0.0    5.0           1.5    3.5    4.0
       0.0320     9.0           0.0    1.0    1.0    4.0           0.0    0.0    5.0           0.5    3.5    4.0
       0.0160     9.0    3.0    0.0    0.0    0.0    9.0           0.0    0.0    5.0           0.0    3.0    3.5475       0.0620     9.0    9.0    0.0    9.0    5.0    9.0           1.0    3.0    7.5           1.5    4.0    4.5
       0.0320     9.0    9.0    0.0    9.0    3.0    9.0           0.0    2.0    6.0           0.5    3.5    4.0
       0.0160     9.0    5.0    0.0    3.0    3.0    9.0           0.0    0.0    4.5           0.5    3.0    4.0476       0.0620     9.0    9.0    0.0    9.0    7.0    9.0           0.0    3.0    6.0           0.0    4.0    4.0
       0.0320     9.0    9.0    0.0    8.0    3.0    9.0           0.0    0.0    5.0           0.0    3.0    3.5
       0.0160     9.0    5.0    0.0    3.0    2.0    9.0           0.0    0.0    4.5           0.0    3.0    3.0
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X477      0.0620      9.0    9.0    2.0    9.0    6.0    9.0           0.0    4.0    7.0           1.5    4.0    5.0
      0.0320      9.0    7.0    0.0    9.0    5.0    9.0           0.0    0.0    5.5           1.0    3.5    4.5
      0.0160      9.0    4.0    0.0    4.0    3.0    9.0           0.0    0.0    5.0           0.0    2.5    4.5478      0.0620      9.0    9.0    3.0    9.0    8.0    9.0           2.0    7.0    8.0           3.0    5.0    5.5
      0.0320      9.0    9.0    1.0    9.0    5.0    9.0           1.0    3.0    8.0           2.5    4.0    4.5
      0.0160      9.0    9.0    0.0    3.0    2.0    9.0           0.0    2.0    7.0           1.0    3.5    4.0479      0.0320      9.0    9.0    8.0    9.0    7.0    9.0           9.0    9.0    8.5           6.0    6.5    9.0
      0.0160      9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    7.0           6.0    6.5    8.0480      0.0620      9.0    9.0    4.0    9.0    5.0    9.0           5.0    5.0    6.0           3.5    4.0    4.5
      0.0320      9.0    7.0    3.0    7.0    3.0    9.0           3.0    4.0    5.5           2.5    3.5    4.5
      0.0160      9.0    7.0    1.0    7.0    1.0    9.0           1.0    1.0    4.5           2.0    2.0    4.5481      0.0620      9.0    9.0    2.0    6.0    5.0    9.0           4.0    3.0    5.0           3.5    3.5    5.0
      0.0320      9.0    9.0    2.0    9.0    2.0    9.0           2.0    2.0    4.5           2.5    3.5    4.5
      0.0160      6.0    4.0    0.0    3.0    1.0    9.0           1.0    1.0    5.0           2.0    2.0    4.0482      0.0320      9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    9.0           5.0    5.5    8.5
      0.0160      9.0    9.0    9.0    9.0    3.0    9.0           9.0    9.0    9.0           4.5    5.0    8.0
                                                  表1(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X483       0.0620      9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           7.0    6.5    8.0
       0.0320      9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    9.0           5.0    5.0    8.0
       0.0160      9.0    9.0    9.0    9.0    4.0    9.0           9.0    9.0    9.0           4.0    4.5    8.0484       0.0620      9.0    9.0    6.0    9.0    4.0    9.0           1.0    4.0    7.0           3.5    4.0    5.0
       0.0320      9.0    7.0    5.0    9.0    3.0    9.0           1.0    4.0    6.5           2.5    3.0    4.5
       0.0160      9.0    7.0    4.0    9.0    1.0    9.0           1.0    6.0    6.0           2.5    3.0    4.0485       0.0620      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           6.5    5.5    8.5
       0.0320      9.0    9.0    7.0    9.0    6.0    9.0           9.0    9.0    9.0           6.0    5.5    8.0
       0.0160      9.0    9.0    9.0    7.0    1.0    9.0           9.0    7.0    9.0           5.0    5.0    8.0486       0.0620      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           3.0    5.5    8.0
       0.0320      9.0    9.0    9.0    9.0    4.0    9.0           9.0    5.0    9.0           4.5    6.0    8.0
       0.0160      9.0    9.0    6.0    9.0    3.0    9.0           9.0    4.0    8.5           3.0    4.0    8.0487       0.0620      9.0    8.0    5.0    9.0    6.0    9.0           6.0    7.0    8.0           7.0    6.5    7.0
       0.0320      9.0    9.0    3.0    9.0    4.0    9.0           3.0    4.0    7.5           6.5    6.0    6.0
       0.0160      9.0    9.0    3.0    9.0    2.0    9.0           3.0    3.0    7.0           6.0    5.0    5.5
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X488       0.0620     9.0    9.0    3.0    9.0    5.0    9.0           6.0    6.0    7.0           6.0    5.5    7.0
       0.0320     9.0    7.0    2.0    7.0    4.0    9.0           3.0    4.0    6.5           5.0    4.5    7.0
       0.0160     9.0    7.0    1.0    4.0    2.0    9.0           3.0    2.0    5.5           3.5    4.0    6.0489       0.0620     9.0    7.0    7.0    9.0    5.0    9.0           4.0    7.0    8.5           5.0    5.0    5.5
       0.0320     9.0    9.0    4.0    9.0    1.0    9.0           4.0    6.0    7.0           4.5    4.5    4.5
       0.0160     9.0    7.0    3.0    9.0    3.0    9.0           3.0    4.0    5.5           3.5    4.0    4.5490       0.0620     9.0    9.0    5.0    9.0    7.0    9.0           3.0    9.0    8.5           6.5    6.5    6.5
       0.0320     9.0    9.0    5.0    9.0    6.0    9.0           4.0    7.0    7.0           6.0    5.5    6.5
       0.0160     9.0    9.0    3.0    7.0    4.0    9.0           3.0    4.0    6.5           5.0    4.5    5.5491       0.0620     9.0    9.0    7.0    9.0    6.0    9.0           4.0    7.0    7.0           7.0    6.5    5.0
       0.0320     9.0    9.0    4.0    9.0    5.0    9.0           4.0    6.0    7.0           5.0    6.0    5.0
       0.0160     9.0    9.0    2.0    9.0    2.0    9.0           2.0    4.0    7.0           3.5    5.0    4.5492       0.0620     9.0    9.0    2.0    9.0    6.0    9.0           6.0    7.0    7.0           7.0    7.0    9.0
       0.0320     9.0    9.0    1.0    9.0    4.0    9.0           6.0    7.0    7.0           4.0    6.0    8.5
       0.0160     9.0    9.0    1.0    9.0    1.0    9.0           4.0    6.0    5.5           3.5    5.0    7.5
                                                  表1(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物      施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号     (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X493        0.0620     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    9.0           6.0    8.5    9.0
        0.0320     9.0    9.0    2.0    9.0    2.0    9.0           9.0    9.0    9.0           4.5    8.5    9.0
        0.0160     9.0    9.0    2.0    9.0    0.0    9.0           9.0    7.0    9.0           4.0    8.0    8.5494        0.0620     9.0    9.0    1.0    9.0    3.0    9.0           9.0    5.0    9.0           3.0    4.5    7.5
        0.0320     9.0    9.0    0.0    9.0    1.0    9.0           9.0    5.0    8.5           2.0    4.5    7.5
        0.0160     8.0    4.0    0.0    9.0    0.0    9.0           2.0    3.0    6.0           0.5    3.5    5.0495        0.0620     9.0    9.0    2.0    9.0    7.0    9.0           1.0    3.0    7.5           2.5    4.0    5.0
        0.0320     9.0    7.0    0.0    9.0    5.0    9.0           0.0    0.0    6.5           1.5    3.0    4.5
        0.0160     9.0    4.0    0.0    9.0    0.0    9.0           0.0    0.0    6.0           1.0    3.0    4.0496        0.0620     9.0    9.0    3.0    9.0    7.0    9.0           1.0    2.0    9.0           2.5    4.0    5.0
        0.0320     9.0    9.0    2.0    9.0    5.0    9.0           0.0    1.0    7.5           1.5    4.0    5.0
        0.0160     9.0    5.0    0.0    9.0    2.0    9.0           0.0    0.0    6.5           0.5    3.0    5.0497        0.0620     9.0    9.0    2.0    9.0    5.0    9.0           1.0    2.0    7.5           1.5    3.5    5.0
        0.0320     9.0    9.0    2.0    9.0    4.0    9.0           0.0    1.0    7.0           1.5    3.5    4.5
        0.0160     9.0    4.0    0.0    4.0    3.0    9.0           0.0           6.5           0.5    3.5    4.0
                                                  表1(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X498       0.0620     9.0    9.0    1.0    9.0    5.0    9.0           1.0    3.0    7.0           2.0    4.0    5.5
       0.0320     9.0    7.0    0.0    9.0    5.0    9.0           1.0           7.0           1.0    4.0    5.0
       0.0160     9.0    4.0    0.0    5.0    3.0    9.0           0.0    0.0    6.0           0.5    4.0    4.5499       0.0820     9.0    9.0    3.0    9.0    9.0    9.0           2.0    8.0    9.0           2.0    4.5    6.5
       0.0320     9.0    9.0    1.0    9.0    9.0    9.0           1.0    7.0    9.0           1.0    4.0    5.0
       0.0160     9.0    8.0    1.0    9.0    6.0    9.0           0.0    3.0    7.5           0.5    4.0    5.0500       0.1250     9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           6.5    6.5    8.0
       0.0620     9.0    9.0    5.0    9.0    5.5    9.0           9.0    9.0    8.8           5.8    5.2    7.6
       0.0320     9.0    9.0    2.0    9.0    3.5    9.0           9.0    7.0    8.6           5.2    4.8    7.2
       0.0160     9.0    9.0    0.5    9.0    1.5    9.0           7.0    2.0    8.6           4.6    4.6    7.2501       0.1250     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    9.0           5.0    5.0    8.0
       0.0620     9.0    9.0    9.0    9.0    5.0    9.0           9.0    7.0    9.0           3.5    4.0    8.0
       0.0320     9.0    9.0    7.0    9.0    3.0    9.0           7.0    6.0    9.0           3.0    3.5    8.0
       0.0160     9.0    9.0    3.0    9.0    2.0    9.0           2.0    1.0    9.0           3.5    4.0    7.5
实施例186
对试验化合物的芽前除草性评估
本发明试验化合物的芽前除草活性以下列试验举例说明，其中由许多种单子叶与双子叶植物的种子分别与盆栽土壤混合，分别种在一品脱杯里的约一英寸土壤表面上。种植后，对杯子喷洒足量的含试验化合物的选定的丙酮水溶液，使每杯中有相当于每公顷约0.0156至0.500公斤试验化合物。经处理的杯子然后置于温室平台上，浇水，根据常规的温室方法照料。处理4至5周后，结束试验，检查各杯，根据实施例185所示的分级系统分级。
所得结果示于下表II。所评估的化合物依实施例185所示的化合物编号说明。
                                               表II
                                      对试验化合物的芽前除草评估
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X1        0.5000      9.0    9.0    9.0    9.0                  9.0    9.0    9.0    7.0           8.0    7.0    7.0
      0.2500      9.0    9.0    9.0    9.0    9.0    8.0    4.0    9.0    9.0    7.5           7.5    6.0    6.5
      0.1250      9.0    9.0    8.0    9.0    5.0    9.0    4.0    9.0    9.0    6.0           6.5    5.0    6.5
      0.0625      9.0    7.5    7.5    9.0           4.0    4.0    7.5    9.0    4.0           5.5    4.0    4.5
      0.0313      5.5    3.5    1.0    9.0    0.0           2.0    7.5    9.0    2.0           4.0    3.0    3.5
      0.0156      9.0    5.0           9.0    0.0    2.0           6.0    9.0    1.0           4.0    2.0    4.02        0.5000      9.0    9.0    2.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    4.0    6.0
      0.2500      9.0    9.0    9.0    9.0    9.0    9.0    9.0    8.3    9.0    8.5    7.0    7.7    4.0    5.6
      0.1250      9.0    9.0    8.0    9.0    9.0    9.0    9.0    8.8    9.0    5.7    9.0    6.7    3.7    4.8
      0.0625      8.8    8.6    5.6    9.0    5.8    7.5    9.0    7.0    8.0    3.5    3.0    6.5    2.7    3.6
      0.0313      7.8    8.2    7.5    9.0    6.0    4.3    4.0    2.6    6.2    1.5    3.0    1.3    1.3    2.1
      0.0157      9.0    3.0    2.0    9.0           0.0           2.0    3.0    0.0                  1.7    2.0
      0.0156      9.0    6.0    4.3    9.0    2.3    3.3           0.7    7.0    1.7           0.7    0.0    1.0
                                                    表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X3       0.5000       9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.0    9.0    9.0
     0.2500       9.0    9.0    9.0    9.0    7.6    9.0    9.0    8.3    9.0    5.0    4.0    6.8    6.3    7.3
     0.1250       9.0    9.0    7.0    9.0    7.3    8.3    4.0    5.5    8.5    4.3    3.0    6.3    4.0    5.7
     0.0630       9.0    9.0    4.0    9.0    9.0    9.0           7.0    9.0    2.0           5.0    7.0    3.0
     0.0625       9.0    8.0    5.5    9.0    4.0    7.3    8.0    4.8    8.3    3.3           4.3    3.0    5.0
     0.0315       9.0    7.0    9.0    9.0    6.0    9.0           6.0    9.0                  0.0    0.0    2.0
     0.0313       8.5    4.7    4.3    9.0    4.0    6.7    9.0    1.3    5.8    1.7    0.0    1.8    1.3    3.5
     0.0158       9.0    9.0    0.0    9.0    0.0    0.0           0.0    7.0    2.0           0.0    0.0    1.0
     0.0157                                   2.0                                                     1.3    3.0
     0.0156       9.0    5.7    4.7    9.0    0.0    2.7           0.3    6.7    2.3           0.3    0.3    1.74       0.5000       9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    7.0    7.0    7.0
     0.2500       9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.0    7.0    7.0
     0.1250       9.0    9.0    6.0    9.0    6.0           7.0    9.0    9.0           9.0    7.0    7.0    7.0
     0.0625       9.0    7.0    7.0    9.0    9.0           4.0    9.0    9.0           9.0    7.0    5.0    7.0
     0.0313       9.0    7.0    7.0    9.0    9.0           2.0    9.0    9.0           3.0    7.0    2.0    3.0
                                              表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X5        0.5000      9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    7.0    6.0    4.0
      0.2500      9.0    9.0    9.0    9.0    6.0           9.0    9.0    9.0           4.0    7.0    4.0    3.0
      0.1250      9.0    8.0    6.0    9.0    9.0           4.0    7.0    9.0           3.0    7.0    8.0    2.0
      0.0625      9.0    4.0    4.0    9.0    2.0           2.0    7.0    9.0           2.0    3.0    3.0    1.0
      0.0313      6.0    2.0    0.0    9.0    2.0           0.0    6.0    9.0           2.0    3.0    1.0    0.06        0.5000      9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0    9.0
      0.2500      9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    8.0    9.0
      0.1250      9.0    7.0    6.5    9.0    9.0    3.0    9.0    6.0    9.0    0.0    7.0    8.0    8.7    6.5
      0.0630      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    7.0           7.0    7.0    8.0
      0.0625      9.0    6.0    5.5    9.0    9.0    3.0    7.0    5.5    6.0    0.0    4.0    7.0    6.3    6.0
      0.0320      9.0    7.4    6.0    9.0    5.3    4.0    7.5    5.6    8.4    2.3    2.0    4.4    5.6    4.2
      0.0315      9.0    9.0    9.0    9.0    8.5    7.5           8.0    9.0    7.0           7.0    6.5    7.5
      0.0313      4.5    4.5    4.5    8.0    9.0    0.0    7.0    4.5    5.5    0.0    2.0    7.0    6.3    5.3
      0.0160      8.0    6.4    4.4    8.8    4.8    1.0    7.5    2.2    7.0    1.3    2.0    2.8    3.0    3.6
      0.0158      9.0    8.0    6.5    9.0    8.5    5.5           6.0    9.0    1.5           4.0    3.5    6.0
      0.0157      3.0    0.0    0.0    5.0           0.0           0.0    0.0    0.0                  3.5    2.3
                                                表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X7       0.5000       9.0    9.0    9.0                         9.0    9.0    9.0                  7.0    7.0    8.0
     0.2500       9.0    9.0    9.0                         9.0    9.0    9.0                  8.0    6.0    7.0
     0.1250       9.0    9.0    9.0                         9.0    9.0    9.0                  8.0    6.0    7.0
     0.0630       9.0    9.0    9.0    9.0    7.0           9.0    9.0    9.0    5.0           6.0    5.0    6.0
     0.0625       9.0    7.0    5.0                         9.0    9.0    9.0                  6.0    5.0    7.0
     0.0315       9.0    9.0    9.0    9.0    0.0           7.0    7.0    9.0                  5.0    2.0    4.0
     0.0313       9.0    7.0    5.0                         3.0    9.0    9.0                  4.0    5.0    5.0
     0.0158       9.0    2.0    9.0    9.0    0.0           9.0    7.0    9.0    3.0           5.0    2.0    2.0
     0.0157       9.0    9.0    9.0                         3.0    7.0    9.0                  5.0    2.0    5.08       0.5000       9.0    9.0    9.0                         9.0    9.0    9.0                  9.0    9.0    9.0
     0.2500       9.0    9.0    9.0                         9.0    9.0    9.0                  9.0    9.0    9.0
     0.1250       9.0    9.0    9.0                         9.0    7.0    9.0                  5.0    7.0    9.0
     0.0630       9.0    9.0    9.0    9.0    5.0           9.0    5.0    9.0    9.0           5.0    2.0    7.0
     0.0625       9.0    9.0    9.0                         9.0    9.0    9.0                  7.0    5.0    4.0
     0.0315       9.0    9.0    9.0    9.0    4.0           9.0    4.0    9.0    9.0           2.0    2.0    5.0
     0.0313       9.0    9.0    5.0                         9.0    5.0    9.0                  5.0    4.0    3.0
     0.0158       9.0    7.0    2.0    9.0    0.0           9.0    0.0    9.0    5.0           2.0    0.0    4.0
     0.0157       9.0    9.0    5.0                         9.0    4.0    7.0                  0.0    5.0    2.0
                                                   表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X9        0.5000      9.0    9.0    9.0                         9.0    9.0    9.0                  9.0    9.0    9.0
      0.2500      9.0    9.0    9.0                         9.0    9.0    9.0                  9.0    9.0    9.0
      0.1250      9.0    9.0    9.0                         9.0    9.0    9.0                  6.0    9.0    6.0
      0.0630      9.0    9.0    9.0    9.0    4.0           9.0    7.0    9.0    7.0           4.0    4.0    6.0
      0.0625      9.0    9.0    9.0                         9.0    5.0    9.0                  5.0    5.0    7.0
      0.0315      9.0    9.0    9.0    9.0    0.0           9.0    0.0    9.0    5.0           0.0    0.0    2.0
      0.0313      9.0    9.0    5.0                         9.0    4.0    6.0                  5.0    4.0    4.0
      0.0158      9.0    9.0    0.0    9.0    0.0           5.0    0.0    9.0    2.0           0.0    0.0    3.0
      0.0157      9.0    9.0    3.0                         5.0    2.0    9.0                  4.0    4.0    5.010       0.5000      9.0    9.0    7.0                         9.0    9.0    9.0                  7.0    6.0    7.0
      0.2500      9.0    9.0    9.0                         9.0    9.0    9.0                  6.0    5.0    5.0
      0.1250      9.0    9.0    9.0                         9.0    8.0    9.0                  5.0    5.0    7.0
      0.0630      9.0    7.0    0.0    9.0    0.0           9.0    3.0    6.0    0.0           0.0    0.0    0.0
      0.0625      9.0    6.0    5.0                         5.0    4.0    9.0                  4.0    4.0    4.0
      0.0315      9.0    2.0           9.0    0.0           0.0    0.0    9.0    0.0           0.0    0.0    0.0
      0.0313      9.0    0.0    9.0                         4.0    3.0    9.0                  2.0    2.0    2.0
      0.0158      0.0    0.0           9.0    0.0           0.0    0.0    5.0    0.0           0.0    0.0    0.0
      0.0157      9.0    0.0    6.0                         5.0    3.0    9.0                  0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X11       0.5000      9.0    9.0    8.0                         9.0    4.0    9.0                  5.0    4.0    3.0
      0.2500      9.0    9.0    3.0                         5.0    0.0    9.0                  0.0    4.0    5.0
      0.1250      9.0    7.0    3.0                         4.0    0.0    7.0                  0.0    3.0    1.0
      0.0625      6.0    6.0    3.0                         2.0    0.0    5.0                  0.0    0.0    1.0
      0.0313      3.0    0.0    0.0                         0.0    0.0    2.0                  0.0    0.0    0.0
      0.0157      1.0    0.0    0.0                         0.0    0.0    0.0                  0.0    0.0    0.012       0.5000      9.0    9.0    9.0                         9.0    9.0    9.0                  7.0    7.0    7.0
      0.2500      9.0    9.0    9.0                         9.0    6.0    9.0                  7.0    5.0    7.0
      0.1250      9.0    9.0    9.0                         9.0    5.0    9.0                  4.0    4.0    7.0
      0.0630      9.0    7.0    5.0    9.0    5.0           9.0    0.0    9.0    5.0           4.0    4.0    3.0
      0.0625      9.0    9.0    9.0                         9.0    0.0    9.0                  0.0    5.0    1.0
      0.0315      9.0    9.0    0.0    9.0    0.0           9.0    0.0    7.0    3.0           0.0    0.0    5.0
      0.0313      9.0    9.0    5.0                         9.0    0.0    7.0                  0.0    4.0    1.0
      0.0158      9.0    0.0           9.0    0.0           9.0    0.0    6.0    4.0           0.0    0.0    1.0
      0.0157      9.0    9.0    0.0                         9.0    0.0    9.0                  0.0    0.0    1.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X13       0.5000      9.0    9.0    9.0                         9.0    9.0    9.0                  7.0    6.0    7.0
      0.2500      9.0    9.0    9.0                         9.0    9.0    9.0                  6.0    4.0    4.0
      0.1250      9.0    9.0    9.0                         9.0    5.0    9.0                  5.0    3.0    4.0
      0.0630      9.0    9.0    9.0    9.0    4.0           5.0    0.0    7.0    3.0           0.0    0.0    0.0
      0.0625      9.0    9.0    4.0                         4.0    0.0    9.0                  0.0    0.0    5.0
      0.0315      9.0    7.0    9.0    9.0    0.0           5.0    0.0    4.0    0.0           0.0    0.0    0.0
      0.0313      9.0    9.0    8.0                         7.0    0.0    7.0                  0.0    2.0    4.0
      0.0158      9.0    7.0    8.0    9.0    0.0           0.0    0.0    5.0    0.0           0.0    0.0    0.0
      0.0157      9.0    6.0    7.0                         4.0    0.0    5.0                  0.0    0.0    0.014       0.2500      9.0    4.5    9.0    9.0    4.5    9.0           2.5    9.0    4.0           6.5    3.0    2.0
      0.1250      9.0    7.0    8.0    9.0    0.5    6.5           2.0    8.5    1.5           3.0    1.0    2.0
      0.0625      9.0    4.5    9.0    9.0    0.0    4.5           1.5    8.0    1.5           1.0    0.5    1.5
      0.0313      6.5    2.5    4.5    9.0    0.0    2.5           0.0    5.0    0.5           0.5    0.5    0.5
      0.0156      6.0    2.0    0.0    9.0    0.0    0.0           0.0    3.5    0.5           0.0    0.0    0.5
                                                表II(续)
                                                                               G             O      T
                A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷) H      L      B      L      P      E      S      G      I      W      A      T      R      X15       0.2500    9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    4.0           7.0    6.0    9.0
      0.1250    9.0    9.0    8.0    9.0    5.5    9.0           7.5    9.0    6.0           6.5    4.0    4.0
      0.0625    9.0    9.0    7.5    9.0    2.0    6.5           3.0    7.5    3.5           4.0    2.0    3.5
      0.0313    9.0    4.5    3.5    9.0    2.0    2.5           2.0    6.5    2.5           1.0    1.0    1.0
      0.0156    6.5    2.5    5.5    9.0    0.0    0.5           0.5    5.0    0.0           1.0    0.0    0.016       0.2500    9.0    9.0    9.0    9.0    9.0    9.0           0.0    7.0    0.0           7.0    1.0    2.0
      0.1250    9.0    5.0    3.0    9.0    5.0    3.0           0.0    0.0    4.0           0.0    0.0    1.0
      0.0625    9.0    4.0    1.0    9.0    0.0    0.0           0.0    2.0    0.0           0.0    0.0    1.0
      0.0313    0.0    0.0    9.0    4.0    0.0    0.0           0.0    7.0    0.0           0.0    0.0    1.0
      0.0156    0.0    0.0    0.0                  0.0           0.0    0.0    0.0           0.0    0.0    0.017       0.2500    9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    6.0           7.0    5.0    4.0
      0.1250    9.0    8.0    9.0    9.0    9.0    9.0           4.0    9.0    6.0           2.0    2.0    2.0
      0.0625    9.0    8.0    7.0    9.0    4.0    0.0           5.0    5.0    2.0           0.0    0.0    3.0
      0.0313    9.0    5.0    2.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156    9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X18       0.2500      9.0    9.0    4.0    9.0    1.0    4.0           5.0    9.0    2.0           0.0    0.0    3.0
      0.1250      9.0    4.0    0.0    9.0    0.0    2.0           3.0    9.0    1.0           2.0    1.0    2.0
      0.0625      9.0    2.0           9.0    5.0    2.0           3.0    9.0    1.0           4.0    2.0    1.0
      0.0313      2.0    2.0    1.0    6.0           0.0           1.0    8.0    2.0           0.0    0.0    0.0
      0.0156             0.0           9.0    0.0    2.0           4.0           1.0           3.0    7.019       0.2500      9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    7.0           7.0    6.0    8.0
      0.1250      9.0    7.0    9.0    9.0    5.0    5.0           6.0    9.0    5.0           5.0    5.0    7.0
      0.0625      9.0    6.0    9.0    9.0    4.0    3.0           0.0    6.0    2.0           0.0    0.0    2.0
      0.0313      9.0    0.0    2.0    9.0    3.0    0.0           0.0    4.0    1.0                  0.0    0.0
      0.0156      3.0    0.0           9.0    0.0    0.0           0.0    4.0    0.0           0.0    0.0    0.020       0.2500      9.0    5.0    7.0    9.0    5.0    3.0           5.0    8.0    1.0           7.0    5.0    4.0
      0.1250      9.0    7.0    0.0    9.0    0.0    2.0           0.0    6.0    0.0           0.0    1.0    1.0
      0.0625      9.0    4.0           7.0    0.0    0.0           0.0    4.0    0.0           0.0    0.0    0.0
      0.0313      4.0    5.0    2.0    4.0    0.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0           0.0    0.0           0.0    1.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O        T
                  A      A      C      C      G      I      I      E      S      L      G      R        R        Z
                  B      M      A      H      A      P      P      C      E      X      L      Y        Z        E
                  U      B      S      E      L      O      O      H      T      M      X      S        A        A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A        W        M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T        R        X21       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    9.0           7.0      7.0      8.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           6.0    9.0    8.0           5.0      5.0      7.0
      0.0625      9.0    7.0    9.0    9.0    6.0    7.0           4.0    7.0    7.0           2.0      2.0      6.0
      0.0313      9.0    5.0    7.0    9.0    3.0    5.0           0.0    3.0    2.0           0.0      0.0      0.0
      0.0156      9.0    3.0    3.0    9.0    0.0    1.0           0.0    2.0    1.0           0.0      0.0      0.022       0.2500      0.0    0.0    9.0    0.0    4.0    0.0           0.0    0.0    2.0           0.0      0.0      1.0
      0.1250      0.0    0.0    0.0           0.0    0.0           0.0    0.0    0.0           0.0      0.0      0.0
      0.0625      0.0    0.0    0.0           0.0    0.0           0.0    0.0    0.0           0.0      0.0      0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0      0.0      0.0
      0.0156      0.0    0.0                  0.0    0.0           0.0    0.0    0.0           0.0      0.0      0.023       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0      9.0      9.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0      9.0      9.0
      0.0625      9.0    9.0    9.0    9.0    9.0    8.0           9.0    9.0    7.5           8.0      8.0      7.0
      0.0313      9.0    8.5    6.0    9.0    7.0    6.5           7.0    9.0    6.5           8.0      7.0      6.0
      0.0157      9.0    8.0    2.0    9.0           0.0           2.0    9.0    2.0                             1.0
      0.0156      9.0    7.0    9.0    9.0    5.0    9.0           6.0    9.0    7.0           4.0      4.0      6.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X24       0.2500      9.0    5.0    4.0    9.0    3.0    9.0           3.0    5.0    1.0           0.0    0.0    2.0
      0.1250      3.0    4.0    4.0    9.0    0.0    0.0           0.0    4.0    0.0           0.0    0.0    1.0
      0.0625      4.0    5.0    2.0    5.0    0.0    0.0           0.0    3.0    1.0           0.0    1.0    2.0
      0.0313      3.0    2.0    0.0    6.0    0.0    0.0           0.0    5.0    2.0           0.0    0.0    0.0
      0.0156      0.0    0.0    1.0    5.0    0.0    0.0           0.0    3.0    1.0           0.0    1.0    0.025       0.2500      9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    9.0           7.0    7.0    7.0
      0.1250      9.0    9.0    9.0    9.0    7.0    6.0           9.0    9.0    5.0           5.0    7.0    7.0
      0.0625      9.0    4.0    9.0    9.0    0.0    5.0           7.0    9.0    1.0           2.0    7.0    1.0
      0.0313      8.0    0.0    9.0    9.0           0.0           2.0    7.0    0.0           0.0    2.0    0.0
      0.0156      9.0    3.0    9.0    9.0    0.0    0.0           2.0    5.0    0.0           0.0    2.0    0.026       0.2500      9.0    9.0    9.0    9.0    4.0    7.0           7.0    9.0    6.0           5.0    5.0    7.0
      0.1250      9.0    9.0    7.0    9.0    7.0    7.0           5.0    9.0    7.0           2.0    2.0    4.0
      0.0625      9.0    9.0    2.0    9.0    8.0    0.0           0.0    9.0    1.0           4.0    2.0    2.0
      0.0313      9.0    0.0    0.0    9.0    5.0    0.0           1.0    9.0    1.0           0.0    0.0    1.0
      0.0156      9.0    0.0           9.0    0.0    2.0           0.0    5.0    1.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X27       0.2500      9.0    9.0    9.0    9.0    2.0    6.0           7.0    9.0    9.0           2.0    5.0    4.0
      0.1250      9.0    9.0    9.0    9.0    5.0    9.0           6.0    9.0    4.0           2.0    4.0    3.0
      0.0825      9.0    2.0    0.0    9.0    0.0    2.0           3.0    9.0    0.0           0.0           4.0
      0.0313      9.0    4.0    9.0    9.0    0.0    2.0           3.0    9.0    0.0           0.0    0.0    1.0
      0.0156      9.0    0.0    0.0    9.0    0.0    0.0           0.0    7.0    0.0           0.0    0.0    0.028       0.2500      9.0    9.0    0.0    9.0    7.0    9.0           8.0    9.0    6.0           5.0    5.0    6.0
      0.1250      9.0    9.0    9.0    9.0    5.0    9.0           4.0    9.0    4.0           5.0    5.0    5.0
      0.0625      9.0    9.0    9.0    9.0           7.0           4.0    9.0    4.0           5.0    5.0    5.0
      0.0313      9.0    4.0    0.0    9.0    0.0    5.0           0.0    9.0    4.0           2.0    2.0    3.0
      0.0156      9.0    9.0    0.0    9.0    0.0    0.0           0.0    4.0    2.0           0.0    0.0    3.029       0.2500      2.0    0.0    0.0    9.0    0.0    0.0           0.0    9.0    1.0           0.0    0.0    2.0
      0.1250      0.0    0.0    0.0    7.0    0.0    0.0           0.0    9.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    9.0    0.0    0.0           0.0    7.0    0.0           0.0    0.0    1.0
      0.0313      0.0    0.0           6.0    0.0    0.0           0.0    4.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           0.0           0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X30       0.2500      9.0    9.0    9.0    9.0    7.0    9.0           7.0    9.0    6.0           6.0    7.0    7.0
      0.1250      9.0    9.0    9.0    9.0    1.0    9.0           6.0    9.0    3.0           5.0    6.0    6.0
      0.0625      7.0    3.0    0.0    9.0    0.0    2.0           1.0    9.0    2.0           4.0    2.0    2.0
      0.0313      9.0    2.0    0.0    9.0    3.0    2.0           0.0    9.0    1.0           2.0    1.0    2.0
      0.0156      9.0    2.0           9.0    0.0    3.0           0.0    7.0    0.0           1.0    0.0    1.031       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    9.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    8.0
      0.0625      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.5           8.0    8.0    8.0
      0.0313      9.0    9.0    6.0    9.0    9.0    7.5           6.5    8.5    6.0           8.0    8.0    7.0
      0.0157      9.0    9.0    0.0    9.0           7.0           7.0    6.0    6.0                         5.0
      0.0156      9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    8.0           8.0    7.0    8.032       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.0           9.0    8.0    8.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    6.0           8.0    7.0    8.0
      0.0625      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    5.0           7.0    7.0    7.0
      0.0313      9.0    9.0    9.0    9.0    8.0    6.0           2.0    7.0                  6.0    2.0    5.0
      0.0156      9.0    5.0    2.0    9.0    7.0    4.0           0.0    5.0    4.0           4.0    2.0    4.0
                                                 表II(续)
                                                                                 G      O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X33       0.2500      9.0    9.0    9.0    9.0    0.0    9.0           9.0    9.0    7.0           7.0    2.0    7.0
      0.1250      9.0    9.0    7.0    9.0    1.0    9.0           7.0    9.0    2.0           6.0    2.0    9.0
      0.0625      9.0    4.0    9.0    9.0           5.0           1.0    9.0                  7.0    4.0    5.0
      0.0313      9.0    4.0    5.0    9.0           4.0           0.0    7.0    4.0           2.0    1.0    2.0
      0.0156      5.0    1.0    9.0    9.0    0.0    3.0           0.0    2.0                  3.0    2.0    3.034       0.2500      1.0    1.0    5.0    1.0    5.0    0.0           0.0    1.0    1.0           1.0    1.0    2.0
      0.1250      0.0    0.0    4.0    2.0    9.0    0.0           0.0    1.0                  1.0    2.0    1.0
      0.0625      0.0    0.0    2.0    7.0    4.0    0.0           0.0    2.0    1.0           1.0    1.0    1.0
      0.0313      0.0    1.0    0.0    0.0    2.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0           2.0    0.0           0.0    0.0    0.0           1.0    0.0    0.035       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    8.0    8.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    9.0    8.0
      0.0625      9.0    9.0    9.0    9.0    8.0    7.0           9.0    9.0    7.0           7.0    7.0    8.0
      0.0313      9.0    9.0    7.0    9.0    7.0    6.0           7.0    9.0    5.0           6.0    6.0    7.0
      0.0156      9.0    8.0    6.0    9.0    7.0    4.0           6.0    7.0    1.0           3.0    3.0    5.0
                                                   表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X36       0.2500      0.0    0.0    0.0    0.0    0.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.1250      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.037       0.2500      1.0    0.0    0.0    3.0    0.0    0.0           0.0    2.0    2.0           0.0    0.0    0.0
      0.1250      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.038       0.2500      0.0    0.0    0.0    3.0    9.0    1.0           0.0    0.0    4.0           1.0    2.0    3.0
      0.1250      0.0    0.0    0.0    5.0    5.0    0.0           0.0    0.0    1.0           1.0    1.0    1.0
      0.0625      0.0    0.0    4.0    0.0    5.0    0.0           0.0    0.0    2.0           2.0    1.0    1.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           2.0    0.0    1.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X39       0.2500      2.0    1.0    0.0    7.0    7.0    1.0           1.0    0.0    3.0           5.0    3.0    5.0
      0.1250      0.0    1.0           5.0    2.0    0.0           0.0    0.0    1.0           5.0    3.0    2.0
      0.0625      0.0    1.0    0.0    0.0    0.0    3.0           1.0    1.0    0.0           6.0    7.0    0.0
      0.0313      1.0    2.0    1.0    5.0    0.0    3.0           0.0    0.0    1.0           5.0    1.0    2.0
      0.0156      1.0    1.0    0.0    0.0    0.0    1.0           0.0    0.0                  6.0    0.0    0.040       0.2500      9.0    9.0    6.0    9.0    9.0    7.0           9.0    9.0    9.0           8.0    7.0    8.0
      0.1250      9.0    7.0    2.0    9.0    9.0    9.0           9.0    9.0    6.0           7.0    7.0    6.0
      0.0625      9.0    7.0    1.0    9.0    7.0    6.0           7.0    9.0    5.0           5.0    6.0    6.0
      0.0313      9.0    6.0    2.0    9.0    7.0    6.0           4.0    9.0    5.0           6.0    1.0    4.0
      0.0156      9.0    0.0    0.0    5.0    0.0    0.0           4.0    9.0    2.0           1.0    3.0    3.041       0.2500      9.0    4.0    1.0    9.0    3.0    5.0           7.0    8.0    2.0           2.0    4.0    5.0
      0.1250      7.0    2.0    5.0    9.0           2.0           6.0    7.0    1.0           1.0    1.0    3.0
      0.0625      3.0    3.0    2.0    5.0           0.0           2.0    5.0    1.0           1.0    1.0    3.0
      0.0313      1.0    1.0    2.0    2.0    3.0    0.0           0.0    0.0    1.0           2.0    1.0    5.0
      0.0156      0.0    0.0    2.0    0.0    3.0    1.0           0.0    0.0    1.0           1.0    0.0    0.0
                                                 表II(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X42       0.2500     9.0    9.0    9.0    9.0    9.0    8.0           8.0    9.0    8.0           8.0    6.0    7.0
      0.1250     9.0    7.0    5.0    9.0    7.0    7.0           7.0    7.0    9.0           5.0    4.0    5.0
      0.0625     9.0    6.0    2.0    9.0    2.0    2.0           4.0    7.0    5.0           4.0    3.0    5.0
      0.0313     7.0    6.0           6.0    1.0    1.0           2.0    4.0    3.0           1.0    1.0    2.0
      0.0156     5.0    1.0    0.0    0.0    1.0    0.0           1.0    1.0    1.0           3.0    1.0    0.043       0.2500     9.0    9.0    4.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.0    8.0
      0.1250     9.0    9.0           9.0    6.0    9.0           8.0    9.0    7.0           7.0    7.0    8.0
      0.0625     8.0    6.0    0.0    9.0    8.0    0.0           9.0    9.0    3.0           4.0    4.0    7.0
      0.0313     9.0    1.0           9.0    0.0    1.0           7.0    9.0    5.0           2.0    1.0    7.0
      0.0156     2.0    0.0    0.0    8.0    1.0    0.0           0.0    5.0                  2.0    0.0    0.044       0.2500     9.0    7.0    9.0    9.0    7.0    9.0           4.0    7.0    9.0           5.0    4.0    5.0
      0.1250     9.0    6.0    5.0    9.0    7.0    6.0           0.0    4.0    5.0           2.0    2.0    3.0
      0.0625     7.0    4.0    0.0    9.0    7.0    1.0           0.0    0.0    3.0           1.0    1.0    1.0
      0.0313     0.0    0.0    0.0    1.0    2.0    0.0           0.0    0.0    5.0           1.0    0.0    0.0
      0.0156     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R       Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z       E
                  U      B      S      E      L      O      O      H      T      M      X      S      A       A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W       M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R       X45       0.2500      9.0    9.0    7.0    9.0    8.5    7.5           8.0    9.0    9.0           6.0    5.5     6.0
      0.1250      9.0    8.0    4.0    9.0    8.5    9.0           7.0    9.0    7.0           5.0    4.5     5.0
      0.0625      9.0    7.5    4.5    8.5    7.0    3.5           7.5    9.0    5.5           5.0    4.0     4.0
      0.0313      9.0    4.5    3.0    9.0    6.5    3.5           5.5    9.0    3.0           4.0    1.5     2.5
      0.0156      5.0    1.5    1.0    9.0    0.5    0.5           0.5    8.0    2.5           1.5    1.5     1.046       0.2500      9.0    8.5    8.0    9.0    9.0    9.0           7.0    9.0    9.0           5.5    4.0     6.5
      0.1250      9.0    8.5    6.0    9.0    5.0    9.0           5.5    9.0    7.0           6.0    4.0     3.5
      0.0625      8.5    8.0    2.5    9.0    2.0    5.5           4.5    8.0    5.5           7.0    4.5     4.0
      0.0313      9.0    4.0    1.5    9.0    6.0    4.5           2.0    8.0    4.5           4.5    5.5     4.0
      0.0156      4.5    2.0    2.0    9.0    1.0    1.0           0.5    7.5    4.0           4.5    3.0     2.547       0.2500      9.0    9.0    6.0    9.0    8.0    9.0           8.0    9.0    9.0           9.0    8.0     9.0
      0.1250      9.0    7.0    7.0    9.0    0.0    6.0           7.0    9.0    7.0           7.0    7.0     7.0
      0.0625      6.0    7.0    4.0    9.0           7.0           4.0    9.0    6.0           6.0    7.0     6.0
      0.0313      9.0    0.0    4.0    5.0    0.0    5.0           1.0    9.0    4.0           4.0    2.0     4.0
      0.0156      0.0    0.0    0.0    5.0    0.0    0.0           0.0    3.0    1.0           2.0    0.0     1.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X48       0.2500      9.0    9.0    5.0    9.0    9.0    7.0           8.0    9.0    9.0           8.0    9.0    8.0
      0.1250      9.0    9.0           9.0    7.0    9.0           4.0    9.0    9.0           8.0    7.0    7.0
      0.0825      7.0    7.0    3.0    9.0    8.0    3.0           2.0    9.0    6.0           8.0    7.0    6.0
      0.0313      9.0    1.0    3.0    2.0    6.0    1.0           0.0    8.0    2.0           5.0    3.0    5.0
      0.0156      0.0    0.0    2.0    0.0    6.0    1.0           0.0    9.0                  3.0    0.0    3.049       0.0630      9.0    9.0    4.0    9.0    4.0           9.0    4.0    7.0    6.0           0.0    0.0    0.0
      0.0315      9.0    9.0           9.0    4.0           0.0    0.0    6.0    0.0           0.0    0.0    0.0
      0.0158      3.0    5.0    0.0    9.0                  0.0    0.0    0.0    0.0           0.0    0.0    0.050       0.1250      9.0    9.0    2.0    9.0           9.0           9.0    9.0    4.0                         2.0
      0.0630      9.0    9.0    9.0    9.0    6.0           9.0    5.0    9.0    8.0           0.0    0.0    0.0
      0.0625      9.0    9.0    2.0    9.0           4.0           5.0    9.0    0.0                         0.0
      0.0315      9.0    5.0    0.0    9.0.   0.0           7.0    0.0    5.0    6.0           0.0    0.0    0.0
      0.0313      9.0    9.0    2.0    9.0           0.0           4.0    7.0    0.0                         0.0
      0.0158      9.0    0.0    0.0    9.0    0.0           0.0    0.0    5.0    5.0           0.0    0.0    0.0
      0.0157      9.0    0.0    0.0    9.0           0.0           0.0    0.0    0.0                         0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X51       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    9.0           7.0    4.0    2.0
      0.1250      9.0    9.0    4.0    9.0    7.0    8.5           8.0    9.0    4.0           0.0    6.0    2.0
      0.0625      9.0    7.0    1.0    9.0    5.0    7.5           5.5    9.0    2.0           0.0    0.0    0.0
      0.0313      9.0    7.0    4.5    9.0    0.0    4.5           2.5    6.5    0.5           0.0    0.0    0.0
      0.0157      9.0    9.0    0.0    9.0           0.0           3.0    5.0    0.0                         0.0
      0.0156      4.0    3.0    0.0    9.0    0.0    0.0           0.0    7.0    0.0           0.0    0.0    0.052       0.2500      9.0    5.0    4.0    9.0    5.0    4.0           0.0    7.0    2.0           0.0    0.0    0.0
      0.1250      4.0    4.0    0.0    9.0    0.0    0.0           0.0    6.0    0.0           0.0    0.0    0.0
      0.0625      1.0    0.0    9.0    9.0    0.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    3.0    9.0    0.0    0.0           0.0    5.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0           0.0           0.0    4.0    0.0           0.0    0.0    0.053       0.2500      9.0    9.0    8.0    9.0    7.0    9.0           9.0    9.0    9.0           7.0    5.0    4.0
      0.1250      9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    6.0           5.0    2.0    4.0
      0.0625      9.0    9.0    4.0    9.0    0.0    5.0           5.0    9.0    4.0           8.0    0.0    2.0
      0.0313      9.0    5.0    0.0    9.0    0.0    0.0           0.0    7.0    0.0           7.0    0.0    0.0
      0.0156      9.0    8.0    3.0    9.0    0.0    3.0           0.0    4.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X54       0.2500      9.0    1.0    9.0    9.0    1.0    9.0           3.0    9.0    0.0           2.0    1.0    2.0
      0.1250      9.0    2.0    9.0    9.0    0.0    5.0           1.0    6.0    0.0           0.0    0.0    1.0
      0.0625      4.0    0.0    9.0    9.0    0.0    0.0           0.0    5.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    9.0    9.0    0.0    0.0           0.0    0.0    2.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.055       0.2500      9.0    7.0    9.0    9.0    0.0    7.0           9.0    9.0    5.0           5.0    0.0    2.0
      0.1250      9.0    5.0    9.0    9.0    0.0    2.0           2.0    7.0    4.0           4.0    0.0    3.0
      0.0625      9.0    5.0    9.0    9.0    0.0    3.0           0.0    9.0    2.0           0.0    0.0    0.0
      0.0313      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    3.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    5.0    0.0           0.0    0.0    0.056       0.2500      9.0    9.0    9.0    9.0    0.0    2.0           4.0    9.0    2.0           0.0    0.0    1.0
      0.1250      9.0    8.0    7.0    9.0    5.0    2.0           5.0    9.0    0.0           0.0    0.0    1.0
      0.0625      9.0    0.0    9.0    9.0    0.0    0.0           0.0    9.0    0.0           0.0    0.0    0.0
      0.0313      4.0    0.0    3.0    9.0    0.0    0.0           0.0    7.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    6.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X57       0.2500      9.0    9.0    9.0    9.0    5.0    7.0           7.0    9.0    7.0           7.0    5.0    7.0
      0.1250      9.0    7.0    9.0    9.0    5.0    6.0           8.0    7.0    5.0           2.0    1.0    3.0
      0.0625      9.0    4.0    9.0    9.0    2.0    9.0           7.0    9.0    0.0           0.0    0.0    0.0
      0.0313      9.0    3.0    9.0    9.0    0.0    5.0           5.0    8.0    0.0           0.0    0.0    0.0
      0.0156      7.0    9.0    5.0    9.0    0.0    0.0           0.0    5.0                  0.0    0.0    0.058       0.2500      9.0    9.0    9.0    9.0    4.0    6.0           8.0    9.0    9.0           6.0    6.0    7.0
      0.1250      9.0    5.0    9.0    9.0    5.0    4.0           5.0    9.0    5.0           2.0    2.0    6.0
      0.0625      6.0    7.0    9.0    9.0    3.0    0.0           0.0    5.0    2.0           0.0    0.0    1.0
      0.0313      9.0    1.0    9.0    9.0    0.0    0.0           0.0    6.0    2.0           0.0    0.0    0.0
      0.0156      5.0    0.0    9.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.059       0.2500      9.0    7.0    9.0    9.0    9.0    9.0           7.0    9.0    5.0           0.0    0.0    3.0
      0.1250      9.0    0.0    2.0    9.0    7.0    0.0           4.0    9.0    0.0           0.0    0.0    2.0
      0.0625      9.0    0.0    9.0    9.0    9.0    0.0           2.0    9.0    0.0           0.0    0.0    1.0
      0.0313      0.0    0.0    0.0    9.0    5.0    0.0           0.0    7.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0           9.0    5.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X60       0.2500      9.0    8.0    9.0    9.0    0.0    0.0           0.0    7.0    1.0           0.0    0.0    1.0
      0.1250      1.0    2.0    2.0    9.0    0.0    0.0           0.0    3.0    1.0           0.0    0.0    0.0
      0.0625      2.0    0.0    0.0    9.0    6.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    9.0    6.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0    2.0    0.0           0.0    0.0    0.0           0.0    0.0    0.061       0.2500      2.0    0.0    9.0    9.0    4.0    0.0           0.0    7.0    0.0           0.0    0.0    5.0
      0.1250      3.0    0.0    3.0    9.0    0.0    0.0           0.0    7.0    0.0           0.0    0.0    0.0
      0.0625      3.0    0.0    4.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0           9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156             0.0           9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.062       0.2500      9.0    9.0    9.0    9.0    6.0    9.0           8.0    9.0    5.0           5.0    2.0    6.0
      0.1250      9.0    9.0    9.0    9.0    0.0    9.0           7.0    9.0    5.0           1.0    1.0    4.0
      0.0625      9.0    9.0    9.0    9.0           9.0           3.0    9.0    5.0           1.0    1.0    4.0
      0.0313      9.0    0.0    9.0    9.0           9.0           1.0    7.0    1.0           0.0    0.0    1.0
      0.0156      9.0    0.0    0.0    9.0    0.0    0.0           0.0    7.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X63       0.2500      9.0    0.0    0.0    9.0    0.0    0.0           1.0    5.0    1.0           0.0    0.0    0.0
      0.1250      9.0    7.0           9.0           1.0           0.0    4.0    1.0           0.0    0.0    0.0
      0.0625      5.0    0.0           9.0    0.0    0.0           0.0    0.0                  0.0    0.0    2.0
      0.0313      0.0    0.0           9.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.0
      0.0156      0.0    0.0           9.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.064       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    2.0    4.0
      0.1250      9.0    9.0    4.0    9.0    6.0    9.0           8.0    8.0    7.0           7.0    1.0    4.0
      0.0625      9.0    9.0    4.0    9.0    4.0    3.0           4.0    9.0    2.0           5.0    0.0    0.0
      0.0313      9.0    7.0    2.0    9.0    2.0    9.0           0.0    4.0    0.0           0.0    0.0    0.0
      0.0156      9.0    5.0    5.0    9.0           0.0           0.0    3.0    0.0           0.0    0.0    0.065       0.2500      9.0    9.0    9.0    9.0    8.0    9.0           8.0    9.0    5.0           8.0    3.0    5.0
      0.1250      9.0    9.0    9.0    9.0    4.0    2.0           7.0    9.0    2.0           2.0    0.0    3.0
      0.0625      9.0    2.0    6.0    9.0    2.0    0.0           5.0    9.0    1.0           2.0    0.0    3.0
      0.0313      4.0    2.0    5.0    9.0    0.0    0.0           2.0    7.0    1.0           3.0    1.0    3.0
      0.0156      9.0    2.0    1.0    9.0    0.0    0.0           1.0    5.0    0.0           2.0    2.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X66       0.2500      9.0    9.0    9.0    9.0    9.0    1.0           9.0    9.0    5.0           5.0    4.0    5.0
      0.1250      9.0    9.0    9.0    9.0    4.0    0.0           9.0    9.0    5.0           4.0    3.0    5.0
      0.0625      9.0    2.0    9.0    9.0    5.0    0.0           5.0    9.0    2.0           4.0    3.0    2.0
      0.0313      9.0    5.0    9.0    9.0    2.0    0.0           3.0    9.0    9.0           1.0    1.0    1.0
      0.0156      9.0    0.0    9.0    9.0    0.0    0.0           2.0    8.0    0.0           3.0    0.0    2.067       0.2500      9.0    8.0    6.0    9.0    5.0    3.0           5.0    9.0    3.0           5.0    2.0    6.0
      0.1250      9.0    5.0    1.0    9.0    5.0    1.0           0.0    9.0    4.0           5.0    3.0    3.0
      0.0625      9.0    2.0    9.0    9.0    7.0    0.0           0.0    9.0    1.0           1.0    2.0    2.0
      0.0313      9.0    3.0    9.0    9.0    0.0    0.0           0.0    8.0    0.0           0.0    0.0    1.0
      0.0156      9.0    1.0    9.0    0.0    0.0    0.0           0.0    7.0    0.0           1.0    0.0    0.068       0.2500      9.0    7.0    9.0    9.0    0.0    5.0           3.0    9.0    0.0           1.0    0.0    2.0
      0.1250      7.0    4.0    2.0    9.0    0.0    0.0           0.0    7.0    1.0           0.0    0.0    0.0
      0.0625      3.0    0.0    3.0    9.0           0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0313      1.0    0.0    0.0    9.0    0.0    1.0           0.0    2.0    1.0           0.0    0.0    0.0
      0.0156      0.0    0.0           9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X69       0.2500      9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    2.0    5.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.0           9.0    1.0    6.0
      0.0625      9.0    9.0    9.0    9.0    6.0    9.0           7.0    9.0    5.0           7.0    1.0    5.0
      0.0313      9.0    9.0    0.0    9.0    0.0    9.0           6.0    9.0                  6.0    1.0    1.0
      0.0156      9.0    7.0    0.0    9.0    0.0    6.0           0.0    7.0    1.0           2.0    3.0    0.070       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    5.0           8.0    2.0    7.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0                  7.0    2.0    4.0
      0.0625      9.0    9.0    9.0    9.0    9.0    9.0           4.0    9.0    4.0           7.0    1.0    3.0
      0.0313      9.0    9.0    9.0    9.0    7.0    4.0           2.0    7.0    4.0           3.0    1.0    1.0
      0.0156      9.0    7.0    0.0    9.0    0.0    5.0           0.0    4.0    6.0           5.0    1.0    0.071       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    4.0    6.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    2.0    4.0
      0.0625      9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    5.0           6.0    2.0    4.0
      0.0313      9.0    7.0    9.0    9.0    3.0    0.0           1.0    9.0    1.0           1.0    1.0    2.0
      0.0156      7.0    5.0    0.0    9.0    3.0                  0.0    5.0    0.0           1.0    1.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X72       0.2500      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    7.0           8.0    4.0    6.0
      0.0625      9.0    9.0    9.0    9.0    6.0    4.0           5.0    9.0    6.0           2.0    1.0    1.0
      0.0313      9.0    9.0    9.0    9.0    0.0    2.0           1.0    5.0    1.0           1.0    1.0    2.0
      0.0156      1.0    1.0    9.0    9.0    0.0    0.0           0.0    4.0    0.0           1.0    0.0    0.073       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.0           8.0    5.0    6.0
      0.1250      9.0    9.0    8.0    9.0    4.0    9.0           9.0    9.0    9.0           7.0    5.0    5.0
      0.0625      9.0    9.0    2.0    9.0    0.0    4.0           3.0    4.0    9.0           6.0    6.0    5.0
      0.0313      9.0    5.0    9.0    9.0    0.0    5.0           0.0    5.0    5.0           4.0    5.0    4.0
      0.0156      9.0    0.0    3.0    9.0    0.0    0.0           0.0           0.0           1.0    1.0    0.074       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    4.0    5.0
      0.1250      9.0    9.0    9.0    9.0    7.0    0.0           9.0    9.0    3.0           6.0    3.0    4.0
      0.0625      9.0    9.0    9.0    9.0    5.0    9.0           7.0    9.0                  5.0    3.0    2.0
      0.0313      9.0    9.0    9.0    9.0    5.0    9.0           4.0    9.0    3.0           4.0    5.0    0.0
      0.0156      9.0    3.0    0.0    9.0    0.0    0.0           0.0    6.0    3.0           1.0    1.0    1.0
                                                 表II(续)
                                                                                  G             O      T
                  A      A      C      C      G      I      I      E       S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C       E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H       T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C       V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G       I      W      A      T      R      X75       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0     9.0    9.0           9.0    3.0    5.0
      0.1250      9.0    9.0    7.0    9.0    7.0    9.0           8.0     7.0    4.0           7.0    3.0    4.0
      0.0625      9.0    9.0    4.0    9.0    6.0    4.0           7.0     9.0    3.0           7.0    3.0    3.0
      0.0313      9.0    9.0    3.0    9.0    6.0    9.0           5.0     9.0                  4.0    2.0    3.0
      0.0156      9.0    5.0    9.0    9.0    0.0    9.0           2.0     7.0    4.0           2.0    6.0    3.076       0.2500      9.0    9.0    9.0    9.0    8.0    9.0           9.0     9.0    9.0           9.0    4.0    4.0
      0.1250      9.0    9.0    2.0    9.0    5.0    9.0           7.0     9.0    5.0           8.0    3.0    5.0
      0.0625      9.0    9.0    9.0    9.0    3.0    5.0           9.0     9.0    4.0           7.0    2.0    4.0
      0.0313      9.0    7.0    4.0    9.0    3.0    9.0           3.0     7.0    5.0           5.0    1.0    4.0
      0.0156      9.0    0.0    2.0    9.0    3.0    3.0           1.0     9.0    0.0           1.0    2.0    1.077       0.5000      9.0    9.0    9.0    9.0    9.0    9.0           9.0     9.0    9.0           8.0    8.0    8.0
      0.2500      9.0    9.0    9.0    9.0    8.3    9.0           6.0     9.0    7.7           8.0    6.3    7.7
      0.1250      9.0    9.0    6.0    9.0    8.3    9.0           4.3     9.0    6.3           7.7    3.7    5.7
      0.0625      9.0    9.0    0.7    9.0    1.5    9.0           0.7     8.3    3.7           5.0    3.3    4.3
      0.0313      9.0    6.7    0.0    9.0    0.0    4.0           0.0     5.3    1.3           2.0    0.0    1.7
      0.0156      7.7    0.0    0.0    7.3    0.0    1.0           0.0     0.0    0.0           0.7    0.0    0.7
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X78       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    6.0           7.0    5.0    8.0
      0.1250      9.0    9.0    0.0    9.0    8.0    9.0           7.0    9.0    5.0           5.0    2.0    7.0
      0.0625      7.0    9.0    0.0    9.0    9.0    3.0           0.0    9.0    1.0           2.0    0.0    6.0
      0.0313             4.0    0.0    9.0    0.0    0.0           0.0    7.0                  0.0    0.0    0.0
      0.0156      5.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.079       0.2500      9.0    9.0    5.0    9.0    5.0    9.0           6.0    9.0    7.0           7.0    3.0    7.0
      0.1250      9.0    9.0    5.0    9.0    4.0    9.0           5.0    9.0    9.0           6.0    1.0    6.0
      0.0625      8.0    7.0    0.0    9.0    4.0    2.0           3.0    7.0    3.0           3.0    0.0    2.0
      0.0313      8.0    9.0    0.0    9.0    0.0    2.0           0.0    7.0    3.0           1.0    0.0    2.0
      0.0156      8.0    9.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.080       0.2500      9.0    9.0    0.0    9.0    9.0    9.0           5.0    9.0    9.0           8.0    4.0    8.0
      0.1250      9.0    9.0    0.0    9.0    9.0    9.0           3.0    9.0    3.0           8.0    2.0    6.0
      0.0625      9.0    9.0    0.0    9.0    0.0    2.0           0.0    9.0    3.0           2.0    0.0    3.0
      0.0313      9.0    0.0    0.0    9.0    0.0                  0.0    6.0    0.0           0.0    0.0    2.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    2.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X81       0.2500      9.0    9.0    5.0    9.0    9.0    9.0           5.0    9.0    9.0           6.0    3.0    8.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    7.0           5.0    1.0    7.0
      0.0625      9.0    6.0    9.0    9.0    3.0    9.0           0.0    5.0    0.0           3.0    0.0    4.0
      0.0313      9.0    9.0    3.0    9.0    3.0    9.0           0.0    2.0    0.0           1.0    0.0    3.0
      0.0156      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           1.0    0.0    0.082       0.2500      9.0    9.0    0.0    9.0    0.0    9.0           5.0    9.0    1.0           5.0    1.0    3.0
      0.1250      9.0    9.0    0.0    9.0    4.0    3.0           4.0    9.0    0.0           2.0    0.0    1.0
      0.0625      9.0    0.0    0.0    9.0    3.0    0.0           0.0    9.0    0.0           0.0    0.0    0.0
      0.0313      5.0    0.0    0.0    9.0    0.0    0.0           0.0    9.0    0.0           0.0    0.0    5.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.083       0.2500      9.0    9.0    9.0    9.0    3.0    9.0           7.0    9.0    9.0           7.0    3.0    7.0
      0.1250      9.0    9.0    3.0    9.0    3.0    9.0           7.0    9.0    5.0           7.0    3.0    5.0
      0.0625      9.0    9.0    3.0    9.0    0.0    9.0           6.0    9.0                  5.0    1.0    5.0
      0.0313      9.0    9.0    0.0    9.0    0.0    9.0           3.0    7.0    5.0           7.0    1.0    5.0
      0.0156      9.0    9.0    0.0    9.0    0.0    0.0           0.0    3.0    5.0           2.0    0.0    5.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X84       0.2500      9.0    9.0    3.0    9.0    2.0    9.0           9.0    9.0    9.0           7.0    1.0    7.0
      0.1250      9.0    9.0    0.0    9.0    0.0    9.0           7.0    9.0    9.0           6.0    0.0    4.0
      0.0625      9.0    9.0    0.0    9.0    0.0    9.0           4.0    9.0    9.0           6.0    0.0    3.0
      0.0313      9.0    0.0    0.0    9.0    0.0    4.0           0.0    0.0    9.0           6.0    0.0    3.0
      0.0156      5.0    0.0    0.0    0.0    0.0    2.0           0.0    0.0    5.0           3.0    0.0    3.085       0.2500      9.0    9.0    0.0    9.0    0.0    7.0           3.0    9.0    3.0           5.0    0.0    6.0
      0.1250      9.0    0.0    0.0    9.0    0.0    3.0           0.0    3.0    3.0           1.0    0.0    3.0
      0.0625      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    3.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    3.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.086       0.2500      9.0    9.0    3.0    9.0    0.0    9.0           9.0    9.0    5.0           7.0    2.0    4.0
      0.1250      9.0    9.0    3.0    9.0    0.0    9.0           7.0    9.0                  7.0    0.0    4.0
      0.0625      9.0    3.0    0.0    9.0    0.0    4.0           3.0    9.0                  7.0    0.0    3.0
      0.0313      4.0    0.0    0.0    9.0    0.0    0.0           0.0    3.0    0.0           3.0    0.0    3.0
      0.0156      3.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X87       0.2500      9.0    9.0    3.0    9.0    6.0    9.0           8.0    9.0    9.0           6.0    2.0    8.0
      0.1250      9.0    0.0    9.0    9.0    9.0    9.0           7.0    9.0    3.0           5.0    1.0    7.0
      0.0625      9.0    0.0    3.0    9.0    0.0    9.0           5.0    7.0                  7.0    0.0    7.0
      0.0313      5.0           0.0    9.0    0.0    9.0           2.0    5.0    3.0           7.0    0.0    3.0
      0.0156      3.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    3.0           2.0    0.0    3.088       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    9.0           7.0    4.0    7.0
      0.1250      9.0    9.0    0.0    9.0    0.0    9.0           4.0    9.0    3.0           3.0    0.0    7.0
      0.0625      9.0    9.0    0.0    9.0    0.0    9.0           3.0    9.0    3.0           1.0    0.0    5.0
      0.0313      9.0    9.0           9.0    0.0    9.0           2.0    9.0    3.0           0.0    0.0    2.0
      0.0156      9.0    3.0    0.0    9.0    0.0    4.0           0.0    3.0    0.0           0.0    0.0    1.089       0.2500      9.0    9.0    2.0    9.0    7.0    4.0           9.0    9.0    6.0           7.0    3.0    6.0
      0.1250      9.0    9.0    0.0    9.0    6.0    9.0           5.0    9.0                  3.0    1.0    6.0
      0.0625      9.0    9.0    0.0    9.0    0.0    0.0           2.0    0.0    3.0           3.0    0.0    2.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           2.0    0.0    2.0
      0.0156      0.0    0.0    0.0           0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X90       0.2500      9.0    9.0    2.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    2.0    5.0
      0.1250      9.0    9.0    0.0    9.0    9.0    9.0           5.0    9.0    9.0           6.0    1.0    4.0
      0.0625      5.0    9.0    0.0    9.0    0.0    9.0           0.0    5.0    2.0           2.0    0.0    3.0
      0.0313      5.0    9.0    0.0    9.0    0.0    3.0           0.0    0.0    1.0           1.0    0.0    1.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0                  0.0    0.0    0.091       0.2500      2.0    2.0    1.0    9.0    3.0    0.0           0.0    9.0    1.0           1.0    0.0    1.0
      0.1250      0.0    0.0    0.0    0.0    0.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.092        0.2500      9.0    9.0    5.0    9.0    4.0    9.0           5.0    9.0    5.0           7.0    7.0    7.0
      0.1250      9.0    9.0    9.0    9.0    4.0    9.0           5.0    9.0                  7.0    3.0    7.0
      0.0625      9.0    9.0    5.0    9.0    2.0    3.0           5.0    6.0    3.0           7.0    1.0    3.0
      0.0313      9.0    4.0    2.0    0.0    0.0    0.0           0.0    0.0                  5.0    0.0    2.0
      0.0158      6.0    4.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           6.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X93       0.2500      9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    6.0           8.0    7.0    9.0
      0.1250      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    3.0           8.0    7.0    9.0
      0.0625      9.0    3.0    6.0    9.0    0.0    9.0           3.0    9.0    3.0           6.0    6.0    4.0
      0.0313      9.0           2.0    9.0    0.0    3.0           2.0    9.0    3.0           1.0    0.0    2.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    6.0    0.0           0.0    0.0    1.094       0.2500      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    2.0           0.0    0.0    0.0
      0.1250      0.0    0.0    0.0    8.0    0.0    0.0           0.0    0.0    2.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0           0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.095       0.2500      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.0           0.0    0.0    2.0
      0.1250      0.0    0.0    0.0           0.0    0.0           0.0    0.0    2.0           0.0    0.0    2.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    2.0           0.0    0.0    2.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X96       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           3.0    8.0    3.0           3.0    9.0    6.0
      0.1250      9.0    0.0    9.0    9.0    0.0    3.0           0.0    6.0    5.0           1.0    4.0    6.0
      0.0625      3.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.0           0.0    0.0    5.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    3.0           0.0    0.0    5.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.097       0.2500      9.0    9.0    6.0    9.0    9.0    9.0           9.0    9.0    5.0           9.0    8.0    7.0
      0.1250      9.0    9.0    6.0    9.0    9.0    9.0           3.0    9.0    5.0           7.0    3.0    5.0
      0.0625      9.0    9.0    0.0    9.0    0.0    0.0           3.0    9.0    5.0           7.0    3.0    5.0
      0.0313      9.0    3.0    0.0    9.0    0.0    0.0           0.0    7.0    2.0           5.0    1.0    5.0
      0.0156      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           3.0    0.0    3.098       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    8.0    8.0
      0.1250      9.0    9.0    9.0    9.0    8.0    9.0           6.5    9.0    8.5           7.5    7.5    6.5
      0.0625      9.0    8.0    7.0    9.0    4.5    7.0           3.0    8.0    8.0           5.0    5.0    4.5
      0.0313      9.0    6.5    6.0    9.0    4.5    4.0           0.0    0.0    6.0           2.5    1.0    0.0
      0.0156      9.0    2.5    0.0    9.0    4.5    1.5           0.0    0.0    2.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X99       0.2500      9.0    7.0    7.0    9.0    0.0    2.0           4.0    6.0    9.0           7.0    5.0    4.0
      0.1250      9.0    2.0    3.0    9.0    0.0    0.0           0.0    2.0    3.0           2.0    3.0    4.0
      0.0625      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0100      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    9.0    9.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    9.0           8.0    9.0    7.5
      0.0625      9.0    9.0    9.0    9.0    8.0    9.0           2.0    5.5    9.0           6.0    6.0    5.5
      0.0313      9.0    7.5    9.0    9.0    5.0    9.0           0.5    5.0    8.0           3.0           2.5
      0.0156      9.0    8.0    0.5    9.0    4.0    4.5           0.0    0.0    4.5           0.5           0.5101      0.2500      9.0    2.0    0.0    9.0    9.0    0.0           0.0    0.0    0.0           8.0    9.0    1.0
      0.1250      3.0    0.0    0.0    9.0    5.0    0.0           0.0    0.0                  0.0    9.0    0.0
      0.0625      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0                  0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X102      0.2500      9.0    9.0    0.0    9.0    5.0    9.0           0.0    6.0    0.0           0.0    0.0    0.0
      0.1250      9.0    7.0    0.0    9.0    6.0    3.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0625      8.0    2.0    0.0           3.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    9.0    0.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0103      0.5000      9.0    9.0    9.0    9.0           9.0           9.0    9.0    3.0                         5.0
      0.2500      9.0    9.0    7.3    9.0    7.5    9.0           8.8    9.0    5.8           8.5    6.5    6.3
      0.1250      9.0    9.0    3.5    9.0    2.5    9.0           8.5    9.0    5.5           6.0    5.0    3.8
      0.0625      9.0    8.3    2.3    9.0    0.5    7.6           4.3    8.8    5.3           4.0    3.0    2.8
      0.0313      9.0    2.5    1.3    9.0    0.5    6.8           1.3    5.8    2.3           0.5    0.5    1.8
      0.0156      6.3    3.7    0.0    9.0    0.0    4.3           0.0    2.0    2.0           1.5    0.5    0.7104      0.2500      9.0    9.0    9.0    8.0    9.0    9.0           5.5    9.0    7.5           8.5    8.5    6.5
      0.1250      9.0    9.0    4.0    9.0    8.0    8.0           0.5    6.0    7.0           5.5    6.5    4.0
      0.0625      9.0    3.5    1.0    8.5    0.5    4.0           0.5    1.5    2.0           5.5    5.5    2.0
      0.0313      5.0    2.0    3.5    7.5    1.0    2.5           0.0    0.0    1.5           5.5    0.5    2.0
      0.0156      6.0    0.0    2.0    7.5    0.0    1.5           0.0    0.0    1.5           1.0    0.5    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X105      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    8.5    7.5
      0.1250      9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    9.0           7.0    7.0    7.0
      0.0625      9.0    9.0    9.0    9.0    6.0    7.5           9.0    9.0    7.5           6.5    6.5    6.0
      0.0313      9.0    7.5    7.0    9.0    4.5    7.5           8.0    9.0    7.5           5.5    5.0    8.0
      0.0156      6.0    6.5    4.5    9.0    3.0    4.5           5.5    9.0    3.0           6.5    4.5    5.0106      0.2500      9.0    2.0    3.0    9.0    7.0    2.0           0.0    2.0    3.0           3.0    0.0    1.0
      0.1250      9.0    1.0    0.0    9.0    5.0    1.0           0.0    2.0    1.0           3.0    0.0    0.0
      0.0625      0.0    0.0    0.0    9.0    5.0                  0.0    0.0    0.0           3.0    0.0    0.0
      0.0313      0.0    0.0    0.0    5.0    0.0    0.0           0.0    0.0    0.0           3.0    0.0    0.0
      0.0156      0.0    0.0    0.0    5.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0107      0.2500      9.0    9.0    7.0    9.0    9.0    9.0           8.0    9.0    7.0           7.0    6.0    7.0
      0.1250      9.0    9.0    5.0    9.0    7.0    8.5           8.0    9.0    3.0           6.0           5.5
      0.0625      8.5    6.0    4.5    9.0    6.0    9.0           6.0    9.0    4.0           5.0    3.0    5.0
      0.0313      4.5    4.0    1.0    9.0    0.0    4.5           2.0    7.5    2.5           3.0    1.0    2.5
      0.0156      1.5    1.0    3.0    8.0    3.0    2.0           0.5    0.5    1.5           1.0    1.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X108      0.2500      9.0    9.0    8.0    9.0    9.0    9.0           7.0    9.0    5.0           6.0    2.0    5.0
      0.1250      9.0    9.0    4.5    9.0    6.0    7.5           5.5    9.0    2.5           7.0    5.0    5.5
      0.0625      8.0    7.0    9.0    9.0    4.0    7.5           3.5    7.5    1.5           6.0    4.0    3.0
      0.0313      8.0    6.0    1.0    9.0    6.0    1.5           0.5    2.5    1.5           0.5    1.0    0.5
      0.0156      1.0    3.5    0.0    9.0    5.0    0.5           0.0    0.5    0.5           0.5    1.0    0.5109      0.2500      9.0    9.0    9.0    9.0    6.0    8.0           9.0    9.0    9.0           8.0    7.0    7.0
      0.1250      9.0    9.0    5.0    9.0    7.0    9.0           8.0    9.0    6.0           5.0    4.0    4.0
      0.0625      7.0    9.0    3.0    9.0    7.0    4.0           7.0    8.0    3.0           6.0    2.0    4.0
      0.0313      4.0    6.0    3.0    9.0    3.0    9.0           4.0    6.0    5.0           7.0    1.0    2.0
      0.0156      2.0    1.0    4.0    9.0    1.0    4.0           2.0    5.0    1.0           3.0    1.0    1.0110      0.2500      9.0    9.0    8.3    9.0    9.0    9.0           8.7    9.0    7.7           7.3    7.5    8.0
      0.1250      9.0    8.7    9.0    9.0    9.0    9.0           8.3    9.0    8.0           6.0    6.0    7.7
      0.0625      9.0    7.3    4.0    9.0    7.0    6.3           8.0    9.0    6.7           6.3    5.5    7.0
      0.0313      9.0    4.7    4.0    9.0    1.5    7.5           6.7    8.7    3.0           3.3    3.5    5.7
      0.0156      8.0    0.7    4.5    9.0    0.0    4.0           3.7    5.3    1.3           1.7    3.0    4.3
                                                   表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X111      0.2500       9.0    9.0    7.0    9.0    9.0    6.0           7.0    9.0    7.0           7.0    6.0    7.0
      0.1250       9.0    9.0    9.0    9.0    7.0    8.0           7.0    9.0    7.0           7.0    6.0    7.0
      0.0625       9.0    9.0    7.0    9.0    7.0    7.0           5.0    7.0    7.0           7.0    4.0    6.0
      0.0313       9.0    7.0    1.0    9.0    6.0    2.0           1.0    5.0    4.0           2.0    1.0    1.0
      0.0156       6.0    6.0    1.0    7.0    2.0    2.0           0.0    3.0    1.0           2.0    1.0    1.0112      0.2500       9.0    2.0    7.0    9.0    4.0    6.0           0.0    7.0    5.0           1.0    1.0    1.0
      0.1250       5.0    2.0    2.0    9.0    4.0    4.0           1.0    6.0    2.0           0.0    0.0    1.0
      0.0625       5.0    0.0    1.0    9.0    3.0    0.0           0.0    1.0    1.0           0.0    0.0    0.0
      0.0313       4.0    0.0    0.0    7.0    3.0    0.0           0.0    1.0    1.0           0.0    1.0    1.0
      0.0156       0.0    0.0    1.0    6.0    2.0    0.0           0.0    1.0    0.0           0.0    0.0    0.0113      0.2500       9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    8.0    8.5
      0.1250       9.0    9.0    7.5    9.0    9.0    9.0           4.5    9.0    9.0           8.5    7.0    8.0
      0.0625       7.5    6.5    4.0    9.0    7.0    9.0           2.0    8.0    2.5           7.0    6.0    5.0
      0.0313       9.0    4.5    1.0    9.0    6.0    7.5           0.0    2.0    0.0           3.0    2.0    3.0
      0.0156       9.0    5.0    0.5    9.0    9.0    9.0           0.0    0.5    1.0           1.0    1.0    2.0
                                                   表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X114      0.5000       9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    8.0    8.0
      0.2500       9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    6.0    8.0
      0.1250       9.0    9.0    6.5    9.0    9.0    9.0           7.5    9.0    9.0           6.0    8.0    7.0
      0.0640       9.0    9.0    6.0    9.0           7.0           8.0    9.0    7.0           7.0           7.0
      0.0625       9.0    9.0    4.5    9.0    6.5    8.0           7.0    8.0    7.0           5.5    7.0    5.5
      0.0320       9.0    9.0    6.0    9.0           6.0           7.0    9.0    6.0           9.0           7.0
      0.0313       8.0    9.0    8.0    9.0    7.0    7.5           6.5    8.0    5.0           4.0    1.0    4.5
      0.0160       9.0    8.0    2.0    9.0           8.0           7.0    8.0    3.0           5.0           7.0
      0.0156       6.0    4.5    2.0    9.0    6.5    9.0           4.5    5.5    6.5           2.0    1.5    2.5115      0.5000       9.0    9.0    5.0    9.0    0.0    9.0           0.0    0.0    2.0           0.0    0.0    3.0
      0.2500       9.0    3.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.1250       0.0    3.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0625       0.0    3.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313       0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156       0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X116      0.5000      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.2500      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.1250      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0117      0.5000      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.2500      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.1250      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0118      0.2500      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.1250      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X119      0.5000      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.5    9.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    8.7
      0.0625      9.0    9.0    2.0    9.0    9.0    9.0           8.7    9.0    9.0           8.3    8.5    8.0
      0.0313      9.0    9.0    1.0    9.0    8.0    9.0           8.0    9.0    8.7           7.7    8.0    8.0
      0.0156      9.0    9.0    0.7    9.0    8.0    9.0           6.3    9.0    6.3           6.3    7.0    7.3120      0.2500      9.0    9.0    6.0    9.0    9.0    7.0           8.0    9.0    7.0           7.0    5.0    7.0
      0.1250      9.0    8.0    6.0    9.0    7.0    7.0           8.0    9.0    9.0           7.0    5.0    7.0
      0.0625      9.0    8.0    5.0    9.0    9.0    4.0           7.0    9.0    7.0           7.0    4.0    6.0
      0.0313      9.0    6.0    2.0    9.0    6.0    4.0           3.0    9.0    5.0           4.0    4.0    3.0
      0.0156      9.0    1.0    5.0    9.0    8.0    2.0           1.0    9.0    6.0           5.0    3.0    3.0121      0.2500      9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    9.0           8.0    7.0    4.0
      0.1250      9.0    9.0    8.0    9.0    9.0    9.0           7.5    9.0    8.0           7.0    7.0    6.0
      0.0625      9.0    9.0    6.5    9.0    6.0    9.0           4.5    8.0    6.0           6.5    2.0    4.5
      0.0313      9.0    9.0    5.0    9.0    5.0    9.0           3.0    7.5    6.0           5.5    2.0    3.5
      0.0156      9.0    8.0    5.5    9.0    5.0    7.0           1.0    3.0    4.5           3.0    6.0    2.5
                                                  表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X122      0.2500       9.0    9.0    6.5    9.0    8.5    9.0           2.5    9.0    7.0           4.0    4.5    4.0
      0.1250       9.0    9.0    6.7    9.0    4.5    9.0           2.3    8.3    5.3           2.7    3.0    3.3
      0.0625       9.0    8.7    3.3    9.0    3.0    4.3           1.0    6.3    3.3           1.0    0.0    1.7
      0.0313       9.0    4.3    3.3    9.0    3.0    4.5           0.3    3.3    2.3           0.7    0.0    1.3
      0.0156       9.0    3.0    1.5    9.0    0.0    3.3           0.3    2.3    2.3           0.3           1.3123      0.2500       9.0    7.5    8.0    9.0    8.0    9.0           1.5    9.0    4.5           1.0    2.5    4.0
      0.1250       9.0    4.5    3.0    9.0    6.0    6.5           0.5    8.0    2.0           2.5    2.5    4.0
      0.0625       9.0    3.5    6.0    9.0    2.5    9.0           0.5    9.0    3.0           1.0    1.5    3.0
      0.0313       9.0    1.5    1.5    9.0    2.0    0.5           0.0    2.0    0.0           1.5           0.5
      0.0156       6.5    1.0    0.5    9.0    2.5    1.0           0.0    0.5    1.0           0.5    0.0    1.0124      0.2500       9.0    9.0    6.5    9.0    9.0    9.0           3.5    9.0    5.0           1.5    1.5    2.5
      0.1250       9.0    5.5    4.0    9.0    4.5    6.5           1.0    9.0    3.5           2.0    1.0    2.5
      0.0625       7.5    6.0    0.0    9.0    3.0    1.0           0.0    4.5    1.0           1.0    1.0    1.0
      0.0313       9.0    1.5    2.5    9.0    2.0    0.0           0.0    2.0    1.0           1.0    0.5    2.0
      0.0156       5.0    0.0    2.5    9.0    0.0    0.0           0.0    2.0    0.0           2.0    0.0    2.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X125      0.5000      9.0    9.0    5.5    9.0    9.0    9.0           9.0    9.0    5.0           9.0    8.0    6.5
      0.2500      9.0    9.0    5.5    9.0    9.0    9.0           6.8    9.0    2.7           5.0    7.5    5.3
      0.1250      9.0    7.5    1.3    8.5    6.0    6.3           3.8    8.5    3.3           5.0    4.0    4.3
      0.0625      9.0    5.8    2.7    9.0    0.0    5.7           1.8    4.5    2.0           4.5    0.0    3.3
      0.0313      8.8    2.6    1.0    8.8    0.0    3.0           0.0    2.8    1.5           2.5    0.0    1.8
      0.0156      5.0    2.7    0.7    7.0    0.0    1.3           0.0    2.0    1.3           1.0    0.0    0.7126      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    7.0           9.0    7.0    7.0
      0.1250      9.0    5.0    7.0    9.0    9.0    9.0           5.0    9.0    6.0           7.0    9.0    4.0
      0.0625      9.0    3.0    2.0    9.0    7.0    6.0           1.0    9.0    9.0           7.0    9.0    4.0
      0.0313      9.0    3.0    7.0    9.0    7.0    3.0           0.0    7.0    7.0           8.0    2.0    1.0
      0.0156      9.0    1.0    7.0    9.0    6.0    0.0           0.0    6.0    2.0           1.0    1.0    1.0127      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           7.5    9.0    7.0           9.0    7.5    7.5
      0.1250      9.0    7.5    4.5    9.0    9.0    8.0           4.5    9.0    6.0           7.5    9.0    7.0
      0.0625      9.0    5.5    4.5    9.0    7.0    7.0           1.5    9.0    4.0           4.5    2.0    5.5
      0.0313      8.0    1.5    4.5    9.0    7.0    1.5           0.5    7.0    3.5           3.0    1.0    4.5
      0.0156      3.5    1.0    1.0    9.0    2.0    0.5           0.5    4.5    1.5           3.0    0.5    0.5
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X128      0.2500      9.0    9.0    8.0    9.0    9.0    9.0           6.5    9.0    7.5           8.0    8.0    8.0
      0.1250      9.0    8.5    4.5    9.0    7.5    9.0           2.0    8.0    4.0           8.0    7.5    6.0
      0.0625      9.0    7.0    7.5    6.0    7.0    9.0           2.5    4.0    4.5           6.5    6.0    4.5
      0.0313      7.5    3.5    2.5    9.0    8.0    4.5           0.0    1.0    2.5           4.0    3.5    1.5
      0.0156      2.0    0.0    0.0    3.0    7.0    2.0           0.5    0.5    2.5           2.0    1.0    3.0129      0.5000      9.0    9.0    9.0    9.0           9.0           9.0    9.0    7.0                         3.0
      0.2500      9.0    8.3    3.5    9.0    8.0    9.0           5.5    9.0    6.3           6.0    6.0    4.8
      0.1250      9.0    5.3    3.8    9.0    8.0    9.0           3.0    9.0    5.3           5.3    6.0    3.3
      0.0625      9.0    3.3    1.7    9.0    3.0    6.3           0.0    4.8    2.8           1.3    3.0    1.8
      0.0313      9.0    0.5    0.0    9.0    0.5    4.8           0.0    2.5    1.5           1.3    2.0    0.8
      0.0156      8.0    0.0    0.3    8.7    0.0    1.3           0.0    1.3    0.7           0.3    0.5    0.0130      0.2500      9.0    8.0    9.0    9.0    5.5    8.0           7.3    8.3    6.7           9.0    7.5    6.3
      0.1250      7.8    7.5    6.0    9.0    7.0    9.0           6.8    8.8    5.8           8.3    8.0    6.5
      0.0625      8.3    4.3    2.3    8.5    7.0    7.3           4.8    7.3    4.3           6.0    4.5    5.3
      0.0313      6.8    2.8    3.0    9.0    3.0    6.8           3.3    6.0    3.0           5.3    4.0    4.5
      0.0156      6.8    0.3    0.0    7.3    0.0    5.3           0.5    1.5    1.0           2.7    2.0    1.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X131      0.2500      8.3    9.0    3.7    9.0    9.0    9.0           8.7    9.0    6.7           8.5    8.0    6.7
      0.1250      9.0    8.8    5.0    9.0    9.0    9.0           7.5    8.5    6.5           8.7    7.0    6.8
      0.0625      9.0    6.0    0.0    9.0    8.0    7.3           5.3    6.8    5.8           7.0    6.0    6.3
      0.0313      9.0    4.5    0.0    9.0    6.0    6.0           3.8    5.0    3.5           6.0    1.0    4.5
      0.0156      6.8    2.0    0.7    7.3    2.0    4.7           1.3    2.8    1.5           2.7    2.0    1.3132      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    8.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           8.5    9.0    9.0           9.0    6.0    7.0
      0.0625      9.0    9.0    8.0    9.0    9.0    9.0           8.0    9.0    9.0           7.0    6.0    4.5
      0.0313      9.0    9.0    9.0    9.0    9.0    9.0           5.5    9.0    9.0           6.0    4.0    4.0
      0.0156      9.0    8.0    5.5    9.0    1.0    9.0           1.5    8.0    9.0           5.0    5.0    3.0133      0.5000      9.0    9.0    9.0    9.0           9.0           9.0    9.0    9.0                         8.0
      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           8.7    9.0    7.0           9.0    7.0    6.7
      0.1250      9.0    9.0    9.0    9.0    7.0    9.0           8.3    9.0    7.5           6.5    7.0    6.0
      0.0625      9.0    8.5    5.5    9.0    1.0    9.0           7.0    9.0    7.8           5.0    9.0    5.0
      0.0313      9.0    6.0    6.8    9.0    1.0    9.0           3.3    7.3    5.5           5.0    9.0    4.3
      0.0156      9.0    2.3    3.3    9.0    0.0    9.0           1.3    7.3    2.3           2.5    6.0    3.7
                                                  表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X134      0.2500       9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    7.0
      0.1250       9.0    9.0    9.0    9.0    6.0    9.0           9.0    9.0    9.0           8.5    6.0    7.0
      0.0625       8.0    9.0    7.5    9.0    1.0    9.0           7.5    9.0    9.0           8.0    5.0    8.0
      0.0313       9.0    9.0    6.0    9.0    0.0    9.0           4.0    9.0    9.0           8.0    4.0    5.0
      0.0156       9.0    7.5    4.5    9.0    1.0    9.0           2.0    5.0    5.0           4.5    5.0    3.0135      0.2500       9.0    9.0    9.0    9.0    5.0    9.0           7.0    9.0    9.0           8.0    9.0    7.0
      0.1250       9.0    9.0    1.0    9.0    5.0    9.0           3.0    9.0    7.0           3.5    3.0    6.0
      0.0625       9.0    8.5    0.0    9.0    5.0    9.0           1.5    9.0    4.5           4.5           4.0
      0.0313       9.0    3.0    0.0    9.0           6.0           0.5    3.5    2.5           4.5    4.0    3.5
      0.0156       9.0    0.0    0.0    9.0    0.0    5.5           0.0    1.5    2.5           1.0    3.0    3.5136      0.2500       7.0    4.0    0.0    9.0    0.0    3.0           0.0    4.0    3.0           1.0    0.0    1.0
      0.1250       5.0    0.0    0.0    7.0    1.0    0.0           0.0    1.0    3.0           1.0           0.0
      0.0625       3.0    2.0    0.0           0.0    0.0           0.0    0.0    1.0           3.0    3.0    0.0
      0.0313       0.0    0.0                  0.0    0.0           0.0    0.0    2.0           6.0           1.0
      0.0156       0.0    1.0    1.0    6.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X137      0.2500       9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    9.0    9.0
      0.1250       9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    9.0           7.0    8.0    9.0
      0.0625       9.0    9.0    7.0    9.0    9.0    9.0           7.0    9.0    9.0           8.0    8.0    8.0
      0.0313       9.0    9.0    7.0    9.0    9.0    9.0           7.0    9.0    8.0           7.0    8.0    8.0
      0.0156       9.0    9.0    2.0    9.0    7.0    9.0           4.0    9.0    5.0           7.0    7.0    6.0138      0.2500       9.0    9.0    7.5    9.0    9.0    9.0           6.5    9.0    9.0           7.0    5.0    6.5
      0.1250       9.0    7.5    7.0    9.0    5.0    9.0           2.0    7.5    8.0           4.0    1.5    3.5
      0.0625       9.0    9.0    5.0    9.0    4.5    8.0           0.0    2.5    2.0           0.5    0.5    2.5
      0.0313       2.0    1.5    0.0    9.0    4.5    4.5           0.0    0.0    2.5           0.5    0.5    1.0
      0.0156       0.5    1.0    0.0    8.5    0.0    4.0           0.0    0.0    1.0           1.5    0.5    0.5139      0.2500       6.0    6.0    1.0    9.0    9.0    3.0           5.0    9.0    4.0           9.0    5.0    1.0
      0.1250       4.0    3.0    1.0    9.0    9.0    1.0           3.0    8.0    6.0           6.0    1.0    1.0
      0.0625       4.0    4.0    1.0    9.0    3.0    2.0           1.0    9.0    5.0           4.0    4.0    1.0
      0.0313       3.0    4.0    0.0    9.0    3.0    1.0           2.0    5.0    1.0           5.0    4.0    1.0
      0.0156       0.0    4.0    0.0    9.0    7.0    1.0           2.0    4.0    1.0           5.0    2.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X140      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.5           9.0    9.0    9.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.5    7.0    8.0
      0.0625      9.0    9.0    6.0    9.0    9.0    9.0           8.7    9.0    7.7           7.5    7.0    7.7
      0.0313      9.0    8.3    5.0    9.0    9.0    8.3           6.7    9.0    7.0           6.5    6.0    6.0
      0.0156      9.0    8.0    3.7    9.0    9.0    8.0           4.0    9.0    5.0           3.5    5.0    5.3141      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    8.0           8.0    9.0    8.0
      0.1250      9.0    9.0    7.8    9.0    9.0    9.0           7.3    8.3    8.0           8.0    7.0    6.5
      0.0625      9.0    8.3    5.0    9.0    8.0    8.5           4.8    8.3    6.7           7.0    6.0    4.8
      0.0313      9.0    7.8    3.5    9.0    8.0    7.3           3.0    5.8    5.8           6.5    3.0    3.5
      0.0156      7.3    6.8    1.5    7.3    6.5    5.5           1.3    3.8    4.0           4.0    1.5    1.3142      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    5.0    7.0
      0.1250      9.0    9.0    5.0    9.0    8.0    9.0           8.0    9.0    9.0           3.0    3.0    5.0
      0.0625      9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    9.0           3.0           4.0
      0.0313      9.0    0.0    9.0    9.0    0.0    9.0           0.0    9.0    6.0           3.0    0.0    0.0
      0.0156      9.0    0.0    5.0    9.0    0.0    9.0           0.0    0.0    0.0           0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物  施用率        T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X143      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           2.0    8.0    0.0           8.0    8.0    5.0
      0.1250      9.0    7.0    6.0    9.0    9.0    9.0           0.0    5.0                  7.0    7.0    1.0
      0.0625      9.0    3.0    0.0    9.0    9.0    1.0           0.0    0.0    0.0           6.0    3.0    0.0
      0.0313      6.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           2.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0144      0.2500      9.0    3.0    8.0    7.0    0.0    9.0           1.0    9.0    0.0           4.0    0.0    0.0
      0.1250      9.0           0.0    7.0    0.0    3.0           0.0    5.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0145      0.2500      9.0    7.0    3.0    9.0    3.0    9.0           3.0    9.0    7.0           3.0    2.0    3.0
      0.1250      9.0    6.0    0.0    9.0           9.0           2.0    9.0    2.0           1.0    1.0    1.0
      0.0625      4.0    2.0           9.0    1.0    2.0           0.0    7.0    1.0           1.0    1.0    0.0
      0.0313      1.0    0.0    0.0    9.0    0.0    0.0           0.0    1.0    0.0           1.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X146      0.2500      9.0    7.0    1.0    9.0    9.0    9.0           3.0    9.0    1.0           4.0    1.0    3.0
      0.1250      9.0    7.0    1.0    9.0    6.0    9.0           0.0    4.0    1.0           1.0    0.0    1.0
      0.0625      9.0    5.0    1.0    9.0    2.0    9.0           0.0    2.0    1.0           1.0    0.0    1.0
      0.0313      9.0    2.0    0.0    9.0           0.0           0.0    0.0    1.0           1.0           1.0
      0.0156      0.0    2.0    0.0    9.0    0.0    0.0           0.0    0.0    1.0           1.0           1.0147      0.2500      9.0    7.0    2.0    7.0    9.0    9.0           0.0    1.0    1.0           4.0    9.0    1.0
      0.1250      9.0    4.0    0.0    9.0    6.0    9.0           0.0    1.0    1.0           1.0    9.0    0.0
      0.0625      9.0    2.0    0.0    9.0           1.0           0.0    0.0    1.0                  4.0    0.0
      0.0313      1.0    2.0    0.0    9.0           0.0           0.0    0.0    2.0           1.0    0.0    1.0
      0.0156      1.0    2.0    0.0    9.0           1.0           0.0    0.0    1.0           0.0    0.0    0.0146      0.2500      9.0    7.0    6.0    9.0    9.0    9.0           2.0    6.0    9.0           7.0    7.0    7.0
      0.1250      9.0    9.0    9.0    9.0    7.0    7.0           0.0    2.0    5.0           5.0    6.0    6.0
      0.0625      9.0    9.0    4.0    9.0           9.0           0.0    2.0    4.0           1.0    4.0    1.0
      0.0313      3.0    3.0    0.0    9.0           9.0           0.0    1.0    1.0           1.0    1.0    1.0
      0.0156             3.0    0.0    5.0    4.0    7.0           0.0    0.0    1.0           1.0    1.0    1.0
                                                 表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X149       0.2500      9.0    3.0    1.0    9.0    9.0    4.0           1.0    5.0    4.0           6.0    2.0    1.0
       0.1250      9.0    3.0    3.0    9.0    5.0    2.0           0.0    4.0    1.0           1.0           0.0
       0.0625      4.0    1.0    1.0    7.0    3.0    1.0           0.0    2.0    2.0           1.0    0.0    1.0
       0.0313      0.0    0.0    2.0    7.0    2.0    0.0           0.0    0.0    1.0           1.0    0.0    0.0
       0.0156      0.0    1.0    1.0    6.0           0.0           0.0    1.0    0.0           1.0    0.0    1.0150       0.2500      9.0    9.0    7.0    9.0    9.0    9.0           7.0    9.0    9.0           7.0    7.0    7.0
       0.1250      9.0    9.0    7.0    9.0    9.0    9.0           3.0    9.0    9.0           6.0    6.0    7.0
       0.0625      9.0    7.0    6.0    9.0    2.0    9.0           1.0    4.0    6.0           7.0    6.0    4.0
       0.0313      9.0    3.0    3.0    9.0    4.0    4.0           1.0    1.0    3.0           4.0    3.0    1.0
       0.0156      9.0    2.0    1.0    9.0    3.0    0.0           0.0    1.0    1.0           4.0    1.0    0.0151       0.5000      0.0    0.0    0.0    9.0    3.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.2500      0.0    0.0    0.0    2.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.1250      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0625      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0313      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X152      0.2500      0.0    3.0    2.0    9.0    0.0    0.0           0.0    0.0    2.0           0.0    0.0    2.0
      0.1250      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0625      0.0    0.0    0.0    7.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0                  0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0153      0.2500      9.0    9.0    9.0    9.0    7.0    9.0           5.0    9.0    3.0           3.0    9.0    6.0
      0.1250      9.0    9.0    4.0    8.0    3.0    9.0           0.0    5.0    3.0           0.0    0.0    4.0
      0.0625      9.0    3.0    0.0    9.0    3.0    2.0           0.0    0.0                  0.0    0.0    0.0
      0.0313      9.0    0.0    0.0    9.0    3.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      9.0    0.0           9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0154      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    9.0           8.0    8.0    7.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           0.0    6.0    7.0           8.0    7.0    5.0
      0.0625      9.0    9.0    4.0    9.0    0.0    9.0           0.0    0.0                  3.0           2.0
      0.0313      3.0    0.0    4.0    0.0    0.0    0.0           0.0    0.0    0.0           3.0    4.0    0.0
      0.0156      0.0    0.0    0.0           0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X155      0.5000      9.0    9.0    9.0    9.0    9.0    9.0           3.0    9.0    9.0           4.0    8.0    8.0
      0.2500      9.0    9.0    9.0    9.0    7.0    9.0           2.0    7.0    9.0           2.0    6.0    2.0
      0.1250      9.0    9.0    9.0    9.0    7.0    9.0           0.0    3.0    9.0           0.0    4.0    0.0
      0.0625      9.0    3.0    2.0    9.0    7.0    9.0           0.0    1.0    5.0           0.0    3.0    0.0
      0.0313      9.0    0.0           0.0    0.0    9.0           0.0    0.0                  0.0    2.0    0.0
      0.0156      9.0    0.0                  0.0    0.0           0.0    0.0    0.0           0.0    1.0    0.0156      0.2500      9.0    6.0    2.0    9.0    7.0    6.0           2.0    6.0    1.0           2.0    1.0    1.0
      0.1250      6.0    2.0           9.0    6.0    3.0           1.0    3.0    1.0           1.0    1.0    1.0
      0.0625      4.0    3.0    1.0    7.0    0.0    1.0           1.0    3.0    1.0           0.0    0.0    0.0
      0.0313      1.0    0.0    0.0           0.0    1.0           0.0    1.0    1.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    0.0    0.0    1.0           0.0    1.0    1.0           0.0    0.0    0.0157      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           6.0    9.0    7.0           7.0    7.0    8.0
      0.1250      9.0    9.0    4.0    9.0    7.0    9.0           4.0    9.0    9.0           8.0    6.0    7.0
      0.0625      9.0    6.0    2.0    6.0    6.0    9.0           3.0    4.0    4.0           6.0    5.0    3.0
      0.0313      9.0    4.0    0.0                  3.0           0.0    1.0    3.0           3.0    2.0    1.0
      0.0156      6.0    2.0    0.0           0.0    3.0           0.0    1.0    2.0           1.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X158      0.2500      9.0    9.0    6.0    9.0    5.0    9.0           7.0    9.0    5.0           5.0    6.0    7.0
      0.1250      9.0    7.0    3.0    9.0    9.0    9.0           5.0    9.0    5.0           2.0    4.0    5.0
      0.0625      9.0    3.0    0.0    9.0    1.0    5.0           2.0    6.0    3.0           1.0    2.0    4.0
      0.0313      9.0    2.0    0.0    9.0    0.0    1.0           1.0    2.0    1.0           1.0    1.0    2.0
      0.0156      3.0    0.0    0.0    9.0    0.0    0.0           0.0    1.0    1.0           0.0    0.0    0.0159      0.2500      9.0    9.0    3.0    9.0    7.0    9.0           5.0    6.0    9.0           4.0    5.0    6.0
      0.1250      9.0    7.0    6.0    9.0    7.0    9.0           1.0    4.0    7.0           2.0    3.0    2.0
      0.0625      9.0    4.0    1.0    9.0    6.0    7.0           0.0    1.0    5.0                  1.0    0.0
      0.0313      9.0    2.0    1.0    9.0    3.0    4.0           0.0    1.0    3.0           0.0    0.0    1.0
      0.0156      5.0    2.0    0.0    9.0    2.0    3.0           1.0    0.0    1.0           0.0    0.0    1.0160      0.2500      4.0    4.0    0.0    9.0    9.0    4.0           0.0    0.0    5.0           2.0    2.0    2.0
      0.1250      3.0    2.0    0.0    9.0    6.0    0.0           0.0    1.0    5.0           0.0    1.0    1.0
      0.0625      1.0    2.0    0.0    9.0    6.0                  0.0    1.0    4.0           1.0    1.0    0.0
      0.0313      1.0    0.0    0.0    9.0    1.0    0.0           1.0    1.0    2.0           1.0    0.0    0.0
      0.0156      0.0    0.0    0.0    5.0    0.0    0.0           0.0    0.0    1.0           0.0    1.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X161      0.2500      9.0    9.0    4.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.0    9.0
      0.1250      9.0    7.0    4.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    5.0    8.0
      0.0625      9.0    6.0    1.0    9.0    6.0    9.0           9.0    9.0    6.0           5.0    5.0    7.0
      0.0313      9.0    3.0    1.0    9.0    6.0    4.0           3.0    9.0    6.0           2.0    3.0    5.0
      0.0156      6.0    2.0    1.0    9.0    3.0    2.0           2.0    7.0    5.0           1.0    0.0    1.0170      0.2500      9.0    9.0    9.0    9.0    8.5    9.0           8.0    9.0    8.0           8.0    8.0    7.0
      0.1250      9.0    9.0    7.5    9.0    6.0    8.0           6.5    9.0    9.0           7.5    2.5    5.5
      0.0625      9.0    8.5    3.5    9.0    0.0    9.0           6.0    9.0    4.5           7.0    2.5    5.5
      0.0313      9.0    4.5    3.5    9.0    2.5    8.0           4.5    9.0    2.5           5.5    2.0    5.0
      0.0156      9.0    2.0    0.5    9.0    0.0    3.0           2.0    4.0    2.0           2.5    2.5    2.5171      0.2500      9.0    6.0    6.0    9.0    3.0    9.0           6.0    9.0    5.0           9.0    4.0    6.0
      0.1250      9.0    7.0    4.0    9.0           4.0           5.0    8.0    5.0           5.0    5.0    6.0
      0.0625      9.0    4.0    4.0    9.0           6.0           4.0    4.0    5.0           6.0           5.0
      0.0313      5.0    4.0    3.0    9.0    5.0    3.0           2.0    4.0    5.0           5.0    3.0    5.0
      0.0156             0.0    2.0    9.0    3.0    3.0           0.0    1.0    4.0           2.0           0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X172      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    7.0    7.0
      0.1250      9.0    9.0    5.0    9.0    9.0    9.0           8.0    9.0    5.0           8.0    6.0    5.0
      0.0625      9.0    9.0    4.0    9.0    7.0    5.0           7.0    9.0                  7.0    7.0    4.0
      0.0313      9.0    7.0    4.0    9.0    3.0    6.0           5.0    8.0    4.0           7.0    5.0    5.0
      0.0156      9.0    6.0    4.0    9.0    5.0    3.0           2.0    4.0    4.0           4.0    2.0    2.0173      0.5000      9.0    9.0    9.0    9.0    7.0    9.0           8.0    9.0    9.0           9.0    8.0    6.0
      0.2500      9.0    9.0    4.0    9.0    8.0    9.0           7.0    9.0    5.0           7.0    8.0    6.5
      0.1250      9.0    6.5    3.5    9.0    7.0    8.0           4.5    8.0    6.0           8.0    5.0    5.5
      0.0625      9.0    5.0    2.5    7.0    2.0    6.5           3.5    7.0    3.5           5.0    3.5    5.0
      0.0313      9.0    3.5    1.5    9.0    2.0    6.5           2.0    3.5    2.0           1.5    1.5    3.5
      0.0156      8.0    1.0    1.5    9.0    2.0    2.0           1.0    1.0    2.5           1.5    1.5    2.5174      0.5000      9.0    9.0    6.0    9.0    9.0    9.0           8.0    8.5    6.5           8.0    9.0    6.5
      0.2500      9.0    9.0    6.3    9.0    8.0    9.0           7.0    8.5    6.3           8.5    5.0    6.0
      0.1250      9.0    7.5    3.0    9.0    5.5    9.0           3.5    7.0    5.0           7.0    4.0    3.8
      0.0625      8.8    6.3    2.0    9.0    4.5    5.0           1.8    3.5    2.8           7.0    3.5    4.5
      0.0313      8.3    4.3    1.3    8.3    1.5    2.3           1.0    2.8    1.8           5.0    3.0    2.8
      0.0156      9.0    2.7    1.0    8.3    0.5    2.0           1.0    2.3    2.0           3.5    2.5    1.7
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X175       0.2500     9.0    9.0    6.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    7.0    7.0
       0.1250     9.0    9.0    6.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    7.0    6.0
       0.0625     9.0    7.0    3.0    9.0    2.0    9.0           5.0    5.0    5.0           6.0    6.0    5.0
       0.0313     9.0    6.0    4.0    9.0    2.0    5.0           4.0    5.0    4.0           5.0    4.0    4.0
       0.0156     9.0    6.0    5.0    7.0    5.0    4.0           3.0    2.0    5.0           7.0    4.0    8.0176       0.5000     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    5.0           9.0    9.0    9.0
       0.2500     9.0    9.0    7.5    9.0    4.5    9.0           7.0    9.0    9.0           8.0    7.5    7.0
       0.1250     9.0    9.0    7.0    9.0    4.5    9.0           7.0    9.0    6.0           8.5    4.5    7.5
       0.0625     9.0    8.0    1.0    9.0    2.0    9.0           3.5    6.0    4.0           8.0    4.0    5.5
       0.0313     9.0    3.5    3.5    9.0    0.5    6.5           1.0    3.5    2.5           6.5    4.0    5.5
       0.0156     9.0    2.0    0.5    9.0    2.5    2.0           0.5    3.0    3.0           3.5    3.0    3.5177       0.2500     9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    6.0    7.0
       0.1250     9.0    9.0    8.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    5.0    7.0
       0.0625     9.0    9.0    6.0    9.0    9.0    8.0           6.0    9.0    6.0           8.0    4.0    7.0
       0.0313     9.0    7.0    6.0    9.0    9.0    9.0           5.0    6.0    5.0           8.0    4.0    7.0
       0.0156     9.0    6.0    6.0    9.0    6.0    9.0           4.0    5.0                  6.0    1.0    5.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X178      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    3.0    7.0
      0.1250      9.0    9.0    5.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    3.0    6.0
      0.0625      9.0    9.0    4.0    9.0    9.0    9.0           6.0    8.0    5.0           6.0    2.0    6.0
      0.0313      9.0    9.0    6.0    9.0    8.0    8.0           5.0    6.0    6.0           7.0    3.0    6.0
      0.0156      9.0    2.0    5.0    9.0    2.0    5.0           2.0    6.0    7.0           7.0    2.0    5.0179      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.5    8.5
      0.1250      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    8.5    8.5
      0.0640      9.0    9.0    7.0    9.0           9.0           9.0    9.0    7.0           8.0           8.0
      0.0625      9.0    9.0    7.0    9.0    9.0    8.0           9.0    9.0    9.0           8.5    8.0    8.0
      0.0320      9.0    9.0    7.0    9.0           7.0           8.0    9.0    7.0           7.0           7.0
      0.0313      9.0    8.0    7.0    9.0    8.0    7.5           8.0    7.5    6.0           7.5    7.0    7.5
      0.0160      9.0    9.0    7.0    9.0           7.0           8.0    9.0    7.0           7.0           7.0
      0.0156      9.0    6.0    2.0    9.0    9.0    2.5           6.0    6.0    5.5           5.5    6.5    7.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X180       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    9.0    9.0
       0.1250     9.0    9.0    6.0    9.0    9.0    9.0           9.0    9.0    8.0           8.0    8.0    9.0
       0.0640     9.0    9.0    7.0    9.0           9.0           9.0    9.0    9.0           9.0           7.0
       0.625      9.0    9.0    6.0    9.0    8.0    9.0           9.0    9.0    9.0           8.0    8.0    8.0
       0.0320     9.0    9.0    5.0    9.0           9.0           8.0    9.0    7.0           7.0           7.0
       0.0313     9.0    9.0    6.0    9.0    7.0    9.0           8.0    8.0    7.0           7.0    7.0    6.0
       0.0160     9.0    9.0    6.0    9.0           9.0           6.0    9.0    7.0           7.0           7.0
       0.0156     9.0    9.0    5.0    9.0    9.0    9.0           7.0    7.0                  7.0    9.0    4.0181       0.2500     9.0    9.0    6.0    9.0    9.0    9.0           8.0    9.0    9.0           9.0    7.0    7.0
       0.1250     9.0    9.0    5.0    9.0    9.0    7.0           8.0    9.0    7.0           7.0    9.0    7.0
       0.0640     9.0    7.0    9.0    9.0           9.0           6.0    9.0    5.0           4.0           7.0
       0.0625     7.0    7.0    5.0    9.0    9.0    6.0           7.0    9.0    7.0           7.0    7.0    6.0
       0.0320     9.0    6.0    0.0    9.0           5.0           7.0    9.0    3.0           5.0           6.0
       0.0313     9.0    6.0    4.0    9.0    2.0    5.0           7.0    8.0    6.0           6.0    6.0    6.0
       0.0160     9.0    4.0    0.0    9.0           1.0           3.0    5.0    2.0           2.0           3.0
       0.0156     9.0    7.0    8.0    9.0    8.0    5.0           5.0    6.0    9.0           4.0    4.0    3.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X182       0.3125     9.0    9.0    3.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    0.0    7.0
       0.1563     9.0    9.0    0.0    9.0    5.0    9.0           6.0    9.0    3.0           4.0    0.0    3.0
       0.0781     9.0    9.0    0.0    9.0    0.0    9.0           0.0    9.0    3.0           4.0    0.0    3.0
       0.0391     9.0    0.0    0.0    9.0    0.0    0.0           0.0    3.0    0.0           0.0    0.0    0.0
       0.0195     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0183       0.3125     9.0    9.0    9.0    9.0    5.0    9.0           9.0    9.0    5.0           7.0    5.0    7.0
       0.1563     9.0    9.0    0.0    9.0    5.0    9.0           8.0    9.0    3.0           7.0    3.0    7.0
       0.0781     9.0    9.0    0.0    9.0    5.0    9.0           6.0    9.0    3.0           7.0    0.0    7.0
       0.0391     9.0    0.0    0.0    9.0    5.0    0.0           3.0    3.0    0.0           1.0    0.0    7.0
       0.0195     0.0    0.0    0.0    9.0    0.0    0.0           0.0    3.0    0.0           0.0    0.0    6.0184       0.3130     9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    2.0    8.0
       0.1565     9.0    9.0    0.0    9.0    9.0    9.0           7.0    9.0    6.0           8.0    0.0    7.0
       0.0783     9.0    9.0    0.0    9.0    5.0    9.0           2.0    7.0    3.0           7.0    0.0    7.0
       0.0391     4.0    4.0    0.0    9.0    5.0    2.0           0.0    2.0    3.0           2.0    0.0    7.0
       0.0196            4.0    0.0    9.0    5.0    2.0           0.0    0.0    1.0           1.0    0.0    7.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X185      0.0840      9.0    9.0    0.0    9.0    0.0    8.0           0.0    7.0    5.0           4.0    0.0    3.0
      0.0320      9.0    5.0    0.0    9.0    0.0    0.0           0.0    6.0    0.0           3.0    0.0    0.0
      0.0160      4.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0186      0.5000      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    3.0    7.0
      0.2500      9.0    9.0    3.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    0.0    7.0
      0.1250      9.0    9.0    3.0    9.0    3.0    9.0           8.0    9.0    7.0           5.0    0.0    6.0
      0.0625      9.0    9.0    3.0    9.0    3.0    9.0           5.0    9.0                  3.0    0.0    5.0
      0.0313      9.0    0.0    3.0    9.0    3.0    0.0           0.0    0.0    4.0           1.0    0.0    5.0
      0.0156      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    4.0           0.0    0.0    5.0187      0.2500      9.0    9.0    9.0    9.0    3.0    9.0           6.0    9.0    9.0           5.0    0.0    7.0
      0.1250      9.0    9.0    3.0    9.0    3.0    9.0           3.0    9.0    5.0           5.0    0.0    6.0
      0.0625      9.0    0.0    0.0    9.0    0.0    0.0           0.0    7.0    3.0           0.0    0.0    6.0
      0.0313      6.0    0.0           9.0    0.0                  0.0    0.0    3.0           0.0    0.0    5.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X168      0.2500      9.0    7.0    4.0    9.0    8.0    7.0           6.0    9.0    5.0           4.0    5.0    5.0
      0.1250      9.0    6.0    3.0    9.0    1.0    9.0           4.0    9.0    5.0           4.0    6.0    5.0
      0.0625      9.0    4.0    3.0    9.0    1.0    2.0           2.0    5.0    4.0           4.0    5.0    4.0
      0.0313      7.0    4.0    9.0    9.0    6.0    5.0           1.0    5.0    5.0           3.0           4.0
      0.0156      2.0    2.0    5.0    9.0    1.0    7.0           1.0    7.0    4.0           5.0           3.0189      0.2500      9.0    9.0    4.0    9.0    7.0    7.0           8.0    9.0    4.0           7.0    7.0    7.0
      0.1250      9.0    4.0    4.0    9.0    4.0    4.0           5.0    9.0    4.0           7.0    5.0    3.0
      0.0625      6.0    4.0           9.0    2.0    4.0           4.0    7.0    5.0           7.0    5.0    3.0
      0.0313      9.0    4.0    2.0    9.0    1.0    2.0           2.0    8.0    3.0           2.0    4.0    2.0
      0.0156      9.0    3.0    2.0    9.0    1.0    1.0           1.0    1.0    3.0           2.0    2.0    3.0190      0.2500      9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    8.0           9.0    7.0    7.0
      0.1250      9.0    9.0    5.5    9.0    7.5    9.0           7.5    9.0    6.5           8.0    5.5    5.5
      0.0625      9.0    9.0    5.5    9.0    7.5    9.0           5.5    9.0    6.5           6.5    3.5    4.5
      0.0313      9.0    8.5    3.0    9.0    6.5    6.5           3.5    6.5    6.0           4.0    4.0    3.0
      0.0156      6.5    3.5    2.0    8.5    3.5    5.0           1.5    3.5    3.5           3.0    2.5    3.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X191       0.2500     9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    8.5           8.0    9.0    7.0
       0.1250     9.0    9.0    6.0    9.0    4.5    9.0           7.0    9.0    8.0           8.0    7.5    4.0
       0.0625     9.0    9.0    5.0    9.0    3.0    9.0           6.0    9.0    9.0           7.5    6.0    4.5
       0.0313     9.0    9.0    5.0    9.0    3.0    6.5           5.0    6.5    5.5           3.5    3.0    2.5
       0.0156     9.0    4.5    3.0    9.0    7.0    6.0           2.0    5.5    4.0           2.0    2.5    2.5192       0.2500     9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    7.0
       0.1250     9.0    9.0    6.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    9.0    6.0
       0.0625     9.0    9.0    5.0    9.0    7.0    9.0           5.0    9.0    6.0           6.0    4.0    6.0
       0.0313     9.0    6.0    6.0    9.0    3.0    6.0           5.0    9.0    5.0           5.0    5.0    5.0
       0.0156     6.0    7.0    6.0    9.0    4.0    5.0           4.0    5.0    5.0           5.0    4.0    4.0193       0.2500     9.0    4.5    3.0    9.0    4.0    5.5           4.0    9.0    3.0           4.5    8.5    2.5
       0.1250     8.0    2.0    1.5    9.0    4.5    3.0           1.5    4.5    3.0           3.5    7.0    2.0
       0.0625     5.0    3.0    2.5    9.0    3.0    4.0           1.0    3.0    3.5           2.5    3.0    2.5
       0.0313     4.5    0.5    6.0    9.0    5.0    1.0           0.5    1.0    3.0           2.0    2.5    1.5
       0.0156     9.0    0.5    1.0    6.5    3.0    4.0           1.0    1.5    3.5           2.0    2.0    1.5
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X194      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    7.0    7.0
      0.1250      9.0    9.0    7.0    9.0    8.0    9.0           8.0    9.0    9.0           8.0    9.0    6.0
      0.0625      9.0    8.0    6.0    9.0    9.0    9.0           7.0    9.0    5.0           7.0    9.0    5.0
      0.0313      9.0    6.0    6.0    9.0    3.0    9.0           6.0    8.0    5.0           6.0    6.0    4.0
      0.0156      9.0    7.0    7.0    9.0    3.0    6.0           2.0    6.0    5.0           5.0    5.0    4.0195      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    8.0
      0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    8.0
      0.0640      9.0    9.0    9.0    9.0           9.0           8.0    9.0    8.0           9.0           8.0
      0.0625      9.0    9.0    9.0    9.0    9.0    7.0           9.0    9.0    9.0           8.0    7.0    8.0
      0.0320      9.0    9.0    9.0    9.0           9.0           9.0    9.0    7.0           9.0           7.0
      0.0313      9.0    9.0    9.0    9.0    7.0    9.0           9.0    9.0    9.0           8.0    7.0    8.0
      0.0160      9.0    9.0    4.0    9.0           7.0           8.0    9.0    7.0           7.0           7.0
      0.0156      9.0    9.0    7.0    9.0           9.0           8.0    9.0    7.0           7.0    7.0    7.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X196      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.5           9.0    9.0    8.0
      0.1250      9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    9.0    8.0
      0.0640      9.0    9.0    6.0    9.0           6.0           9.0    9.0    9.0           8.0           7.0
      0.0625      9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    9.0           6.0    8.0    7.0
      0.0320      9.0    6.0    5.0    9.0           9.0           8.0    8.0    9.0           7.0           7.0
      0.0313      9.0    8.0    8.0    9.0    6.0    9.0           7.5    8.5    7.5           7.0    7.0    6.5
      0.0160      9.0    9.0                  9.0    4.0           7.0    9.0    5.0           7.0           6.0
      0.0156      9.0    7.5    3.5    9.0    6.0    6.5           7.0    7.0    4.5           8.0    8.0    5.5197      0.2500      9.0    9.0    2.5    9.0    4.5    9.0           1.0    9.0    5.0           3.5    8.5    2.5
      0.1250      5.5    6.5    2.0    9.0    4.5    4.5           0.0    4.5    0.0           1.5    0.0    2.0
      0.0625      2.5    1.0    0.0    9.0    0.0    0.0           0.0    1.5    1.0           1.5    0.0    0.0
      0.0313      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0198      0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
      0.1250      9.0    9.0    8.0    9.0    7.0    9.0           9.0    9.0    9.0           9.0    9.0    8.5
      0.0625      9.0    9.0    5.0    9.0    0.0    9.0           9.0    9.0    5.0           8.0    9.0    8.0
      0.0313      9.0    9.0    6.0    9.0    0.0    8.0           7.0    8.5    4.5           7.5    7.0    7.0
      0.0156      9.0    4.0    2.0    9.0    0.0    3.5           2.5    3.5    4.0           4.5    3.0    5.5
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X199       0.2500     9.0    6.0    2.0    9.0    9.0    4.0           9.0    9.0    9.0           6.0    6.0    8.0
       0.1250     9.0    7.5    3.0    9.0    9.0    6.5           7.0    9.0    7.0           6.0    6.0    7.0
       0.0625     7.5    6.0    2.5    9.0    7.0    3.5           5.0    6.5    4.5           3.5    1.0    6.5
       0.0313     9.0    3.0    2.5    9.0    0.0    2.5           2.5    4.5    2.0           2.5    0.0    5.0
       0.0156     4.5    2.5    0.0    9.0    0.0    1.5           0.0    2.0    1.5           1.0    0.0    2.0200       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.1250     9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    9.0    9.0
       0.0625     9.0    9.0    9.0    9.0    9.0    9.0           7.5    8.5    9.0           7.5    8.0    8.0
       0.0313     9.0    9.0    4.5    9.0    0.0    9.0           5.0    8.0    9.0           7.0           7.5
       0.0156     9.0    6.0    1.0    9.0    0.0    7.0           2.0    3.5    5.0           4.5    2.0    3.5201       0.2500     9.0    9.0    8.0    9.0    9.0    9.0           9.0    9.0    8.5           8.0    8.0    8.5
       0.1250     9.0    9.0    7.5    9.0    9.0    9.0           9.0    9.0    8.5           8.0    8.0    7.5
       0.0625     9.0    8.5    7.5    9.0    9.0    5.5           8.5    9.0    8.0           7.0    7.0    7.5
       0.0313     8.0    6.5    3.0    9.0    0.0    3.5           4.0    8.5    4.5           6.0    5.0    7.0
       0.0156     8.5    4.0    5.0    9.0    0.0    3.0           2.0    4.0    4.0           4.0    4.0    5.0
                                                   表II(续)
                                                                                  G      O      T
                  A       A      C      C      G      I      I      E      S      L      G      R      R     Z
                  B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T       E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H       L      B      L      P      E      S      G      I      W      A      T      R      X202       0.2500     9.0     9.0    8.0    9.0    9.0    9.0           8.0    8.5    9.0           8.5    8.0    8.0
       0.1250     9.0     9.0    8.0    9.0    8.0    9.0           4.5    9.0    6.5           7.0    7.0    4.0
       0.0625     9.0     8.5    3.5    9.0    6.0    7.0           1.5    3.5    5.0           4.5    2.0    4.0
       0.0313     9.0     5.0    3.5    9.0    4.5    4.5           0.0    2.0    3.5           3.0    2.5    1.0
       0.0156     6.5     2.0    0.5    9.0    6.0    4.5           0.0    1.0    3.0           0.5    4.0    0.5203       0.2500     9.0     9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    8.3
       0.1250     9.0     9.0    6.8    9.0    9.0    9.0           9.0    9.0    7.8           8.7    9.0    8.3
       0.0625     9.0     9.0    5.5    9.0    9.0    8.3           7.5    9.0    7.8           8.7    9.0    7.3
       0.0313     8.8     8.3    5.7    9.0    4.0    6.0           5.0    8.0    6.3           7.0    8.0    5.5
       0.0156     7.5     6.0    0.5    8.8    4.5    4.3           2.5    4.8    4.0           3.7    5.0    2.8204       0.2500     9.0     8.5    7.5    9.0    9.0    9.0           9.0    9.0    7.5           9.0    9.0    7.5
       0.1250     8.3     9.0    6.0    9.0    8.0    9.0           8.7    9.0    6.7           8.0    7.0    6.7
       0.0625     9.0     6.7    5.0    9.0    9.0    6.0           6.3    9.0    6.0           7.5    6.0    5.7
       0.0313     9.0     5.3    1.3    9.0    7.0    5.3           4.3    6.0    4.0           6.5    6.0    5.3
       0.0156     6.0     0.7    0.0    6.0    9.0    2.0           1.7    1.0    3.3           7.0    6.0    3.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X205       0.2500     9.0    9.0    7.5    9.0    9.0    9.0           9.0    9.0    9.0           8.0    9.0    8.0
       0.1250     9.0    9.0    7.5    9.0    9.0    9.0           8.5    9.0    8.0           8.0    8.0    7.5
       0.0625     9.0    8.0    4.5    9.0    8.0    9.0           6.5    9.0    7.0           6.0    7.0    7.0
       0.0313     8.5    7.5    5.5    9.0    0.0    8.0           7.0    7.0    6.5           6.0    9.0    6.5
       0.0156     7.0    3.0    1.0    8.0    2.0    5.5           3.0    3.0    4.0           7.0    9.0    4.0206       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    7.5
       0.1250     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    7.0
       0.0625     9.0    7.5    5.5    9.0    4.0    8.0           9.0    9.0    6.5           7.0    9.0    7.0
       0.0313     9.0    6.5    5.5    9.0    5.0    7.5           7.0    9.0    7.5           7.0    9.0    7.0
       0.0156     8.0    4.5    5.5    9.0    1.0    7.0           5.0    5.5    4.5           0.0    2.0    4.0207       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
       0.1250     9.0    9.0    9.0    9.0    8.0    9.0           9.0    9.0    9.0           8.5    9.0    8.5
       0.0625     9.0    9.0    6.0    9.0    9.0    9.0           9.0    9.0    8.0           8.0    9.0    8.0
       0.0313     9.0    8.5    5.0    9.0    4.0    9.0           7.5    9.0    7.0           7.0    9.0    7.0
       0.0156     9.0    8.0    3.5    9.0    2.0    9.0           5.0    6.0    8.0           6.0    5.0    4.5
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X208       0.1250     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.0           8.0    7.0    8.0
       0.0625     9.0    7.0    9.0    9.0    9.0    9.0           7.0    9.0    6.0           7.0    9.0    6.0
       0.0313     6.0    6.0    4.0    9.0    9.0    4.0           4.0    9.0    9.0           7.0    9.0    5.0
       0.0156     7.0    5.0    9.0    9.0    0.0    6.0           2.0    7.0    2.0           2.0    9.0    3.0209       0.2500     9.0    9.0    5.0    9.0    9.0    9.0           9.0    9.0    5.0           8.0    7.0    8.0
       0.1250     9.0    9.0    3.0    9.0    0.0    9.0           7.0    9.0                  7.0    5.0    7.0
       0.0625     9.0    6.0    1.0    9.0           9.0           6.0    9.0    4.0           6.0           7.0
       0.0313     9.0    2.0    1.0    9.0    2.0    9.0           4.0    4.0    3.0           5.0    4.0    4.0
       0.0156     2.0    1.0    0.0    9.0    0.0    1.0           0.0    4.0    1.0           1.0    3.0    1.0210       0.2500     9.0    9.0    3.0    9.0    9.0    9.0           7.0    9.0    9.0           9.0    8.0    8.0
       0.1250     9.0    8.0    9.0    9.0    7.0    9.0           4.0    9.0    9.0           6.0    6.0    7.0
       0.0625     9.0    9.0    9.0    9.0    2.0    4.0           4.0    9.0    7.0           4.0    4.0    5.0
       0.0313     9.0    2.0    7.0    9.0    0.0    0.0           3.0    9.0    0.0           0.0    1.0    4.0
       0.0156     0.0    0.0    5.0    9.0    0.0    0.0           0.0    3.0    0.0           0.0           0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X211       0.1250     9.0    9.0    9.0    9.0    7.0    5.0           3.0    9.0    6.0           1.0    0.0    7.0
       0.0625     9.0    0.0    0.0    9.0    3.0    9.0           0.0    3.0    1.0           0.0    0.0    6.0
       0.0313     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    3.0
       0.0156     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0212       0.2500     9.0    9.0    0.0    9.0    9.0    9.0           8.0    9.0    9.0           9.0    6.0    9.0
       0.1250     9.0    9.0    0.0    9.0    6.0    9.0           3.0    9.0    7.0           9.0    6.0    6.0
       0.0625     8.0    5.0    0.0    9.0    0.0    9.0           0.0    0.0    7.0           7.0    3.0    6.0
       0.0313     7.0    4.0    0.0    9.0    0.0    3.0           0.0    0.0    1.0           2.0    1.0    2.0
       0.0156     7.0    0.0    0.0    7.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.0213       0.5000     9.0    9.0    9.0    9.0    7.0    9.0           7.0    9.0    9.0           7.0    7.0    7.0
       0.2500     9.0    9.0    7.0    9.0    7.0    9.0           7.0    9.0    6.0           7.0    7.0    7.0
       0.1250     9.0    6.0    1.0    9.0    3.0    9.0           4.0    6.0    3.0           6.0    6.0    5.0
       0.0625     6.0    3.0    1.0    9.0    2.0    5.0           2.0    4.0    1.0           5.0    4.0    4.0
       0.0313     1.0    0.0    1.0    4.0    1.0    0.0           0.0    4.0    1.0           1.0    0.0    1.0
                                                  表II(续)
                                                                                   G             O      T
                   A       A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B       M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U       B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T       E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H       L      B      L      P      E      S      G      I      W      A      T      R      X214       0.5000      9.0     7.0    6.0    9.0    9.0    9.0           5.0    9.0    6.0           7.0    4.0    6.0
       0.2500      7.0     6.0    4.0    9.0    7.0    6.0           3.0    9.0    6.0           4.0    3.0    6.0
       0.1250              4.0    0.0    4.0    7.0    3.0           0.0    6.0    4.0           2.0    1.0    2.0
       0.0625              2.0    0.0           1.0    3.0           0.0           2.0           1.0    1.0    1.0
       0.0313      1.0     1.0    0.0                  0.0           0.0    1.0    1.0           0.0    0.0    1.0215       0.5000      1.0     5.0    1.0    9.0    5.0    1.0           1.0    2.0    1.0           1.0    4.0    1.0
       0.2500      0.0     2.0    0.0    9.0    4.0                  0.0    0.0    1.0           0.0    0.0    1.0
       0.1250      2.0     1.0    0.0    4.0    2.0    1.0           0.0    0.0    1.0           1.0    0.0    1.0
       0.0625      0.0     0.0    1.0           1.0    0.0           0.0    0.0    1.0           0.0    1.0    0.0
       0.0313      0.0     0.0    0.0           1.0    1.0           0.0    0.0    1.0           1.0    1.0    0.0216       0.5000      9.0     7.0    5.0    9.0    6.0    6.0           5.0    9.0    6.0           7.0    4.0    7.0
       0.2500      9.0     4.0    2.0    9.0    2.0    6.0           2.0    7.0    3.0           4.0    1.0    4.0
       0.1250      9.0     3.0    1.0    9.0    1.0    6.0           1.0    6.0    2.0           3.0    2.0    4.0
       0.0625      6.0     0.0    0.0    9.0    1.0    2.0           0.0    6.0    3.0           1.0           1.0
       0.0313      1.0     1.0    0.0    5.0    1.0    1.0           0.0    3.0    0.0           1.0    1.0    1.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X217       0.5000     9.0    7.0    9.0    9.0    9.0    9.0           7.0    9.0    7.0           7.0    7.0    9.0
       0.2500     9.0    6.0    6.0    9.0    9.0    9.0           6.0    9.0    6.0           7.0    4.0    7.0
       0.1250     9.0    4.0    4.0    9.0    9.0    5.0           6.0    9.0    6.0           6.0    1.0    5.0
       0.0625     6.0    1.0    1.0    9.0    5.0    2.0           1.0    5.0    4.0           1.0    1.0    1.0
       0.0313            1.0           9.0    5.0    2.0           0.0    6.0    1.0           0.0    0.0    0.0218       0.5000     9.0    3.0    3.0    9.0    7.0    6.0           3.0    6.0    3.0           2.0           1.0
       0.2500     6.0    3.0    1.0    9.0    9.0                  2.0    4.0    1.0           1.0    2.0    0.0
       0.1250     1.0    0.0    2.0    9.0    4.0    0.0           0.0    2.0                  1.0    0.0    1.0
       0.0625     0.0    0.0    0.0    7.0           0.0           0.0    1.0    0.0           1.0    0.0    1.0
       0.0313     0.0    0.0    0.0    9.0           0.0           0.0    1.0    0.0           0.0    0.0    0.0219       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    8.0    7.5
       0.1250     9.0    8.0    7.0    9.0    7.0    8.5           8.0    9.0    5.5           7.0    7.0    7.0
       0.0625     9.0    7.5    3.0    9.0    0.0    9.0           6.5    9.0    3.5           7.0    7.0    6.0
       0.0313     9.0    3.5    3.0    9.0    0.0    5.5           5.5    7.5    1.0           4.0    4.0    5.0
       0.0156     8.0    2.5    2.0    7.5    0.0    7.5           1.0    7.0    1.5           2.0    2.0    4.5
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X220       0.2500     9.0    9.0    9.0    9.0    9.0    9.0           8.0    9.0    5.0           9.0    8.0    8.0
       0.1250     9.0    9.0    9.0    9.0    3.0    9.0           7.0    9.0    2.0           6.0    7.0    6.0
       0.0625     9.0    4.0    0.0    9.0    0.0    9.0           0.0    9.0    2.0           6.0    3.0    5.0
       0.0313     7.0    2.0    0.0    9.0    0.0    0.0           0.0    9.0    2.0           6.0    1.0    0.0
       0.0156     7.0    0.0           9.0    0.0    0.0           0.0    8.0    0.0           2.0    0.0    0.0221       0.2500     9.0    9.0    0.0    9.0    9.0    9.0           2.0    9.0    3.0           1.0    1.0    5.0
       0.1250     9.0    9.0    0.0    9.0    7.0    0.0           2.0    9.0                  1.0    1.0    5.0
       0.0625     9.0    5.0    0.0    9.0    0.0    0.0           0.0    9.0    3.0           0.0    0.0    5.0
       0.0313     9.0    0.0    0.0    9.0    0.0    0.0           0.0    9.0    0.0           0.0    0.0    3.0
       0.0156     4.0    0.0    0.0    9.0    0.0    0.0           0.0    9.0    0.0           0.0    0.0    0.0222       0.2500     9.0    9.0    4.0    9.0    0.0    0.0           2.0    9.0    9.0           1.0    1.0    6.0
       0.1250     9.0    4.0    0.0    9.0    0.0    9.0           0.0    9.0    5.0           1.0    0.0    1.0
       0.0625     3.0           0.0    9.0    0.0    3.0           0.0    9.0    3.0           0.0    0.0    1.0
       0.0313     2.0    0.0    0.0    9.0    0.0    0.0           0.0    7.0    2.0           0.0    0.0    1.0
       0.0156     0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X223       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    9.0
       0.1250      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    7.0    8.0
       0.062       9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    9.0           7.0    6.0    7.0
       0.0313      9.0    9.0    0.0    9.0    9.0    7.0           6.0    9.0    4.0           4.0    5.0    7.0224       0.5000      9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.0    9.0
       0.2500      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    9.0           8.0    6.0    8.0
       0.1250      9.0    9.0    3.0    9.0    9.0    9.0           9.0    9.0    6.5           6.0    5.0    7.0
       0.0625      9.0    7.0    2.0    9.0    9.0    9.0           7.5    9.0    7.0           7.0    5.0    7.0
       0.0313      9.0    5.0    1.5    9.0    7.0    6.0           7.0    9.0    4.5           6.0    3.0    6.5
       0.0156      9.0    2.0    0.0    9.0                         4.0    7.0    2.0                         4.0225       0.5000      9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    7.0           8.0    9.0    9.0
       0.2500      9.0    9.0    9.0    9.0    9.0    9.0           7.0    9.0    9.0           7.0    6.0    7.0
       0.1250      9.0    9.0    9.0    9.0    9.0    9.0           5.0    9.0    6.0           6.0    6.0    7.0
       0.0625      9.0    9.0    6.0    9.0    9.0    9.0           4.0    7.0                         3.0    6.0
       0.0313      9.0    6.0    3.0    9.0    9.0    9.0           2.0    4.0    2.0           3.0    1.0    4.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X226      0.2500      9.0    9.0    0.0    9.0    0.0    9.0           0.0    9.0    5.0           0.0    0.0    5.0
      0.1250      9.0    9.0    0.0    9.0    0.0    9.0           0.0    0.0    3.0           0.0    0.0    5.0
      0.0625      9.0    3.0    0.0    9.0    0.0    3.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      4.0    3.0    0.0    9.0    0.0                  0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    3.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0227      0.2500      9.0    9.0    4.0    9.0    0.0    9.0           0.0    0.0    9.0           2.0    2.0    3.0
      0.1250      7.0    9.0    0.0    9.0    0.0    0.0           0.0    0.0    4.0           0.0    0.0    3.0
      0.0625      9.0    4.0           9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0228      0.2500      3.0    4.0    4.0    9.0    0.0    3.0           0.0    0.0    3.0           0.0    0.0    4.0
      0.1250      3.0    0.0    9.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0
      0.0625      7.0    0.0    0.0    7.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0313      0.0    0.0    0.0    5.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0156      0.0    0.0    0.0           0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X229       0.2500     9.0    2.0    3.0    9.0    0.0    3.0           0.0    0.0    2.0           0.0    0.0    0.0
       0.1250     0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0           0.0
       0.0625     0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0313     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0156     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0230       0.2500     9.0    9.0    9.0    9.0    5.0    9.0           0.0    0.0    5.0           0.0    2.0    4.0
       0.1250     9.0    9.0    0.0    9.0    5.0    9.0           0.0    0.0    5.0           0.0    2.0    4.0
       0.0625     9.0    0.0    0.0    9.0    0.0    9.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0313     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0156     9.0                  9.0    0.0    0.0           0.0    0.0    0.0           0.0           0.0231       0.2500     9.0    9.0    0.0    9.0    5.0    9.0           2.0    2.0    3.0           3.0    6.0    4.0
       0.1250     9.0    9.0    0.0    9.0    0.0    9.0           0.0    0.0    3.0           1.0    1.0    2.0
       0.0625     9.0    5.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0313     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
       0.0156     0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X232     0.2500       9.0    9.0    9.0    9.0    9.0    9.0           2.0    9.0    5.0           0.0    0.0    4.0
     0.1250       9.0    9.0    9.0    9.0    0.0    9.0           2.0    7.0    5.0           0.0    0.0    4.0
     0.0625       9.0    9.0    3.0    9.0    0.0    9.0           0.0    7.0    0.0           0.0    0.0    3.0
     0.0313       9.0    4.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    3.0
     0.0156       9.0    0.0    0.0    9.0    0.0                  0.0    0.0    0.0           0.0    0.0    3.0233     0.2500       9.0    4.0    0.0    9.0    0.0    0.0           0.0    0.0    5.0           0.0    0.0    5.0
     0.1250       9.0           0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0625       0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0313       0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0156       0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0234     0.2500       9.0    9.0    2.0    9.0    0.0    9.0           0.0    9.0    3.0           4.0    0.0    6.0
     0.1250       9.0    6.0    2.0    9.0    0.0    9.0           0.0    0.0                  0.0    0.0    4.0
     0.0625       9.0    0.0    2.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0313       9.0    0.0           9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0156       0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物      施用率    T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X235       0.2500     9.0    7.0    2.0    9.0    0.0    3.0           0.0    0.0    2.0           0.0    0.0    4.0
       0.1250     7.0           0.0    9.0    0.0                  0.0           0.0           0.0    0.0    4.0
       0.0625     9.0    0.0    0.0    9.0    0.0                  0.0    0.0    0.0           0.0    0.0    0.0
       0.0313     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0                         0.0
       0.0156     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0236       0.2500     9.0    1.0    3.0    9.0    5.0    1.0           1.0    3.0    2.0           1.0    4.0    3.0
       0.1250     9.0    1.0    0.0    9.0    1.0    0.0           0.0    3.0    2.0           1.0    0.0    2.0
       0.0625     9.0    0.0    1.0    9.0    0.0    0.0           0.0    1.0    1.0           1.0    0.0    1.0
       0.0313     9.0    0.0    0.0    7.0    0.0    0.0           0.0    2.0    1.0           1.0    0.0    0.0
       0.0156     2.0    0.0    0.0           0.0    0.0           0.0    0.0    0.0           0.0    1.0    0.0237       0.2500     9.0    9.0    2.0    9.0    9.0    9.0           5.0    9.0    5.0           2.0    3.0    4.0
       0.1250     9.0    2.0    1.0    9.0    6.0    2.0           1.0    9.0    2.0           1.0    1.0    1.0
       0.0625     4.0    0.0    0.0    9.0    1.0    0.0           0.0    1.0    2.0           0.0    0.0    1.0
       0.0313     3.0    0.0    0.0    9.0    0.0    1.0           0.0    0.0    0.0           0.0    0.0    1.0
       0.0156     0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    1.0
                                                       表II(续)
                                                                              G           O      T
                 A      A      C     C     G     I      I      E      S       L      G    R      R       Z
                 B      M      A     H     A     P      P      C      E       X      L    Y      Z       E
                 U      B      S     E     L     O      O      H      T       M      X    S      A       A化合物    施用率     T      E      O     A     A     H      S      C      V       A      M    A      W       M编号  (公斤/公顷)   H      L      B     L     P     E      S      G      I       W      A    T      R       X238      0.2500    9.0    9.0    3.0   9.0   9.0   9.0           7.0    9.0    9.0          6.0    6.0     7.0
      0.1250    9.0    9.0    2.0   9.0   6.0   9.0           5.0    9.0    5.0          4.0    3.0     7.0
      0.0625    6.0    7.0    1.0   9.0   3.0   9.0           1.0    9.0    9.0          1.0    1.0     4.0
      0.0313           4.0    0.0   9.0   3.0   0.0           1.0    9.0    3.0          1.0    1.0     2.0
      0.0156    3.0    3.0    0.0   0.0   0.0   0.0           1.0    1.0    2.0          0.0    0.0     1.0239      0.2500    9.0    9.0    9.0   9.0   9.0   9.0           7.0    9.0    9.0          7.0    6.0     7.0
      0.1250    9.0    9.0    6.0   9.0   9.0   9.0           6.0    9.0    9.0          7.0    5.0     7.0
      0.0625    9.0    4.0    3.0   9.0   7.0   9.0           2.0    4.0    4.0          4.0    3.0     5.0
      0.0313    9.0    2.0    0.0   9.0         9.0           1.0    3.0    1.0          0.0    1.0     0.0
      0.0156    2.0    1.0    0.0   9.0   0.0   4.0           0.0    1.0    0.0          0.0    1.0     0.0245      0.2500    0.0    0.0    0.0   0.0   0.0   0.0           0.0    0.0    2.0          0.0    0.0     0.0
      0.1250    0.0    0.0    0.0   0.0   0.0   0.0           0.0    0.0    2.0          0.0    0.0     0.0
      0.0625    0.0    0.0    0.0   0.0   0.0   0.0           0.0    0.0    0.0          0.0    0.0     0.0
      0.0313    0.0    0.0    0.0   0.0   0.0   0.0           0.0    0.0    0.0          0.0    0.0     0.0
      0.0156    0.0    0.0    0.0   0.0   0.0   0.0           0.0    0.0    0.0          0.0    0.0     0.0
                                                     表II(续)
                                                                                 G            O      T
                  A      A      C      C      G      I      I      E      S      L      G     R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L     Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X     S      A      A化合物   施用率       T      E      O      A      A      H      S      C      V      A      M     A      W      M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A     T      R      X246      0.2500     9.0    0.0    3.0    9.0    0.0    9.0           3.0    6.0    4.0          1.0    7.0    3.0
      0.1250     9.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    4.0          0.0    0.0    3.0
      0.0625     0.0    0.0    0.0           0.0    0.0           0.0    0.0    2.0          0.0    0.0    2.0
      0.0313     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    1.0          0.0    0.0    2.0
      0.0156     0.0    0.0    0.0           0.0    0.0           0.0    0.0    1.0          0.0    0.0    0.0256      0.2500     9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0          9.0    9.0    9.0
      0.1250     9.0    9.0    8.3    9.0    9.0    9.0           9.0    9.0    9.0          8.0    9.0    8.7
      0.0620     9.0    9.0    9.0    9.0           9.0           9.0    9.0    9.0          8.0           9.0
      0.0320     8.6    9.0    6.0    9.0           9.0           9.0    9.0    9.0          8.0           9.0
      0.0160     8.0    9.0    9.0    9.0           9.0           9.0    9.0    9.0          5.0           5.0257      0.2500     9.0    9.0    4.5    9.0    9.0    9.0           5.0    9.0    8.0          7.0    9.0    7.5
      0.1250     9.0    9.0    1.5    9.0    3.0    9.0           3.0    8.5    5.5          4.5    3.0    2.0
      0.0620     9.0    6.5    0.0    9.0    0.0    6.0           1.0    1.0    4.5          3.5    3.0    0.0
      0.0320     4.5    3.0    0.0    9.0    0.0    5.0           0.0    0.0    2.0          0.0    2.0    0.0
      0.0160     4.5    1.0    0.0    9.0    0.0    1.5           0.0    0.0    0.0          0.0    0.0    0.0
                                                        表II(续)
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率        T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)     H      L      B      L      P      E      S      G      I      W      A      T      R      X258     0.2500       9.0    9.0    8.3    9.0    7.0    8.0           6.7    9.0    7.3           6.3    7.5    7.0
     0.1250       9.0    9.0    4.3    9.0    3.5    8.0           3.0    9.0    3.7           3.7    5.5    3.3
     0.0620       9.0    9.0    1.3    9.0    0.5    7.3           1.7    4.7    3.0           2.0    2.5    1.7
     0.0320       4.7    3.7    0.0    9.0    0.0    4.7           0.7    4.0    0.7           1.0    0.0    0.0
     0.0160       4.0    1.0    0.0    9.0    0.0    2.0           0.0    0.3    0.0           0.7    0.0    0.0259     0.2500       9.0    9.0    7.0    9.0    0.0    9.0           3.5    9.0    9.0           7.0    6.0    6.0
     0.1250       9.0    6.5    3.5    9.0    0.0    9.0           1.5    7.0    6.0           6.5    4.0    1.5
     0.0620       4.5    5.5    0.0    9.0    0.0    5.5           3.0    1.0    0.0           1.0    0.0    0.0
     0.0320       1.0    1.0    0.0    7.0    0.0    7.5           0.5    2.0    0.0           0.0    0.0    0.0
     0.0160       0.0    0.0    0.0    9.0    0.0    1.5           0.0    1.5    0.0           0.0    0.0    0.0260     0.2500       9.0    6.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.1250       9.0    3.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0620       9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0320       0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0160       0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                     表II(续)
                                                                              G             O      T
               A      A      C      C      G      I      I      E      S      L      G      R      R      Z
               B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
               U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物  施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X261    0.2500    9.0    9.0    9.0    9.0    9.0    9.0           0.0    9.0    9.0           3.0    2.0    7.0
    0.1250    9.0    5.0    0.0    9.0    9.0    7.0           0.0    0.0    3.0           0.0    0.0    2.0
    0.0620    9.0    0.0    0.0    9.0    0.0    9.0           0.0    0.0    0.0           0.0    0.0    0.0
    0.0320    0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
    0.0160    0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0262    0.5000    9.0    9.0    9.0    9.0           9.0           4.0    9.0    9.0           4.0           6.0
    0.2500    9.0    6.5    7.5    9.0           9.0           4.5    8.5    8.5           4.0    6.0    5.0
    0.1250    9.0    6.0    5.0    9.0           9.0           1.5    8.0    6.0           1.5    4.0    1.0
    0.0620    9.0    5.0    3.5    9.0           8.0           0.0    2.0    3.0           1.0    3.0    0.5
    0.0320    8.0    1.0    1.0    9.0           4.5           0.0    1.5    1.0           0.5    0.0    0.0
    0.0160    0.0    0.0    0.0    9.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0263    0.5000    9.0    9.0    7.0    9.0           9.0           3.0    6.0    9.0           4.0           5.0
    0.2500    9.0    5.5    6.5    9.0           9.0           1.0    3.0    6.0           0.0    3.0    2.5
    0.1250    9.0    4.0    2.0    9.0           9.0           0.0    1.5    3.0           0.0    0.0    0.0
    0.0620    9.0    2.0    1.0    9.0           4.0           0.0    1.0    1.0           0.0    0.0    0.0
    0.0320    9.0    1.0    0.5    8.0           0.0           0.0    1.0    0.5           0.0    0.0    0.0
    0.0160    9.0    0.0    0.0    4.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                     表II(续)
                                                                               G             O      T
                  A     A      C     C      G      I      I      E      S      L      G      R      R      Z
                  B     M      A     H      A      P      P      C      E      X      L      Y      Z      E
                  U     B      S     E      L      O      O      H      T      M      X      S      A      A化合物   施用率       T     E      O     A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H     L      B     L      P      E      S      G      I      W      A      T      R      X264      0.2500     9.0   8.0    8.0   9.0           9.0           8.0    9.0    8.5           7.5    8.0    6.5
      0.1250     9.0   9.0    5.5   9.0           9.0           6.5    9.0    8.0           5.5    7.0    4.5
      0.0620     9.0   9.0    1.0   9.0           7.0           3.5    9.0    4.5           2.5    4.0    4.0
      0.0320     7.5   4.0    1.0   9.0           5.5           0.5    3.0    1.0           1.0    0.0    1.0
      0.0160     7.5   2.0    1.0   7.5           0.0           0.0    1.5    0.0           0.5    0.0    1.0265      0.2500     9.0   0.0    0.0   9.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.1250     8.0   0.0    0.0   9.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0620     0.0   0.0    0.0   9.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0320     0.0   0.0    0.0   0.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0266      0.5000     9.0   9.0    7.0   9.0           9.0           9.0    9.0    7.0           7.0           6.0
      0.2500     9.0   9.0    1.0   9.0           9.0           7.0    9.0    4.6           7.0    8.0    4.5
      0.1250     9.0   6.0    1.0   9.0           6.5           1.0    5.0    3.0           3.5    3.0    3.0
      0.0620     2.0   1.0    1.0   7.5           1.0           1.5    2.0    0.5           1.0    0.0    1.0
      0.0320     2.5   0.5    1.0   1.0           0.0           0.5    2.5    0.0           0.0    0.0    0.5
      0.0160     0.0   0.0    0.0   0.0           0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                        表II(续)
                                                                                 G           O      T
                 A      A      C      C      G      I      I      E      S       L      G    R      R      Z
                 B      M      A      H      A      P      P      C      E       X      L    Y      Z      E
                 U      B      S      E      L      O      O      H      T       M      X    S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V       A      M    A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I       W      A    T      R      X267      0.2500    9.0    3.0    0.0    9.0           9.0           9.0     9.0    3.0         0.0    0.0    6.0
      0.1250    9.0    1.0    0.0    9.0           0.0           0.0     9.0    0.0         0.0    0.0    0.0
      0.0620    9.0    9.0    0.0    9.0           0.0           0.0     0.0    0.0         0.0    0.0    0.0
      0.0320    0.0    0.0    0.0    9.0           0.0           0.0     0.0    0.0         0.0    0.0    0.0
      0.0160    0.0    0.0    0.0    9.0           0.0           0.0     0.0    0.0         0.0    0.0    0.0268      0.5000    9.0    9.0    9.0    9.0           9.0           9.0     9.0    9.0         9.0           9.0
      0.2500    9.0    9.0    9.0    9.0    9.0    9.0           8.8     9.0    9.0         8.8    8.0    9.0
      0.1250    9.0    9.0    5.3    9.0    9.0    9.0           7.3     9.0    9.0         7.5    5.0    8.3
      0.0620    9.0    9.0    3.8    9.0    8.0    9.0           6.5     8.0    4.8         5.5    3.0    5.3
      0.0320    9.0    7.0    0.8    8.8    3.0    9.0           3.3     6.3    3.3         3.3    1.0    3.0
      0.0160    9.0    8.0    0.3    9.0    5.0    7.7           2.3     6.7    2.0         2.3    1.0    2.7269      0.2500    0.0    0.0    0.0    9.0           0.0           0.0     0.0    0.0         0.0    0.0    0.0
      0.1250    0.0    0.0    0.0    9.0           0.0           0.0     0.0    0.0         0.0    0.0    0.0
      0.0620    0.0    0.0    0.0    9.0           0.0           0.0     0.0    0.0         0.0    0.0    0.0
      0.0320    0.0    0.0    0.0    0.0           0.0           0.0     0.0    0.0         0.0    0.0    0.0
                                                        表II(续)
                                                                                       G             O        T
                  A       A       C      C      G     I      I      E         S        L      G      R        R         Z
                  B       M       A      H      A     P      P      C         E        X      L      Y        Z         E
                  U       B       S      E      L     O      O      H         T        M      X      S        A         A化合物     施用率     T       E       O      A      A     H      S      C         V        A      M      A        W         M编号   (公斤/公顷)   H       L       B      L      P     E      S      G         I        W      A      T        R         X270       0.5000    9.0     9.0     9.0    9.0          9.0           4.0       9.0      4.0           4.0                5.0
       0.2500    9.0     9.0     1.5    8.5          9.0           2.0       8.0      2.5           1.0      0.0       5.0
       0.1250    9.0     9.0     0.0    9.0          8.0           1.0       5.5      2.0           1.0      0.0       3.0
       0.0620    9.0     8.0     0.0    9.0          4.5           0.0       3.5      1.0           1.0      0.0       1.0
       0.0320    9.0     2.5     0.0    6.0          0.0           0.0       1.0      0.0           1.0      0.0       0.0
       0.0160    0.0     0.0     0.0    0.0          0.0           0.0       0.0      0.0           0.0      0.0       0.0271       0.2500    9.0     9.0     3.0    9.0          9.0           9.0       9.0      7.0           9.0      8.0       9.0
       0.1250    9.0     9.0     9.0    9.0          9.0           8.0       9.0      6.0           6.0      3.0       6.5
       0.0620    9.0     6.0     2.0    9.0          5.5           3.0       9.0      1.5           2.5      1.0       2.0
       0.0320    9.0     4.5     2.0    9.0          5.0           2.5       6.5      2.0           2.0      0.0       2.5
       0.0160    4.0     2.0     2.0    3.5          1.5           1.0       2.0      1.0           0.0      0.0       0.0272       0.5000    9.0     3.0     0.0    9.0   7.0    2.0           0.0       0.0      0.0           0.0      0.0       0.0
       0.2500    3.0     0.0     0.0    2.0   7.0    0.0           0.0       0.0      0.0           0.0      0.0       0.0
       0.1250    2.0     0.0     0.0    0.0   0.0    0.0           0.0       0.0      0.0           0.0      0.0       0.0
       0.0620    0.0     0.0     0.0    0.0   0.0    0.0           0.0       0.0      0.0           0.0      0.0       0.0
                                                         表II(续)
                                                                               G             O      T
                A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)  H      L      B      L      P      E      S      G      I      W      A      T      R      X273      0.2500   9.0    9.0    0.0    9.0    9.0    9.0           0.0    9.0    3.0           3.0    0.0    0.0
      0.1250   9.0    9.0    0.0    9.0    0.0    2.0           0.0    7.0    0.0           0.0    0.0    0.0
      0.0620   9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0320   0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0160   0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0274      0.2500   9.0    3.0    0.0    9.0    9.0    5.0           7.0    9.0    0.0           3.0    0.0    0.0
      0.1250   9.0           0.0    9.0    0.0    0.0           3.0    9.0    0.0           0.0    0.0    0.0
      0.0620   9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0320   0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0275      0.2500   9.0    9.0    5.0    9.0    0.0    9.0           9.0    9.0    0.0           4.0    3.0    0.0
      0.1250   9.0    0.0    0.0    9.0    0.0    3.0           4.0    7.0    0.0           0.0    0.0    0.0
      0.0620   9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0320   0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0160   0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                    表II(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物   施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X276      0.2500    9.0    9.0    7.0    9.0    9.0    9.0           8.0    9.0    9.0           8.0    8.0    7.0
      0.1250    9.0    7.0    3.0    9.0    9.0    9.0           0.0    9.0    2.0           4.0    5.0    6.0
      0.0620    9.0    2.0    0.0    9.0    7.0    0.0           0.0    9.0    0.0           0.0    0.0    0.0
      0.0320    9.0    1.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0160    9.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0277      0.2500    9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0
      0.1250    9.0    9.0    6.5    9.0    9.0    9.0           9.0    9.0    8.5           8.0    8.0    8.5
      0.0620    9.0    8.0    3.0    9.0    9.0    5.5           9.0    9.0    6.0           7.0    7.0    8.0
      0.0320    9.0    6.5    1.0    9.0    8.0    3.0           6.0    9.0    4.5           4.0    5.0    6.0
      0.0160    9.0    4.0    0.0    9.0    0.0    1.5           2.5    9.0    2.5           1.5    2.0    3.5278      0.2500    9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    7.0           9.0    8.0    9.0
      0.1250    9.0    9.0    1.0    9.0    9.0    9.0           9.0    9.0    5.0           8.0    7.0    9.0
      0.0620    9.0    5.0    0.0    9.0    9.0    9.0           0.0    9.0    5.0           0.0    3.0    3.0
      0.0320    9.0    3.0    0.0    9.0    9.0    2.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0160    0.0    0.0    0.0    3.0    3.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                        表II(续)
                                                                                  G                 O        T
                  A      A      C      C      G      I      I      E      S       L        G        R        R       Z
                  B      M      A      H      A      P      P      C      E       X        L        Y        Z       E
                  U      B      S      E      L      O      O      H      T       M        X        S        A       A化合物    施用率      T      E      O      A      A      H      S      C      V       A        M        A        W       M编号  (公斤/公顷)    H      L      B      L      P      E      S      G      I       W        A        T        R       X279      0.2500     9.0    9.0    0.0    9.0    9.0    9.0           2.0    9.0     3.0               7.0      7.0     7.0
      0.1250     9.0    9.0    0.0    9.0    4.0    3.0           0.0    9.0     1.0               1.0      2.0     5.0
      0.0620     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0     0.0               0.0      0.0     0.0
      0.0320     9.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0     0.0               0.0      0.0     0.0
      0.0160     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0     0.0               0.0      0.0     0.0280      0.2500     9.0    7.0    7.0    9.0    1.0    9.0           9.0    9.0     8.0               7.0      2.0     8.0
      0.1250     9.0    9.0    4.0    9.0    0.0    4.0           9.0    9.0     2.0               6.0      1.0     2.0
      0.0620     7.0    7.0    1.0    9.0    0.0    0.0           0.0    0.0     1.0               0.0      0.0     2.0
      0.0320            1.0    0.0    9.0    0.0    0.0           0.0    0.0     0.0               0.0      0.0     0.0
      0.0160     0.0    0.0    0.0    2.0    0.0    0.0           0.0    0.0     0.0               0.0      0.0     0.0281      0.2500     9.0    9.0    5.0    9.0    9.0    9.0           7.0    9.0     9.0               7.0      7.0     8.0
      0.1250     9.0    9.0    2.0    9.0    6.0    9.0           4.0    9.0     6.0               5.0      2.0     7.0
      0.0620     9.0    6.0    0.0    9.0    2.0    9.0                  7.0     2.0               1.0      1.0     1.0
      0.0320     1.0    4.0    0.0    9.0    0.0    0.0           0.0    0.0     0.0               1.0      1.0     1.0
      0.0160     0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0     0.0               0.0      0.0     0.0
                                                             表II(续)
                                                                                       G                   O        T
                  A       A       C      C       G       I      I      E      S        L        G          R        R         Z
                  B       M       A      H       A       P      P      C      E        X        L          Y        Z         E
                  U       B       S      E       L       O      O      H      T        M        X          S        A         A化合物     施用率     T       E       O      A       A       H      S      C      V        A        M          A        W         M编号   (公斤/公顷)   H       L       B      L       P       E      S      G      I        W        A          T        R         X282       0.5000    8.0     5.0     4.0    9.0             7.0           0.0    2.0      2.0                 2.0                0.0
       0.2500    2.0     0.0     0.0    2.5     0.0     2.0           0.0    2.0      0.0                 0.0      0.0       0.5
       0.1250    0.0     0.0     0.0    2.5     0.0     0.0           0.0    0.0      0.0                 0.0      0.0       0.5
       0.0620    0.0     0.0     0.0    0.0     0.0     0.0           0.0    0.0      0.0                 0.0      0.0       0.0283       0.5000    9.0     7.0     7.0    9.0             9.0           9.0    9.0      6.0                 9.0                6.0
       0.2500    8.0     5.0     3.0    9.0     4.0     4.5           1.0    5.5      2.0                 5.0      6.0       2.5
       0.1250    8.0     3.0     1.5    7.0     1.0     2.5           0.0    4.5      1.0                 1.0      3.0       2.0
       0.0620    3.5     1.5     0.0    2.0     0.0     0.0           0.5    0.0      0.0                 0.0      1.0       0.0
       0.0320    0.0     0.0     0.0    0.0     0.0     0.0           0.0    0.0      0.0                 0.0      0.0       0.0284       0.2500    4.0     2.0     0.0    9.0     2.0     1.0           1.0    1.0      0.0                 0.0      1.0       2.0
       0.1250            0.0     0.0    1.0     0.0     0.0           0.0    0.0      0.0                 0.0      0.0       0.0
       0.0620    0.0     0.0     0.0    0.0     0.0     0.0           0.0    0.0      0.0                 0.0      0.0       0.0285       0.5000    9.0     9.0     5.0    9.0             9.0           9.0    9.0      9.0                 9.0                9.0
       0.2500    9.0     8.0     2.5    9.0     9.0     9.0           9.0    9.0      6.5                 8.0      7.0       8.5
       0.1250    9.0     6.0     1.5    9.0     9.0     8.0           8.5    9.0      5.0                 6.0      6.0       6.5
       0.0620    9.0     4.0     1.0    9.0     7.0     6.0           5.0    9.0      4.0                 5.0      5.0       7.0
       0.0320    5.0     2.0     1.0    9.0     2.0     4.0           1.0    6.0      2.0                 1.0      1.0       3.0
       0.0160    5.0     0.0     0.0    6.0     2.0     0.0           0.0    0.0      0.0                 0.0      0.0       1.0
                                                       表II(续)
                                                                                 G             O      T
                 A      A       C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M       A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B       S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E       O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L       B      L      P      E      S      G      I      W      A      T      R      X286     0.2500     9.0    5.5     0.0    9.0    2.0    4.0           1.0    6.5    0.5           0.5    0.0    1.0
     0.1250     4.5    1.0     0.0    6.5    0.0    0.0           0.0    1.5    0.0           0.0    1.0    0.0
     0.0620     0.5    0.0     0.0    0.5    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0320     0.0    0.0     0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0287     0.2500     9.0    7.0     0.0    9.0    1.0    5.0           7.0    9.0    5.0           4.0    4.0    5.0
     0.1250     9.0    4.0     0.0    9.0    0.0    1.0           3.0    6.0    2.0           2.0    4.0    4.0
     0.0620     6.0    3.0     0.0    9.0    0.0    0.0           1.0    5.0    0.0           0.0    0.0    1.0
     0.0320     1.0    0.0     0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0160     0.0    0.0     0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0288     0.2500     9.0    9.0     1.0    9.0    9.0    9.0           5.0    9.0    5.0           4.0    9.0    9.0
     0.1250     9.0    9.0     0.0    9.0    0.0    9.0           4.0    5.0    3.0           1.0    3.0    9.0
     0.0620     9.0    6.0     0.0    9.0    0.0    9.0           0.0    0.0    0.0           0.0    0.0    2.0
     0.0320     5.0    2.0     0.0    9.0    0.0    9.0           0.0    0.0    0.0           1.0    0.0    1.0
     0.0160            2.0     0.0    5.0    0.0    1.0           0.0    1.0    0.0           0.0    0.0    0.0
                                                            表II(续)
                                                                                                   G                   O         T
                      A       A       C      C      G       I         I         E         S        L        G          R         R         Z
                      B       M       A      H      A       P         P         C         E        X        L          Y         Z         E
                  U       B       S      E      L       O         O         H         T        M        X          S         A         A化合物   施用率       T       E       O      A      A       H         S         C         V        A        M          A         W         M编号  (公斤/公顷)    H       L       B      L      P       E         S         G         I        W        A          T         R         X289      0.2500      9.0     5.0     0.0    9.0    0.0     9.0                 0.0       0.0      1.0                 0.0       0.0       0.0
          0.1250      9.0     1.0     0.0    9.0    0.0     2.0                 1.0       1.0      0.0                 0.0       0.0       0.0
          0.0620      2.0     0.0     0.0    9.0            0.0                 0.0       0.0      0.0                 0.0       0.0       0.0
          0.0320      0.0     0.0     0.0    0.0    0.0     0.0                 1.0       0.0      0.0                 0.0       0.0       0.0
          0.0160      0.0     0.0     0.0    0.0    0.0     0.0                 0.0       0.0      0.0                 0.0       0.0       1.0290      0.2500      5.0     2.0     0.0    9.0    0.0     1.0                 1.0       3.0      1.0                 0.0       0.0       1.0
          0.1250      3.0     0.0     0.0    9.0    0.0     0.0                 1.0       1.0      0.0                 0.0       0.0       0.0
          0.0620      1.0     0.0     0.0    1.0    0.0     0.0                 0.0       0.0      0.0                 0.0       0.0       1.0
          0.0320      0.0     0.0     0.0           0.0     0.0                 0.0       0.0      0.0                 0.0       0.0       1.0291      0.2500      9.0     9.0     0.0    9.0    9.0     9.0                 0.0       9.0      2.0                 7.0       7.0       4.0
          0.1250      9.0     7.0     0.0    9.0    3.0     5.0                 0.0       0.0      0.0                 3.0       5.0       3.0
          0.0620      9.0     3.0     0.0    9.0    3.0     2.0                 0.0       0.0      0.0                 0.0       3.0       0.0
          0.0320      0.0     0.0     0.0    0.0    3.0     0.0                 0.0       0.0      0.0                 0.0       0.0       0.0
          0.0160      0.0     0.0     0.0           3.0     0.0                 0.0       0.0      0.0                 0.0       0.0       0.0
                                                             表II(续)
                                                                                     G                 O      T
                  A      A      C      C      G      I       I       E       S       L        G        R      R       Z
                  B      M      A      H      A      P       P       C       E       X        L        Y      Z       E
                  U      B      S      E      L      O       O       H       T       M        X        S      A       A化合物     施用率     T      E      O      A      A      H       S       C       V       A        M        A      W       M编号   (公斤/公顷)   H      L      B      L      P      E       S       G       I       W        A        T      R       X292       0.2500    9.0    8.0    6.0    9.0    5.0    9.0             0.0     3.0     3.0               3.0    8.0     9.0
       0.1250    9.0    2.0    0.0    6.0    5.0    3.0             0.0     0.0     0.0               0.0    7.0     9.0
       0.0620    0.0    0.0    0.0    0.0    0.0    0.0             0.0     0.0     0.0               0.0    0.0     0.0293       0.2500    9.0    9.0    8.0    9.0    9.0    9.0             0.0     5.0     3.0               7.0    8.0     8.0
       0.1250    9.0    5.0    0.0    9.0    0.0    3.0             0.0     0.0     0.0               4.0    6.0     4.0
       0.0620    0.0    0.0    0.0    0.0    0.0    0.0             0.0     0.0     0.0               0.0    0.0     0.0294       0.2500    9.0    3.0    0.0    9.0    9.0    3.0             0.0     0.0     2.0               3.0    5.0     6.0
       0.1250    9.0    3.0    0.0    9.0    0.0    3.0             0.0     0.0     1.0               3.0    3.0     1.0
       0.0620    9.0    1.0    0.0    7.0    0.0    2.0             0.0     0.0     0.0               0.0    0.0     0.0
       0.0320    3.0    0.0    0.0    0.0    0.0    0.0             0.0     0.0     0.0               0.0    0.0     0.0
       0.0160    0.0    0.0    0.0           0.0    0.0             0.0     0.0     0.0               0.0    0.0     0.0295       0.2500    9.0    9.0    9.0    9.0    9.0    9.0             0.0     0.0     0.0               3.0    5.0     4.0
       0.1250    9.0    5.0    2.0    9.0    3.0    9.0             0.0     0.0     0.0               0.0    4.0     2.0
       0.0620    9.0    1.0    0.0    0.0    0.0    2.0             0.0     0.0     0.0               0.0    0.0     0.0
       0.0320    0.0    0.0    0.0    0.0    0.0    0.0             0.0     0.0     0.0               0.0    0.0     0.0
                                                           表II(续)
                                                                                              G                   O       T
                    A       A       C      C       G       I         I         E         S        L        G          R       R         Z
                    B       M       A      H       A       P         P         C         E        X        L          Y       Z         E
                U       B       S      E       L       O         O         H         T        M        X          S       A         A化合物   施用率     T       E       O      A       A       H         S         C         V        A        M          A       W         M编号 (公斤/公顷)   H       L       B      L       P       E         S         G         I        W        A          T       R         X296      0.2500    9.0     5.0     0.0    9.0     9.0     9.0                 0.0       0.0      4.0                 7.0     7.0       5.0
          0.1250    9.0     2.0     0.0    0.0     0.0     3.0                 0.0       0.0      0.0                 4.0     5.0       3.0
          0.0620    7.0     1.0     0.0    0.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0
          0.0320    0.0     0.0     0.0    0.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0297      0.2500    9.0     7.0     2.0    9.0     5.0     5.0                 0.0       6.0      0.0                 3.0     4.0       3.0
          0.1250    7.0     6.0     0.0    9.0     5.0     3.0                 0.0       0.0      0.0                 1.0     1.0       0.0
          0.0620    7.0     1.0     0.0    9.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0
          0.0320            0.0     0.0    0.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0298      0.2500    9.0     3.0     3.0    9.0     3.0     8.0                 0.0       4.0      2.0                 3.0     3.0       4.0
          0.1250    9.0     3.0     0.0    9.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0
          0.0620    0.0     0.0     0.0    9.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0
          0.0320    0.0     0.0     0.0    0.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0299      0.2500    9.0     8.0     3.0    9.0     5.0     6.0                 0.0       2.0      2.0                 2.0     2.0       3.0
          0.1250    9.0     2.0     0.0    9.0     0.0     1.0                 0.0       0.0      0.0                 0.0     0.0       0.0
          0.0820    0.0     0.0     0.0    4.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0
          0.0320    0.0     0.0     0.0    0.0     0.0     0.0                 0.0       0.0      0.0                 0.0     0.0       0.0
                                                    表II(续)
                                                                                                   G                   O        T
                    A       A       C       C       G       I        I          E         S        L        G          R        R         Z
                    B       M       A       H       A       P        P          C         E        X        L          Y        Z         E
                U       B       S       E       L       O        O          H         T        M        X          S        A         A化合物   施用率     T       E       O       A       A       H        S          C         V        A        M          A        W         M编号  (公斤/公顷)  H       L       B       L       P       E        S          G         I        W        A          T        R         X300      0.5000    9.0     9.0     9.0     9.0             9.0                 9.0       9.0      4.0                 9.0                7.0
          0.2500    9.0     9.0     4.3     9.0     8.5     8.3                 9.0       9.0      4.3                 8.0      7.0       5.3
          0.1250    9.0     9.0     3.3     9.0     8.5     7.7                 5.3       9.0      1.7                 4.0      5.5       4.7
          0.0620    8.0     6.3     0.3     9.0     8.5     3.3                 1.3       8.0      0.0                 1.3      3.5       1.0
          0.0320    7.7     1.7     0.0     9.0     4.0     1.7                 0.0       0.7      0.0                 1.7      0.0       0.3
          0.0160    4.5     0.0     0.0     9.0     0.0     0.0                 0.0       0.0      0.0                 0.0      0.0       0.0301      0.2500    9.0     9.0     0.0     9.0     9.0     2.0                 8.0       9.0      3.0                 0.0      6.0       4.0
          0.1250    9.0     0.0     0.0     9.0     9.0     0.0                 7.0       9.0      0.0                 0.0      2.0       4.0
          0.0620    9.0     0.0     0.0     9.0     9.0     0.0                 0.0       7.0      0.0                 0.0      0.0       0.0
          0.0320    4.0     0.0     0.0     4.0     0.0     0.0                 0.0       2.0      0.0                 0.0      0.0       0.0
          0.0160    0.0     0.0     0.0     3.0     0.0     0.0                 0.0       0.0      0.0                 0.0      0.0       0.0302      0.2500    9.0     9.0     0.0     9.0     9.0     9.0                 9.0       9.0      5.0                 6.0      7.0       8.0
          0.1250    9.0     9.0             9.0     0.0     9.0                 9.0       9.0      4.0                 4.0      6.0       7.0
          0.0620    9.0     3.0     0.0     9.0     0.0     3.0                 6.0       9.0      3.0                 3.0      6.0       6.0
          0.0320    9.0     3.0     0.0     9.0     0.0     1.0                 3.0       9.0      3.0                 0.0     .0.0       5.0
                                                         表II(续)
                                                                                      G              O       T
                  A       A       C       C       G       I      I      E      S      L      G       R       R      Z
                  B       M       A       H       A       P      P      C      E      X      L       Y       Z      E
                  U       B       S       E       L       O      O      H      T      M      X       S       A      A化合物    施用率      T       E       O       A       A       H      S      C      V      A      M       A       W      M编号  (公斤/公顷)    H       L       B       L       P       E      S      G      I      W      A       T       R      X303      0.2500     9.0     9.0     8.0     9.0     9.0     9.0           8.0    9.0    5.0            7.0     7.0    8.0
      0.1250     9.0     9.0     0.0     9.0     0.0     3.0           8.0    9.0    4.0                    5.0    7.0
      0.0620     9.0     7.0     0.0     9.0     0.0     3.0           7.0    9.0    2.0            1.0     4.0    6.0
      0.0320     0.0     0.0     0.0     9.0     0.0     0.0           0.0    4.0    0.0            0.0     1.0    4.0
      0.0160     0.0     0.0     0.0     9.0     0.0     0.0           0.0    0.0    0.0            0.0     0.0    1.0304      0.2500     9.0     7.0     4.0     9.0     9.0     9.0           0.0    9.0    7.0            4.0     0.0    3.0
      0.1250     9.0     4.0     1.0     9.0     9.0     4.0           0.0    1.0    4.0            0.0     0.0    1.0
      0.0620     7.0     2.0     0.0     3.0     7.0     3.0           0.0    0.0    3.0            0.0     0.0    0.0
      0.0320     3.0     1.0     0.0     0.0     0.0     0.0           0.0    0.0    0.0            0.0     0.0    0.0
      0.0160     0.0     0.0     0.0     0.0     0.0     0.0           0.0    0.0    0.0            0.0     0.0    0.0305      0.5000     9.0     9.0     9.0     9.0             9.0           5.0    9.0    8.5            7.0            7.0
      0.2500     9.0     9.0     9.0     9.0     9.0     9.0           2.0    8.3    7.7            4.7     3.0    5.7
      0.1250     9.0     7.7     8.0     9.0     9.0     8.3           0.0    6.3    7.0            2.3     3.0    4.0
      0.0620     9.0     4.7     5.3     9.0     0.0     6.3           0.0    4.0    5.7            1.3     1.0    2.7
      0.0320     6.7     2.3     3.0     6.0     0.0     3.0           0.0    0.0    3.0            0.7     0.0    0.7
      0.0160     3.5     1.5     0.0     3.5     0.0     1.5           0.0    0.0    1.0            0.0     0.0    0.0
                                                    表II(续)
                                                                                              G                 O        T
                      A       A       C       C       G       I        I        E        S        L        G        R        R        Z
                      B       M       A       H       A       P        P        C        E        X        L        Y        Z        E
                  U       B       S       E       L       O        O        H        T        M        X        S        A        A化合物    施用率      T       E       O       A       A       H        S        C        V        A        M        A        W        M编号  (公斤/公顷)    H       L       B       L       P       E        S        G        I        W        A        T        R        X306      0.2500      9.0     0.0     0.0     9.0     0.0     1.0               0.0      0.0      1.0               0.0      4.0      0.0
          0.1250      0.0     0.0     0.0     0.0     0.0     0.0               0.0      0.0      0.0               0.0      0.0      0.0307      0.2500      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      9.0               9.0      8.0      9.0
          0.1250      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      8.3               8.0      7.5      8.7
          0.0620      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      8.3               7.3      5.5      7.7
          0.0320      9.0     9.0     6.0     9.0     8.0     9.0               7.7      9.0      7.7               7.0      1.5      7.3
          0.0160      9.0     9.0     3.3     9.0     4.5     5.7               3.7      8.3      4.7               4.7      1.0      3.3308      0.2500      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      9.0               9.0      9.0      9.0
          0.1250      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      9.0               9.0      8.7      8.8
          0.0620      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      9.0               8.8      8.0      8.8
          0.0320      9.0     9.0     8.3     9.0     9.0     8.8               8.3      8.8      9.0               7.8      5.7      8.0
          0.0160      9.0     8.8     4.4     9.0     8.5     7.6               5.4      8.4      8.0               5.8      4.5      6.0309      0.2500      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      9.0               9.0      9.0      9.0
          0.1250      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      9.0               9.0      8.0      9.0
          0.0620      9.0     9.0     9.0     9.0     9.0     9.0               9.0      9.0      9.0               9.0      6.0      8.5
          0.0320      9.0     9.0     7.5     9.0     9.0     9.0               8.0      9.0      8.0               7.0      4.0      7.0
          0.0160      9.0     9.0     6.5     9.0     0.0     9.0               3.5      8.0      6.5               5.5      2.0      4.5
                                                                 表II(续)
                                                                                               G              O      T
                    A        A        C      C      G       I         I         E         S        L       G      R      R        Z
                    B        M        A      H      A       P         P         C         E        X       L      Y      Z        E
                U        B        S      E      L       O         O         H         T        M       X      S      A        A化合物   施用率     T        E        O      A      A       H         S         C         V        A       M      A      W        M编号 (公斤/公顷)   H        L        B      L      P       E         S         G         I        W       A      T      R        X310     0.2500     9.0      9.0      4.0    9.0    9.0     9.0                 9.0       9.0      5.0            8.0    7.0      7.0
         0.1250     9.0      7.0      0.0    9.0    9.0     3.0                 3.0       9.0      3.0            8.0    7.0      5.0
         0.0620     9.0      4.0      0.0    5.0    9.0     1.0                 0.0       8.0      0.0            3.0    1.0      2.0
         0.0320     9.0      1.0      0.0           0.0     1.0                 0.0       0.0      0.0            0.0    1.0      0.0
         0.0160     9.0      0.0      0.0    0.0    0.0     0.0                 0.0       0.0      0.0            0.0    0.0      0.0311     0.2500     9.0      9.0      4.0    4.0    9.0     9.0                 7.0       9.0      4.0            8.0    7.0      6.0
         0.1250     9.0      4.0      4.0           0.0     4.0                 0.0       8.0      4.0            6.0    3.0      3.0
         0.0620     0.0      0.0      0.0    0.0    0.0     0.0                 0.0       0.0      0.0            0.0    0.0      0.0312     0.2500     9.0      9.0      0.0    9.0    9.0     9.0                 9.0       9.0      9.0            9.0    7.0      6.0
         0.1250     9.0      9.0             9.0    0.0     9.0                 9.0       9.0      9.0            8.0    2.0      6.0
         0.0620     9.0      9.0      0.0    9.0    0.0     9.0                 9.0       9.0      3.0            5.0    0.0      4.0
         0.0320     9.0      3.0      0.0    9.0    0.0     2.0                 7.0       7.0      3.0            5.0    0.0      3.0
         0.0160     9.0      0.0      0.0    9.0    0.0     0.0                 3.0       0.0      0.0            0.0             0.0
                                                      表II(续)
                                                                                          G             O      T
                     A       A       C       C       G       I       I      E      S      L      G      R      R      Z
                     B       M       A       H       A       P       P      C      E      X      L      Y      Z      E
                     U       B       S       E       L       O       O      H      T      M      X      S      A      A化合物     施用率        T       E       O       A       A       H       S      C      V      A      M      A      W      M编号   (公斤/公顷)      H       L       B       L       P       E       S      G      I      W      A      T      R      X313       0.2500       9.0     9.0     3.0     9.0     9.0     9.0            9.0    9.0    9.0           8.0    3.0    4.0
       0.1250       9.0     4.0     0.0     9.0     0.0     4.0            9.0    9.0    3.0           4.0    0.0    0.0
       0.0620       9.0     0.0     0.0     9.0     0.0     0.0            0.0    9.0    0.0           0.0    0.0    0.0
       0.0320       4.0     0.0     0.0     9.0     0.0                    0.0    0.0    0.0           0.0    0.0    0.0
       0.0160       0.0     0.0     0.0     0.0     0.0     0.0            0.0    0.0    0.0           0.0    0.0    0.0314       0.2500       9.0     9.0     9.0     9.0     9.0     9.0            9.0    9.0    9.0           5.0    9.0    9.0
       0.1250       9.0     9.0     9.0     9.0     9.0     9.0            9.0    9.0    9.0           5.0    9.0    7.0
       0.0620       9.0     7.0     0.0     9.0     9.0     9.0            2.0    7.0    2.0           0.0    3.0    4.0
       0.0320       9.0     7.0     0.0     9.0     0.0     9.0            0.0    7.0    0.0           0.0    0.0    0.0
       0.0160       9.0     2.0     0.0     9.0     0.0     9.0            0.0    0.0    0.0           0.0    0.0    0.0315       0.5000       9.0     9.0     5.0     9.0             9.0            9.0    9.0    9.0           7.0           5.0
       0.2500       9.0     9.0     2.5     9.0     9.0     9.0            9.0    9.0    9.0           7.5    8.0    3.5
       0.1250       9.0     7.0     0.0     9.0     9.0     7.5            4.5    8.5    5.0           5.5    8.0    2.0
       0.0620       7.0     2.5     0.0     9.0     0.0     6.5            0.0    3.0    3.0           2.5    1.0    0.5
       0.0320       6.0     0.0     0.0     2.0     0.0     4.0            0.0    0.0    2.0           0.5    1.0    0.0
       0.0160       0.0     0.0     0.0     0.0     0.0     0.0            0.0    0.0    0.0           0.0    0.0    0.0
                                                  表II(续)
                                                                                                        G                    O        T
                     A       A        C       C       G       I          I          E         S         L          G         R        R         Z
                     B       M        A       H       A       P          P          C         E         X          L         Y        Z         E
                 U       B        S       E       L       O          O          H         T         M          X         S        A         A化合物   施用率      T       E        O       A       A       H          S          C         V         A          M         A        W         M编号 (公斤/公顷)    H       L        B       L       P       E          S          G         I         W          A         T        R         X316      0.2500     9.0     9.0      9.0     9.0     9.0     9.0                   9.0       9.0       6.0                  7.0      4.0       7.0
          0.1250     9.0     9.0      7.0     9.0     0.0     9.0                   7.0       9.0       6.0                  5.0      2.0       4.0
          0.0620     9.0     6.0      1.0     9.0             3.0                   2.0       6.0       2.0                  2.0      1.0       3.0
          0.0320     9.0     4.0      1.0     9.0     0.0     3.0                   1.0       6.0                            1.0      1.0       1.0
          0.0160     9.0     0.0      0.0     9.0     0.0     0.0                   0.0       0.0       1.0                  0.0      0.0       1.0317      0.2500     9.0     9.0      8.0     9.0     9.0     9.0                   9.0       9.0       9.0                  9.0      9.0       8.5
          0.1250     9.0     9.0      7.5     9.0     9.0     9.0                   9.0       9.0       8.0                  7.5      7.0       7.5
          0.0620     9.0     9.0      3.5     9.0     7.0     6.5                   9.0       9.0       8.0                  7.0      6.0       7.5
          0.0320     9.0     9.0      2.5     9.0     0.0     6.0                   8.0       9.0       5.5                  5.0      3.0       7.0
          0.0160     9.0     7.5      0.0     8.0     0.0     4.0                   6.5       9.0       3.0                  4.0      2.0       4.5318      0.5000     9.0     9.0      9.0     9.0             9.0                   9.0       9.0       9.0                  9.0                7.0
          0.2500     9.0     9.0      9.0     9.0     9.0     9.0                   9.0       9.0       8.0                  7.5      7.0       7.5
          0.1250     9.0     9.0      9.0     9.0     9.0     8.0                   9.0       9.0       9.0                  6.5      6.0       7.5
          0.0620     9.0     9.0      9.0     9.0     9.0     7.0                   9.0       9.0       7.0                  6.5      2.0       6.5
          0.0320     9.0     7.0      2.5     9.0     0.0     5.5                   8.0       9.0       6.5                  3.5      1.0       6.5
          0.0160     9.0     3.5      2.0     9.0     0.0     3.0                   4.0       9.0       4.0                  3.5      1.0       6.5
                                                     表II(续)
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号  (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X319      0.2500    9.0    9.0    1.0    9.0    9.0    9.0           9.0    9.0    9.0           6.0    5.0    2.0
      0.1250    9.0    3.0    0.0    9.0    9.0    4.0           2.0    5.0    0.0           4.0    4.0    2.0
      0.0620    1.0    1.0    0.0    9.0    7.0    1.0           1.0           3.0           1.0    1.0    1.0
      0.0320    0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    1.0           0.0    0.0    0.0
      0.0160    0.0    0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0320      0.2500    9.0    9.0    1.0    9.0    9.0    7.0           9.0    9.0    4.0           7.0    7.0    2.0
      0.1250    9.0    1.0    0.0    9.0    9.0    2.0           2.0    4.0    2.0           5.0    5.0    2.0
      0.0620    3.0    1.0    1.0    9.0    7.0    0.0           0.0    1.0    2.0           1.0    1.0    1.0
      0.0320    0.0    1.0    0.0    4.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.0160    0.0    0.0    0.0    0.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0321      0.5000    9.0    9.0    9.0    9.0           9.0           9.0    9.0    9.0           9.0           9.0
      0.2500    9.0    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    8.0    8.5
      0.1250    9.0    9.0    6.5    9.0    9.0    9.0           9.0    9.0    8.0           7.0    7.0    7.0
      0.0620    9.0    9.0    5.5    9.0    7.0    8.0           7.0    9.0    6.0           5.5    6.0    6.0
      0.0320    9.0    8.5    1.5    9.0    9.0    6.0           5.0    7.0    3.5           3.5    5.0    4.0
      0.0160    9.0    7.0    1.0    9.0    5.0    0.0           0.0    2.0    1.0           1.0    1.0    1.0
                                                         表II(续)
                                                                                    G             O      T
                A       A       C       C       G       I      I      E      S      L      G      R      R      Z
                B       M       A       H       A       P      P      C      E      X      L      Y      Z      E
                U       B       S       E       L       O      O      H      T      M      X      S      A      A化合物  施用率      T       E       O       A       A       H      S      C      V      A      M      A      W      M编号(公斤/公顷)     H       L       B       L       P       E      S      G      I      W      A      T      R      X322    0.2500      9.0     9.0     6.0     9.0     9.0     7.0           2.0    9.0    6.0           6.0    9.0    7.0
   0.1250      9.0     8.0     3.5     9.0     9.0     7.5           2.0    9.0    5.5           3.5    3.0    5.5
   0.0620      7.0     5.0     2.5     9.0     1.0     4.0           0.0    2.0    3.5           1.5    1.0    2.5
   0.0320      6.5     1.5     0.0     9.0     1.0     2.0           0.0    1.0    2.0           1.0    0.0    1.5
   0.0160      3.0     0.5     0.0     3.0     1.0     1.5           0.0    1.0    0.0           0.0    0.0    0.5323    0.5000      9.0     9.0     0.5     9.0     9.0     9.0           9.0    9.0    7.5           6.5    7.0    6.5
   0.2500      9.0     9.0     0.3     9.0     9.0     9.0           9.0    9.0    4.0           5.7    5.2    3.7
   0.1250      9.0     8.9     1.8     9.0     8.0     9.0           6.7    9.0    2.3           4.7    4.6    1.9
   0.0620      9.0     4.9     0.3     9.0     4.3     8.6           4.0    8.6    1.6           2.6    1.2    0.7
   0.0320      6.2     2.7     0.2     7.3     5.0     6.7           1.8    4.3    0.3           0.7    0.3    0.2
   0.0160      3.8     2.3     0.0     4.2     2.5     3.5           0.2    1.0    0.5           0.2    0.2    0.2324    0.2500      9.0     9.0     9.0     9.0     9.0     9.0           9.0    9.0    9.0           9.0    9.0    9.0
   0.1250      9.0     9.0     9.0     9.0     0.0     9.0           9.0    9.0    9.0           9.0    9.0    9.0
   0.0620      9.0     9.0     9.0     9.0     0.0     9.0           7.0    9.0    8.5           7.0    9.0    8.5
   0.0320      9.0     8.0     3.0     9.0     0.0     9.0           1.0    7.0    5.0           3.5    3.0    6.0
   0.0160      9.0     7.0     3.0     9.0     0.0     4.5           1.0    3.5    3.5           2.0    1.0    2.5
                                                   表II(续)
                                                                                  G             O      T
                 A     A      C       C       G       I      I      E      S      L      G      R      R      Z
                 B     M      A       H       A       P      P      C      E      X      L      Y      Z      E
                 U     B      S       E       L       O      O      H      T      M      X      S      A      A化合物  施用率       T     E      O       A       A       H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H     L      B       L       P       E      S      G      I      W      A      T      R      X325      0.5000     9.0   9.0    9.0     9.0             9.0           9.0    9.0    9.0           9.0           7.0
     0.2500     9.0   9.0    9.0     9.0     9.0     9.0           9.0    9.0    9.0           6.5    4.0    7.0
     0.1250     9.0   8.0    6.0     9.0     8.0     7.5           8.0    9.0    6.5           5.0    0.0    5.5
     0.0620     9.0   8.5    3.0     9.0     0.0     4.0           4.0    4.5    3.0           2.0    0.0    2.5
     0.0320     6.5   4.0    0.0     9.0     0.0     2.0           2.0    3.0    1.0           2.0    0.0    1.0
     0.0160     0.0   0.0    0.0     9.0     0.0     0.0           0.0    0.0    0.0           0.0    0.0    0.0326      0.5000     9.0   9.0    4.0     9.0             9.0           9.0    9.0    9.0           8.0           7.0
     0.2500     9.0   9.0    3.0     9.0     9.0     9.0           9.0    9.0    4.5           6.0    1.0    2.5
     0.1250     9.0   9.0    3.0     9.0     0.0     9.0           7.0    9.0    3.0           4.0    0.0    1.0
     0.0620     4.5   6.5    0.0     9.0     0.0     2.5           3.0    4.5    2.0           1.0    0.0    0.5
     0.0320     4.5   2.5    0.0     9.0     0.0     0.0           0.0    2.0    0.0           0.0    0.0    0.0
     0.0160     0.0   0.0    0.0     9.0     0.0     0.0           0.0    0.0    0.0           0.0    0.0    0.0327      0.2500     9.0   5.0    0.0     9.0     0.0     5.0           7.0    9.0    3.0           0.0    2.0    7.0
     0.1250     9.0   0.0    0.0     9.0     0.0     0.0           3.0    9.0    1.0           0.0    1.0    3.0
     0.0620     9.0   0.0    0.0     9.0     0.0     0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0320     0.0   0.0    0.0     9.0     0.0     0.0           0.0    0.0    0.0           0.0    0.0    0.0
     0.0160     0.0   0.0    0.0     9.0     0.0     0.0           0.0    0.0    0.0           0.0    0.0    0.0
                                                        表II(续)
                                                                                            G               O      T
                  A       A       C       C       G       I       I       E        S        L       G       R      R      Z
                  B       M       A       H       A       P       P       C        E        X       L       Y      Z      E
                  U       B       S       E       L       O       O       H        T        M       X       S      A      A化合物    施用率      T       E       O       A       A       H       S       C        V        A       M       A      W      M编号   (公斤/公顷)   H       L       B       L       P       E       S       G        I        W       A       T      R      X328      0.2500     9.0     5.0     0.0     9.0     0.0     9.0             0.0      9.0      3.0             0.0    0.0    0.0
      0.1250     9.0     3.0     0.0     9.0     0.0     0.0             0.0      9.0      2.0             0.0    0.0    0.0
      0.0620     9.0     0.0     0.0     9.0     0.0     0.0             0.0      0.0      2.0             0.0    0.0    0.0
      0.0320     3.0     0.0     0.0     9.0     0.0     0.0             0.0      0.0      0.0             0.0    0.0    0.0
      0.0160     0.0     0.0     0.0     9.0     0.0     0.0             0.0      0.0      0.0             0.0    0.0    0.0329      0.2500     9.0     9.0     8.5     9.0     9.0     9.0             9.0      9.0      8.0             8.0    7.0    7.5
      0.1250     9.0     9.0     9.0     9.0     9.0     9.0             7.0      9.0      9.0             6.5    6.0    7.0
      0.0620     9.0     8.0     7.0     9.0     6.0     8.0             4.5      9.0      7.5             5.0    4.0    6.5
      0.0320     9.0     7.0     2.0     9.0     1.0     4.0             1.0      2.5      6.0             2.5    2.0    2.5
      0.0160     9.0     3.0     0.5     9.0     1.0     2.5             0.0      1.5      5.0             1.5    1.0    1.5330      0.2500     9.0     9.0     2.0     9.0     9.0     6.0             5.0      9.0      7.0             6.0    5.0    7.0
      0.1250     9.0     7.0             9.0     9.0     2.0             1.0      7.0      7.0             3.0    3.0    5.0
      0.0620     9.0     1.0     1.0     9.0     0.0     1.0             0.0      4.0      4.0             0.0    0.0    1.0
      0.0320     3.0     1.0     0.0     9.0     0.0     1.0             0.0      0.0      1.0             0.0    0.0    0.0
      0.0160     1.0     0.0     0.0     3.0     0.0     0.0             0.0      0.0      0.0             0.0    0.0    0.0
                                                                  表II(续)
                                                                                           G             O      T
                  A       A       C       C       G       I       I       E       S        L      G      R      R      Z
                  B       M       A       H       A       P       P       C       E        X      L      Y      Z      E
                  U       B       S       E       L       O       O       H       T        M      X      S      A      A化合物    施用率      T       E       O       A       A       H       S       C       V        A      M      A      W      M编号  (公斤/公顷)    H       L       B       L       P       E       S       G       I        W      A      T      R      X331      0.2500     3.0     2.0     0.0     9.0     0.0     0.0             0.0     0.0     0.0            0.0    0.0    0.0
      0.1250     3.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.0            0.0    0.0    0.0
      0.0620     0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.0            0.0    0.0    0.0332      0.5000     9.0     9.0     9.0     9.0             9.0             9.0     9.0     9.0            9.0           5.0
      0.2500     9.0     9.0     6.0     9.0     9.0     8.5             9.0     9.0     5.0            6.5    1.0    4.5
      0.1250     9.0     9.0     4.0     9.0     9.0     7.0             7.5     9.0     3.0            5.5    0.0    1.5
      0.0620     8.0     8.0     0.0     9.0     8.0     3.0             1.5     5.5     1.0            3.5    0.0    0.5
      0.0320     4.5     0.0     0.0     9.0     0.0     1.5             0.0     2.5     0.0            1.5    0.0    0.0
      0.0160     0.0     0.0     0.0     0.0     0.0     0.0             0.0     0.0     0.0            0.0    0.0    0.0333      0.5000     9.0     9.0     2.0     9.0             9.0             9.0     9.0     4.0            6.0           5.0
      0.2500     9.0     9.0     5.5     9.0     9.0     7.5             9.0     9.0     4.0            4.0    5.0    7.0
      0.1250     8.0     8.0     1.5     9.0     9.0     4.5             7.5     7.5     2.0            1.5    3.0    6.5
      0.0620     7.5     4.0     1.5     9.0     0.0     2.0             7.5     7.5     0.5            1.0    3.0    5.5
      0.0320     7.0     1.5     0.0     9.0     0.0     1.5             6.5     7.0     0.5            0.0    0.0    3.0
      0.0160     3.0     0.0     0.0     9.0     0.0     2.0             0.0     7.0     1.0            0.0    0.0    3.0
                                                         表II(续)
                                                                                          G               O      T
                   A       A       C       C       G       I       I       E      S       L       G       R      R      Z
                   B       M       A       H       A       P       P       C      E       X       L       Y      Z      E
                   U       B       S       E       L       O       O       H      T       M       X       S      A      A化合物    施用率       T       E       O       A       A       H       S       C      V       A       M       A      W      M编号   (公斤/公顷)    H       L       B       L       P       E       S       G      I       W       A       T      R      X334       0.2500     9.0     9.0     1.5     9.0     9.0     9.0             7.5     9.0    2.0             4.5    3.0    4.0
       0.1250     9.0     8.5     1.5     9.0     5.0     9.0             1.0     8.0    1.5             1.5    1.0    1.5
       0.0620     9.0     6.5     0.0     9.0     1.0     7.5             1.0     3.5    0.5             0.5    1.0    0.5
       0.0320     8.0     2.0     0.0     8.0     0.0     3.5             0.0     1.0    0.0             0.0    0.0    0.0
       0.0160     7.0     0.5     0.0     7.5     0.0     1.5             0.0     1.0    0.0             0.0    0.0    0.5335       0.5000     9.0     9.0     9.0     9.0             9.0             9.0     9.0    9.0             9.0           9.0
       0.2500     9.0     9.0     9.0     9.0     9.0     9.0             9.0     9.0    7.5             8.5    8.0    8.3
       0.1250     9.0     9.0     8.3     9.0     2.7     9.0             8.8     9.0    5.8             7.3    5.0    8.0
       0.0620     9.0     9.0     7.8     9.0     2.3     9.0             4.3     8.8    4.0             6.3    3.3    4.3
       0.0320     9.0     6.3     1.8     9.0     0.0     5.5             1.3     4.8    2.0             4.3    1.0    1.5
       0.0160     8.5     2.8     0.0     7.8     0.3     4.0             0.5     3.0    0.5             2.3    0.0    0.5336       0.2500     9.0     9.0     7.0     9.0     8.0     9.0             8.5     9.0    9.0             7.5    6.0    6.0
       0.1250     9.0     9.0     6.0     9.0     2.0     9.0             8.0     9.0    7.0             6.0    6.0    6.5
       0.0620     9.0     8.0     4.0     9.0     4.0     4.5             4.5     9.0    5.0             5.5    3.0    5.5
       0.0320     9.0     3.5     2.0     9.0     0.0     3.0             1.5     2.5    2.0             3.5    1.0    3.0
       0.0160     6.5     0.0     0.0     7.5     0.0     2.5             0.0     0.0    0.0             1.5    0.0    1.0
                                                          表II(续)
                                                                                       G             O      T
                  A       A       C       C       G       I       I      E      S      L      G      R      R      Z
                  B       M       A       H       A       P       P      C      E      X      L      Y      Z      E
                  U       B       S       E       L       O       O      H      T      M      X      S      A      A化合物    施用率      T       E       O       A       A       H       S      C      V      A      M      A      W      M编号   (公斤/公顷)   H       L       B       L       P       E       S      G      I      W      A      T      R      X337      0.5000     9.0     9.0     9.0     9.0             9.0            9.0    9.0    8.0           8.0           7.0
      0.2500     9.0     9.0     9.0     9.0     9.0     8.0            9.0    9.0    7.5           7.0    5.0    6.0
      0.1250     9.0     9.0     7.5     9.0     9.0     8.0            6.0    9.0    6.0           5.5    2.0    2.5
      0.0620     9.0     8.0     3.5     9.0     4.0     3.5            1.5    3.5    2.5           2.0    1.0    1.5
      0.0320     6.5     2.0     3.0     9.0     3.0     2.0            0.0    2.0    0.5           0.5    0.0    1.0
      0.0160     0.0     0.5     2.5     9.0     5.0     1.0            0.0    0.0    0.5           0.0    0.0    0.5338      0.2500     9.0     9.0     7.0     9.0     9.0     9.0            9.0    9.0    9.0           8.0    8.0    7.0
      0.1250     9.0     9.0     5.0     9.0     6.0     6.0            7.0    9.0    7.0           6.0    5.0    5.0
      0.0620     9.0     7.0     2.0     9.0     6.0     5.0            4.0    9.0    5.0           4.0    1.0    3.0
      0.0320     9.0     6.0     0.0     9.0     1.0     1.0            0.0    6.0    3.0           1.0    1.0    1.0
      0.0160     9.0     1.0     0.0     9.0     1.0     0.0            0.0    1.0    1.0           0.0    0.0    0.0339      0.2500     9.0     9.0     9.0     9.0     9.0     9.0            9.0    9.0    9.0           8.5    8.0    8.0
      0.1250     9.0     9.0     9.0     9.0     9.0     9.0            9.0    9.0    9.0           8.5    7.0    7.5
      0.0620     9.0     9.0     8.0     9.0     9.0     8.0            6.5    9.0    7.0           7.0    6.0    6.5
      0.0320     9.0     8.0     3.0     9.0     2.0     9.0            3.0    6.5    4.5           3.0    1.0    2.0
      0.0160     9.0     5.0     0.5     9.0     2.0     3.0            1.5    3.0    2.0           1.0    0.0    1.0
                                  表II(续)
                                                                                         G              O       T
                 A       A       C       C       G       I       I       E       S       L       G      R       R      Z
                 B       M       A       H       A       P       P       C       E       X       L      Y       Z      E
                 U       B       S       E       L       O       O       H       T       M       X      S       A      A化合物    施用率     T       E       O       A       A       H       S       C       V       A       M      A       W      M编号  (公斤/公顷)   H       L       B       L       P       E       S       G       I       W       A      T       R      X340      0.2500    9.0     9.0     9.0     9.0     9.0     9.0             9.0     9.0     9.0            9.0     8.0    9.0
      0.1250    9.0     9.0     9.0     9.0     9.0     9.0             9.0     9.0     8.0            7.5     7.0    8.0
      0.0620    9.0     9.0     7.0     9.0     9.0     7.5             8.0     9.0     8.0            6.0     5.0    6.0
      0.0320    9.0     9.0     4.5     9.0     9.0     6.5             4.0     9.0     4.5            4.5     2.0    3.5
      0.0160    9.0     7.0     1.0     9.0     1.0     5.0             2.0     7.0     3.5            2.0     1.0    1.5341      0.5000    9.0     9.0     9.0     9.0             9.0             9.0     9.0     9.0            7.0            6.0
      0.2500    9.0     9.0     9.0     9.0     9.0     9.0             9.0     9.0     8.8            5.2     3.5    5.8
      0.1250    9.0     9.0     8.9     9.0     8.2     8.8             8.1     9.0     8.0            4.1     2.2    3.4
      0.0620    9.0     8.6     6.0     9.0     6.0     9.0             6.1     7.9     5.4            2.5     0.8    2.4
      0.0320    8.3     6.6     4.4     9.0     3.2     6.8             3.2     6.1     3.0            1.9     0.5    1.4
      0.0160    6.4     4.2     0.8     8.5     1.5     4.1             0.5     2.6     1.1            0.6     0.2    0.3342      0.2500    9.0     5.0     1.0     9.0     0.0     2.0             2.0     4.0     1.0            1.0     2.0    1.0
      0.1250    9.0     2.0     0.0     9.0     1.0     0.0             0.0     0.0     0.0            0.0     0.0    0.0
      0.0620    9.0     1.0     0.0     9.0     0.0                     0.0     0.0     0.0            0.0     0.0    0.0
      0.0320    2.0     0.0     0.0     9.0     0.0     0.0             0.0     0.0     0.0            0.0     1.0    0.0
      0.0160    1.0     0.0     0.0     5.0     0.0     0.0             0.0     0.0     1.0            0.0     0.0    1.0
                                                         表II(续)
                                                                                         G              O      T
                  A       A       C       C       G       I      I       E       S       L       G      R      R      Z
                  B       M       A       H       A       P      P       C       E       X       L      Y      Z      E
                  U       B       S       E       L       O      O       H       T       M       X      S      A      A化合物    施用率      T       E       O       A       A       H      S       C       V       A       M      A      W      M编号  (公斤/公顷)    H       L       B       L       P       E      S       G       I       W       A      T      R      X343     0.5000      9.0     9.0     5.0     9.0             9.0            9.0     9.0     9.0            5.0           5.0
     0.2500      9.0     9.0     5.5     9.0     1.0     7.5            7.0     9.0     3.5            5.0    2.0    4.5
     0.1250      9.0     9.0     3.5     9.0     1.0     5.0            6.5     9.0     2.5            4.0    2.0    3.0
     0.0620      9.0     8.0     1.0     9.0     0.0     3.0            1.5     5.5     1.0            1.0    1.0    1.5
     0.0320      9.0     6.0     0.0     8.0     0.0                    0.5     0.5     1.0            0.5    1.0    0.5
     0.0160      6.5     3.5     0.5     9.0     0.0     0.5            0.5     0.5     0.5            0.0    0.0    0.5344     0.5000      9.0     9.0     9.0     9.0             9.0            9.0     9.0     9.0            7.0           7.0
     0.2500      9.0     9.0     9.0     9.0     9.0     9.0            9.0     9.0     9.0            6.5    7.0    6.0
     0.1250      9.0     9.0     7.5     9.0     8.0     8.0            6.5     9.0     5.0            6.0    3.0    5.5
     0.0620      9.0     8.0     5.5     9.0     0.0     9.0            5.5     9.0     3.0            3.5    2.0    3.5
     0.0320      9.0     7.0     1.5     9.0     0.0     5.5            2.0     7.5     1.5            3.5    2.0    2.0
     0.0160      9.0     4.5     0.5     9.0     0.0     1.0            1.0     4.5     1.0            2.0    1.0    1.5345     0.2500      9.0     9.0     4.0     9.0     9.0     9.0            9.0     9.0     9.0            0.0    6.0    9.0
     0.1250      9.0     9.0     0.0     9.0     9.0     9.0            8.0     9.0     2.0            0.0    1.0    6.0
     0.0620      9.0     9.0             9.0     9.0     0.0            7.0     9.0     1.0            0.0    0.0    1.0
     0.0320      9.0     0.0     0.0     9.0     9.0     0.0.           2.0     9.0     0.0            0.0    0.0    0.0
                                                   表II(续)
                                                                                           G             O      T
                   A       A       C       C       G       I       I       E        S      L      G      R      R      Z
                   B       M       A       H       A       P       P       C        E      X      L      Y      Z      E
                   U       B       S       E       L       O       O       H        T      M      X      S      A      A化合物     施用率      T       E       O       A       A       H       S       C        V      A      M      A      W      M编号   (公斤/公顷)    H       L       B       L       P       E       S       G        I      W      A      T      R      X346      0.2500      0.0     7.0                     0.0             4.0     5.0      6.0    0.0           0.0    2.0    0.0
      0.0620      0.0     0.0                     0.0             0.0     0.0      0.0    0.0           0.0    0.0    0.0347      0.5000      9.0     9.0     9.0     9.0             9.0             9.0      9.0    9.0           9.0           7.0
      0.2500      9.0     9.0     3.0     9.0     9.0     9.0             9.0      9.0    8.0           6.0    2.0    4.0
      0.1250      9.0     9.0     3.0     9.0     9.0     9.0             9.0      9.0    4.5           4.5    0.0    3.0
      0.0620      9.0     6.0     3.0     9.0     0.0     6.5             5.0      4.5    2.5           3.0    0.0    1.0
      0.0320      9.0     4.5     1.5     4.5     0.0     4.5             3.5      4.0    2.5           1.0    0.0    0.5
      0.0160      4.5     2.0     0.0     9.0     0.0     3.5             0.0      1.0    1.0           1.0    0.0    0.5348      0.5000      9.0     9.0     9.0     9.0             9.0             9.0      9.0    5.0           7.0           9.0
      0.2500      9.0     9.0     3.0     9.0     9.0     9.0             9.0      9.0    1.5           5.5    4.0    4.0
      0.1250      9.0     9.0     6.0     9.0     0.0     5.5             9.0      9.0    1.5           2.5    1.0    3.0
      0.0620      9.0     6.5     2.5     9.0     0.0     3.0             3.0      3.5    1.5           2.0    0.0    1.0
      0.0320      4.5     3.5     2.0     9.0     0.0     2.0             2.0      1.5    1.0           0.5    0.0    0.5
      0.0160      4.5     1.5     0.0     9.0     0.0     0.0             0.0      0.0    0.0           0.0    0.0    0.0
                                                 表II(续)
                                                                                     G             O      T
                    A        A      C      C      G      I      I      E      S      L      G      R      R      Z
                    B        M      A      H      A      P      P      C      E      X      L      Y      Z      E
                    U        B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率       T        E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)     H        L      B      L      P      E      S      G      I      W      A      T      R      X349      0.2500       9.0      9.0    4.0    9.0    9.0    9.0           9.0    9.0    7.0           8.0    4.0    7.0
      0.1250       9.0      9.0    4.0    9.0    9.0    7.0           9.0    9.0    7.0           7.0    4.0    3.0
      0.0620       9.0      3.0    0.0    9.0    9.0    5.0           7.0    9.0    1.0           6.0    1.0    0.0
      0.0320       9.0      0.0    0.0    9.0    0.0    3.0           0.0    0.0    1.0           0.0    0.0    0.0
      0.0160       0.0      0.0    0.0    9.0    0.0    0.0           0.0    0.0    0.0           0.0    0.0    0.0350      0.2500       9.0      9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    8.5
      0.1250       9.0      9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           8.5    9.0    8.0
      0.0620       9.0      9.0    9.0    9.0    9.0    9.0           9.0    9.0    8.5           8.5    9.0    7.5
      0.0320       9.0      9.0    7.0    9.0    9.0    9.0           9.0    9.0    8.5           7.5    9.0    7.5
      0.0160       9.0      9.0    3.5    9.0    9.0    8.0           8.0    9.0    7.5           7.0    7.0    7.0351      0.2500       9.0      9.0    6.5    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    8.5
      0.1250       9.0      9.0    7.5    9.0    9.0    9.0           9.0    9.0    8.0           8.5    9.0    8.0
      0.0620       9.0      9.0    7.5    9.0    9.0    9.0           8.5    9.0    9.0           7.5    9.0    7.5
      0.0320       9.0      9.0    4.5    9.0    8.0    8.5           7.5    9.0    6.5           8.0    7.0    7.0
      0.0160       9.0      5.0    0.0    9.0    8.0    5.0           4.0    9.0    3.0           4.0    2.0    6.0
                                                   表II(续)
                                                                                         G               O        T
                    A       A       C       C       G      I        I      E      S      L       G       R        R      Z
                    B       M       A       H       A      P        P      C      E      X       L       Y        Z      E
                    U       B       S       E       L      O        O      H      T      M       X       S        A      A化合物      施用率      T       E       O       A       A      H        S      C      V      A       M       A        W      M编号    (公斤/公顷)    H       L       B       L       P      E        S      G      I      W       A       T        R      X352       0.2500      9.0     9.0     2.5     9.0     0.0   9.0             4.5    3.5    8.0             3.0      0.0    3.5
       0.1250      9.0     9.0     3.5     9.0     0.0   9.0             0.5    2.5    7.0             2.5      0.0    1.0
       0.0620      9.0     9.0     1.5     9.0     0.0   9.0             0.0    0.0    3.5             2.0      0.0    1.0
       0.0320      9.0     4.0     1.5     9.0     0.0   9.0             0.0    0.0    1.5             1.0      0.0    1.0
       0.0160      4.0     0.0     0.0     7.5     0.0   7.0             0.0    0.0    1.0             0.0      0.0    0.0353       0.5000      9.0     9.0     5.0     9.0           9.0             3.0    6.0    3.0             4.0      3.0    3.0
       0.2500      9.0     9.0     5.0     9.0           9.0             1.0    1.0    2.0             1.0      1.0    3.0
       0.1250      9.0     9.0     1.0     9.0           6.0             1.0    1.0    1.0             1.0      1.0    1.0
       0.0620      7.0     0.0     0.0     9.0           3.0             0.0    0.0    0.0             0.0      0.0    0.0
       0.0320              1.0     0.0     9.0           1.0             0.0    0.0    0.0             0.0      0.0    0.0
       0.0160      0.0     1.0     0.0     9.0           0.0             0.0    0.0    0.0             0.0      0.0    0.0354       0.5000      9.0     9.0     6.0     9.0           9.0             9.0    9.0    7.0             8.0      7.0    9.0
       0.2500      9.0     9.0     5.0     9.0           7.5             9.0    9.0    8.0             6.5      7.0    7.0
       0.1250      9.0     9.0     4.5     9.0           7.0             9.0    9.0    7.0             6.0      3.0    6.0
       0.0620      9.0     9.0     4.5     9.0           5.5             7.0    9.0    5.0             5.5      1.0    5.5
       0.0320      9.0     7.0     4.0     8.5           3.0             3.0    8.0    3.5             2.0      1.0    3.5
       0.0160      5.5     3.0     1.0     9.0           2.0             0.0    3.5    3.0             1.0      0.0    2.0
                                               表II(续)
                                                                                       G             O      T
                   A       A       C       C      G      I       I      E       S      L      G      R      R      Z
                   B       M       A       H      A      P       P      C       E      X      L      Y      Z      E
                   U       B       S       E      L      O       O      H       T      M      X      S      A      A化合物      施用率     T       E       O       A      A      H       S      C       V      A      M      A      W      M编号    (公斤/公顷)   H       L       B       L      P      E       S      G       I      W      A      T      R      X355       0.5000     9.0     9.0     6.0     9.0           9.0            9.0     9.0    3.0           6.0    1.0    6.0
       0.2500     9.0     9.0     1.0     9.0           5.0            8.0     9.0    3.0           5.0    1.0    3.0
       0.1250     9.0     4.0     1.0     9.0           2.0            1.0     3.0    2.0           1.0    1.0    1.0
       0.0620     9.0     4.0     0.0     9.0           0.0            0.0     0.0    1.0           1.0    1.0    1.0
       0.0320     0.0     0.0     0.0     9.0           0.0            0.0     0.0    1.0           0.0    0.0    1.0
       0.0160     0.0     0.0     0.0     1.0           0.0            0.0     0.0    0.0           0.0    1.0    1.0356       0.5000     9.0     9.0     8.0     9.0           9.0            2.5     6.5    8.0           3.0    3.0    4.5
       0.2500     9.0     9.0     3.0     9.0           9.0            0.0     2.0    6.5           1.5    1.0    3.0
       0.1250     9.0     9.0     3.0     9.0           7.0            0.0     0.5    3.0           1.0    1.0    2.0
       0.0620     9.0     9.0     2.0     8.0           5.5            0.0     0.0    1.5           0.0    0.0    1.0
       0.0320     7.5     2.5     2.0     9.0           3.5            0.0     0.0    1.0           0.0    0.0    0.0
       0.0160     6.5     2.0     1.0     9.0           1.0            0.0     0.0    0.0           0.0    0.0    0.0357       0.5000     9.0     9.0     4.0     9.0           9.0            1.0     2.0    3.0           1.0    1.0    2.0
       0.2500     9.0     9.0     1.0     9.0           4.0            0.0     0.0    2.0           1.0    2.0    2.0
       0.1250     1.0     3.0     0.0     9.0           0.0            0.0     0.0    1.0           1.0    1.0    2.0
       0.0620     2.0     2.0     0.0     9.0           0.0            0.0     0.0    0.0           0.0    0.0    0.0
       0.0320     1.0     0.0     0.0     9.0           0.0            0.0     0.0    0.0           0.0    0.0    0.0
       0.0160     0.0     0.0     0.0     7.0           1.0            0.0     0.0    1.0           0.0           1.0
                                                         表II(续)
                                                                                    G             O       T
                  A       A       C       C       G       I      I      E     S     L      G      R       R       Z
                  B       M       A       H       A       P      P      C     E     X      L      Y       Z       E
                  U       B       S       E       L       O      O      H     T     M      X      S       A       A化合物     施用率     T       E       O       A       A       H      S      C     V     A      M      A       W       M编号   (公斤/公顷)   H       L       B       L       P       E      S      G     I     W      A      T       R       X358      0.5000     9.0     9.0     3.0     9.0     8.0     9.0           0.0   3.0   3.0           1.0     1.0     2.0
      0.2500     9.0     5.0     0.0     9.0     7.0     9.0           0.0   0.0   2.0           0.0     0.0     0.0
      0.1250     3.0     3.0     0.0     8.0     0.0     1.0           0.0   0.0   0.0           0.0     0.0     0.0
      0.0620     1.0     1.0     0.0     3.0     0.0     0.0           0.0   0.0   0.0           0.0     0.0     0.0
      0.0320     0.0     0.0     0.0     0.0     0.0     0.0           0.0   0.0   0.0           0.0     0.0     0.0
      0.0160     0.0     0.0     0.0     0.0     0.0     0.0           0.0   0.0   0.0           0.0     0.0     0.0359      0.5000     9.0     9.0     9.0     9.0     9.0     9.0           9.0   9.0   5.3           6.7     5.5     6.7
      0.2500     9.0     9.0     7.5     9.0     8.5     9.0           9.0   9.0   3.5           7.3     3.7     6.3
      0.1250     9.0     9.0     4.3     9.0     8.0     8.5           7.8   8.5   2.5           6.0     1.7     4.5
      0.0620     9.0     9.0     2.0     9.0     6.0     9.0           5.5   6.8   1.8           4.0     1.0     3.0
      0.0320     9.0     8.3     0.7     9.0     1.0     7.0           2.8   4.8   1.3           2.3     1.0     1.5
      0.0160     7.5     6.3     1.5     9.0     0.5     1.8           1.0   2.0   0.5           1.5     0.7     1.0360      0.5000     9.0     9.0     3.0     9.0     9.0     7.0           7.5   9.0   4.0           7.5     6.0     6.5
      0.2500     9.0     9.0     3.0     9.0     9.0     3.5           5.0   8.0   3.0           4.0     3.0     4.0
      0.1250     8.0     7.0     2.5     9.0     9.0     3.5           3.0   7.5   2.0           2.0     1.0     3.0
      0.0620     6.5     4.5     0.0     9.0     9.0     1.5           1.0   4.5   0.0           0.5     1.0     1.5
      0.0320     1.5     0.0     0.0     4.5     7.0     1.0           0.0   1.0   0.5           0.0     0.0     1.5
      0.0160     0.0     0.5     0.0     0.0     9.0     0.0           0.0   0.0   0.5           0.0     0.0     0.5
                                                 表II(续)
                                                                                        G             O      T
                    A       A       C       C       G       I      I      E      S      L      G      R      R      Z
                    B       M       A       H       A       P      P      C      E      X      L      Y      Z      E
                    U       B       S       E       L       O      O      H      T      M      X      S      A      A化合物    施用率        T       E       O       A       A       H      S      C      V      A      M      A      W      M编号  (公斤/公顷)      H       L       B       L       P       E      S      G      I      W      A      T      R      X361      0.5000       9.0     0.0     2.0     9.0     9.0     0.0           2.0    4.0    0.0           1.0    1.0    2.0
      0.2500       0.0     1.0     0.0     6.0     9.0     0.0           0.0    0.0    0.0           0.0    0.0    0.0
      0.1250       0.0     4.0     0.0             4.0     0.0           0.0    0.0    0.0           0.0    1.0    1.0
      0.0620       0.0     0.0     0.0             5.0     0.0           0.0    1.0    0.0           0.0    0.0    0.0
      0.0320       0.0     1.0     0.0     0.0     0.0     0.0           0.0    0.0    1.0           0.0    0.0    0.0
      0.0160       0.0     0.0     0.0     0.0     0.0     0.0           0.0    1.0    0.0           0.0           0.0362      0.5000       9.0     9.0     9.0     9.0     9.0     9.0           9.0    9.0    4.5           7.0    8.0    6.5
      0.2500       9.0     9.0     3.5     9.0     0.0     9.0           9.0    9.0    4.0           5.0    7.0    5.0
      0.1250       9.0     9.0     2.0     9.0     0.0     9.0           5.5    9.0    3.5           3.0    3.0    1.5
      0.0620       9.0     9.0     0.0     9.0     0.0     9.0           2.5    8.5    1.0           1.5    0.0    1.0
      0.0320       9.0     7.0     0.0     6.5     0.0     9.0           0.0    4.0    1.0           0.5    0.0    1.0
      0.0160       9.0     2.5     0.0     7.0     0.0     9.0           0.0    2.0    0.0           0.0    0.0    0.0363      0.5000       9.0     9.0     8.0     9.0     9.0     9.0           9.0    9.0    6.5           9.0    9.0    8.0
      0.2500       9.0     9.0     6.7     9.0     9.0     9.0           7.3    9.0    2.7           7.7    8.0    6.7
      0.1250       9.0     7.7     5.3     9.0     9.0     9.0           2.3    8.7    0.7           4.7    5.0    5.7
      0.0620       9.0     5.7     3.7     9.0     0.0     7.3           0.7    3.7    0.0           3.0    0.0    2.3
      0.0320       8.0     2.7     0.7     5.7     0.0     2.3           0.0    1.3    0.0           1.3    0.0    0.7
      0.0160       4.5     0.0     0.0     5.0     0.0     2.0           0.0    1.0    0.0           0.0    0.0    0.0
                                                       表II(续)
                                                                                       G             O      T
                   A       A       C       C       G       I      I      E      S      L      G      R      R      Z
                   B       M       A       H       A       P      P      C      E      X      L      Y      Z      E
                   U       B       S       E       L       O      O      H      T      M      X      S      A      A化合物    施用率       T       E       O       A       A       H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H       L       B       L       P       E      S      G      I      W      A      T      R      X364      0.5000      9.0     9.0     9.0     9.0     9.0     9.0           9.0    9.0    7.5           9.0    9.0    8.0
      0.2500      9.0     9.0     7.0     9.0     9.0     9.0           9.0    9.0    5.3           8.7    9.0    7.0
      0.1250      9.0     9.0     8.0     9.0     9.0     9.0           8.3    9.0    4.0           8.0    8.0    7.0
      0.0620      9.0     9.0     5.3     9.0     9.0     9.0           3.3    9.0    1.3           7.0    6.0    4.7
      0.0320      9.0     5.7     3.3     9.0     0.0     8.3           0.7    5.0    0.0           2.3    0.0    1.7
      0.0160      8.3     4.3     2.0     7.7     0.0     5.7           0.0    1.0    0.0           1.3    0.0    1.0365      0.5000      9.0     9.0     4.0     9.0     9.0     9.0           9.0    9.0    6.0           9.0    9.0    9.0
      0.2500      9.0     9.0     1.0     9.0     9.0     9.0           9.0    9.0    5.0           8.0    8.0    8.0
      0.1250      9.0     9.0     1.0     9.0     0.0     9.0           2.0    9.0    4.0           5.0    4.0    8.0
      0.0620      9.0     7.0     0.0     9.0     0.0     3.0           0.0    8.0    0.0           0.0    0.0    7.0
      0.0320      4.0     2.0     0.0     9.0     0.0     1.0           0.0    3.0    0.0           0.0    0.0    2.0
      0.0160      4.0     0.0     0.0     4.0     0.0     1.0           0.0    0.0    0.0           0.0    0.0    0.0366      0.2500      9.0     9.0     9.0     9.0     9.0     9.0           9.0    9.0    9.0           9.0    9.0    9.0
      0.1250      9.0     9.0     9.0     9.0     9.0     9.0           9.0    9.0    9.0           8.7    9.0    8.7
      0.0620      9.0     9.0     9.0     9.0     9.0     9.0           9.0    9.0    9.0           8.0    8.5.   8.3
      0.0320      9.0     9.0     8.3     9.0     8.0     9.0           9.0    9.0    8.3           7.3    7.0    8.0
      0.0160      9.0     8.7     6.3     9.0     0.0     9.0           8.0    9.0    6.7           6.3    7.0    7.7
                                       表II(续)
                                                                                    G      O      T
                  A      A      C       C       G       I      I      E      S      L      G      R      R      Z
                  B      M      A       H       A       P      P      C      E      X      L      Y      Z      E
                  U      B      S       E       L       O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O       A       A       H      S      C      V      A      M      A      W      M编号  (公斤/公顷)    H      L      B       L       P       E      S      G      I      W      A      T      R      X367    0.5000       9.0    9.0    5.0     9.0             9.0           8.0    9.0    9.0           7.0           4.0
    0.2500       9.0    8.5    2.5     9.0     9.0     6.0           3.0    9.0    7.5           6.0    7.0    2.5
    0.1250       8.0    6.0    3.0     9.0     4.0     3.0           0.0    4.0    3.0           4.5    4.0    2.0
    0.0620       6.0    1.5    2.0     9.0     3.0     1.5           0.0    1.0    1.5           2.0    1.0    1.0
    0.0320       0.0    0.0    2.0     2.5             1.5           0.0    0.5    1.5           1.5    0.0    1.0
    0.0160       0.0    0.0    1.5     1.0     0.0     1.5           0.0    0.0    1.0           0.0    0.0    0.5368    0.5000       9.0    9.0    9.0     9.0             9.0           9.0    9.0    6.0           8.0           7.0
    0.2500       9.0    9.0    9.0     9.0     9.0     9.0           8.0    9.0    5.0           7.5    7.0    6.5
    0.1250       9.0    9.0    4.5     9.0     9.0     9.0           5.0    8.0    3.0           7.0    6.0    6.0
    0.0620       9.0    8.0    1.0     9.0     9.0     7.5           1.5    7.0    1.5           5.5    4.0    4.0
    0.0320       9.0    4.0    3.0     9.0     2.0     9.0           0.0    5.5    0.5           3.0    1.0    2.5
    0.0160       9.0    2.0    2.0     7.5     1.0     5.5           0.0    2.0    0.5           1.5    0.0    0.0369    0.5000       9.0    9.0    9.0     9.0             9.0           9.0    9.0    9.0           9.0           7.0
    0.2500       9.0    9.0    8.3     9.0     9.0     9.0           9.0    9.0    5.3           8.0    7.0    7.7
    0.1250       9.0    9.0    8.0     9.0     9.0     9.0           7.0    8.3    3.3           6.7    6.0    6.7
    0.0620       8.3    8.0    6.0     9.0     6.0     9.0           2.3    7.7    2.3           4.3    1.5    4.7
    0.0320       8.3    7.0    2.3     9.0     3.5     6.0           0.0    2.3    1.7           2.0    0.0    1.7
    0.0160       6.3    4.7    2.5     8.3     2.0     4.0           0.0    0.7    0.7           0.7    0.0    0.7
                                                 表II(续)
                                                                                       G             O      T
                  A       A      C       C       G      I       I       E      S       L      G      R      R      Z
                  B       M      A       H       A      P       P       C      E       X      L      Y      Z      E
                  U       B      S       E       L      O       O       H      T       M      X      S      A      A化合物    施用率      T       E      O       A       A      H       S       C      V       A      M      A      W      M编号   (公斤/公顷)   H       L      B       L       P      E       S       G      I       W      A      T      R      X370      0.5000     9.0     9.0    7.0     9.0            9.0             9.0     9.0    9.0           8.0           4.0
      0.2500     9.0     8.7    0.0     9.0     9.0    9.0             9.0     9.0    5.7           7.3    6.0    2.7
      0.1250     9.0     8.0    0.0     9.0     9.0    9.0             3.7     5.7    1.3           6.3    1.0    2.0
      0.0620     8.7     4.0    0.0     9.0     9.0    9.0             2.0     4.7    2.7           3.3    1.0    1.3
      0.0320     4.0     1.7    0.0     9.0     9.0    6.0             0.0     1.7    1.3           1.0    0.0    0.0
      0.0160     3.0     0.0    0.3     1.7     6.0    4.0             0.0     1.0    0.7           0.7    0.0    0.0371      0.2500     9.0     9.0    6.0     9.0     9.0    9.0             6.5     9.0    4.5           8.0    7.0    7.0
      0.1250     9.0     8.5    4.0     9.0     9.0    7.5             3.5     8.0    1.5           5.0    3.0    4.5
      0.0620     9.0     6.5    0.0     9.0     9.0    5.5
实施例187
在水稻田条件下稻子对移植后施用的耐受力和对发芽前杂草的控制
按下列方法测定移植的稻对移植后施用除草剂的耐受性：取二株十天大的稻秧苗(堤伯内品种(Tebonnet))移植至在直径10.5公分且没有排水孔的32盎斯塑胶容器内的砂质壤土中。移植后，容器内灌水，水位保持在土表面上1.5至3公分。移植3天后，用含试验化合物的选定的水/丙酮50/50v/v混合物处理容器里灌水的土表面，使之相当于约0.0313至0.500公斤/公顷活性成份。经处理的容器置于温室平台上，浇水，使水位保持上述程度，并根据一般温室方法照料。处理3至4周后，结束试验，检查各容器，根据实施例185的分级系统为除草效果分级，所得数据示于表III。所评估的化合物按实施例185所示的化合物编号说明。
按下列方法测定水稻田条件下的芽前除草活性：取植物种子或繁殖器官种植在含于直径10.5公分且没有排水孔的32盎斯塑胶容器内砂质壤土土表0.5公分中。向这些容器中加水，实验期间均保持在土表以上1.5至3公分。试验化合物含于水/丙酮50/50v/v混合物中直接滴注至灌溉水中，使之相当于约0.0313至0.500公斤/公顷活性成份。经处理的容器置于温室平台上，并根据常规温室方法照料。处理3至4周后，结束试验，检查各容器，根据实施例185的分级系统为除草效果分级。所得数据示于表III。所评估的化合物按实施例185的化合物编号说明。
本实施例采用的植物品种系以字头缩写、俗名及学名表示。
在稻子耐受性/芽前杂草控制评估中采用的植物品种字头缩写      俗名                   学名ECHORC        水包禾(加州种)         Echinochloa oryzoides(Ard.)Fritsch.CYPIR         碎米莎草               Cyperus iriaCYPSE         水莎草                 Cyperus serotinus，Rottb.MOOVA         鸭舌草                 Monochoria vaginalis，Presl.SAGPY         矮慈姑                 Sagittaria pygmaea，L.ORYSAT        稻，堤伯内种           Oryza sativa，(L.)Tebonnet
                                               表III
                                      水稻田条件-移植后的稻子
                                             发芽前的杂草
                  E                                                      O
                  C          C          C          M          S          R
                  H          Y          Y          O          A          Y
                  O          P          P          O          G          S化合物   施用率       R          I          S          V          P          A编号  (公斤/公顷)    C          R          E          A          Y          T1     0.5000       9.0        9.0        8.0        9.0        8.5        7.0
    0.2500       9.0        9.0        9.0        9.0        8.3        7.7
    0.1250       9.0        9.0        6.0        9.0        6.7        5.3
    0.0625       9.0        9.0        3.0        9.0        5.0        4.7
    0.0313       9.0        9.0        1.3        9.0        3.3        4.72     0.5000       9.0        9.0        0.0        9.0        9.0        9.0
    0.2500       9.0        9.0        0.0        9.0        4.0        5.0
    0.1250       9.0        9.0        0.0        9.0        2.0        3.0
    0.0625       9.0        9.0        0.0        9.0        0.0        3.0
    0.0313       9.0        8.0        0.0        7.0        0.0        2.03     0.5000       9.0        9.0        4.0        9.0        9.0        4.0
    0.2500       9.0        9.0        2.0        9.0        8.0        4.0
    0.1250       9.0        9.0        0.0        9.0        6.0        3.0
    0.0625       9.0        9.0        0.0        9.0        2.0        2.0
    0.0313       9.0        9.0        0.0        9.0        0.0        2.04     0.5000       9.0        9.0        9.0        9.0        9.0        8.0
    0.2500       9.0        9.0        9.0        9.0        9.0        8.0
    0.1250       9.0        9.0        9.0        9.0        6.0        7.0
    0.0625       9.0        9.0        2.0        9.0        2.0        7.0
    0.0313       9.0        9.0                   9.0        2.0        4.05     0.5000       9.0        9.0        7.0        9.0        7.0        7.0
    0.2500       9.0        9.0        8.0        9.0        7.0        5.0
    0.1250       9.0        9.0        6.0        9.0        2.0        4.0
    0.0625       9.0        9.0        2.0        9.0        0.0        3.0
    0.0313       9.0        9.0        0.0        9.0        0.0        2.0
                                     表III(续)
                    E                                            O
                    C        C        C        M        S        R
                    H        Y        Y        O        A        Y
                    O        P        P        O        G        S化合物     施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T6        0.5000      9.0      9.0      9.0      9.0      9.0      8.0
       0.2500      9.0      9.0      9.0      9.0      7.0      8.0
       0.1250      8.0      9.0      7.0      9.0      7.0      8.0
       0.0625      6.0      9.0      4.0      9.0      4.0      8.07        0.5000      9.0      9.0      9.0      9.0      9.0      9.0
       0.2500      9.0      9.0      7.0      9.0      9.0      7.0
       0.1250      9.0      9.0      8.0      9.0      9.0      7.0
       0.0625      9.0      9.0      7.0      9.0      8.0      8.0
       0.0313      9.0      9.0      7.0      9.0      6.0      6.08        0.5000      9.0      9.0      9.0      9.0      9.0      9.0
       0.2500      9.0      9.0      9.0      9.0      9.0      9.0
       0.1250      9.0      9.0      9.0      9.0      9.0      9.0
       0.0625      9.0      9.0      9.0      9.0      9.0      7.0
       0.0313      9.0      9.0      4.0      9.0      6.0      7.09        0.5000      9.0      9.0      9.0      9.0      9.0      9.0
       0.2500      9.0      9.0      9.0      9.0      8.0      8.0
       0.1250      9.0      9.0      9.0      9.0      8.0      7.0
       0.0625      9.0      9.0      4.0      9.0      2.0      7.0
       0.0313      9.0      9.0      2.0      9.0      0.0      6.010        0.5000      9.0      9.0      7.0      9.0      9.0      7.0
       0.2500      9.0      9.0      7.0      9.0      9.0      7.0
       0.1250      9.0      9.0      7.0      9.0      9.0      6.0
       0.0625      9.0      9.0      7.0      9.0      8.0      6.0
       0.0313      9.0      9.0      4.0      9.0      2.0      4.0
                                   表III(续)
                     E                                                      O
                     C          C          C          M          S          R
                     H          Y          Y          O          A          Y
                     O          P          P          O          G          S化合物    施用率         R          I          S          V          P          A编号  (公斤/公顷)       C          R          E          A          Y          T11      0.5000        9.0        9.0        7.0        9.0        9.0        3.0
      0.2500        8.0        9.0        2.0        9.0        2.0        3.0
      0.1250        8.0        9.0        2.0        9.0        0.0        2.0
      0.0625        7.0        9.0        2.0        9.0        0.0        2.012      0.5000        9.0        9.0        7.0        9.0        9.0        9.0
      0.2500        9.0        9.0        7.0        9.0        9.0        8.0
      0.1250        9.0        9.0        8.0        9.0        4.0        7.0
      0.0625        9.0        9.0        7.0        9.0        2.0        7.0
      0.0313        9.0        9.0        6.0        9.0        0.0        4.013      0.5000        9.0        9.0        7.0        9.0        9.0        9.0
      0.2500        9.0        9.0        7.0        9.0        8.0        7.0
      0.1250        9.0        9.0        7.0        9.0        6.0        7.0
      0.0625        9.0        9.0        2.0        9.0        2.0        6.0
      0.0313        9.0        9.0        0.0        9.0        0.0        4.014      0.2500        7.5        8.0        2.0        9.0        0.0        3.5
      0.1250        6.5        6.0        1.0        9.0        0.0        2.5
      0.0625        5.0        4.0        0.0        9.0        0.0        2.0
      0.0313        4.0        2.0        0.0        9.0        0.0        2.016      0.2500        5.0        6.0        0.0        9.0        0.0        4.0
      0.1250        3.5        4.0        0.0        9.0        0.0        2.5
      0.0625        1.0        2.0        0.0        4.0        0.0        1.5
      0.0313        1.0        0.0        0.0        2.0        0.0        1.017      0.2500        8.0        9.0        8.0        9.0        8.0        4.0
      0.1250        7.5        8.0        2.0        9.0        2.0        2.5
      0.0625        5.5        8.0        0.0        9.0        0.0        3.0
      0.0313        4.0        4.0        0.0        8.0        0.0        2.0
                                表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T18     0.2500      9.0      9.0      8.0      9.0      0.0      9.0
     0.1250      9.0      9.0      9.0      9.0      0.0      4.0
     0.0625      9.0      9.0      9.0      9.0      0.0      3.0
     0.0313      9.0      9.0      6.0      9.0      0.0      3.019     0.2500      6.5      8.0      2.0      9.0      0.0      2.5
     0.1250      5.0      8.0      0.0      9.0      0.0      2.0
     0.0625      3.5      4.0      0.0      9.0      0.0      1.5
     0.0313      2.0      2.0      0.0      8.0      0.0      1.020     0.2500      0.0      2.0      0.0      4.0      0.0      1.0
     0.1250      0.0      1.0      0.0      2.0      0.0      0.5
     0.0625      0.0      0.0      0.0      0.0      0.0      0.5
     0.0313      0.0      0.0      0.0      0.0      0.0      0.521     0.2500      4.7      1.0      0.0      9.0      0.0      4.3
     0.1250      2.7      0.5      0.0      7.5      0.0      2.3
     0.0625      0.7      0.0      0.0      6.0      0.0      2.0
     0.0313      0.0      0.0      0.0      4.0      0.0      1.722     0.2500      9.0      9.0      9.0      9.0      9.0      2.5
     0.1250      9.0      9.0      7.0      9.0      4.0      2.5
     0.0625      9.0      9.0      7.0      9.0      2.0      2.0
     0.0313      9.0      9.0      2.0      9.0      0.0      2.023     0.2500      9.0      9.0      9.0      9.0      9.0      8.5
     0.1250      8.5      9.0      8.0      9.0      9.0      8.0
     0.0625      7.0      9.0      7.0      9.0      6.0      6.5
     0.0313      4.5      7.0      4.0      9.0      4.0      5.524     0.2500      7.0      8.0      4.0      9.0      0.0      4.0
     0.1250      2.0      6.0      1.0      9.0      0.0      3.0
     0.0625      0.0      2.0      0.0      8.0      0.0      2.0
     0.0313      0.0      0.0      0.0      4.0      0.0      2.0
                              表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物    施用率     R        I        S        V        P        A编号  (公斤/公顷)   C        R        E        A        Y        T25     0.2500     9.0      9.0      8.0      9.0      4.0      7.0
     0.1250     9.0      9.0      7.0      9.0      1.0      7.0
     0.0625     9.0      9.0      2.0      9.0      0.0      6.0
     0.0313     7.0      9.0      0.0      9.0      0.0      4.026     0.2500     9.0      9.0      9.0      9.0      9.0      9.0
     0.1250     9.0      9.0      2.0      9.0      2.0      6.0
     0.0625     9.0      8.0      4.0      9.0      0.0      4.0
     0.0313     7.0      6.0      0.0      9.0      0.0      3.027     0.2500     9.0      9.0      2.0      9.0      4.0      6.0
     0.1250     9.0      6.0      0.0      9.0      2.0      5.0
     0.0625     7.0      4.0      0.0      9.0      0.0      3.0
     0.0313     6.0      2.0      0.0      8.0      0.0      2.028     0.2500     9.0      9.0      4.0      9.0      8.0      9.0
     0.1250     9.0      6.0      0.0      9.0      4.0      7.0
     0.0625     9.0      4.0      0.0      9.0      2.0      4.0
     0.0313     8.0      2.0      0.0      8.0      0.0      3.029     0.2500     9.0      9.0      4.0      9.0      0.0      4.0
     0.1250     9.0      9.0      4.0      9.0      0.0      4.0
     0.0625     9.0      7.0               9.0      0.0      3.0
     0.0313     7.0      4.0      0.0      8.0      0.0      2.030     0.2500     9.0      8.0      2.0      9.0      7.0      3.5
     0.1250     9.0      8.0      4.0      9.0      2.0      3.0
     0.0625     8.5      6.0      0.0      9.0      0.0      3.0
     0.0313     6.5      2.0      0.0      9.0      0.0      2.031     0.2500     9.0      9.0      9.0      9.0      9.0      8.0
     0.1250     9.0      9.0      8.0      9.0      9.0      7.5
     0.0625     8.5      9.0      7.0      9.0      7.0      8.0
     0.0313     7.0      9.0      7.0      9.0      4.0      7.5
                             表III(续)
                    E                                   O
                    C      C       C      M      S      R
                    H      Y       Y      O      A      Y
                    O      P       P      O      G      S化合物     施用率       R      I       S      V      P      A编号   (公斤/公顷)     C      R       E      A      Y      T32       0.2500      7.5    9.0     7.0    9.0    9.0    4.5
       0.1250      4.5    8.0     2.0    9.0    2.0    4.0
       0.0625      3.5    6.0     0.0    9.0    0.0    2.5
       0.0313      2.0    4.0     0.0    8.0    0.0    1.533       0.2500      9.0    4.0     0.0    9.0    0.0    3.5
       0.1250      9.0    2.0     0.0    9.0    0.0    3.0
       0.0625      8.5    0.0     0.0    9.0    0.0    3.0
       0.0313      7.5    0.0     0.0    9.0    0.0    2.034       0.2500      4.5    0.0     0.0    0.0    0.0    0.0
       0.1250      3.5    0.0     0.0    0.0    0.0    0.0
       0.0625      2.5    0.0     0.0    0.0    0.0    0.0
       0.0313      2.0    0.0     0.0    0.0    0.0    0.035       0.2500      9.0    9.0     7.0    9.0    9.0    5.0
       0.1250      7.5    9.0     7.0    9.0    2.0    4.0
       0.0625      6.5    8.0     2.0    9.0    0.0    2.5
       0.0313      4.5    4.0     0.0    9.0    0.0    2.036       0.2500      0.0                                 1.0
       0.1250      0.0                                 1.0
       0.0625      0.0                                 1.0
       0.0313      0.0                                 1.037       0.2500      9.0                                 1.0
       0.1250      8.0                                 1.0
       0.0625      7.0                                 1.0
       0.0313      4.0                                 0.038       0.2500      2.0    0.0     0.0    0.0    0.0    0.0
       0.1250      1.0    0.0     0.0    0.0    0.0    0.0
       0.0625      0.0    0.0     0.0    0.0    0.0    0.0
       0.0313      0.0    0.0     0.0    0.0    0.0    0.0
                                            表III(续)
                     E                                                            O
                     C           C           C           M           S            R
                     H           Y           Y           O           A            Y
                     O           P           P           O           G            S化合物    施用率         R           I           S           V           P            A编号   (公斤/公顷)      C           R           E           A           Y            T39      0.2500        0.0         0.0         0.0         0.0         0.0          0.0
      0.1250        0.0         0.0         0.0         0.0         0.0          0.0
      0.0625        0.0         0.0         0.0         0.0         0.0          0.0
      0.0313        0.0         0.0         0.0         0.0         0.0          0.040      0.2500        9.0         9.0         9.0         9.0         6.0          4.0
      0.1250        9.0         9.0         9.0         9.0         2.0          3.0
      0.0625        9.0         4.0         4.0         9.0         0.0          3.0
      0.0313        9.0         2.0         2.0         9.0         0.0          2.041      0.2500        6.0         2.0         0.0         9.0         0.0          0.0
      0.1250        2.0         1.0         0.0         4.0         0.0          0.0
      0.0625        0.0         0.0         0.0         2.0         0.0          0.0
      0.0313        0.0         0.0         0.0         0.0         0.0          0.042      0.2500        0.0         0.0         0.0         0.0         0.0          0.0
      0.1250        0.0         0.0         0.0         0.0         0.0          0.0
      0.0625        0.0         0.0         0.0         0.0         0.0          0.0
      0.0313        0.0         0.0         0.0         0.0         0.0          0.043      0.2500        8.0         0.0         0.0         9.0         0.0          3.0
      0.1250        2.0         0.0         0.0         9.0         0.0          3.0
      0.0625        0.0         0.0         0.0         9.0         0.0          2.0
      0.0313        0.0         0.0         0.0         6.0         0.0          1.044      0.2500        0.0         0.0         0.0         0.0         0.0          0.0
      0.1250        0.0         0.0         0.0         0.0         0.0          0.0
      0.0625        0.0         0.0         0.0         0.0         0.0          0.0
      0.0313        0.0         0.0         0.0         0.0         0.0          0.045      0.2500        9.0         9.0         9.0         9.0         6.0          3.0
      0.1250        9.0         9.0         9.0         9.0         4.0          3.0
      0.0625        9.0         9.0         2.0         9.0         0.0          2.0
      0.0313        9.0         6.0                     9.0         0.0          2.0
                                 表III(续)
                 E                                       O
                 C       C       C       M       S       R
                 H       Y       Y       O       A       Y
                 O       P       P       O       G       S化合物    施用率     R       I       S       V       P       A编号  (公斤/公顷)   C       R       E       A       Y       T46      0.2500    9.0     9.0     2.0     9.0     7.0     3.0
      0.1250    9.0     9.0             9.0     2.0     2.0
      0.0625    9.0     6.0     0.0     9.0     0.0     1.0
      0.0313    9.0     2.0     0.0     9.0     0.0     1.047      0.2500    5.0     1.0     2.0     9.0     0.0     6.0
      0.1250    3.5     0.0     1.0     5.5     0.0     4.0
      0.0625    1.5     0.0     0.0     4.5     0.0     2.5
      0.0313    0.0     0.0     0.0     4.5     0.0     1.548      0.2500    6.0     0.0             9.0     0.0     6.0
      0.1250    2.0     0.0     0.0     9.0     0.0     4.0
      0.0625    0.0     0.0     0.0     9.0     0.0     2.0
      0.0313    0.0     0.0     0.0     6.0     0.0     2.049      0.2500    8.0     8.0     0.0     9.0     0.0     2.0
      0.1250    6.0     2.0     0.0     9.0     0.0     1.0
      0.0625    4.0     0.0     0.0     9.0     0.0     1.0
      0.0313    0.0     0.0     0.0     4.0     0.0     1.050      0.2500    9.0     6.0     0.0     9.0     0.0     3.0
      0.1250    9.0     2.0     0.0     9.0     0.0     2.0
      0.0625    9.0     2.0     0.0     9.0     0.0     2.0
      0.0313    9.0     0.0     0.0     9.0     0.0     2.051      0.2500    9.0     9.0     9.0     9.0     9.0     9.0
      0.1250    9.0     9.0     7.0     9.0     4.0     9.0
      0.0625    7.0     8.0     2.0     9.0     2.0     9.0
      0.0313    4.0     7.0     0.0     9.0     2.0     7.052      0.2500    7.0     0.0             9.0     0.0     0.0
      0.1250    4.0                     9.0     0.0     0.0
      0.0625    2.0     0.0     0.0     9.0     0.0     0.0
      0.0313    0.0     0.0     0.0     8.0     0.0     0.0
                                表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T53      0.2500      9.0      9.0      0.0      9.0      0.0      7.0
      0.1250      6.0      9.0      0.0      9.0      0.0      5.0
      0.0625      2.0      6.0      0.0      9.0      0.0      4.0
      0.0313      0.0      2.0      0.0      8.0      0.0      2.054      0.2500      9.0      9.0      2.0      9.0      0.0      6.0
      0.1250      7.0      7.0      1.0      9.0      0.0      3.0
      0.0625      6.0      4.0      0.0      9.0      0.0      2.0
      0.0313      2.0      2.0      0.0      8.0      0.0      2.055      0.2500      9.0      9.0      0.0      9.0      0.0      6.0
      0.1250      9.0      6.0      0.0      9.0      0.0      3.0
      0.0625      7.0      2.0      0.0      9.0      0.0      1.0
      0.0313      5.0      0.0      0.0      7.0      0.0      2.056      0.2500      9.0      9.0      2.0      9.0      0.0      6.0
      0.1250      9.0      9.0      2.0      9.0      0.0      3.0
      0.0625      9.0      9.0      0.0      9.0      0.0      2.0
      0.0313      9.0      6.0      0.0      9.0      0.0      1.057      0.2500      9.0      9.0      0.0      9.0      0.0      6.0
      0.1250      9.0      9.0      0.0      9.0      0.0      5.0
      0.0625      9.0      9.0      0.0      9.0      0.0      4.0
      0.0313      9.0      9.0      0.0      9.0      0.0      3.058      0.2500      9.0      9.0      0.0      9.0      0.0      5.0
      0.1250      9.0      9.0      0.0      9.0      0.0      3.0
      0.0625      9.0      9.0      0.0      9.0      0.0      2.0
      0.0313      9.0      9.0      0.0      9.0      0.0      2.059      0.2500      9.0      9.0      0.0      9.0      0.0      4.0
      0.1250      9.0      8.0      0.0      9.0      0.0      4.0
      0.0625      9.0      7.0      0.0      9.0      0.0      3.0
      0.0313      9.0      7.0      0.0      9.0      0.0      2.0
                                     表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)    C        R        E        A        Y        T60      0.2500      9.0      0.0      0.0      9.0      0.0      0.0
      0.1250      8.0      0.0      0.0      9.0      0.0      0.0
      0.0625      4.0      0.0      0.0      9.0      0.0      0.0
      0.0313      2.0      0.0      0.0      9.0      0.0      0.061      0.2500      8.0      2.0      0.0      9.0      0.0      0.0
      0.1250      8.0      2.0      0.0      9.0      0.0      0.0
      0.0625      7.0      0.0      0.0      8.0      0.0      0.0
      0.0313      4.0      0.0      0.0      8.0      0.0      0.062      0.2500      9.0      9.0      9.0      9.0      7.0      9.0
      0.1250      9.0      9.0      2.0      9.0      4.0      9.0
      0.0625      9.0      6.0      1.0      9.0      1.0      9.0
      0.0313      6.0      4.0      0.0      9.0      0.0      4.063      0.2500      9.0      9.0      0.0      9.0      0.0      3.0
      0.1250      9.0      9.0      0.0      9.0      0.0      2.0
      0.0625      9.0      8.0      0.0      9.0      0.0      2.0
      0.0313      9.0      7.0      0.0      9.0      0.0      1.064      0.2500      9.0      7.0      0.0      9.0      0.0      7.0
      0.1250      8.0      7.0      0.0      9.0      0.0      4.0
      0.0625      8.0      4.0      0.0      9.0      0.0      3.0
      0.0313      6.0      2.0      0.0      9.0      0.0      3.065      0.2500      0.0      0.0      0.0      0.0      0.0      0.0
      0.1250      0.0      0.0      0.0      0.0      0.0      0.0
      0.0625      0.0      0.0      0.0      0.0      0.0      0.0
      0.0313      0.0      0.0      0.0      0.0      0.0      0.066      0.2500      9.0      9.0      9.0      9.0      2.0      2.0
      0.1250      9.0      9.0      9.0      9.0      0.0      2.0
      0.0625      9.0      9.0      2.0      9.0      0.0      1.0
      0.0313      9.0      8.0      0.0      9.0      0.0      1.0
                                  表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T67      0.2500      9.0      0.0      6.0      9.0      0.0      1.0
      0.1250      9.0      0.0      1.0      9.0      0.0      1.0
      0.0625      8.0      0.0      0.0      9.0      0.0      0.5
      0.0313      5.5      0.0      0.0      8.0      0.0      0.568      0.2500      9.0      9.0      7.0      9.0      2.0      1.0
      0.1250      9.0      9.0               9.0      2.0      1.5
      0.0625      9.0      9.0      7.0      9.0      0.0      1.0
      0.0313      7.5      7.0      6.0      9.0      0.0      0.569      0.2500      9.0      7.0      9.0      9.0      9.0      8.0
      0.1250      9.0      4.0      2.0      9.0      2.0      6.5
      0.0625      9.0      2.0      0.0      9.0      0.0      5.0
      0.0313      9.0      0.0      0.0      9.0      0.0      3.570      0.2500      9.0      9.0      0.0      9.0      2.0      6.5
      0.1250      9.0      9.0      0.0      9.0      1.0      6.0
      0.0625      8.0      7.0      0.0      9.0      0.0      4.5
      0.0313      4.0      2.0      0.0      9.0      0.0      3.071      0.2500      9.0      2.0      9.0      9.0      4.0      7.0
      0.1250      8.5      0.0      2.0      9.0      0.0      5.5
      0.0625      7.5      0.0      0.0      9.0      0.0      3.5
      0.0313      5.5      0.0      0.0      8.0      0.0      2.072      0.2500      9.0      7.0      9.0      9.0      4.0      7.0
      0.1250      8.5      4.0      2.0      9.0      0.0      6.0
      0.0625      8.0      0.0      2.0      9.0      0.0      5.0
      0.0313      7.5      0.0      0.0      9.0      0.0      4.073      0.2500      9.0      8.0      9.0      9.0      2.0      6.0
      0.1250      9.0      8.0      2.0      9.0      0.0      4.0
      0.0625      6.5      6.0      0.0      9.0      0.0      3.0
      0.0313      8.0      2.0      0.0      9.0      0.0      2.5
                                    表III(续)
                  E                                          O
                  C      C        C        M        S        R
                  H      Y        Y        O        A        Y
                  O      P        P        O        G        S化合物    施用率      R      I        S        V        P        A编号  (公斤/公顷)    C      R        E        A        Y        T74      0.2500     9.0    8.0      6.0      9.0      0.0      7.0
      0.1250     9.0    7.0      2.0      9.0      0.0      5.0
      0.0625     7.5    2.0      0.0      9.0      0.0      4.0
      0.0313     6.5    0.0      0.0      8.0      0.0      2.575      0.2500     9.0    7.0      0.0      9.0      4.0      8.0
      0.1250     8.5    4.0      0.0      9.0      0.0      5.0
      0.0625     9.0    2.0      0.0      9.0      0.0      3.0
      0.0313     6.5    0.0      0.0      9.0      0.0      2.076      0.2500     9.0    9.0      2.0      9.0      9.0      5.5
      0.1250     9.0    9.0      1.0      9.0      2.0      3.5
      0.0625     8.5    6.0      0.0      9.0      0.0      2.5
      0.0313     8.0    4.0      0.0      8.0      0.0      2.577      0.2500     9.0                                        7.0
      0.1250     9.0                                        7.0
      0.0625     9.0                                        4.0
      0.0313     9.0                                        3.078      0.2500     9.0                                        4.0
      0.1250     9.0                                        4.0
      0.0625     9.0                                        4.0
      0.0313     9.0                                        3.079      0.2500     9.0                                        4.0
      0.1250     9.0                                        4.0
      0.0625     9.0                                        4.0
      0.0313     9.0                                        3.080      0.2500     9.0                                        4.0
      0.1250     9.0                                        3.0
      0.0625     9.0                                        3.0
      0.0313     9.0                                        4.0
                                   表III(续)
                   E                                  O
                   C      C      C      M      S      R
                   H      Y      Y      O      A      Y
                   O      P      P      O      G      S化合物     施用率      R      I      S      V      P      A编号   (公斤/公顷)    C      R      E      A      Y      T81      0.2500      9.0                                4.0
      0.1250      9.0                                4.0
      0.0625      9.0                                4.0
      0.0313      9.0                                4.082      0.2500      9.0                                3.0
      0.1250      9.0                                3.0
      0.0625      9.0                                2.0
      0.0313      9.0                                1.083      0.2500      9.0                                5.0
      0.1250      9.0                                6.0
      0.0625      9.0                                5.0
      0.0313      9.0                                3.084      0.2500      9.0                                7.0
      0.1250      9.0                                4.0
      0.0625      9.0                                3.0
      0.0313      9.0                                3.085      0.2500      9.0                                1.0
      0.1250      9.0                                0.0
      0.0625      9.0                                0.0
      0.0313      8.0                                0.086      0.2500      9.0                                3.0
      0.1250      9.0                                2.0
      0.0625      9.0                                3.0
      0.0313      9.0                                2.087      0.2500      9.0                                4.0
      0.1250      9.0                                4.0
      0.0625      9.0                                3.0
      0.0313      9.0                                3.0
                                表III(续)
                   E                                       O
                   C       C       C       M       S       R
                   H       Y       Y       O       A       Y
                   O       P       P       O       G       S化合物    施用率       R       I       S       V       P       A编号   (公斤/公顷)    C       R       E       A       Y       T88      0.2500      9.0                                     7.0
      0.1250      9.0                                     6.0
      0.0625      9.0                                     4.0
      0.0313      9.0                                     3.089      0.2500      9.0                                     5.0
      0.1250      9.0                                     4.0
      0.0625      9.0                                     3.0
      0.0313      9.0                                     4.090      0.2500      9.0                                     7.0
      0.1250      9.0                                     6.0
      0.0625      9.0                                     6.0
      0.0313      9.0                                     4.091      0.2500      9.0                                     1.0
      0.1250      9.0                                     0.0
      0.0625      9.0                                     0.0
      0.313       9.0                                     0.092      0.2500      9.0                                     6.0
      0.1250      9.0                                     6.0
      0.0625      6.0                                     5.0
      0.0313      4.0                                     3.093      0.2500      9.0     7.0     9.0     9.0             7.0
      0.1250      8.0     4.0     9.0     9.0     7.0     6.0
      0.0625      8.0     2.0     2.0     9.0     0.0     4.0
      0.0313      7.0     0.0             9.0     0.0     4.094      0.2500      7.0     7.0     0.0     9.0     0.0     0.0
      0.1250      4.0     4.0     0.0     9.0     0.0     1.0
      0.0625      2.0     2.0     0.0     9.0     0.0     0.0
      0.0313      0.0     0.0     0.0     6.0     0.0     0.0
                                 表III(续)
                E                                            O
                C        C        C        M        S        R
                H        Y        Y        O        A        Y
                O        P        P        O        G        S化合物  施用率      R        I        S        V        P        A编号 (公斤/公顷)   C        R        E        A        Y        T95   0.2500      0.0      8.0      0.0      9.0      0.0      4.0
   0.1250      0.0      2.0      0.0      6.0      0.0      2.0
   0.0625      0.0      0.0      0.0      2.0      0.0      2.0
   0.0313      0.0      0.0      0.0      0.0      0.0      0.096   0.2500      7.0      0.0      2.0      9.0      0.0      2.0
   0.1250      4.0      0.0      0.0      9.0      0.0      3.0
   0.0625      4.0      0.0      0.0      9.0      0.0      2.0
   0.0313      2.0      0.0      0.0      8.0      0.0      2.097   0.2500      8.5      0.0      0.0      9.0      0.0      5.5
   0.1250      7.5      0.0      0.0      4.0      0.0      4.0
   0.0625      5.5      0.0      0.0      2.0      0.0      2.5
   0.0313      5.5      0.0      0.0      0.0      0.0      1.598   0.2500      6.5      6.0      0.0      9.0      0.0      7.0
   0.1250      6.5      6.0      0.0      9.0      0.0      7.0
   0.0625      5.0      4.0      0.0      4.0      0.0      6.0
   0.0313      3.0      0.0      0.0      2.0      0.0      4.099   0.2500      4.5      2.0      0.0      9.0      0.0      3.5
   0.1250      4.5      0.0      0.0      8.0      0.0      2.5
   0.0625      3.0      0.0      0.0               0.0      1.5
   0.0313      1.0      0.0      0.0      2.0      0.0      0.5100   0.2500      0.0      0.0      0.0      9.0      0.0      3.0
   0.1250      0.0      0.0      0.0      8.0      0.0      3.0
   0.0625      0.0      0.0      0.0      8.0      0.0      2.0
   0.0313      0.0      0.0      0.0      6.0      0.0      2.0101   0.2500      0.0      0.0      0.0      9.0      0.0      1.0
   0.1250      0.0      0.0      0.0      4.0      0.0      0.0
   0.0625      0.0      0.0      0.0      0.0      0.0      0.0
   0.0313      0.0      0.0      0.0      0.0      0.0      0.0
                               表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T102      0.2500      0.0      0.0      0.0      4.0      0.0      2.0
      0.1250      0.0      0.0      0.0      2.0      0.0      1.0
      0.0625      0.0      0.0      0.0      0.0      0.0      0.0
      0.0313      0.0      0.0      0.0      0.0      0.0      0.0103      0.2500      6.0      0.0      0.0      9.0      0.0      4.0
      0.1250      4.0      0.0      0.0      9.0      0.0      4.0
      0.0625      2.0      0.0      0.0      9.0      0.0      3.0
      0.0313      0.0      0.0      0.0      8.0      0.0      2.0104      0.2500      0.0      0.0      0.0      9.0      0.0      4.0
      0.1250      0.0      0.0      0.0      8.0      0.0      3.0
      0.0625      0.0      0.0      0.0      7.0      0.0      2.0
      0.0313      0.0      0.0      0.0      7.0      0.0      2.0105      0.2500      9.0      9.0      9.0      9.0      9.0      8.0
      0.1250      9.0      9.0      9.0      9.0      9.0      8.0
      0.0625      9.0      8.0      7.0      9.0      4.0      6.0
      0.0313      9.0      8.0      7.0      9.0      2.0      6.0106      0.2500      0.0      4.0      0.0      8.0      0.0      0.0
      0.1250      0.0      2.0      0.0      8.0      0.0      0.0
      0.0625      0.0      0.0      0.0      4.0      0.0      0.0
      0.0313      0.0      0.0      0.0      2.0      0.0      0.0107      0.2500      4.0      6.0      0.0      9.0      0.0      6.0
      0.1250      1.0      2.0      0.0      9.0      0.0      5.0
      0.0625      0.0      0.0      0.0      9.0      0.0      3.0
      0.0313      0.0      0.0      0.0      9.0      0.0      2.0108      0.2500      0.0      0.0      0.0      8.0      0.0      0.0
      0.1250      0.0      0.0      0.0      4.0      0.0      0.0
      0.0625      0.0      0.0      0.0      0.0      0.0      0.0
      0.0313      0.0      0.0      0.0      0.0      0.0      0.0
                                表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物   施用率        R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T109     0.2500       7.0      8.0      0.0      9.0      0.0      4.0
     0.1250       4.0      4.0      0.0      9.0      0.0      4.0
     0.0625       2.0      0.0      0.0      9.0      0.0      2.0
     0.0313       0.0      0.0      0.0      9.0      0.0      2.0110     0.2500       7.0      7.0      0.0      9.0      0.0      6.0
     0.1250       4.0      2.0      0.0      9.0      0.0      5.0
     0.0625       1.0      0.0      0.0      9.0      0.0      4.0
     0.0313       0.0      0.0      0.0      9.0      0.0      3.0112     0.2500       0.0      0.0      0.0      0.0      0.0      0.0
     0.1250       0.0      0.0      0.0      0.0      0.0      0.0
     0.0625       0.0      0.0      0.0      0.0      0.0      0.0
     0.0313       0.0      0.0      0.0      0.0      0.0      0.0114     0.2500       6.0      9.0      6.0      8.0      6.0      7.0
     0.1250       4.0      9.0      2.0      9.0      6.0      7.0
     0.0625       0.0      9.0      0.0      9.0      2.0      6.0
     0.0313       0.0      9.0      0.0      9.0      0.0      4.0116     0.2500       0.0      0.0      0.0      8.0      0.0      0.0
     0.1250       0.0      0.0      0.0      8.0      0.0      0.0
     0.0625       0.0      0.0      0.0      2.0      0.0      0.0
     0.0313       0.0      0.0      0.0      0.0      0.0      0.0117     0.2500       0.0      0.0      0.0      4.0      0.0      0.0
     0.1250       0.0      0.0      0.0      2.0      0.0      0.0
     0.0625       0.0      0.0      0.0      0.0      0.0      0.0
     0.0313       0.0      0.0      0.0      0.0      0.0      0.0118     0.2500       0.0      0.0      0.0      0.0      0.0      0.0
     0.1250       0.0      0.0      0.0      0.0      0.0      0.0
     0.0625       0.0      0.0      0.0      0.0      0.0      0.0
     0.0313       0.0      0.0      0.0      0.0      0.0      0.0
                            表III(续)
                    E                                            O
                    C        C        C        M        S        R
                    H        Y        Y        O        A        Y
                    O        P        P        O        G        S化合物    施用率        R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T119       0.2500      9.0      9.0      9.0      9.0      9.0      9.0
       0.1250      9.0      9.0      8.0      9.0      8.0      9.0
       0.0625      9.0      9.0      4.0      9.0      8.0      8.0
       0.0313      4.0      9.0      2.0      9.0      6.0      7.0121       0.2500      9.0      4.0      4.0      9.0      0.0      9.0
       0.1250      8.0      2.0      2.0      9.0      0.0      6.0
       0.0625      7.0      0.0      0.0      9.0      0.0      4.0
       0.0313      6.0      0.0      0.0      9.0      0.0      3.0122       0.2500      9.0      0.0      0.0      9.0      0.0      4.0
       0.1250      8.0      0.0      0.0      9.0      0.0      4.0
       0.0625      7.0      0.0      0.0      8.0      0.0      3.0
       0.0313      4.0      0.0      0.0      6.0      0.0      2.0128       0.2500      0.0      0.0      0.0      9.0      0.0      0.0
       0.1250      0.0      0.0      0.0      7.0      0.0      0.0
       0.0625      0.0      0.0      0.0      4.0      0.0      0.0
       0.0313      0.0      0.0      0.0      2.0      0.0      0.0129       0.2500      2.0      7.0      0.0      9.0      0.0      3.0
       0.1250      1.0      7.0      0.0      9.0      0.0      3.0
       0.0625      0.0      4.0      0.0      9.0      0.0      2.0
       0.0313      0.0      0.0      0.0      8.0      0.0      1.0130       0.2500      2.0      6.0      0.0      9.0      0.0      7.0
       0.1250      0.0      2.0      0.0      9.0      0.0      7.0
       0.0625      0.0      0.0      0.0      9.0      0.0      4.0
       0.0313      0.0      0.0      0.0      9.0      0.0      3.0131       0.2500      4.0      8.0      0.0      9.0      0.0      7.0
       0.1250      0.0      2.0      0.0      9.0      0.0      6.0
       0.0625      0.0      0.0      0.0      9.0      0.0      3.0
       0.0313      0.0      0.0      0.0      8.0      0.0      2.0
                                  表III(续)
                      E                                  O
                      C      C      C      M      S      R
                      H      Y      Y      O      A      Y
                      O      P      P      O      G      S化合物   施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T132     0.2500          9.0    9.0    2.0           4.0    9.0
     0.1250          9.0    9.0    2.0    0.0    2.0    6.0
     0.0625          6.0    9.0    0.0    0.0    0.0    3.0
     0.0313          4.0    9.0    0.0    0.0    0.0    3.0133     0.2500          9.0    9.0    0.0    2.0    0.0    5.0
     0.1250          6.0    9.0    0.0    1.0    0.0    4.0
     0.0625          2.0    9.0    0.0    0.0    0.0    3.0
     0.0313          1.0    9.0    0.0    0.0    0.0    2.0134     0.2500          8.0    9.0    9.0    7.0    4.0    9.0
     0.1250          9.0    9.0    4.0    4.0    2.0    7.0
     0.0625          9.0    9.0    4.0    4.0    2.0    4.0
     0.0313          6.0    9.0    2.0    2.0    2.0    3.0135     0.2500          6.0    9.0    0.0    0.0    0.0    4.0
     0.1250          2.0    9.0    0.0    0.0    0.0    3.0
     0.0625          0.0    8.0    0.0    0.0    0.0    3.0
     0.0313          0.0    6.0    0.0    0.0    0.0    2.0136     0.2500          0.0    0.0    0.0    0.0    0.0    0.0
     0.1250          0.0    0.0    0.0    0.0    0.0    0.0
     0.0625          0.0    0.0    0.0    0.0    0.0    0.0
     0.0313          0.0    0.0    0.0    0.0    0.0    0.0137     0.2500          7.0    9.0    6.0    4.0    4.0    8.0
     0.1250          2.0    9.0    0.0    2.0    0.0    8.0
     0.0625          0.0    9.0    0.0    0.0    0.0    7.0
     0.0313          0.0    9.0    0.0    0.0    0.0    4.0138     0.1250          0.0    8.0    0.0    0.0    0.0    3.0
     0.0625          0.0    6.0    0.0    0.0    0.0    3.0
     0.0313          0.0    2.0    0.0    0.0    0.0    2.0
                                   表III(续)
                       E                                  O
                       C      C      C      M      S      R
                       H      Y      Y      O      A      Y
                       O      P      P      O      G      S化合物  施用率             R      I      S      V      P      A编号  (公斤/公顷)          C      R      E      A      Y      T139    0.1250             9.0    9.0    4.0    8.0    0.0    4.0
   0.0625             6.0    9.0    0.0    6.0    0.0    4.0
   0.0313             4.0    9.0    0.0    2.0    0.0    3.0140    0.1250             6.0    9.0    0.0    2.0    0.0    8.0
   0.0625             4.0    9.0    0.0    2.0    0.0    7.0
   0.0313             2.0    9.0    0.0    2.0    0.0    6.0141    0.1250             2.0    9.0    0.0    0.0    0.0    3.0
   0.0625             1.0    4.0    0.0    0.0    0.0    3.0
   0.0313             0.0    2.0    0.0    0.0    0.0    2.0142    0.2500             9.0    8.0    9.0    9.0    0.0    9.0
   0.1250             9.0    6.0    2.0    9.0    0.0    7.0
   0.0625             9.0    6.0    0.0    9.0    0.0    6.0
   0.0313             9.0    4.0    0.0    9.0    0.0    3.0143    0.2500             6.0    0.0    0.0    9.0    0.0    4.0
   0.1250             2.0    0.0    0.0    9.0    0.0    3.0
   0.0625             0.0    0.0    0.0    9.0    0.0    3.0
   0.0313             0.0    0.0    0.0    9.0    0.0    3.0144    0.2500             9.0    8.0    0.0    9.0    0.0    2.0
   0.1250             9.0    4.0    0.0    9.0    0.0    2.0
   0.0625             6.0    2.0    0.0    4.0    0.0    2.0
   0.0313             2.0    0.0    0.0    2.0    0.0    1.0170    0.2500             9.0    6.0    0.0    9.0    0.0    8.0
   0.1250             9.0    4.0    0.0    9.0    0.0    6.0
   0.0625             9.0    0.0    0.0    2.0    0.0    5.0
   0.0313             9.0    0.0    0.0    0.0    0.0    3.0
                               表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T171    0.2500           9.0    2.0    0.0    9.0    0.0    2.0
   0.1250           9.0    2.0    0.0    9.0    0.0    1.0
   0.0625           9.0    0.0    0.0    9.0    0.0    0.0
   0.0313           8.5    0.0    0.0    9.0    0.0    0.0172    0.2500           9.0    4.0    2.0    9.0    0.0    8.0
   0.1250           9.0    4.0    1.0    9.0    0.0    6.0
   0.0625           9.0    2.0    0.0    9.0    0.0    3.5
   0.0313           6.5    2.0    0.0    9.0    0.0    2.5173    0.2500           9.0    2.0           9.0    0.0    3.5
   0.1250           6.5    1.0    0.0    9.0    0.0    3.0
   0.0625           4.5    0.0    0.0    9.0    0.0    2.5
   0.0313           2.0    0.0    0.0    8.0    0.0    2.0174    0.2500           8.5    2.0    0.0    9.0    0.0    4.0
   0.1250           6.5    2.0    0.0    9.0    0.0    2.5
   0.0625           5.5    2.0    0.0    9.0    0.0    2.5
   0.0313           4.5    1.0    0.0    9.0    0.0    1.5175    0.2500           8.0    2.0    0.0    9.0    0.0    6.0
   0.1250           8.0    1.0    0.0    9.0    0.0    5.0
   0.0625           7.5    6.0    0.0    9.0    0.0    3.5
   0.0313           6.5    0.0    0.0    8.0    0.0    2.5176    0.2500           8.0    8.0    0.0    9.0    0.0    6.5
   0.1250           8.0    4.0    0.0    9.0    0.0    5.0
   0.0625           5.5    2.0    0.0    9.0    0.0    3.5
   0.0313           4.5    2.0    0.0    9.0    0.0    2.5177    0.2500           9.0    4.0    8.0    9.0    0.0    6.5
   0.1250           9.0    4.0    7.0    9.0    0.0    4.5
   0.0625           6.5    2.0    0.0    9.0    0.0    3.5
   0.0313           3.0    0.0    0.0    9.0    0.0    2.5
                               表III(续)
                      E                                  O
                      C      C      C      M      S      R
                      H      Y      Y      O      A      Y
                      O      P      P      O      G      S化合物  施用率            R      I      S      V      P      A编号  (公斤/公顷)         C      R      E      A      Y      T178    0.2500            8.5    2.0    0.0    9.0    0.0    6.0
   0.1250            7.5    1.0    0.0    9.0    0.0    5.0
   0.0625            7.5    0.0    0.0    9.0    0.0    3.5
   0.0313            4.0    0.0    0.0    9.0    0.0    2.5179    0.2500            9.0    6.0    6.0    9.0    4.0    9.0
   0.1250            9.0    6.0    6.0    9.0    0.0    8.5
   0.0625            8.0    4.0    2.0    9.0    0.0    8.0
   0.0313            4.5    2.0    0.0    9.0    0.0    6.5180    0.2500            8.5    8.0    6.0    9.0    0.0    8.5
   0.1250            8.0    7.0    4.0    9.0    0.0    8.0
   0.0625            5.0    4.0    0.0    9.0    0.0    7.5
   0.0313            3.5    2.0    0.0    9.0    0.0    6.0181    0.2500            9.0    9.0    8.0    9.0    0.0    7.0
   0.1250            9.0    9.0    7.0    9.0    0.0    6.0
   0.0625            8.5    9.0    7.0    9.0    0.0    5.0
   0.0313            8.5    7.0    4.0    9.0    0.0    3.5182    0.0630            9.0    9.0    4.0    9.0    4.0    9.0
   0.0315            9.0    9.0    2.0    9.0    4.0    7.0183    0.0630            9.0    9.0    0.0    9.0    0.0    9.0
   0.0315            9.0    9.0    0.0    9.0    0.0    8.0184    0.0630            9.0    4.0    6.0    9.0    4.0    9.0
   0.0315            9.0    1.0    2.0    9.0    2.0    7.0185    0.0630            0.0    0.0    0.0    9.0    0.0    0.0
   0.0315            0.0    0.0    0.0    9.0    0.0    0.0186    0.0630            9.0    9.0    9.0    9.0    9.0    9.0
   0.0315            9.0    9.0    9.0    9.0    9.0    9.0
                                    表III(续)
                       E                                    O
                       C        C      C      M      S      R
                       H        Y      Y      O      A      Y
                       O        P      P      O      G      S化合物  施用率             R        I      S      V      P      A编号  (公斤/公顷)          C        R      E      A      Y      T187    0.2500             9.0      4.0    0.0    9.0    0.0    6.0
   0.1250             6.0      2.0    0.0    9.0    0.0    3.0
   0.0625             2.0      0.0    0.0    9.0    0.0    3.0
   0.0313             0.0      0.0    0.0    8.0    0.0    2.0188    0.2500             8.0      0.0           9.0    0.0    2.0
   0.1250             2.0      0.0           9.0    0.0    2.0
   0.0625             0.0      0.0           9.0    0.0    1.0
   0.0313             0.0      0.0    0.0    9.0    0.0    1.0189    0.2500             0.0      0.0    0.0    8.0    0.0    0.0
   0.1250             0.0      0.0    0.0    2.0    0.0    0.0
   0.0625             0.0      0.0    0.0    0.0    0.0    0.0
   0.0313             0.0      0.0    0.0    0.0    0.0    0.0190    0.2500             8.0      4.0    0.0    9.0    0.0    7.0
   0.1250             7.0      2.0    0.0    9.0    0.0    4.0
   0.0625             4.0      0.0    0.0    9.0    0.0    3.0
   0.0313             2.0      0.0    0.0    9.0    0.0    2.0191    0.2500             7.0      4.0           9.0    0.0    6.0
   0.1250             4.0      2.0    0.0    9.0    0.0    3.0
   0.0625             2.0      0.0    0.0    9.0    0.0    2.0
   0.0313             0.0      0.0    0.0    9.0    0.0    1.0192    0.2500             9.0      7.0           9.0    9.0    4.0
   0.1250             9.0      2.0    0.0    9.0    2.0    3.0
   0.0625             4.0      0.0    0.0    9.0    0.0    2.0
   0.0313             1.0      0.0    0.0    9.0    0.0    1.0193    0.2500             0.0      0.0    0.0    9.0    0.0    1.0
   0.1250             0.0      0.0    0.0    9.0    0.0    0.0
   0.0625             0.0      0.0    0.0    4.0    0.0    0.0
   0.0313             0.0      0.0    0.0    2.0    0.0    0.0
                              表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T194    0.2500           9.0    0.0    0.0    9.0    0.0    4.0
   0.1250           6.0    0.0    0.0    9.0    0.0    3.0
   0.0625           2.0    0.0    0.0    9.0    0.0    3.0
   0.0313           0.0    0.0    0.0    9.0    0.0    2.0195    0.2500           9.0    9.0    7.0    9.0    2.0    9.0
   0.1250           6.0    4.0    2.0    9.0    1.0    9.0
   0.0625           3.0    2.0    0.0    9.0    0.0    7.0
   0.0313           2.0    0.0    0.0    9.0    0.0    6.0196    0.2500           4.0    4.0    9.0    9.0    0.0    8.0
   0.1250           4.0    1.0    6.0    9.0    0.0    8.0
   0.0625           2.0    0.0    4.0    9.0    0.0    6.0
   0.0313           0.0    0.0    2.0    9.0    0.0    4.0198    0.2500           9.0    7.0    8.0    9.0    4.0    9.0
   0.1250           9.0    4.0    4.0    9.0    2.0    8.0
   0.0625           6.0    2.0    2.0    9.0    0.0    7.0
   0.0313           4.0    0.0    0.0    9.0    0.0    4.0199    0.2500           7.0    8.0    0.0    9.0    0.0    8.0
   0.1250           7.0    4.0    0.0    9.0    0.0    6.0
   0.0625           4.0    2.0    0.0    9.0    0.0    4.0
   0.0313           2.0    0.0    0.0    8.0    0.0    3.0200    0.2500           9.0    8.0    7.0    9.0    4.0    9.0
   0.1250           6.0    7.0    2.0    9.0    0.0    9.0
   0.0625           2.0    6.0    0.0    9.0    0.0    7.0
   0.0313           0.0    4.0    0.0    9.0    0.0    7.0202    0.2500           2.0    9.0    0.0    0.0    0.0    6.0
   0.1250           2.0    9.0    0.0    0.0    0.0    5.0
   0.0625           1.0    9.0    0.0    0.0    0.0    4.0
   0.0313           1.0    9.0    0.0    0.0    0.0    3.0
                                   表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T203    0.2500           4.0    9.0    6.0    8.0    4.0    7.0
   0.1250           2.0    9.0    2.0    2.0    2.0    6.0
   0.0625           0.0    9.0    0.0    0.0    0.0    6.0
   0.0313           0.0    9.0    0.0    0.0    0.0    4.0204    0.2500           9.0    9.0    7.0    7.0    0.0    7.0
   0.1250           4.0    9.0    2.0    4.0    0.0    7.0
   0.0625           2.0    9.0    0.0    2.0    0.0    4.0
   0.0313           0.0    9.0    0.0    0.0    0.0    3.0206    0.2500           9.0    9.0    7.0    4.0    4.0    9.0
   0.1250           2.0    9.0    7.0    1.0    1.0    7.0
   0.0625           2.0    9.0    2.0    0.0    0.0    6.0
   0.0313           0.0    9.0    0.0    0.0    0.0    5.0207    0.2500           5.5    8.5    6.0    7.5    1.0    7.5
   0.1250           2.0    8.5    1.0    5.5    0.0    7.0
   0.0625           1.5    6.5    0.0    4.5    0.0    6.0
   0.0313           1.0    5.5    0.0    4.0    0.0    5.0208    0.2500           0.0    9.0    0.0    4.0    0.0    5.0
   0.1250           0.0    9.0    0.0    2.0    0.0    3.0
   0.0625           0.0    9.0    0.0    2.0    0.0    3.0
   0.0313           0.0    9.0    0.0    0.0    0.0    2.0209    0.1250           2.0    8.0    0.0    0.0    0.0    4.0
   0.0625           2.0    4.0    0.0    0.0    0.0    3.0
   0.0313           1.0    2.0    0.0    0.0    0.0    3.0210    0.2500           9.0    7.0    0.0    9.0    0.0    7.0
   0.1250           9.0           0.0    9.0    0.0    6.0
   0.0625           9.0    7.0    0.0    9.0    0.0    4.0
   0.0313           9.0    2.0    0.0    9.0    0.0    3.0
                              表III(续)
                       E                                  O
                       C      C      C      M      S      R
                       H      Y      Y      O      A      Y
                       O      P      P      O      G      S化合物  施用率             R      I      S      V      P      A编号  (公斤/公顷)          C      R      E      A      Y      T211    0.2500             9.0    4.0    0.0    9.0    0.0    3.0
   0.1250             7.0    4.0    0.0    9.0    0.0    2.0
   0.0625             4.0    0.0    0.0    9.0    0.0    2.0
   0.0313             2.0    0.0    0.0    9.0    0.0    2.0212    0.2500             4.0    2.0    0.0    9.0    0.0    7.0
   0.1250             2.0    0.0    0.0    9.0    0.0    6.0
   0.0625             0.0    0.0    0.0    8.0    0.0    4.0
   0.0313             0.0    0.0    0.0    4.0    0.0    3.0213    0.2500             0.0           0.0    2.0    0.0    7.0
   0.1250             0.0    0.0    0.0    0.0    0.0    6.0
   0.0625             0.0    0.0    0.0    0.0    0.0    4.0
   0.0313             0.0    0.0    0.0    0.0    0.0    3.0214    0.2500             0.0    7.0    0.0    9.0    0.0    5.0
   0.1250             0.0    7.0    0.0    9.0    0.0    3.0
   0.0625             0.0    4.0    0.0    9.0    0.0    2.0
   0.0313             0.0    2.0    0.0    8.0    0.0    2.0217    0.2500             0.0    0.0    0.0    7.0    0.0    4.0
   0.1250             0.0    0.0    0.0    7.0    0.0    3.0
   0.0625             0.0    0.0    0.0    4.0    0.0    2.0
   0.0313             0.0    0.0    0.0    2.0    0.0    2.0218    0.2500             4.0    0.0    0.0    9.0    0.0    3.0
   0.1250             2.0    0.0    0.0    9.0    0.0    3.0
   0.0625             0.0    0.0    0.0    9.0    0.0    2.0
   0.0313             0.0    0.0    0.0    8.0    0.0    1.0223    0.2500             9.0    9.0    8.0    9.0    9.0    9.0
   0.1250             8.0    7.0    6.0    9.0    6.0    8.0
   0.0625             6.0    7.0    4.0    9.0    2.0    8.0
   0.0313             6.0    4.0    0.0    9.0    0.0    7.0
                          表III(续)
                    E                                  O
                    C      C      C      M      S      R
                    H      Y      Y      O      A      Y
                    O      P      P      O      G      S化合物  施用率          R      I      S      V      P      A编号(公斤/公顷)         C      R      E      A      Y      T224    0.2500          9.0    8.0    7.0    9.0    8.0    9.0
   0.1250          9.0    8.0    2.0    9.0    4.0    8.0
   0.0625          9.0    7.0    0.0    9.0    2.0    7.0
   0.0313          6.0    4.0    0.0    9.0    0.0    6.0225    0.2500          7.0    7.0    0.0    9.0    0.0    7.0
   0.1250          4.0    2.0    0.0    9.0    0.0    6.0
   0.0625          2.0    0.0    0.0    8.0    0.0    4.0
   0.0313          0.0    0.0    0.0    8.0    0.0    3.0245    0.2500          0.0    0.0    0.0    0.0    0.0    0.0
   0.1250          0.0    0.0    0.0    0.0    0.0    0.0
   0.0625          0.0    0.0    0.0    0.0    0.0    0.0
   0.0313          0.0    0.0    0.0    0.0    0.0    0.0246    0.2500          9.0    4.0           9.0    2.0    2.0
   0.1250          9.0    4.0    0.0    9.0    2.0    2.0
   0.0625          7.0    2.0    0.0    9.0    0.0    1.0
   0.0313          6.0    0.0    0.0    9.0    0.0    0.0256    0.2500          9.0    9.0    9.0    9.0    8.0    9.0
   0.1250          7.0    9.0    6.0    9.0    4.0    8.0
   0.0620          3.0    9.0    2.0    9.0    0.0    8.0
   0.0320          1.0    8.0    0.0    8.0    0.0    6.0257    0.2500          0.0    6.0           9.0    0.0    2.0
   0.1250          0.0    4.0           9.0    0.0    1.0
   0.0620          0.0    2.0    0.0    9.0    0.0    0.0
   0.0320          0.0    0.0    0.0    8.0    0.0    0.0258    0.2500          0.0    8.0           9.0    0.0    4.0
   0.1250          0.0    7.0    0.0    9.0    0.0    3.0
   0.0620          0.0    2.0    0.0    9.0    0.0    2.0
   0.0320          0.0    0.0    0.0    9.0    0.0    2.0
                              表III(续)
                    E                                  O
                    C      C      C      M      S      R
                    H      Y      Y      O      A      Y
                    O      P      P      O      G      S化合物  施用率          R      I      S      V      P      A编号  (公斤/公顷)       C      R      E      A      Y      T259    0.2500          2.0    4.0           9.0    0.0    3.0
   0.1250          0.0    4.0           9.0    0.0    2.0
   0.0620          0.0    2.0    0.0    9.0    0.0    1.0
   0.0320          0.0    0.0    0.0    6.0    0.0    1.0260    0.2500          0.0    0.0    0.0    0.0    0.0    0.0261    0.2500          0.0    2.0    0.0    3.0    0.0    0.0
   0.1250          2.0    5.5    4.5    6.0    0.0    0.0
   0.0620          2.0    4.5    4.5    4.5    0.0    0.0
   0.0320          2.5    4.0    4.5    4.5    0.0    0.0262    0.2500          3.0    9.0    0.0    9.0    0.0    3.0
   0.1250          0.0    6.0    0.0    9.0    0.0    0.0
   0.0620          0.0    0.0    0.0    0.0    0.0    0.0263    0.2500          2.0    9.0    9.0    9.0    0.0    4.0
   0.1250          0.0    9.0    9.0    6.0    0.0    0.0
   0.0620          0.0    7.0    9.0    0.0    0.0    0.0
   0.0320          0.0    4.0    9.0    0.0    0.0    0.0264    0.2500          2.0    5.0    9.0    9.0    0.0    5.0
   0.1250          0.0    5.0    9.0    9.0    0.0    0.0
   0.0620          0.0    5.0    4.0    9.0    0.0    0.0
   0.0320          0.0    5.0    4.0    9.0    0.0    0.0265    0.2500          0.0    3.0    0.0    9.0    0.0    0.0
   0.1250          0.0    0.0    0.0    9.0    0.0    0.0
   0.0620          0.0    0.0    0.0    9.0    0.0    0.0
   0.0320          0.0    0.0    0.0    9.0    0.0    0.0266    0.2500          0.0    9.0    3.0    9.0    0.0    0.0
   0.1250          0.0    5.0    0.0    9.0    0.0    0.0
   0.0620          0.0    5.0    0.0    9.0    0.0    0.0
   0.0320          0.0    5.0    0.0    9.0    0.0    0.0
                                表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T267    0.2500           9.0    9.0    9.0    9.0    5.0    6.0
   0.1250           9.0    9.0    5.5    9.0    3.0    4.5
   0.0620           9.0    8.0    0.0    9.0    1.0    3.0
   0.0320           9.0    8.0    0.0    7.5    0.0    2.0268    0.2500           4.5    7.5    9.0    9.0    4.0    7.5
   0.1250           4.5    6.0    9.0    9.0    1.0    5.0
   0.0620           3.0    3.0    5.5    9.0    1.0    4.0
   0.0320           1.0    1.0    1.0    7.5    0.0    3.5269    0.5000           4.0    0.0    0.0    9.0    0.0    0.0
   0.2500           0.0    0.0    0.0    0.0    0.0    0.0270    0.5000           9.0    9.0    3.0    9.0    5.0    2.0
   0.2500           9.0    9.0    9.0    9.0    0.0    8.0
   0.1250           4.3    9.0    7.0    9.0    0.0    7.0
   0.0620           2.7    9.0    0.0    9.0.   0.0    4.0
   0.0320           1.3    8.0    0.0    9.0    0.0    4.0271    0.5000           0.0    0.0    0.0    9.0    0.0    0.0
   0.2500           0.0    0.0    0.0    9.0    0.0    3.0
   0.1250           0.0    0.0    0.0    4.0    0.0    2.0
   0.0620           0.0    0.0    0.0    0.0    0.0    1.0272    0.5000           0.0    0.0    0.0    0.0    0.0    0.0273    0.5000           9.0    4.0    9.0    9.0    0.0    3.0
   0.2500           9.0    9.0    7.0    9.0    6.0    4.0
   0.1250           6.0    9.0           9.0    0.0    3.0
   0.0620           5.1    9.0    0.0    9.0    0.0    2.0
   0.0320           3.9    6.0    0.0    9.0    0.0    0.0
                                    表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T274    0.5000           9.0    2.0    9.0    9.0    4.0    7.0
   0.2500           9.0    9.0    9.0    9.0    9.0    8.0
   0.1250           5.9    9.0    8.0    9.0    4.0    4.0
   0.0620           4.1    8.0    2.0    9.0    0.0    4.0
   0.0320           3.3    7.0    0.0    9.0    0.0    2.0275    0.5000           7.0    0.0    0.0    9.0    0.0    5.0
   0.2500           9.0    7.0    9.0    9.0    9.0    4.0
   0.1250           4.1    6.0    9.0    9.0    3.0    3.0
   0.0620           3.9    4.0    9.0    9.0    0.0    0.0
   0.0320           3.7    0.0    9.0    6.0    0.0    0.0276    0.5000           9.0    9.0    7.0    9.0    9.0    9.0
   0.2500           9.0    9.0    7.0    9.0    9.0    7.0
   0.1250           7.9    9.0    8.0    9.0    9.0    6.0
   0.0620           7.7    9.0    2.0    9.0    9.0    5.0
   0.0320           4.0    8.0    2.0    9.0    8.0    4.0277    0.5000           9.0    9.0    9.0    9.0    9.0    9.0
   0.2500           9.0    9.0    9.0    9.0    9.0    8.0
   0.1250           9.0    9.0    9.0    9.0    9.0    7.0
   0.0620           8.6    9.0    9.0    9.0    8.0    7.0
   0.0320           7.0    9.0    2.0    9.0    6.0    5.0278    0.5000           9.0    9.0    9.0    9.0    9.0    8.0
   0.2500           8.0    9.0    4.0    9.0    2.0    7.0
   0.1250           7.4    7.0    2.0    9.0    0.0    4.0
   0.0620           6.1    2.0    0.0    8.0    0.0    3.0
   0.0320           0.0    0.0    0.0    6.0    0.0    2.0
                              表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T279    0.5000           7.0    9.0    5.0    9.0    9.0    6.0
   0.2500           6.0    6.0           9.0    4.0    4.0
   0.1250           6.1    2.0    0.0    8.0    0.0    4.0
   0.0620           5.7    0.0    0.0           0.0    3.0
   0.0320           0.0    0.0    0.0           0.0    2.0280    0.5000           9.0    9.0    3.0    9.0    9.0    9.0
   0.2500           9.0    9.0    2.0    9.0    9.0    8.0
   0.1250           7.6    8.0    0.0    9.0    2.0    7.0
   0.0620           5.7    6.0    0.0    9.0    0.0    3.0
   0.0320           0.0    2.0    0.0    9.0    0.0    3.0281    0.5000           7.0    9.0    9.0    9.0    9.0    4.0
   0.2500           9.0    9.0    9.0    9.0    8.0    6.0
   0.1250           7.1    9.0    9.0    9.0    2.0    4.0
   0.0620           5.9    8.0    9.0    9.0    0.0    2.0
   0.0320           0.0    4.0    9.0    9.0    0.0    0.0282    0.5000           0.0    9.0    0.0    9.0    0.0    0.0
   0.2500           0.0    8.0    0.0    9.0    0.0    4.0
   0.1250           1.9    8.0    0.0    9.0    0.0    4.0
   0.0620           0.0    8.0    0.0    9.0    0.0    3.0
   0.0320           0.0    4.0    0.0    6.0    0.0    2.0283    0.5000           6.0    9.0    0.0    9.0    9.0    4.0
   0.2500           6.0    9.0           9.0           5.0
   0.1250           3.4    8.0           9.0    0.0    4.0
   0.0620           3.4    4.0           8.0    0.0    2.0
   0.0320           0.0    0.0           2.0    0.0    2.0284    0.2500           0.0    9.0    9.0    9.0    0.0    0.0
   0.1250           0.0    9.0    2.0    9.0    0.0    0.0
   0.0620           0.0    9.0    0.0    9.0    0.0    0.0
   0.0320           0.0    4.0    0.0    4.0    0.0    0.0
                                   表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T285    0.2500           7.0    9.0    0.0    9.0    3.0    7.0
   0.1250           7.0    9.0    0.0    9.0    0.0    7.0
   0.0620           7.0    9.0    0.0    9.0    0.0    7.0
   0.0320           3.0    5.0    0.0    4.0    0.0    3.0286    0.2500           8.0    9.0    0.0    9.0    0.0    2.0
   0.1250           3.0    7.0    0.0    9.0    0.0    1.0
   0.0620           0.0    7.0    0.0    9.0    0.0    0.0
   0.0320           0.0    3.0    0.0    9.0    0.0    0.0287    0.2500           7.0    9.0    4.0    9.0    0.0    5.0
   0.1250           5.0    9.0    0.0    9.0    0.0    3.0
   0.0620           2.0    9.0    0.0    9.0    0.0    3.0
   0.0320           0.0    0.0    0.0    9.0    0.0    0.0288    0.2500           5.0    6.0    0.0    6.0    0.0    2.0
   0.1250           4.0    4.0    0.0    3.0    0.0    1.0
   0.0620           0.0    0.0    0.0    0.0    0.0    0.0
   0.0320           0.0    0.0    0.0    0.0    0.0    0.0289    0.2500           4.0    9.0    0.0    9.0    0.0    0.0
   0.1250           3.0    9.0    0.0    9.0    0.0    0.0
   0.0620           2.0    0.0    0.0    0.0    0.0    0.0
   0.0320           0.0    0.0    0.0    0.0    0.0    0.0290    0.2500           7.0    6.0    0.0    7.0    0.0    0.0
   0.1250           3.0    6.0    0.0    7.0    0.0    0.0
   0.0620           0.0    6.0    0.0    7.0    0.0    0.0
   0.0320           0.0    6.0    0.0    0.0    0.0    0.0291    0.2500           0.0    9.0           9.0    0.0    0.0
   0.1250           0.0    9.0           9.0    0.0    0.0
   0.0620           0.0    0.0           9.0    0.0    0.0
   0.0320           0.0    0.0           0.0    0.0    0.0
                                  表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号(公斤/公顷)          C      R      E      A      Y      T292    0.2500           0.0    9.0           9.0    5.0    0.0
   0.1250           0.0    9.0           9.0    0.0    0.0
   0.0620           0.0    9.0           9.0    0.0    0.0
   0.0320           0.0    9.0           9.0    0.0    0.0293    0.2500           0.0    9.0           9.0    6.0    0.0
   0.1250           0.0    9.0           9.0    0.0    0.0
   0.0620           0.0    9.0           9.0    0.0    0.0
   0.0320           0.0    9.0           9.0    0.0    0.0294    0.2500           0.0    9.0           9.0    0.0    0.0
   0.1250           0.0    3.0           9.0    0.0    0.0
   0.0620           0.0    0.0           9.0    0.0    0.0
   0.0320           0.0    0.0           9.0    0.0    0.0295    0.2500           0.0    9.0           9.0    6.0    0.0
   0.1250           0.0    9.0           9.0    0.0    0.0
   0.0620           0.0    0.0           0.0    0.0    0.0296    0.2500           4.0    7.0           9.0    7.0    2.0
   0.1250           2.0    7.0           9.0    5.0    0.0
   0.0620           0.0    7.0           9.0    0.0    0.0
   0.0320           0.0    6.0           9.0    0.0    0.0297    0.2500           4.0    9.0           9.0    9.0    2.0
   0.1250           3.0    7.0           9.0    3.0    0.0
   0.0620           0.0    5.0           9.0    0.0    0.0
   0.0320           0.0    4.0           9.0    0.0    0.0298    0.2500           3.0    9.0           9.0    9.0    0.0
   0.1250           0.0    9.0           9.0    3.0    0.0
   0.0620           0.0    9.0           9.0    0.0    0.0
   0.0320           0.0    3.0           9.0    0.0    0.0
                                  表III(续)
                     E                                   O
                     C      C      C      M      S       R
                     H      Y      Y      O      A       Y
                     O      P      P      O      G       S化合物  施用率           R      I      S      V      P       A编号(公斤/公顷)          C      R      E      A      Y       T299    0.2500           5.0    9.0           9.0    7.0     5.0
   0.1250           2.0    9.0           9.0    3.0     3.0
   0.0620           0.0    7.0           9.0    0.0     0.0
   0.0320           0.0    3.0           7.0    0.0     0.0300    0.2500           9.0    9.0           9.0    7.0     5.0
   0.1250           7.0    9.0           9.0    6.0     4.0
   0.0620           6.0    6.0           9.0    5.0     4.0
   0.0320           3.0    3.0           9.0    2.0     2.0301    0.2500           9.0    9.0    9.0    9.0    8.5     3.5
   0.1250           9.0    9.0    9.0    9.0    7.0     2.5
   0.0620           9.0    9.0    9.0    9.0    4.5     1.0
   0.0320           9.0    9.0    9.0    9.0    2.0     1.0302    0.2500           8.5    8.5    6.0    9.0    9.0     8.0
   0.1250           8.0    8.5    4.5    9.0    9.0     7.0
   0.0620           5.0    8.0    4.5    7.0    0.0     4.5
   0.0320           4.0    8.0    4.5    7.0    0.0     1.0303    0.2500           9.0    8.5    6.0    9.0    9.0     7.5
   0.1250           9.0    8.5    5.0    9.0    8.5     5.0
   0.0620           7.5    8.0    4.0    9.0    2.0     4.5
   0.0320           2.5    8.0    0.0    7.0    2.0     2.0304    0.2500           0.0    9.0    0.0    9.0    0.0     4.0
   0.1250           0.0    9.0    0.0    7.0    0.0     4.0
   0.0620           0.0    4.0    0.0    7.0    0.0     2.0
   0.0320           0.0    0.0    0.0    0.0    0.0     0.0305    0.2500           0.0    0.0    0.0    0.0    0.0     0.0306    0.2500           0.0    0.0    0.0    0.0    0.0     0.0
                                   表III(续)
                     E                                  O
                     C      C      C      M      S      R
                     H      Y      Y      O      A      Y
                     O      P      P      O      G      S化合物  施用率           R      I      S      V      P      A编号  (公斤/公顷)        C      R      E      A      Y      T307    0.2500           9.0    7.5    9.0    9.0    9.0    9.0
   0.1250           8.5    6.5    7.0    9.0    6.5    8.5
   0.0620           5.0    6.5    3.5    8.0    1.0    6.0
   0.0320           6.0    6.5    0.0    6.0    0.0    5.0308    0.2500           9.0    0.0    9.0    0.0    9.0    7.0
   0.1250           6.0    0.0    3.0    0.0    3.0    6.0
   0.0620           5.0    0.0    0.0    0.0    0.0    5.0
   0.0320           5.0    0.0    0.0    0.0    0.0    5.0309    0.2500           7.0    9.0    7.0    9.0    8.0    7.0
   0.1250           4.0    9.0    0.0    9.0    4.0    5.0
   0.0620           2.0    9.0    0.0    6.0    3.0    4.0
   0.0320           1.0    9.0    0.0    6.0    2.0    3.0310    0.2500           3.0    9.0    0.0    9.0    0.0    3.0
   0.1250           2.0    9.0    0.0    9.0    0.0    2.0
   0.0620           0.0    9.0    0.0    9.0    0.0    0.0
   0.0320           0.0    9.0    0.0    9.0    0.0    0.0311    0.2500           0.0    9.0    0.0    9.0    0.0    2.0
   0.1250           0.0    9.0    0.0    9.0    0.0    2.0
   0.0620           0.0    9.0    0.0    9.0    0.0    0.0
   0.0320           0.0    0.0    0.0    0.0    0.0    0.0312    0.2500           9.0    9.0    6.0    9.0    6.5    7.5
   0.1250           9.0    9.0    4.5    9.0    5.5    7.0
   0.0620           6.5    6.5    3.5    6.0    2.0    6.5
   0.0320           6.0    4.5    0.0    4.5    0.0    5.0313    0.2500           9.0    9.0    2.0    9.0    3.0    4.0
   0.1250           6.0    9.0    0.0    9.0    0.0    3.0
   0.0620           5.0    0.0    0.0    9.0    0.0    1.0
   0.0320           4.0    0.0    0.0    0.0    0.0    0.0
                                表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物  施用率        R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T314      0.2500      9.0      9.0      0.0      9.0      0.0      5.0
     0.1250      9.0      9.0      0.0      9.0      0.0      4.0
     0.0620      5.0      9.0      0.0      9.0      0.0      3.0
     0.0320      5.0      9.0      0.0      9.0      0.0      3.0315      0.2500      3.0      9.0      3.0      9.0      4.0      2.0
     0.1250      0.0      5.0      3.0      9.0      3.0      0.0
     0.0620      0.0      0.0      0.0      9.0      0.0      0.0
     0.0320      0.0      0.0      0.0      9.0      0.0      0.0316      0.2500      9.0      6.0      0.0      9.0      3.0      4.0
     0.1250      9.0      7.5      4.5      9.0      1.0      4.5
     0.0620      9.0      7.5      4.5      9.0      3.0      4.0
     0.0320      5.5      8.5      1.0      8.0      0.0      4.5318      0.2500      5.0      6.0      9.0      9.0      4.0      9.0
     0.1250      5.0      5.0      0.0      9.0      0.0      5.0
     0.0620      3.0      2.0      0.0      6.0      0.0      5.0
     0.0320      0.0      0.0      0.0      4.0      0.0      5.0319      0.2500      9.0      9.0      6.0      9.0      9.0      7.0
     0.1250      9.0      9.0      6.0      9.0      9.0      6.0
     0.0620      7.0      9.0      6.0      9.0      6.0      6.0
     0.0320      3.0      3.0      4.0      9.0      6.0      5.0320      0.2500      2.5      8.0               9.0      5.0      2.5
     0.1250      0.0      5.5               3.0      2.5      2.0
     0.0620      0.0      2.0               0.0      2.5      2.0
     0.0320      0.0      0.0               0.0      1.0      1.5321      0.2500      8.0      9.0      9.0      9.0      8.5      9.0
     0.1250      6.5      8.5      9.0      9.0      8.5      9.0
     0.0620      5.0      7.5      1.0      9.0      6.5      8.0
     0.0320      4.0      4.0      0.0      8.0      5.5      8.0
                                表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号   (公斤/公顷)    C        R        E        A        Y        T322      0.2500      9.0      9.0      9.0      9.0      9.0      7.0
     0.1250      9.0      7.0      6.0      9.0      3.0      5.0
     0.0620      9.0      6.0      5.0      9.0      3.0      5.0
     0.0320      9.0      4.0      5.0      5.0      3.0      5.0323      0.2500      8.0      8.0      7.5      9.0      9.0      7.5
     0.1250      8.0      8.0      6.5      9.0      3.5      6.0
     0.0620      6.5      4.5      6.0      9.0      3.5      5.0
     0.0320      4.5      3.5      5.0      8.0      0.0      3.5324      0.2500      6.0      9.0      7.0      9.0      9.0      9.0
     0.1250      5.0      9.0      3.0      9.0      9.0      7.0
     0.0620      4.0      9.0      0.0      9.0      3.0      4.0
     0.0320      0.0      9.0      0.0      9.0      0.0      3.0325      0.2500      9.0      9.0      9.0      9.0      9.0      4.0
     0.1250      9.0      9.0      7.3      9.0      6.3      3.7
     0.0620      9.0      8.7      9.0      9.0      4.3      3.0
     0.0320      7.7      8.0      4.7      8.0      4.0      2.7326      0.2500      9.0      9.0      7.5      9.0      9.0      5.5
     0.1250      9.0      7.0      4.5      9.0      5.5      5.5
     0.0620      8.5      7.0      4.5      9.0      1.0      5.5
     0.0320      5.5      6.0      4.0      9.0      0.0      5.5327      0.2500      9.0      9.0      9.0      9.0      7.5      4.0
     0.1250      9.0      9.0      5.5      9.0      5.5      3.5
     0.0620      9.0      9.0      5.5      9.0      5.5      2.5
     0.0320      9.0      9.0      1.0      9.0      3.0      3.0328      0.2500      9.0      9.0      9.0      9.0      4.5      4.5
     0.1250      9.0      9.0      7.5      9.0      4.5      4.0
     0.0620      9.0      9.0      6.0      9.0      3.0      3.0
     0.0320      9.0      9.0      6.0      9.0      2.5      2.0
                                 表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T329      0.2500      3.0      0.0      0.0      9.0      4.0      3.0
     0.1250      3.0      0.0      0.0      9.0      4.0      3.0
     0.0620      3.0      0.0      0.0      9.0      4.0      3.0
     0.0320      2.0      0.0      0.0      9.0      3.0      3.0330      0.2500      9.0      6.0      5.0      9.0      0.0      7.0
     0.1250      9.0      6.0      5.0      9.0      0.0      7.0
     0.0620      7.0      0.0      5.0      9.0      0.0      7.0
     0.0320      7.0      0.0      5.0      9.0      0.0      7.0331      0.2500      8.0      9.0      0.0      9.0      0.0      1.0
     0.1250      4.0      5.0      0.0      9.0      0.0      0.0
     0.0620      2.0      0.0      0.0      9.0      0.0      0.0
     0.0320      0.0      0.0      0.0      9.0      0.0      0.0332      0.2500      9.0      9.0      7.5      9.0      9.0      7.5
     0.1250      9.0      9.0      4.5      9.0      6.5      5.5
     0.0620      8.5      9.0      4.5      9.0      3.5      5.5
     0.0320      6.5      9.0      4.0      9.0      3.0      5.5333      0.2500      9.0      9.0      7.5      9.0      9.0      7.0
     0.1250      9.0      9.0      7.5      9.0      8.5      7.0
     0.0620      9.0      9.0      7.0      9.0      8.0      6.0
     0.0320      9.0      9.0      7.0      9.0      5.5      4.0334      0.2500      3.0      6.0      2.0               4.0      3.0
     0.1250      0.0      6.0      2.0               4.0      3.0
     0.0620      0.0      5.0      0.0               0.0      0.0
     0.0320      0.0      3.0      0.0               0.0      0.0335      0.2500      9.0      2.0      6.0               4.0      7.0
     0.1250      7.0      2.0      6.0               4.0      5.0
     0.0620      7.0      0.0      0.0               0.0      4.0
     0.0320      6.0      0.0      0.0               0.0      3.0
                                  表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物  施用率       R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T336     0.2500      9.0      9.0      3.0      9.0      9.0      9.0
    0.1250      9.0      4.0      2.0      9.0      1.0      4.5
    0.0620      9.0      1.0      0.0      9.0      0.0      4.5
    0.0320      6.5      0.0      0.0      9.0      0.0      2.0337     0.2500      6.0      9.0      9.0               3.0      3.0
    0.1250      6.0      6.0      0.0               0.0      3.0
    0.0620      2.0      0.0      0.0               0.0      3.0
    0.0320      2.0      0.0      0.0               0.0      3.0338     0.2500      9.0      8.0      5.0               5.0      6.0
    0.1250      4.0      3.0      0.0               2.0      3.0
    0.0620      2.0      3.0      0.0               2.0      0.0
    0.0320      2.0      3.0      0.0               0.0      0.0339     0.2500      6.0      7.0      9.0               9.0      9.0
    0.1250      4.0      7.0      6.0               5.0      9.0
    0.0620      0.0      4.0      0.0               5.0      7.0
    0.0320      0.0      4.0      0.0               5.0      5.0340     0.2500      9.0      9.0      7.0               7.0      9.0
    0.1250      9.0      7.0      6.0               5.0      7.0
    0.0620      6.0      5.0      3.0               4.0      6.0
    0.0320      5.0      2.0      3.0               4.0      5.0341     0.2500      8.5      4.0      3.5      9.0      4.5      3.5
    0.1250      8.0      3.5      2.5      9.0      4.5      3.0
    0.0620      5.5      2.0      0.0      9.0      4.5      2.5
    0.0320      3.0      1.0      0.0      7.0      1.0      1.5342     0.2500      7.0      8.0      9.0               2.0      3.0
    0.1250      7.0      4.0      0.0               0.0      2.0
    0.0620      4.0      0.0      0.0               0.0      0.0
    0.0320      4.0      0.0      0.0               0.0      0.0
                                表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物  施用率        R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T343      0.2500      9.0      6.0      6.0               3.0      4.0
     0.1250      7.0      0.0      4.0               0.0      3.0
     0.0620      6.0      0.0      3.0               0.0      2.0
     0.0320      3.0      0.0      0.0               0.0      0.0344      0.2500      9.0      9.0      6.0               6.0      9.0
     0.1250      7.0      7.0      6.0               3.0      5.0
     0.0620      7.0      6.0      6.0               0.0      5.0
     0.0320      4.0      6.0      6.0               0.0      2.0345      0.2500      9.0      9.0      9.0      9.0      9.0      6.0
     0.1250      9.0      9.0      4.5      9.0      9.0      5.5
     0.0620      9.0      9.0      9.0      9.0      9.0      5.5
     0.0320      9.0      9.0      5.0      9.0      4.5      5.5347      0.2500      9.0      9.0      7.0               5.0      9.0
     0.1250      9.0      9.0      4.0               4.0      7.0
     0.0620      9.0      9.0      0.0               3.0      6.0
     0.0320      7.0      7.0      0.0               2.0      3.0348      0.2500      9.0      9.0      0.0               9.0      5.0
     0.1250      7.0      6.0      0.0               7.0      4.0
     0.0620      6.0      0.0      0.0               6.0      3.0
     0.0320      6.0      0.0      0.0               4.0      2.0349      0.2500      7.0      7.0      4.0               6.0      7.0
     0.1250      6.0      7.0      4.0               5.0      7.0
     0.0620      5.0      4.0      4.0               5.0      5.0
     0.0320      5.0      0.0      4.0               4.0      4.0350      0.2500      9.0      9.0      9.0      9.0      9.0      9.0
     0.1250      8.0      9.0      8.5      9.0      7.5      9.0
     0.0620      7.5      5.0      8.5      9.0      7.0      9.0
     0.0320      6.0      4.0      7.5      9.0      5.5      9.0
                                 表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物    施用率      R        I        S        V        P        A编号   (公斤/公顷)    C        R        E        A        Y        T351      0.2500      7.0      9.0      8.0               7.0      9.0
     0.1250      6.0      7.0      6.0               7.0      7.0
     0.0620      6.0      7.0      6.0               6.0      7.0
     0.0320      5.0      6.0      0.0               5.0      7.0352      0.2500      9.0      9.0      0.0      9.0      9.0      3.0
     0.1250      6.5      7.5      1.0      9.0      9.0      2.5
     0.0620      4.0      6.5      0.0      9.0      5.0      1.0
     0.0320      2.5      2.0      0.0      6.0      2.5      0.5353      0.2500      3.0      3.0      2.5      8.0      0.0      4.0
     0.1250      2.5      1.0      1.5      8.0      0.0      3.5
     0.0620      2.0      0.0      0.0      6.5      0.0      3.0
     0.0320      0.0      0.0      0.0      3.5      0.0      2.5354      0.2500      9.0      9.0      9.0      9.0      9.0      9.0
     0.1250      9.0      9.0      9.0      9.0.     9.0      9.0
     0.0620      9.0      9.0      9.0      9.0      9.0      8.0
     0.0320      9.0      8.3      8.0      9.0      6.3      7.3355      0.2500      9.0      5.0      5.0      9.0      9.0      5.0
     0.1250      9.0      6.5      3.5      9.0      4.5      5.5
     0.0620      9.0      4.5      1.0      9.0      4.5      3.0
     0.0320      7.0      4.5      0.0      9.0      2.0      2.5356      0.2500      9.0      9.0      6.5      9.0      8.0      2.0
     0.1250      6.5      9.0      5.0      9.0      5.5      4.5
     0.0620      5.0      9.0      0.0      9.0      4.5      2.5
     0.0320      3.5      6.5      0.0      7.5      4.5      0.5357      0.2500      7.0      6.0      0.0      9.0      4.0      3.0
     0.1250      5.0      2.0      0.0      9.0      0.0      2.0
     0.0620      5.0      0.0      0.0      9.0      0.0      2.0
     0.0320      4.0      0.0      0.0      9.0      0.0      2.0
                                    表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T358     0.2500      5.0      7.0      0.0      9.0      6.0      3.0
    0.1250      5.0      0.0      0.0      9.0      6.0      3.0
    0.0620      5.0      0.0      0.0      9.0      5.0      3.0
    0.0320      4.0      0.0      0.0      9.0      5.0      2.0359     0.5000      9.0      9.0               9.0      5.0      9.0
    0.2500      9.0      9.0      9.0      9.0      4.5      9.0
    0.1250      9.0      8.5      9.0      9.0      1.8      8.8
    0.0620      9.0      7.5      6.0      9.0      0.5      7.3
    0.0320      8.5      6.3      9.0      8.8      0.0      6.5360     0.5000      9.0      9.0               9.0      9.0      9.0
    0.2500      7.5      9.0      9.0      9.0      9.0      9.0
    0.1250      5.0      9.0      0.0      4.5      4.5      3.5
    0.0620      2.0      2.5      0.0      4.5      4.5      2.0
    0.0320      0.0      0.0      0.0      4.5      1.5      1.0361     0.5000      4.0      6.0               9.0      5.0      3.0
    0.2500      4.0      6.0               9.0      5.0      5.0
    0.1250      0.0      0.0               9.0      5.0      4.0
    0.0620      0.0      0.0               9.0      4.0      0.0
    0.0320      0.0      0.0               9.0      4.0      0.0362     0.5000      9.0      9.0      9.0      9.0      9.0      8.0
    0.2500      9.0      7.0      9.0      9.0      9.0      6.0
    0.1250      7.0      5.0      9.0      9.0      9.0      4.0
    0.0620      7.0      5.0      9.0      9.0      9.0      4.0
    0.0320      4.0      3.0      6.0      9.0      9.0      4.0363     0.5000      7.0      8.0      7.0      9.0      9.0      9.0
    0.2500      6.0      7.0      7.0      9.0      9.0      7.0
    0.1250      5.0      7.0      5.0      9.0      7.0      6.0
    0.0620      4.0      7.0      0.0      9.0      5.0      5.0
    0.0320      3.0      6.0      0.0      9.0      3.0      4.0
                           表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T364     0.5000      7.0      9.0      7.0      9.0      9.0      9.0
    0.2500      6.0      9.0      6.0      9.0      9.0      9.0
    0.1250      6.0      9.0      5.0      9.0      5.0      6.0
    0.0620      5.0      7.0      3.0      9.0      4.0      5.0
    0.0320      3.0      7.0      3.0      9.0      4.0      4.0365     0.5000      9.0      9.0      9.0      9.0      6.0      6.0
    0.2500      9.0      9.0      9.0      9.0      5.0      5.0
    0.1250      9.0      6.0      4.0      9.0      5.0      5.0
    0.0620      6.0      6.0      4.0      9.0      5.0      5.0
    0.0320      4.0      4.0      4.0      9.0      3.0      3.0366     0.5000      9.0      9.0      9.0      9.0      9.0      9.0
    0.2500      9.0      9.0      9.0      9.0      9.0      9.0
    0.1250      9.0      9.0      9.0      9.0      9.0      9.0
    0.0620      8.5      9.0      8.0      9.0      8.0      9.0
    0.0320      8.0      8.5      8.0      9.0      7.0      7.5367     0.2500      6.0      9.0      9.0      9.0      9.0      6.0
    0.1250      3.0      7.0      9.0      9.0      5.0      5.0
    0.0620      0.0      5.0      9.0      9.0      2.0      0.0
    0.0320      0.0      0.0      0.0      9.0      0.0      0.0368     0.2500      8.0      9.0      8.0      9.0      9.0      7.0
    0.1250      7.0      9.0      7.0      9.0      9.0      6.0
    0.0620      7.0      9.0      4.0      9.0      6.0      5.0
    0.0320      3.0      7.0      0.0      9.0      5.0      5.0369     0.2500      8.0      9.0      9.0      9.0      9.0      7.0
    0.1250      6.0      9.0      4.0      9.0      9.0      7.0
    0.0620      3.0      7.0      3.0      9.0      6.0      6.0
    0.0320      3.0      7.0      0.0      9.0      0.0      6.0
                            表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物  施用率       R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T370     0.2500      7.0      9.0      9.0      9.0      9.0      5.0
    0.1250      6.0      9.0      7.0      9.0      7.0      4.0
    0.0620      4.0      7.0      4.0      9.0      3.0      4.0
    0.0320      3.0      4.0      0.0      7.0      0.0      3.0371     0.2500      7.0      9.0      9.0      9.0      9.0      9.0
    0.1250      6.0      9.0      6.0      9.0      9.0      6.0
    0.0620      4.0      6.0      0.0      9.0      4.0      6.0
    0.0320      3.0      4.0      0.0      9.0      3.0      5.0372     0.2500      9.0      9.0      9.0      9.0      9.0      9.0
    0.1250      9.0      9.0      8.5      9.0      9.0      8.0
    0.0620      9.0      9.0      5.0      9.0      9.0      8.0
    0.0320      9.0      8.5      1.0      9.0      8.5      6.0373     0.2500      9.0      9.0      8.0      9.0      9.0      8.0
    0.1250      9.0      9.0      7.5      9.0      9.0      6.0
    0.0620      9.0      9.0      5.0      9.0      8.5      6.5
    0.0320      6.5      6.5      2.0      9.0      5.5      5.5374     0.2500      6.0      9.0      5.0      9.0      9.0      7.0
    0.1250      4.0      9.0      0.0      9.0      6.0      6.0
    0.0620      3.0      9.0      0.0      9.0      3.0      4.0
    0.0320      3.0      6.0      0.0      9.0      2.0      4.0375     0.2500      9.0      9.0      7.0      9.0      9.0      6.0
    0.1250      9.0      6.0      4.0      9.0      9.0      4.0
    0.0620      6.0      4.0      0.0      9.0      9.0      4.0
    0.0320      6.0      3.0      0.0      9.0      7.0      2.0376     0.2500      9.0      9.0      8.0      9.0      9.0      8.5
    0.1250      6.5      9.0      5.5      9.0      9.0      6.0
    0.0620      5.5      8.0      4.0      9.0      8.5      6.0
    0.0320      3.0      3.0      3.0      9.0      8.0      4.0
                                表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物  施用率       R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T377     0.2500      9.0      8.0      8.5      9.0      9.0      9.0
    0.1250      7.0      4.5      5.0      9.0      8.5      8.0
    0.0620      5.0      3.0      3.0      9.0      4.0      6.5
    0.0320      2.0      2.0      1.0      9.0      0.0      5.5378     0.2500      9.0      9.0      9.0      9.0      9.0      9.0
    0.1250      9.0      9.0      9.0      9.0      9.0      9.0
    0.0620      9.0      9.0      9.0      9.0      9.0      9.0
    0.0320      9.0      9.0      9.0      9.0      9.0      9.0379     0.2500      8.0      9.0      8.5      9.0      9.0      9.0
    0.1250      7.5      9.0      8.5      9.0      9.0      9.0
    0.0620      5.0      7.5      6.5      9.0      6.5      8.5
    0.0320      2.0      5.5      2.5      9.0      3.5      7.0380     0.2500      9.0      9.0      8.0      9.0      9.0      6.5
    0.1250      9.0      9.0      8.0      9.0      4.0      5.0
    0.0620      9.0      9.0      3.5      9.0      0.0      4.0
    0.0320      9.0      9.0      3.5      9.0      0.0      2.5381     0.2500      6.0      8.0      7.0      8.0      7.0      7.0
    0.1250      4.0      8.0      7.0      8.0      6.0      6.0
    0.0620      3.0      7.0      4.0      7.0      5.0      3.0
    0.0320      0.0      6.0      0.0      6.0      3.0      3.0382     0.2500      7.0      9.0      7.0      9.0      9.0      5.0
    0.1250      4.0      7.0      7.0      9.0      7.0      6.0
    0.0620      3.0      6.0      0.0      9.0      4.0      6.0
    0.0320      0.0      5.0      0.0      9.0      3.0      5.0383     0.2500      8.0      8.0      9.0      9.0      9.0      6.5
    0.1250      7.5      7.0      7.5      9.0      9.0      6.0
    0.0620      6.5      7.0      5.5      9.0      7.5      4.5
    0.0320      4.0      2.5      4.5      9.0      3.0      3.5
                                 表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物  施用率       R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T384     0.2500      6.0      8.0      7.0      9.0      6.0      6.0
    0.1250      4.0      8.0      7.0      9.0      6.0      7.0
    0.0620      4.0      7.0      7.0      9.0      6.0      4.0
    0.0320      2.0      4.0      7.0      9.0      5.0      4.0385     0.2500      6.0      9.0      7.0      9.0      9.0      7.0
    0.1250      3.0      6.0      7.0      9.0      9.0      7.0
    0.0620      3.0      6.0      6.0      9.0      0.0      5.0
    0.0320      0.0      4.0      6.0      9.0      0.0      3.0386     0.2500      5.0      9.0      7.0      9.0      9.0      5.0
    0.1250      4.0      9.0      7.0      9.0      9.0      5.0
    0.0620      3.0      9.0      7.0      9.0      7.0      5.0
    0.0320      0.0      7.0      3.0      9.0      4.0      5.0387     0.2500      3.0      7.0      5.0      9.0      6.0      2.0
    0.1250      0.0      6.0      5.0      9.0      5.0      2.0
    0.0620      0.0      5.0      5.0      9.0      4.0      0.0
    0.0320      0.0      0.0      2.0      4.0      3.0      0.0388     0.2500      6.0      9.0      6.0      9.0      7.0      6.0
    0.1250      5.0      7.0               9.0      4.0      4.0
    0.0620      2.0      7.0               9.0      4.0      4.0
    0.0320      0.0      4.0      6.0      9.0      3.0      3.0389     0.2500      7.0      9.0      8.0      9.0      9.0      5.0
    0.1250      4.0      7.0      7.0      9.0      7.0      4.0
    0.0620      4.0      5.0               9.0      4.0      4.0
    0.0320      3.0      5.0      0.0      7.0      3.0      3.0390     0.5000      9.0      9.0      6.0      9.0      9.0      5.0
    0.2500      9.0      9.0      9.0      9.0      8.0      6.5
    0.1250      8.0      7.0      4.0      9.0      8.0      6.0
    0.0620      7.0      4.0               9.0      5.5      5.5
    0.0320      5.5      1.0      2.5      9.0      2.5      4.0
                                  表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T391     0.5000      6.0      9.0      3.0      9.0      9.0      3.0
    0.2500      4.0      6.0      0.0      9.0      7.0      3.0
    0.1250      2.0      4.0      0.0      9.0      7.0      3.0
    0.0620      0.0      3.0      0.0      9.0      6.0      2.0
    0.0320      0.0      3.0      0.0      6.0      6.0      2.0392     0.2500      9.0      7.0      0.0      9.0      0.0
    0.1250      9.0      3.0      0.0      7.0      0.0
    0.0620      7.0      0.0      0.0      7.0      0.0
    0.0320      5.0      0.0      0.0      6.0      0.0393     0.2500      9.0      6.0      6.0      9.0      4.0
    0.1250      4.0      3.0      3.0      8.0      3.0
    0.0620      4.0      3.0      0.0      8.0
    0.0320      2.0      0.0      0.0      7.0      0.0394     0.2500      6.0      7.0      2.0      9.0      0.0
    0.1250      4.0      5.0      0.0      9.0      0.0
    0.0620      0.0      3.0      0.0      8.0      0.0
    0.0320      0.0      0.0      0.0      8.0395     0.2500      3.0      3.0      0.0      9.0      5.0
    0.1250      2.0      0.0      0.0      9.0      4.0
    0.0620      0.0      0.0      0.0      9.0      2.0
    0.0320      0.0      0.0      0.0      9.0      0.0396     0.2500      9.0      9.0      6.0      9.0      8.0
    0.1250      9.0      9.0      0.0      9.0      8.0
    0.0620      9.0      8.0      0.0      9.0      7.0
    0.0320      9.0      7.0      0.0      9.0      7.0397     0.2500      9.0      9.0      0.0      9.0      5.0
    0.1250      9.0      9.0      0.0      9.0      5.0
    0.0620      9.0      7.0               9.0      5.0
    0.0320      9.0      6.0      0.0      9.0      4.0
                                    表III(续)
                  E                                       O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T398      0.2500      8.0      8.0      3.0      9.0      3.0
     0.1250      3.0      6.0      3.0      9.0      0.0
     0.0620      2.0      3.0      0.0      9.0      0.0
     0.0320      0.0      0.0      0.0      6.0      0.0399      0.2500      3.0      8.0      0.0      9.0      0.0
     0.1250      2.0      7.0      0.0      8.0      0.0
     0.0620      0.0      2.0      0.0      7.0      0.0
     0.0320      0.0      0.0      0.0      6.0      0.0400      0.2500      0.0      9.0      0.0      9.0      0.0
     0.1250      0.0      9.0      0.0      7.0      0.0
     0.0620      0.0      3.0      0.0      7.0      0.0
     0.0320      0.0      3.0      0.0      6.0      0.0401      0.2500      6.0      6.0      3.0      9.0      3.0      5.0
     0.1250      2.0      5.0      0.0      7.0      2.0      4.0
     0.0620      0.0      4.0      0.0      7.0      0.0      4.0
     0.0320      0.0      3.0               6.0      0.0      3.0402      0.2500      4.0      7.0      5.0      9.0      3.0      4.0
     0.1250      3.0      3.0      0.0      9.0      0.0      2.0
     0.0620      0.0      2.0      0.0      7.0      0.0      0.0
     0.0320      0.0      0.0      7.0      0.0      0.0403      0.2500      4.0      9.0      4.0      9.0      9.0
     0.1250      4.0      7.0      2.0      9.0      9.0
     0.0620      2.0      6.0      0.0      6.0      9.0
     0.0320      0.0      5.0      0.0      7.0      3.0404      0.2500      7.0      6.0      0.0      6.0      0.0      2.0
     0.1250      6.0      2.0      0.0      5.0      0.0      0.0
     0.0620      3.0      0.0      0.0      5.0      0.0      0.0
     0.0320      0.0      0.0      0.0      4.0      0.0      0.0
                           表III(续)
                E                                            O
                C        C        C        M        S        R
                H        Y        Y        O        A        Y
                O        P        P        O        G        S化合物   施用率     R        I        S        V        P        A编号  (公斤/公顷)   C        R        E        A        Y        T405      0.2500    9.0      8.0      0.0      7.0      6.0      2.0
     0.1250    9.0      7.0      0.0      7.0      5.0      2.0
     0.0060    7.0      4.0      0.0      6.0      0.0      0.0
     0.0320    7.0      4.0      0.0      6.0      0.0      0.0406      0.2500    7.0      7.0      6.0      9.0      4.0      4.0
     0.1250    7.0      4.0      3.0      9.0      4.0      2.0
     0.0620    6.0      4.0      0.0      7.0      4.0      0.0
     0.0320    6.0      0.0      0.0      4.0      3.0      0.0407      0.2500    7.0      9.0      7.0      9.0      7.0      5.0
     0.1250    7.0      9.0      5.0      9.0      6.0      3.0
     0.0620    3.0      4.0      0.0      7.0      2.0      2.0
     0.0320    0.0      3.0      0.0      6.0      0.0      0.0408      0.2500    7.0      9.0      6.0      9.0      6.0      3.0
     0.1250    6.0      9.0      5.0      9.0      4.0      2.0
     0.0620    3.0      9.0      0.0      9.0      0.0      2.0
     0.0320    2.0      6.0      0.0      7.0      0.0      0.0409      0.2500    9.0      9.0      9.0      9.0      9.0      9.0
     0.1250    9.0      9.0      9.0      9.0      7.0      7.0
     0.0620    4.0      9.0      5.0      9.0      4.0      5.0
     0.0320    3.0      7.0      2.0      9.0      2.0      3.0410      0.2500    9.0      9.0      9.0      9.0      9.0      7.0
     0.1250    9.0      9.0      9.0      9.0      9.0      5.0
     0.0620    0.0      9.0      5.0      9.0      7.0      3.0
     0.0320    0.0      9.0      2.0      9.0      3.0      0.0411      0.2500    6.0      9.0      9.0      9.0               5.0
     0.1250    0.0      3.0      7.0      9.0               2.0
     0.0620    0.0      2.0      2.0      9.0               0.0
     0.0320    0.0      0.0      0.0      9.0               0.0
                                  表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T412      0.2500               8.0      6.0      9.0               4.0
     0.1250      0.0      4.0      4.0      9.0               2.0
     0.0620      0.0      0.0      0.0      9.0               0.0
     0.0320      0.0      0.0      0.0      7.0               0.0413      0.2500      6.0      7.0      9.0      9.0               9.0
     0.1250      0.0      5.0      5.0      9.0               7.0
     0.0620      0.0      2.0      3.0      9.0               5.0
     0.0320      0.0      0.0      0.0      7.0               3.0414      0.2500      7.0      9.0      9.0      7.0               9.0
     0.1250      2.0      6.0               7.0               5.0
     0.0620      0.0      2.0               7.0               5.0
     0.0320      0.0      0.0      0.0                        5.0415      0.2500      9.0      6.0               8.0               9.0
     0.1250      3.0      2.0               5.0               5.0
     0.0620      0.0      0.0      0.0      5.0               4.0
     0.0320      0.0      0.0      0.0      5.0               3.0416      0.2500      9.0      8.0      3.0      9.0               9.0
     0.1250      3.0      4.0      0.0      7.0               9.0
     0.0620      3.0      4.0      0.0      7.0               7.0
     0.0320      0.0      4.0      0.0      7.0               6.0417      0.2500      3.0      6.0               9.0               3.0
     0.1250      3.0      5.0      3.0      9.0               0.0
     0.0620      0.0      4.0               6.0               0.0
     0.0320      0.0      4.0               6.0               0.0418      0.2500      3.0      0.0      0.0      0.0               3.0
     0.1250      1.0      0.0               0.0               2.0
     0.0620      0.0      0.0      0.0      0.0               0.0
                               表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T419      0.2500     7.0      6.0      0.0      5.0               3.0
     0.1250     2.0      3.0      0.0      4.0               1.0
     0.0620     0.0      0.0      0.0      0.0               0.0420      0.2500     7.0      6.0      0.0      9.0      3.0      5.0
     0.1250     7.0      6.0               9.0      2.0      3.0
     0.0620     7.0      4.0               9.0      0.0      2.0
     0.0320     7.0      2.0               9.0      0.0      0.0421      0.2500     9.0      9.0      4.0      9.0      2.0      2.0
     0.1250     7.0      8.0               7.0      0.0      0.0
     0.0620     5.0      6.0               6.0      0.0      0.0
     0.0320     5.0      2.0               5.0      0.0      0.0422      0.2500     9.0      9.0               9.0      6.0      3.0
     0.1250     9.0      9.0               9.0      3.0      2.0
     0.0620     6.0      6.0      5.0      9.0      0.0      0.0
     0.0320     5.0      5.0      0.0      7.0      0.0      0.0423      0.2500     9.0      9.0      9.0      9.0      9.0      7.0
     0.1250     9.0      9.0      9.0      9.0      9.0      7.0
     0.0620     9.0      7.0      9.0      9.0      9.0      6.0
     0.0320     6.0      6.0      9.0      9.0      9.0      5.0424      0.2500     3.0      7.0      3.0      9.0      0.0      2.0
     0.1250     3.0      6.0      3.0      9.0      0.0      0.0
     0.0620     0.0      5.0               9.0      0.0      0.0
     0.0320     0.0      4.0               7.0      0.0      0.0425      0.2500     9.0      9.0      3.0      9.0      4.0      8.0
     0.1250     9.0      6.0      3.0      9.0      3.0      7.0
     0.0620     9.0      0.0      3.0      7.0      0.0      6.0
     0.0320     6.0      0.0      0.0      6.0      0.0      4.0
                                 表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物  施用率        R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T426      0.2500      9.0      9.0      2.0               4.0      6.0
     0.1250      5.0      7.0      0.0               4.0      4.0
     0.0620      5.0      7.0      0.0               2.0      2.0
     0.0320      5.0      5.0      0.0               0.0      2.0427      0.2500      9.0      9.0      4.0               9.0      3.0
     0.1250      9.0      7.0                        6.0      1.0
     0.0620      7.0      7.0      0.0               5.0      0.0
     0.0320      7.0      7.0      0.0               4.0      0.0428      0.2500      9.0      7.0               9.0      6.0      6.0
     0.1250      6.0      4.0               9.0      2.0      6.0
     0.0620      3.0      2.0      0.0      9.0      0.0      2.0
     0.0320      2.0      0.0      0.0      9.0      0.0      0.0429      0.2500      9.0      9.0      1.0      9.0      3.0      3.0
     0.1250      9.0      8.3      1.0      9.0      2.3      2.3
     0.0620      9.0      7.7      1.0      9.0      2.3      2.0
     0.0320      9.0      7.3      0.0      9.0      2.0      1.3430      0.2500      9.0      6.0      7.0      9.0      7.0      3.0
     0.1250      7.0      7.0      2.0      9.0      6.0      4.0
     0.0620      5.0      6.0      0.0      9.0               2.0
     0.0320      5.0      2.0      0.0      9.0               3.0431      0.2500      9.0      9.0      9.0      9.0      9.0      6.5
     0.1250      8.5      9.0      7.5      9.0      7.5      5.0
     0.0620      9.0      9.0      4.0      9.0      5.5      5.5
     0.0320      8.0      8.0      0.0      9.0      3.5      3.5432      0.2500      9.0      9.0      9.0      9.0      8.5      7.5
     0.1250      9.0      9.0      6.5      9.0      7.5      6.5
     0.0620      9.0      9.0      3.5      9.0      3.5      6.0
     0.0320      9.0      8.0      0.0      9.0      0.0      6.0
                                    表III(续)
                      E                                                O
                      C          C          C        M        S        R
                      H          Y          Y        O        A        Y
                      O          P          P        O        G        S化合物     施用率         R          I          S        V        P        A编号    (公斤/公顷)       C          R          E        A        Y        T433        0.2500        9.0        9.0        7.5      9.0      7.0      7.5
       0.1250        9.0        9.0        7.5      9.0      6.0      5.0
       0.0620        9.0        8.5        6.0      9.0      4.5      4.0
       0.0320        8.0        5.5        0.0      8.5      2.0      2.0434        0.2500        9.0        8.0        7.0      9.0      6.0      7.0
       0.1250        7.0        7.0        4.0      9.0      5.0      6.0
       0.0620        7.0        3.0                 9.0      4.0      6.0
       0.0320        6.0        3.0        4.0      9.0      4.0      4.0435        0.2500        9.0        3.0        2.0      9.0      6.0      2.0
       0.1250        7.0        2.0        3.0      9.0      0.0      2.0
       0.0620        7.0        0.0        0.0      9.0      0.0      1.0
       0.0320        5.0        0.0                 9.0      0.0      2.0436        0.2500        9.0        7.0        6.0      9.0      3.0      6.0
       0.1250        9.0        7.0                 9.0      2.0      7.0
       0.0620        9.0        2.0        6.0      9.0      0.0      5.0
       0.0320        6.0        0.0        4.0      9.0      0.0      3.0437        0.2500        8.0        6.0        7.0      9.0      7.0      7.0
       0.1250        7.0        4.0        3.0      9.0      4.0      6.0
       0.0620        7.0        0.0        2.0      9.0      3.0      5.0
       0.0320        5.0        0.0        0.0      9.0      0.0      4.0438        0.2500        9.0        9.0        9.0      9.0      9.0      8.0
       0.1250        9.0        8.5        7.0      9.0      8.5      7.0
       0.0620        8.0        6.5        9.0      8.5      3.5      5.0
       0.0320        7.0        4.5        4.5      8.0      2.0      4.0439        0.2500        6.0        5.0        0.0      7.0      3.0      0.0
       0.1250        6.0        4.0        0.0      7.0      0.0      0.0
       0.0620        3.0        3.0        0.0      6.0      0.0      0.0
       0.0320        2.0        1.0        0.0      5.0      0.0      0.0
                              表III(续)
                E                                            O
                C        C        C        M        S        R
                H        Y        Y        O        A        Y
                O        P        P        O        G        S化合物   施用率     R        I        S        V        P        A编号  (公斤/公顷)   C        R        E        A        Y        T440      0.2500    9.0      9.0      9.0      9.0      9.0      4.0
     0.1250    9.0      9.0      9.0      9.0      7.0      4.0
     0.0620    7.0      9.0      9.0      9.0      6.0      4.0
     0.0320    5.0      5.0      6.0      7.0      4.0      3.0441      0.2500    3.0      9.0      7.0      9.0      6.0      3.0
     0.1250    0.0      9.0      4.0      9.0      3.0      2.0
     0.0620    0.0      6.0      0.0      9.0      2.0      0.0
     0.0320    0.0      4.0               9.0      0.0      0.0442      0.2500    9.0      9.0      4.5      9.0      4.0      3.3
     0.1250    9.0      8.7      0.0      9.0      2.0      1.7
     0.0620    9.0      6.3      0.0      8.3      1.7      1.3
     0.0320    8.3      4.3      0.0      6.0      1.3      0.3443      0.2500    9.0      7.0               7.0      5.0      8.0
     0.1250    7.0      7.0      0.0      7.0      4.0      5.0
     0.0620    5.0      6.0      0.0      6.0      3.0      4.0
     0.0320    6.0      4.0      0.0      5.0      3.0      3.0444      0.2500    9.0      9.0      9.0      9.0      9.0      8.5
     0.1250    8.5      9.0      9.0      9.0      7.0      9.0
     0.0620    6.0      8.0      9.0      9.0      6.0      6.5
     0.0320    3.5      7.5      3.5      8.0      4.5      4.5445      0.2500    9.0      9.0      8.5      9.0      9.0      8.0
     0.1250    9.0      9.0      8.0      9.0      8.5      7.0
     0.0620    8.5      8.0      8.5      9.0      8.0      6.5
     0.0320    8.5      6.5      7.5      9.0      4.5      5.0446      0.2500    9.0      9.0      9.0      9.0      9.0      9.0
     0.1250    7.0      9.0      9.0      9.0      9.0      9.0
     0.0620    6.0      9.0      9.0      9.0      9.0      7.0
     0.0320    6.0      9.0      9.0      9.0      9.0      6.0
                                  表III(续)
                E                                            O
                C        C        C        M        S        R
                H        Y        Y        O        A        Y
                O        P        P        O        G        S化合物   施用率     R        I        S        V        P        A编号  (公斤/公顷)   C        R        E        A        Y        T447      0.2500    9.0      9.0      4.0      9.0      9.0      7.0
     0.1250    7.0      7.0               9.0      5.0      5.0
     0.0620    6.0      6.0      0.0      9.0      4.0      4.0
     0.0320    4.0      4.0      0.0      7.0      4.0      4.0448      0.2500    9.0      9.0      6.5      9.0      3.5      4.0
     0.1250    9.0      9.0      4.5      9.0      2.5      4.0
     0.0620    9.0      9.0      4.5      9.0      1.5      4.0
     0.0320    9.0      8.5      4.5      9.0      0.0      3.5449      0.2500    9.0      9.0      4.0      9.0      6.0      9.0
     0.1250    9.0      8.0               9.0      4.0      3.0
     0.0620    7.0      5.0               7.0      4.0      3.0
     0.0320    5.0      4.0      2.0      7.0      2.0      2.0450      0.2500    9.0      9.0               9.0      9.0      9.0
     0.1250    6.0      9.0               9.0      6.0      5.0
     0.0620    2.0      7.0               7.0      5.0      4.0
     0.0320    0.0      6.0      0.0      7.0      5.0      3.0451      0.2500    7.0      9.0      0.0      9.0      9.0      6.0
     0.1250    6.0      7.0               9.0      6.0      6.0
     0.0620    0.0      5.0      0.0      9.0      5.0      4.0
     0.0320    0.0      5.0               9.0      4.0      4.0452      0.2500    7.0      9.0      7.0      9.0      2.0      7.0
     0.1250    3.0      9.0               9.0      0.0      6.0
     0.0620    3.0      6.0               9.0      0.0      5.0
     0.0320    0.0      4.0      0.0      9.0      0.0      3.0453      0.2500    9.0      9.0      9.0      9.0      9.0      9.0
     0.1250    9.0      9.0      9.0      9.0      9.0      9.0
     0.0620    9.0      9.0      9.0      9.0      9.0      9.0
     0.0320    9.0      9.0      9.0      9.0      9.0      9.0
                                    表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物    施用率     R        I        S        V        P        A编号   (公斤/公顷)   C        R        E        A        Y        T454       0.2500    7.0      9.0      8.0      9.0      6.0      5.0
      0.1250    6.0      6.0      4.0      9.0      3.0      5.0
      0.0620    3.0      1.0      0.0      7.0      2.0      2.0
      0.0320    3.0      0.0      0.0      2.0      0.0      2.0455       0.2500    9.0      9.0      9.0      9.0      9.0      9.0
      0.1250    9.0      9.0      8.0      9.0      7.0      9.0
      0.0620    9.0      7.0      6.0      7.0      6.0      8.0
      0.0320    9.0      6.0      2.0      6.0      4.0      6.0456       0.2500    9.0      6.0      4.0      9.0      4.0      9.0
      0.1250    7.0      6.0      2.0      9.0      2.0      8.0
      0.0620    6.0      4.0      0.0      9.0      0.0      8.0
      0.0320    4.0      0.0      0.0      7.0      0.0      7.0457       0.2500    9.0      7.0      0.0      7.0      3.0      3.0
      0.1250    9.0      5.0      0.0      7.0      3.0      0.0
      0.0620    7.0      3.0      0.0      4.0      0.0      0.0
      0.0320    5.0      0.0      0.0      2.0      0.0      0.0458       0.2500    8.0      7.0      6.0      9.0      8.0      5.0
      0.1250    7.0      7.0      9.0      9.0      6.0      5.0
      0.0620    6.0      4.0               6.0      2.0      3.0
      0.0320    5.0      0.0      2.0      4.0      2.0      3.0459       0.2500    9.0      4.0      3.0      7.0      0.0      5.0
      0.1250    9.0      4.0      0.0      7.0      0.0      5.0
      0.0620    7.0      2.0      0.0      5.0      0.0      4.0
      0.0320    7.0      0.0      0.0      3.0      0.0      2.0460       0.2500    9.0      3.0      0.0      4.0      3.0      5.0
      0.1250    9.0      3.0      0.0      4.0      3.0      4.0
      0.0620    7.0      2.0               4.0      0.0      4.0
      0.0320    6.0      0.0               3.0      0.0      4.0
                                   表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T461      0.2500      9.0      9.0      7.0      9.0      6.0      6.0
     0.1250      9.0      9.0               9.0      4.0      5.0
     0.0620      9.0      9.0               7.0      3.0      5.0
     0.0320      9.0      6.0      0.0      7.0      2.0      5.0462      0.2500      9.0      9.0               9.0      6.0      6.0
     0.1250      9.0      9.0               9.0      5.0      9.0
     0.0620      9.0      9.0      3.0      9.0      4.0      5.0
     0.0320      9.0      9.0               9.0      1.0      5.0463      0.2500      9.0      9.0      7.0      9.0      7.0      6.0
     0.1250      9.0      9.0      6.0      9.0      5.0      5.0
     0.0620      6.0      6.0               9.0      3.0      2.0
     0.0320      2.0      5.0      2.0      7.0      0.0      0.0464      0.2500      9.0      5.0      7.0      6.0      4.0      4.0
     0.1250      6.0      3.0      0.0      9.0      6.0      2.0
     0.0620               3.0      0.0      9.0      0.0      2.0
     0.0320      6.0      0.0      0.0      7.0      0.0      0.0465      0.2500      9.0      8.0      9.0      9.0      6.0      5.0
     0.1250      7.0      3.0      7.0      6.0      5.0      4.0
     0.0620      6.0      0.0      4.0      3.0      5.0      3.0
     0.0320      6.0      0.0      0.0      2.0      2.0      2.0466      0.2500      7.0      9.0      1.0      9.0      7.0      9.0
     0.1250      5.0      7.0               9.0      3.0      7.0
     0.0620      4.0      3.0               7.0      0.0      5.0
     0.0320      2.0      3.0               7.0      0.0      4.0467      0.2500      9.0      9.0      9.0      9.0      7.0      5.0
     0.1250      9.0      6.0      9.0      9.0      3.0      4.0
     0.0620      7.0      5.0      7.0      9.0      0.0      2.0
     0.0320      6.0      2.0      6.0      7.0      0.0      2.0
                                      表III(续)
                     E                                          O
                     C       C         C       M        S       R
                     H       Y         Y       O        A       Y
                     O       P         P       O        G       S化合物    施用率         R       I         S       V        P       A编号   (公斤/公顷)       C       R         E       A        Y       T468       0.2500        9.0     5.0       5.0     5.0      5.0     5.0
      0.1250        9.0     6.0       7.0     7.0      4.0     5.0
      0.0620        7.0     6.0       6.0     6.0      4.0     3.0
      0.0320        7.0     5.0       2.0     5.0      3.0     3.0469       0.2500        9.0     7.0       6.0     8.0      3.0     1.5
      0.1250        9.0     6.5       9.0     5.0      2.5     0.0
      0.0620        9.0     1.5       4.5     4.5      1.5     0.0
      0.0320        7.0     0.0       0.0     2.0      0.0     0.0470       0.2500        9.0     7.0       4.5     3.0      1.5     1.5
      0.1250        9.0     6.0       0.0     2.0      0.0     1.0
      0.0620        9.0     0.0       0.0     2.0      0.0     0.0
      0.0320        8.5     0.0       0.0     1.5      0.0     0.0471       0.2500        9.0     9.0       7.0     9.0      7.0     5.0
      0.1250        6.0     9.0               9.0      5.0     5.0
      0.0620        3.0     6.0               7.0      3.0     3.0
      0.0320        0.0     6.0       3.0     6.0      0.0     2.0472       0.2500        4.0     6.0       9.0     7.0      3.0     6.0
      0.1250        4.0     5.0       6.0     7.0      2.0     3.0
      0.0620        3.0     4.0               6.0      0.0     1.0
      0.0320        3.0     4.0       0.0     5.0      0.0     0.0473       0.2500        4.0     8.0       5.0     7.0      3.0     5.0
      0.1250        2.0     6.0               7.0      2.0     4.0
      0.0620        2.0     4.0       0.0     6.0      0.0     2.0
      0.0320        1.0     2.0       0.0     4.0      0.0     0.0474       0.2500        0.0     6.0       0.0     9.0      0.0     3.0
      0.1250        0.0     4.0       0.0     7.0      0.0     2.0
      0.0620        0.0     5.0       0.0     3.0      0.0     0.0
      0.0320        0.0     2.0       0.0     2.0      0.0     0.0
                                     表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T475      0.2500      3.0      9.0      7.0      9.0      7.0      9.0
     0.1250      2.0      9.0      5.0      9.0      6.0      3.0
     0.0620      0.0      6.0               9.0      4.0      0.0
     0.0320      0.0      4.0      0.0      9.0      0.0      0.0476      0.2500      3.0      9.0      6.0      9.0      5.0      6.0
     0.1250      2.0      9.0      3.0      6.0      4.0      4.0
     0.0620      2.0      4.0               6.0      2.0      3.0
     0.0320      0.0      4.0      0.0      5.0      0.0      2.0477      0.2500      3.0      6.0      3.0      7.0      2.0      6.0
     0.1250      2.0      5.0               6.0      0.0      4.0
     0.0620      0.0      4.0      3.0      3.0      0.0      4.0
     0.0320      0.0      4.0      3.0      3.0      0.0      3.0478      0.2500      9.0      9.0      9.0      9.0      9.0      9.0
     0.1250      7.0      9.0      9.0      9.0      9.0      9.0
     0.0620      6.0      9.0      7.0      9.0      6.0      9.0
     0.0320      4.0      4.0      6.0      7.0      6.0      7.0479      0.2500      9.0      9.0      9.0      9.0      8.0      9.0
     0.1250      9.0      5.0      9.0      9.0      6.0      9.0
     0.0620      7.0      0.0      7.0      7.0      5.0      5.0
     0.0320      7.0      0.0      0.0      0.0      3.0      5.0480      0.2500      6.0      9.0               9.0      6.0      6.0
     0.1250      5.0      9.0      3.0      9.0      5.0      5.0
     0.0620      2.0      9.0               9.0      3.0      5.0
     0.0320      0.0      6.0      3.0      7.0      0.0      4.0481      0.2500      9.0      9.0      6.0      9.0               7.0
     0.1250      9.0      6.0               7.0      0.0      2.0
     0.0620      2.0      2.0               7.0      0.0      0.0
     0.0320      0.0      0.0               6.0      0.0      0.0
                                         表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T482       0.2500      9.0      6.0               7.0      7.0      7.0
      0.1250      9.0      0.0               6.0      5.0      6.0
      0.0620      7.0      0.0               5.0      4.0      2.0
      0.0320      4.0      0.0               4.0      3.0      0.0483       0.2500      7.0      6.0      6.0      9.0      5.0      6.0
      0.1250      7.0      5.0               9.0      3.0      5.0
      0.0620      7.0      2.0      4.0      9.0      0.0      3.0
      0.0320      6.0      0.0               7.0      0.0      3.0484       0.2500      9.0      9.0               9.0               6.0
      0.1250      7.0      6.0               9.0               6.0
      0.0620      4.0      4.0               9.0               5.0
      0.0320      5.0      4.0      0.0      7.0      5.0      5.0485       0.2500      9.0      6.0               8.0      3.0      5.0
      0.1250      6.0      5.0               7.0      0.0      4.0
      0.0620      6.0      4.0      0.0      6.0      0.0      2.0
      0.0320      4.0      2.0      0.0      4.0      0.0      0.0486       0.2500      9.0      6.0      3.0      9.0      6.0      6.0
      0.1250      7.0      6.0               7.0      3.0      5.0
      0.0620      6.0      5.0      0.0      6.0      0.0      3.0
      0.0320      4.0      4.0      0.0      5.0      0.0      0.0487       0.2500      9.0      9.0      3.0      9.0      7.0      7.0
      0.1250      7.0      6.0               9.0      6.0      6.0
      0.0620      7.0      5.0               9.0      5.0      3.0
      0.0320      6.0      4.0               7.0      4.0      2.0488       0.2500      0.0      5.0               9.0      0.0      4.0
      0.1250      0.0      4.0      0.0      9.0      0.0      4.0
      0.0620      0.0      3.0      0.0      9.0      0.0      3.0
      0.0320      0.0      3.0               7.0      0.0      3.0
                                     表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T489       0.2500      9.0      9.0      9.0      9.0      9.0      6.0
      0.1250      9.0      9.0      9.0      9.0      9.0      6.0
      0.0620      7.0      9.0      7.0      9.0      9.0      6.0
      0.0320      7.0      6.0      6.0      9.0      6.0      5.0490       0.2500      9.0      9.0      9.0      9.0      9.0      9.0
      0.1250      9.0      9.0      9.0      9.0      9.0      8.5
      0.0620      9.0      9.0      9.0      9.0      9.0      9.0
      0.0320      8.0      9.0      9.0      9.0      6.0      7.5491       0.2500      9.0      9.0      9.0      9.0      9.0      7.5
      0.1250      9.0      9.0      9.0      9.0      9.0      8.0
      0.0620      9.0      9.0      9.0      9.0      5.5      6.5
      0.0320      9.0      7.5      7.0      9.0      5.0      5.0492       0.2500      9.0      5.0      0.0      7.0      2.0      3.0
      0.1250      6.0      4.0               7.0      0.0      2.0
      0.0620      6.0      4.0               6.0      0.0      2.0
      0.0320      4.0      4.0               6.0      0.0      2.0493       0.2500      9.0      9.0      9.0      9.0      3.0      3.0
      0.1250      9.0      7.0      9.0      7.0      0.0      3.0
      0.0620      5.0      6.0               7.0      0.0      2.0
      0.0320      4.0      4.0               5.0      0.0      2.0494       0.2500      3.0      5.0      3.0      6.0      3.0      0.0
      0.1250      3.0      5.0      0.0      5.0      0.0      0.0
      0.0620      2.0      4.0               4.0      0.0      0.0
      0.0320      0.0      3.0               4.0      0.0      0.0495       0.2500      7.0      9.0               9.0               7.0
      0.1250      5.0      7.0               9.0      3.0      5.0
      0.0620      4.0      6.0               7.0      0.0      4.0
      0.0320      3.0      6.0               7.0      0.0      2.0
                                    表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T496      0.2500      7.0      9.0      7.0      8.0      6.0      5.0
     0.1250      6.0      7.0               6.0      3.0      3.0
     0.0620      4.0      7.0               6.0      0.0      3.0
     0.0320      4.0      0.0               0.0      0.0      0.0497      0.2500      7.0      9.0      9.0      9.0      6.0      8.0
     0.1250      4.0      9.0      6.0      9.0      2.0      7.0
     0.0620      0.0      6.0               7.0      0.0      3.0
     0.0320      0.0      5.0               6.0      0.0      0.0498      0.2500      6.0      9.0               8.0      6.0      6.0
     0.1250      5.0      9.0      0.0      7.0      3.0      3.0
     0.0620      3.0      5.0               5.0      0.0      2.0
     0.0320      0.0      2.0               4.0      0.0      0.0499      0.2500      9.0      9.0      9.0      9.0      9.0      9.0
     0.1250      9.0      9.0      9.0      9.0      9.0      7.5
     0.0620      9.0      9.0      9.0      9.0      9.0      8.0
     0.0320      7.5      8.0      9.0      8.0      8.0      6.5500      0.2500      9.0      9.0      0.0      9.0      9.0      2.0
     0.1250      7.0      6.0      0.0      9.0      7.0      2.0
     0.0620      6.0      6.0      0.0      9.0      7.0      2.0
     0.0320      4.0      6.0      0.0      7.0      5.0      2.0501      0.2500      7.0      6.0      5.0      9.0      6.0      4.0
     0.1250      5.0      4.0      3.0      7.0      5.0      3.0
     0.0620      5.0      2.0      0.0      6.0      3.0      1.0
     0.0320      4.0      0.0      0.0      6.0      2.0      0.0502      0.2500      7.0      9.0      5.0      9.0      9.0      6.0
     0.1250      5.0      9.0               7.0      5.0      5.0
     0.0620      3.0      6.0      2.0      6.0      2.0      2.0
     0.0320      3.0      4.0      0.0      6.0      0.0      2.0
                                  表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T503     0.2500      6.0      7.0      6.0      9.0      8.0      6.0
    0.1250      6.0      9.0      5.0      9.0      4.0      7.0
    0.0620      4.0      6.0               9.0      3.0      3.0
    0.0320      2.0      0.0               7.0      0.0      1.0504     0.2500      7.0      9.0               9.0      7.0      5.0
    0.1250      6.0      9.0      0.0      9.0               3.0
    0.0620      3.0      7.0      0.0      8.0
    0.0320      2.0      4.0      0.0      6.0      0.0      3.0505     0.2500      9.0      4.0               8.0      4.0      6.0
    0.1250      7.0      3.0      0.0      7.0      2.0      4.0
    0.0620      6.0               0.0      7.0      2.0      4.0
    0.0320      6.0      0.0               7.0      0.0      4.0506     0.2500      9.0      9.0      7.0      9.0      4.5      2.0
    0.1250      9.0      9.0      4.5      9.0      3.0      1.5
    0.0620      9.0      8.0      4.5      9.0      3.0      1.5
    0.0320      7.5      6.5      4.5      8.0      2.5      1.5507     0.2500      7.0      9.0               9.0      9.0      5.0
    0.1250      4.0      9.0               9.0      9.0      7.0
    0.0620      2.0      6.0               9.0      9.0      5.0
    0.0320      2.0      5.0      0.0      9.0      7.0      3.0508     0.2500      9.0      9.0               9.0      9.0      6.0
    0.1250      6.0      7.0               9.0      9.0      5.0
    0.0620      5.0      7.0               9.0      6.0      2.0
    0.0320      2.0      6.0      0.0      9.0      5.0      0.0509     0.2500      7.0      7.0      7.0      9.0      6.0      7.0
    0.1250      2.0      4.0      0.0      4.0      3.0      3.0
    0.0620      0.0      0.0      0.0      0.0      0.0      0.0
                                  表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T510     0.2500      9.0      8.0      5.0      9.0      6.0      8.0
    0.1250      9.0      7.0      3.0      9.0      5.0      4.0
    0.0620      9.0      3.0      0.0      7.0      4.0      2.0
    0.0320      9.0      0.0      0.0      6.0      3.0      0.0511     0.2500      7.0      7.0      3.0               7.0      6.0
    0.1250      5.0      2.0      3.0               0.0      5.0
    0.0620      2.0      0.0      0.0               0.0      4.0
    0.0320      0.0      0.0      0.0               0.0      3.0512     0.2500      9.0      5.0      0.0      9.0      4.0      2.0
    0.1250      9.0      5.0      0.0      9.0      2.0      1.0
    0.0620      7.0      2.0      0.0      9.0      0.0      0.0
    0.0320      7.0      0.0      0.0      9.0      0.0      0.0513     0.2500      8.0      9.0      9.0      9.0      9.0      9.0
    0.1250      7.0      6.0      9.0      9.0      9.0      9.0
    0.0620      5.0      4.0      9.0      9.0      9.0      7.0
    0.0320      0.0      4.0      9.0      9.0      9.0      9.0514     0.2500      8.0      7.0      0.0      9.0      0.0      4.0
    0.1250      2.0      2.0      0.0      9.0      0.0      1.0
    0.0620      1.0      0.0      0.0      9.0      0.0      2.0
    0.0320      0.0      0.0      0.0      9.0      0.0      2.0515     0.2500      9.0      7.0      0.0      9.0      0.0      6.0
    0.1250      8.0      4.0      0.0      9.0      0.0      4.0
    0.0620      6.0      2.0      0.0      9.0      0.0      2.0
    0.0320      2.0      0.0      0.0      9.0      0.0      0.0516     0.2500      0.0      2.0      0.0      9.0      0.0      3.0
    0.1250      0.0      0.0      0.0      8.0      0.0      2.0
    0.0620      0.0      0.0      0.0      6.0      0.0      1.0
    0.0320      0.0      0.0      0.0      4.0      0.0      0.0
                                  表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T517      0.2500      9.0      7.0      0.0      9.0      0.0      3.0
     0.1250      8.0      5.5      4.5      9.0      0.0      1.5
     0.0620      9.0      6.5      4.5      9.0      0.0      0.0
     0.0320      9.0      5.5      3.0      9.0      0.0      0.0518      0.2500      7.0      4.0      0.0      9.0      0.0      4.0
     0.1250      4.0      2.0      0.0      9.0      0.0      4.0
     0.0620      2.0      2.0      0.0      7.0      0.0      2.0
     0.0320      0.0      0.0      0.0      4.0      0.0      1.0519      0.2500      9.0      6.0      0.0      9.0      0.0      4.0
     0.1250      6.5      2.0      0.0      9.0      0.0      4.5
     0.0620      4.0      0.0      0.0      9.0      0.0      4.0
     0.0320      2.0      0.0      0.0      9.0      0.0      2.0520      0.2500      9.0      4.0      0.0      9.0      0.0      3.0
     0.1250      8.5      2.0      0.0      9.0      0.0      4.5
     0.0620      8.0      0.0      0.0      9.0      0.0      3.5
     0.0320      6.5      0.0      0.0      9.0      0.0      2.0521      0.2500      4.0      2.0      0.0      9.0      0.0      0.0
     0.1250      4.0      0.0      0.0      9.0      0.0      0.0
     0.0620      2.0      0.0      0.0      9.0      0.0      0.0
     0.0320      2.0      0.0      0.0      6.0      0.0      0.0522      0.2500      9.0      2.0      0.0      9.0      0.0      4.5
     0.1250      8.0      0.0      0.0      9.0      0.0      4.0
     0.0620      6.5      0.0      0.0      9.0      0.0      4.0
     0.0320      5.5      0.0      0.0      9.0      0.0      2.5523      0.2500      9.0      8.0      9.0      9.0      0.0      7.0
     0.1250      8.0      4.0      2.0      9.0      0.0      5.5
     0.0620      8.0      2.0      0.0      9.0      0.0      4.5
     0.0320      6.0      0.0      0.0      8.0      0.0      4.5
                                        表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T524      0.2500      9.0      7.0      6.0      9.0      0.0      9.0
     0.1250      9.0      4.0      2.0      9.0      0.0      7.0
     0.0620      9.0      2.0      0.0      9.0      0.0      4.0
     0.0320      7.0      2.0      0.0      9.0      0.0      2.0525      0.2500      9.0      4.0      0.0      9.0      0.0      4.0
     0.1250      9.0      2.0      0.0      9.0      0.0      2.0
     0.0620      7.0      2.0      0.0      9.0      0.0      2.0
     0.0320      6.0      0.0      0.0      9.0      0.0      0.0526      0.2500      6.0      9.0      0.0      9.0      0.0      3.0
     0.1250      4.0      7.0      0.0      9.0      0.0      2.0
     0.0620      2.0      4.0      0.0      9.0      0.0      2.0
     0.0320      2.0      2.0      0.0      8.0      0.0      1.0527      0.2500      9.0      4.0      0.0      9.0      0.0      4.0
     0.1250      9.0      4.0      0.0      9.0      0.0      2.5
     0.0620      8.0      2.0      0.0      9.0      0.0      2.5
     0.0320      3.0      2.0      0.0      9.0      0.0      2.0528      0.2500      9.0      9.0      0.0      9.0      3.0      9.0
     0.1250      9.0      5.0      0.0      9.0      1.5      7.0
     0.0620      9.0      5.0      0.0      9.0      0.0      3.5
     0.0320      9.0      4.5      0.0      9.0      1.0      1.5529      0.2500      9.0      0.0      0.0      0.0      9.0      9.0
     0.1250      9.0      3.0      0.0      3.0      9.0      3.0
     0.0620      9.0      3.0      0.0      3.0      9.0      0.0
     0.0320      7.0      3.0      0.0      3.0      9.0      0.0530      0.2500      9.0      9.0      0.0      9.0      9.0      9.0
     0.1250      9.0      9.0      0.0      9.0      3.0      3.0
     0.0620      9.0      9.0      0.0      9.0      0.0      0.0
     0.0320      9.0      0.0      0.0      9.0      0.0      0.0
                                        表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T532      0.2500      9.0      4.0      3.0      9.0      3.0      9.0
     0.1250      9.0      4.0      3.0      9.0      3.0      3.0
     0.0620      9.0      0.0      0.0      9.0      0.0      0.0
     0.0320      9.0      0.0      0.0      9.0      0.0      0.0532      0.2500      9.0      9.0      0.0      9.0      9.0      2.0
     0.1250      9.0      9.0      0.0      9.0      0.0      0.0
     0.0620      9.0      9.0      0.0      9.0      0.0      0.0
     0.0320      9.0      9.0      0.0      9.0      0.0      0.0533      0.2500      9.0      9.0      9.0      9.0      4.0      8.0
     0.1250      9.0      4.0      3.0      9.0      0.0      5.0
     0.0620      9.0      3.0      0.0      9.0      0.0      4.5
     0.0320      7.5      2.0      0.0      9.0      0.0      3.0534      0.2500      9.0      9.0      0.0      9.0      0.0      4.5
     0.1250      9.0      3.0      0.0      9.0      0.0      4.0
     0.0620      4.5      3.0      0.0      9.0      0.0      4.0
     0.0320      3.5      0.0      0.0      4.0      0.0      2.0535      0.2500      4.0      9.0      5.0      9.0      3.0      9.0
     0.1250      3.0      9.0      5.0      9.0      3.0      4.0
     0.0620      3.0      6.0      3.0      9.0      0.0      3.0
     0.0320      0.0      0.0      0.0      6.0      0.0      0.0536      0.2500      9.0      4.0      0.0      9.0      0.0      4.0
     0.1250      5.0      0.0      0.0      9.0      0.0      1.0
     0.0620      4.0      0.0      0.0      9.0      0.0      0.0
     0.0320      3.0      0.0      0.0      9.0      0.0      0.0
                                       表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T537     0.5000      9.0      9.0      0.0      9.0      0.0      0.0
    0.2500      9.0      4.0      0.0      9.0      0.0      0.0
    0.1250      5.0      1.0      0.0      9.0      0.0      0.0
    0.0620      4.4      0.0      0.0      9.0      0.0      0.0
    0.0320      3.4      0.0      0.0      9.0      0.0      0.0538     0.5000      9.0      9.0      0.0      9.0      0.0      1.0
    0.2500      9.0      0.0      0.0      9.0      0.0      1.0
    0.1250      4.7      0.0      0.0      9.0      0.0      1.0
    0.0620      3.4      0.0      0.0      9.0      0.0      0.0
    0.0320      2.1      0.0      0.0      9.0      0.0      0.0539     0.5000      9.0      9.0      2.0      9.0      9.0      5.0
    0.2500      7.0      8.0      0.0      9.0      4.0      1.0
    0.1250      4.7      6.0      0.0      9.0      1.0      1.0
    0.0620      3.0      2.0      0.0      9.0      0.0      1.0
    0.0320      2.1      0.0      0.0      8.0      0.0      0.0540     0.5000      9.0      9.0      3.0      9.0      0.0      3.0
    0.2500      9.0      9.0      0.0      9.0      0.0      1.0
    0.1250      4.7      9.0      0.0      9.0      0.0      0.0
    0.0620      3.4      8.0      0.0      9.0      0.0      0.0
    0.0320      2.3      6.0      0.0      8.0      0.0      0.0541     0.5000      6.0      9.0      0.0      9.0      0.0      2.0
    0.2500      4.0      6.0      0.0      9.0      0.0      0.0
    0.1250      0.0      4.0      0.0      9.0      0.0      0.0
    0.0620      0.0      3.0      0.0      9.0      0.0      0.0542     0.5000      9.0      9.0      0.0      9.0      9.0      2.0
    0.2500      8.0      4.0               9.0      0.0      0.0
    0.1250      4.3      2.0      0.0      9.0      0.0      0.0
    0.0620      2.7      0.0      0.0      9.0      0.0      0.0
    0.0320      1.7      0.0      0.0      7.0      0.0      0.0
                                  表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T543       0.5000      9.0      3.0      0.0      9.0      0.0      2.0
      0.2500      7.0      8.0      0.0      9.0      0.0      2.0
      0.1250      4.0      7.0      0.0      9.0      0.0      1.0
      0.0620      2.9      6.0      0.0      9.0      0.0      0.0
      0.0320      2.1      2.0      0.0      9.0      0.0      0.0544       0.5000      9.0      9.0      4.0      9.0      9.0      8.0
      0.2500      9.0      9.0      9.0      9.0      9.0      9.0
      0.1250      6.4      9.0      7.0      9.0      8.0      9.0
      0.0620      5.6      9.0               9.0      4.0      9.0
      0.0320      5.4      9.0      9.0      9.0      7.0      4.0545       0.5000      9.0      9.0      6.0      9.0      9.0      9.0
      0.2500      9.0      7.0      9.0      9.0      7.0      9.0
      0.1250      7.0      6.0      9.0      9.0      4.0      4.0
      0.0620      6.6      5.0      0.0      7.0      0.0      2.0
      0.0320      5.6      4.0      0.0      6.0      0.0      2.0546       0.5000      9.0      2.0      0.0      9.0      9.0      6.0
      0.2500      9.0      9.0      9.0      9.0      9.0      7.0
      0.1250      4.6      6.0      9.0      7.0      4.0      4.0
      0.0620      4.3      4.0      0.0      7.0      0.0      3.0
      0.0320      4.1      3.0      0.0      6.0      0.0      2.0547       0.5000      9.0      9.0      0.0      9.0      3.0      3.0
      0.2500      9.0      9.0      7.0      9.0      7.0      4.0
      0.1250      5.6      9.0      8.0      9.0      4.0      4.0
      0.0620      5.4      7.0      8.0      9.0      4.0      3.0
      0.0320      5.4      7.0      6.0      9.0      2.0      2.0548       0.5000      6.0      0.0      9.0      9.0      0.0      4.0
      0.2500      9.0      9.0      9.0      9.0      4.0      6.0
      0.1250      4.9      8.0      9.0      9.0      2.0      4.0
      0.0620      3.7      6.0      9.0      9.0      0.0      2.0
      0.0320      2.9      2.0               8.0      0.0      3.0
                                      表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T549       0.5000      9.0      9.0      9.0      9.0      0.0      2.0
      0.2500      9.0      9.0      9.0      9.0      4.0      4.0
      0.1250      5.1      9.0      2.0      9.0      4.0      4.0
      0.0620      3.6      9.0      0.0      9.0      0.0      4.0
      0.0320      3.0      7.0      0.0      9.0      0.0      4.0550       0.5000      9.0      5.0      9.0      9.0      0.0      0.0
      0.2500      9.0      7.0      0.0      9.0      0.0      0.0
      0.1250      5.9      8.0      0.0      9.0      0.0      0.0
      0.0620      5.9      8.0      0.0      9.0      0.0      0.0
      0.0320      4.7      2.0      0.0      9.0      0.0      0.0551       0.5000      9.0      9.0      0.0      9.0      2.0      4.0
      0.2500      7.0      2.0      0.0      9.0      0.0      3.0
      0.1250      7.0      0.0      0.0      9.0      0.0      3.0
      0.0620      4.0      0.0      0.0      0.0      0.0      0.0552       0.5000      9.0      9.0      9.0      9.0      5.0      4.0
      0.2500      9.0      9.0      9.0      9.0      0.0      7.0
      0.1250      4.7      7.0      4.0      9.0      0.0      6.0
      0.0620      3.7      8.0               8.0      0.0      6.0
      0.0320      2.6      6.0      0.0      6.0      0.0      4.0553       0.5000      7.0      4.0      9.0      9.0      0.0      4.0
      0.2500      9.0      9.0      2.0      9.0      0.0      6.0
      0.1250      6.4      7.0               9.0      0.0      4.0
      0.0620      2.1      6.0      0.0      9.0      0.0      4.0
      0.0320      1.3      2.0      0.0      7.0      0.0      3.0554       0.5000      7.0      5.0      9.0      9.0      0.0      6.0
      0.2500      9.0      9.0      9.0      9.0      9.0      7.0
      0.1250      5.7      9.0      4.0      9.0      0.0      6.0
      0.0620      4.1      7.0      0.0      9.0      0.0      4.0
      0.0320      3.0      2.0      0.0      9.0      0.0      4.0
                                   表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物     施用率      R        I        S        V        P        A编号    (公斤/公顷)    C        R        E        A        Y        T555       0.5000      9.0      3.0      9.0      9.0      0.0      3.0
      0.2500      9.0      9.0      8.0      9.0      7.0      9.0
      0.1250      4.6      9.0      8.0      9.0      2.0      8.0
      0.0620      2.3      6.0      6.0      9.0      0.0      6.0
      0.0320      1.6      4.0      4.0      9.0      0.0      6.0556       0.5000      9.0      3.0      0.0      9.0      3.0      5.0
      0.2500      9.0      9.0      9.0      9.0      4.0      9.0
      0.1250      4.4      7.0      9.0      9.0      6.0      8.0
      0.0620      3.6      2.0      2.0      9.0      0.0      7.0
      0.0320      2.9      0.0      2.0      9.0      0.0      4.0557       0.5000      9.0      9.0      5.0      9.0      4.0      9.0
      0.2500      9.0      9.0      9.0      9.0      4.0      9.0
      0.1250      6.3      9.0      6.0      9.0      2.0      8.0
      0.0620      5.1      8.0               9.0      0.0      8.0
      0.0320      4.3      4.0      0.0      9.0      0.0      6.0558       0.5000      9.0      9.0      9.0      9.0      4.0      9.0
      0.2500      9.0      9.0      9.0      9.0      8.0      9.0
      0.1250      7.0      8.0      9.0      9.0      4.0      9.0
      0.0620      4.7      6.0               9.0      2.0      7.0
      0.0320      4.3      2.0               9.0      2.0      4.0559       0.5000      9.0      4.0      9.0      9.0      0.0      2.0
      0.2500      6.0      0.0      9.0      9.0      0.0      2.0
      0.1250      3.0      0.0      0.0      9.0      0.0      1.0
      0.0620      3.0      0.0      0.0      9.0      0.0      1.0560       0.5000      7.0      3.0      9.0      9.0      0.0      2.0
      0.2500      9.0      9.0      9.0      9.0      0.0      4.0
      0.1250      4.6      7.0      7.0      9.0      0.0      2.0
      0.0620      3.0      2.0      2.0      9.0      0.0      3.0
      0.0320      2.0      0.0      0.0      8.0      0.0      3.0
                               表III(续)
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号   (公斤/公顷)   C        R        E        A        Y        T561       0.5000    9.0      6.0      9.0      9.0      0.0      2.0
      0.2500    9.0      9.0      0.0      9.0      3.0      4.5
      0.1250    6.4      8.5      0.0      9.0      1.0      3.5
      0.0620    4.8      6.0      0.0      9.0      0.0      4.0
      0.0320    3.6      3.0      0.0      9.0      0.0      2.5562       0.5000    9.0      3.0      9.0      9.0      0.0      6.0
      0.2500    9.0      9.0      9.0      9.0      7.0      9.0
      0.1250    5.1      9.0      9.0      9.0      5.0      4.0
      0.0620    5.1      7.0      4.0      9.0      0.0      3.0
      0.0320    2.7      2.0               9.0      0.0      2.0563       0.5000    9.0      9.0      0.0      9.0      4.0      4.0
      0.2500    9.0      6.0      4.0      9.0      2.0      7.0
      0.1250    5.6      6.0      0.0      9.0      0.0      7.0
      0.0620    5.1      2.0      0.0      9.0      0.0      7.0
      0.0320    3.6      0.0      0.0      8.0      0.0      4.0564       0.2500    7.0      9.0      4.0      9.0      0.0      0.0
      0.1250    5.0      7.0      0.0      9.0      0.0      0.0
      0.0620    4.0      6.0      0.0      9.0      0.0      0.0
      0.0320    4.0      6.0      0.0      9.0      0.0      0.0565       0.2500    0.0      6.0      0.0      9.0      0.0      3.0
      0.1250    0.0      6.0      0.0      9.0      0.0      2.0
      0.0620    0.0      3.0      0.0      9.0      0.0      0.0
      0.0320    0.0      0.0      0.0      9.0      0.0      0.0566       0.2500    6.0      9.0      3.0      9.0      9.0      6.0
      0.1250    3.0      0.0      0.0      9.0      0.0      5.0
      0.0620    3.0      0.0      0.0      9.0      0.0      3.0
      0.0320    3.0      0.0      0.0      9.0      0.0      2.0
                                   表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物    施用率      R        I        S        V        P        A编号   (公斤/公顷)    C        R        E        A        Y        T567      0.2500      4.0      9.0      0.0      9.0      0.0      2.0
     0.1250      2.0      4.0      0.0      9.0      0.0      1.0
     0.0620      0.0      9.0      0.0      3.0      0.0      0.0
     0.0320      0.0      4.0      0.0      0.0      0.0      0.0568      0.2500      6.0      7.0      0.0      9.0      0.0      3.0
     0.1250      5.0      5.0      0.0      9.0      0.0      1.0
     0.0620      3.0      0.0      0.0      9.0      0.0      0.0
     0.0320      0.0      0.0      0.0      0.0      0.0      0.0569      0.2500      5.0      0.0      0.0      6.0      9.0      1.0
     0.1250      5.0      0.0      0.0      6.0      0.0      0.0
     0.0620      4.0      0.0      0.0      6.0      0.0      0.0
     0.0320      2.0      0.0      0.0      4.0      0.0      0.0570      0.2500      6.0      9.0      0.0      9.0      0.0      3.0
     0.1250      4.0      0.0      0.0      0.0      0.0      2.0
     0.0620      2.0      0.0      0.0      0.0      0.0      1.0
     0.0320      0.0      0.0      0.0      0.0      0.0      0.0571      0.2500      6.0      9.0      0.0      9.0      0.0      2.0
     0.1250      3.0      3.0      0.0      7.0      0.0      1.0
     0.0620      2.0      3.0      0.0      6.0      0.0      0.0
     0.0320      0.0      0.0      0.0      0.0      0.0      0.0572      0.2500      6.0      5.0      2.0      9.0      3.0      6.0
     0.1250      2.0      2.0      0.0      6.0      0.0      3.0
     0.0620      0.0      0.0      0.0      6.0      0.0      1.0
     0.0320      0.0      0.0      0.0      0.0      0.0      0.0573      0.2500      7.0      5.0      4.0      9.0      2.0      1.0
     0.1250      7.0      5.0      0.0      9.0      0.0      0.0
     0.0620      7.0      3.0      0.0      9.0      0.0      0.0
     0.0320      6.0      0.0      0.0      9.0      0.0      0.0
                                 表III(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T574       0.2500      9.0      7.0      6.5      9.0      6.0      8.0
      0.1250      8.5      6.0      4.5      9.0      2.0      6.5
      0.0620      6.5      5.5      2.0      9.0      1.0      4.5
      0.0320      4.0      2.0      0.0      9.0      0.0      3.0575       0.2500      9.0      6.0      2.0      9.0      3.0      2.0
      0.1250      6.0      4.0      0.0      9.0      0.0      0.0
      0.0620      5.0      0.0      0.0      4.0      0.0      0.0
      0.0320      2.0      0.0      0.0      4.0      0.0      0.0576       0.2500      9.0      5.0      4.0      9.0      4.0      9.0
      0.1250      7.0      3.0      0.0      9.0      3.0      7.0
      0.0620      7.0      3.0      0.0      9.0      0.0      7.0
      0.0320      6.0      0.0      0.0      7.0      0.0      4.0577       0.2500      9.0      9.0      3.0               6.0      9.0
      0.1250      7.0      7.0      3.0               6.0      5.0
      0.0620      7.0      4.0      3.0               6.0      5.0
      0.0320      6.0      2.0      0.0               4.0      4.0578       0.2500      9.0      7.0      9.0               9.0      7.0
      0.1250      7.0      5.0      6.0               6.0      6.0
      0.0620      6.0      5.0      6.0               6.0      5.0
      0.0320      5.0      4.0      3.0               3.0      4.0579       0.2500      5.0      6.0      0.0      9.0      2.0      3.0
      0.1250      4.0      4.0      0.0      7.0      0.0      3.0
      0.0620      4.0      0.0      0.0      7.0      0.0      2.0
      0.0320      2.0      0.0      0.0      6.0      0.0      0.0580       0.2500      9.0      9.0      8.5      9.0      8.5      6.5
      0.1250      9.0      9.0      9.0      9.0      8.0      4.0
      0.0620      9.0      9.0      9.0      9.0      8.0      4.0
      0.0320      8.5      3.0      5.5      4.5      5.5      1.5
                                      表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物   施用率       R        I        S        V        P        A编号  (公斤/公顷)     C        R        E        A        Y        T581      0.2500      9.0      9.0      8.0      9.0      9.0      7.0
     0.1250      9.0      9.0      6.0      9.0      9.0      6.0
     0.0620      8.5      4.5      1.5      4.5      9.0      3.5
     0.0320      6.0      3.0      1.0      4.5      3.0      1.5582      0.2500      9.0      6.0      7.0      7.0      6.0      3.0
     0.1250      7.0      6.0      0.0      7.0      6.0      0.0
     0.0620      7.0      4.0      0.0      7.0      5.0      0.0
     0.0320      6.0      3.0      0.0      7.0      5.0      0.0583      0.2500      9.0      9.0      9.0      9.0      9.0      9.0
     0.1250      9.0      9.0      9.0      9.0      9.0      9.0
     0.0620      7.5      9.0      9.0      9.0      9.0      7.0
     0.0320      3.0      9.0      8.5      6.0      9.0      5.0584      0.2500      9.0      9.0      0.0      9.0      2.0      3.5
     0.1250      9.0      9.0               9.0      4.0      1.0
     0.0620      9.0      6.0      0.0      8.0      1.5      1.0
     0.0320      6.0      1.5      0.0      3.0      0.0      0.0585      0.2500      9.0      9.0      3.0      9.0      2.5      1.5
     0.1250      8.5      9.0      0.0      4.5      2.0      1.5
     0.0620      8.5      8.5      0.0      3.5      1.5      1.5
     0.0320      5.0      2.5      0.0      3.5      0.0      1.0586      0.2500      9.0      9.0      4.5      9.0      0.0      2.0
     0.1250      9.0      9.0      4.5      9.0      0.0      2.0
     0.0620      9.0      8.5      0.0      6.5      0.0      2.0
     0.0320      8.0      8.0      0.0      9.0      0.0      1.0587      0.2500      9.0      9.0               9.0      5.0      5.0
     0.1250      9.0      9.0      0.0      9.0      5.0      4.0
     0.0620      7.0      8.0               5.0      2.0      4.0
     0.0320      7.0      4.0      0.0      5.0      0.0      4.0
                                      表III(续)
                    E                                            O
                    C        C        C        M        S        R
                    H        Y        Y        O        A        Y
                    O        P        P        O        G        S化合物     施用率       R        I        S        V        P        A编号    (公斤/公顷)     C        R        E        A        Y        T588        0.2500      7.0      6.0      5.0      8.0      0.0      3.0
       0.1250      9.0      6.0      5.0      7.0      0.0      3.0
       0.0620      7.0      2.0      0.0               0.0      3.0
       0.0320      4.0      0.0      0.0               0.0      0.0589        0.2500      4.0      4.0               9.0      3.0      0.0
       0.1250      4.0      3.0      0.0      8.0      2.0      0.0
       0.0620      4.0      2.0      0.0      8.0      2.0      0.0
       0.0320      4.0      0.0      0.0      7.0      0.0      0.0590        0.2500      9.0      9.0      5.0      9.0      9.0      6.0
       0.1250      6.0      7.0               7.0      8.0      5.0
       0.0620      5.0      7.0               7.0      4.0      5.0
       0.0320      3.0      2.0      0.0               3.0      3.0591        0.2500      9.0      7.0               9.0      7.0      5.0
       0.1250      7.0      7.0      0.0      9.0      7.0      4.0
       0.0620      3.0      4.0               9.0      3.0      4.0
       0.0320      3.0      3.0      0.0      7.0      0.0      2.0592        0.2500      5.0      6.0               9.0               4.0
       0.1250      4.0      4.0      0.0      9.0      3.0      4.0
       0.0620      3.0      3.0               9.0      3.0      2.0
       0.0320      0.0      2.0      0.0      8.0      0.0      2.0593        0.2500      0.0      5.0      0.0      7.0      0.0      0.0
       0.1250      0.0      4.0      0.0      7.0      0.0      0.0
       0.0620      0.0      3.0               7.0      0.0      0.0
       0.0320      0.0      3.0                        0.0      0.0594        0.2500      7.0      9.0               9.0               3.0
       0.1250      6.0      5.0               9.0      5.0      2.0
       0.0620      5.0      5.0               7.0      4.0      2.0
       0.0320      3.0      3.0      0.0      6.0      2.0      1.0
                                     表III(续)
                  E                                            O
                  C        C        C        M        S        R
                  H        Y        Y        O        A        Y
                  O        P        P        O        G        S化合物    施用率      R        I        S        V        P        A编号   (公斤/公顷)    C        R        E        A        Y        T595      0.2500      4.0      4.0                        0.0      2.0
     0.1250      3.0      2.0      0.0               0.0      0.0
     0.0620      0.0      0.0                        0.0      0.0596      0.2500      7.0      0.0      0.0      9.0      6.0      6.0
     0.1250      5.0      0.0      0.0      7.0      2.0      4.0
     0.0620      4.0      0.0      0.0      4.0      0.0      3.0
     0.0320      0.0      0.0      0.0      3.0      0.0      0.0597      0.2500      9.0      0.0      0.0      4.0      0.0      0.0
     0.1250      7.0      0.0      0.0               0.0      0.0
     0.0620      6.0      0.0      0.0      4.0      0.0      0.0
     0.0320      4.0      0.0      0.0               0.0      0.0598      0.2500      0.0      3.0      0.0      7.0      0.0      3.0
     0.1250      0.0      2.0               7.0      0.0      3.0
     0.0620      0.0      0.0                        0.0      0.0
     0.0320      0.0      0.0      0.0               0.0      0.0599      0.2500      4.0      3.0      0.0      7.0      0.0      5.0
     0.1250      0.0                                 0.0      3.0
     0.0620      0.0      0.0      0.0      7.0      0.0      3.0
     0.0320      0.0      0.0               6.0      0.0      2.0600      0.2500      2.0      2.0      0.0      7.0      0.0      4.0
     0.1250      0.0      0.0               7.0      0.0      4.0
     0.0620      0.0      0.0      0.0      6.0      0.0      3.0
     0.0320      0.0      0.0      0.0      6.0      0.0      3.0601      0.2500      6.0      4.0      3.0      9.0      0.0      7.0
     0.1250      2.0      4.0      0.0      9.0      0.0      6.0
     0.0620      0.0      0.0      0.0      7.0      0.0      5.0
     0.0320      0.0      0.0      0.0      6.0      0.0      4.0
                                表III(续)
                    E                                            O
                    C        C        C        M        S        R
                    H        Y        Y        O        A        Y
                    O        P        P        O        G        S化合物     施用率       R        I        S        V        P        A编号    (公斤/公顷)     C        R        E        A        Y        T602        0.2500      9.0      5.0      9.0      9.0      3.0
       0.1250      9.0      5.0      7.0      8.0      0.0
       0.0620      5.0      3.0      0.0      7.0      0.0
       0.0320      0.0      3.0               7.0      0.0603        0.2500      8.0      7.0      9.0      9.0      4.0
       0.1250      6.0      6.0      8.0      9.0      2.0
       0.0620      4.0                        7.0      0.0
       0.0320      0.0      5.0      0.0      7.0      0.0604        0.2500      9.0      6.0      0.0      8.0      0.0
       0.1250      7.0      4.0      0.0      7.0      0.0
       0.0620      7.0      3.0      0.0      6.0      0.0
       0.0320      7.0      0.0      0.0      5.0      0.0605        0.2500      7.0      7.0      0.0      9.0      7.0
       0.1250      7.0      7.0      0.0      9.0      5.0
       0.0620      4.0      3.0      0.0      9.0      4.0
       0.0320      4.0      1.0      0.0      9.0      4.0606        0.2500      6.0      9.0      2.0      9.0      4.0
       0.1250      5.0      6.0      2.0      7.0      3.0
       0.0620      5.0      6.0      2.0      7.0
       0.0320      5.0      4.0      0.0      6.0      0.0607        0.2500      9.0      5.0      0.0      9.0      3.0      3.0
       0.1250      9.0      5.0      0.0      9.0      0.0      2.0
       0.0620      7.0      2.0      0.0      7.0      0.0      0.0
       0.0320      4.0      0.0               6.0      0.0      0.0
实施例188
在水稻田条件下稻子对移植后施用的耐受性及芽后杂草控制
用水灌注含有3至5公分高的杂草及1.5至2.5叶龄的稻秧苗的塑胶容器。实验期间的水位均保持在土表以上1.5至3公分。试验化合物含在水/丙酮v/v50/50混合物中直接加至灌溉水中，使其相当于约0.0313至0.500公斤/公顷活性成份。经处理的容器置于温室平台上，根据常规温室方法照料。处理3至4周后，结束试验，检查各容器，根据实施例185的分级系统为除草效果分级。结果综述于表IV。所评估的化合物按实施例185所示的化合物编号说明。
                                      表IV
                 E                                            O
                 C        C        C        M        S        R
                 H        Y        Y        O        A        Y
                 O        P        P        O        G        S化合物   施用率      R        I        S        V        P        A编号  (公斤/公顷)    C        R        E        A        Y        T1       0.5000      9.0      9.0      6.5      6.5      3.0      7.0
    0.2500      8.0      9.0      5.5      5.5      1.0      6.0
    0.1250      6.5      9.0      3.0      4.5      0.0      4.0
    0.0625      2.5      4.0      1.0      1.0      0.0      3.0
    0.0313      1.0      0.0      1.0      0.0      0.0      3.02       0.5000      9.0      9.0      0.0      9.0      4.0      8.0
    0.2500      9.0      9.0      0.0      9.0      2.0      7.0
    0.1250      7.0      9.0      0.0      9.0      0.0      3.0
    0.0625      4.0      9.0      0.0      9.0      0.0      2.0
    0.0313      4.0      9.0      0.0      9.0      0.0      2.03       0.5000      4.0      9.0      0.0      9.0      0.0      3.0
    0.2500      2.0      9.0      0.0      9.0      0.0      3.0
    0.1250      0.0      9.0      0.0      9.0      0.0      3.0
    0.0625      0.0      9.0      0.0      9.0      0.0      2.0
    0.0313      0.0      9.0      0.0      9.0      0.0      2.04       0.5000      9.0      9.0      9.0      9.0      9.0      8.0
    0.2500      9.0      9.0      7.0      9.0      9.0      8.0
    0.1250      9.0      9.0      7.0      9.0      6.0      7.0
    0.0625      9.0      9.0      4.0      9.0      2.0      4.0
    0.0313      7.0      8.0      2.0      8.0      3.0      3.05       0.5000      9.0      9.0      0.0      9.0      8.0      8.0
    0.2500      9.0      9.0      0.0      9.0      6.0      6.0
    0.1250      6.0      9.0      0.0      9.0      4.0      4.0
    0.0625      7.0      9.0      0.0      9.0      2.0      2.0
    0.0313      2.0      9.0      0.0      9.0      2.0      2.06       0.5000      9.0      9.0      9.0      9.0      9.0      9.0
    0.2500      9.0      9.0      7.0      9.0      8.0      9.0
    0.1250      9.0      9.0      7.0      9.0      6.0      9.0
    0.0625      7.0      9.0      2.0      9.0      4.0      4.0
    0.0313      4.0      9.0      0.0      9.0      2.0      4.0
                                   表IV(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T7         0.5000      9.0      9.0      8.0      9.0      9.0      8.0
      0.2500      9.0      9.0      9.0      9.0      9.0      7.0
      0.1250      9.0      9.0      9.0      9.0      4.0      7.0
      0.0625      9.0      9.0      6.0      9.0      2.0      7.0
      0.0313      9.0      9.0      2.0      9.0      0.0      7.08         0.5000      9.0      9.0      9.0      9.0      9.0      9.0
      0.2500      9.0      9.0      7.0      9.0      9.0      8.0
      0.1250      9.0      9.0      7.0      9.0      4.0      6.0
      0.0625      9.0      9.0      2.0      9.0      4.0      6.0
      0.0313      6.0      9.0      0.0      9.0      2.0      4.09         0.5000      9.0      9.0      9.0      9.0      9.0      9.0
      0.2500      9.0      9.0      7.0      9.0      9.0      9.0
      0.1250      9.0      9.0      2.0      9.0      2.0      7.0
      0.0625      4.0      9.0      0.0      9.0      0.0      6.0
      0.0313      0.0      9.0      0.0      9.0      0.0      4.010        0.5000      9.0      9.0      7.0      9.0      4.0      4.0
      0.2500      9.0      9.0      6.0      9.0      4.0      3.0
      0.1250      9.0      9.0      2.0      9.0      4.0      4.0
      0.0625      9.0      9.0      0.0      9.0      2.0      2.0
      0.0313      7.0      9.0      0.0      9.0      2.0      2.011        0.5000      7.0      9.0      0.0      9.0      7.0      1.0
      0.2500      4.0      9.0      0.0      9.0      4.0      1.0
      0.1250      2.0      9.0      0.0      9.0      0.0      0.0
      0.0625      0.0      9.0      0.0      9.0      0.0      0.0
      0.0313      0.0      8.0      0.0      9.0      0.0      0.012        0.5000      9.0      9.0      2.0      9.0      9.0      7.0
      0.2500      9.0      9.0               9.0      4.0      7.0
      0.1250      6.0      9.0               9.0      0.0      7.0
      0.0625      2.0      9.0      0.0      9.0      0.0      4.0
      0.0313      0.0      9.0      0.0      9.0      0.0      4.0
                                       表IV(续)
                    E                                            O
                    C        C        C        M        S        R
                    H        Y        Y        O        A        Y
                    O        P        P        O        G        S化合物     施用率       R        I        S        V        P        A编号    (公斤/公顷)     C        R        E        A        Y        T13        0.5000       9.0      9.0      2.0      9.0      9.0      7.0
      0.2500       8.0      9.0      4.0      9.0      2.0      4.0
      0.1250       6.0      9.0      2.0      9.0      2.0      4.0
      0.0625       2.0      9.0      0.0      9.0      0.0      2.0
      0.0313       0.0      9.0      0.0      9.0      0.0      2.049        0.2500       9.0      6.0      0.0      9.0      0.0      0.0
      0.1250       9.0      4.0      0.0      9.0      0.0      0.050        0.2500       9.0      9.0      0.0      9.0      0.0      0.0
      0.1250       9.0      9.0      0.0      9.0      0.0      0.063        0.5000       4.0               0.0      9.0      0.0      0.0
      0.2500       2.0               0.0      9.0      0.0      0.0
      0.1250       0.0               0.0      2.0      0.0      0.0261       0.2500       0.0      6.0      0.0      9.0      0.0      0.0
      0.1250       0.0      6.0      0.0      9.0      0.0      0.0
      0.0620       0.0      6.0      0.0      9.0      0.0      0.0
      0.0320       0.0      5.0      0.0      9.0      0.0      0.0267       0.2500       9.0      9.0      0.0      9.0      0.0      7.0
      0.1250       9.0      9.0      0.0      9.0      0.0      6.0
      0.0620       8.0      9.0      0.0      9.0      0.0      5.0
      0.0320       4.0      9.0      0.0      9.0      0.0      2.0327       0.2500       9.0      9.0      2.0      9.0      4.0      4.0
      0.1250       9.0      9.0      0.0      9.0      4.0      5.0
      0.0620       7.0      9.0      0.0      9.0      0.0      3.0
      0.0320       9.0      9.0      0.0      9.0      0.0      2.0328       0.2500       9.0      9.0      6.0      9.0      6.0      4.0
      0.1250       9.0      9.0      6.0      9.0      2.0      4.0
      0.0620       9.0      9.0      2.0      9.0      0.0      4.0
      0.0320       7.0      9.0      0.0      9.0      0.0      2.0
                                    表IV(续)
                   E                                            O
                   C        C        C        M        S        R
                   H        Y        Y        O        A        Y
                   O        P        P        O        G        S化合物    施用率       R        I        S        V        P        A编号   (公斤/公顷)     C        R        E        A        Y        T333       0.2500      9.0      9.0      8.0      9.0      4.0      6.0
      0.1250      9.0      9.0      4.0      9.0      4.0      6.0
      0.0620      9.0      9.0      2.0      9.0      2.0      5.0
      0.0320      9.0      9.0      0.0      9.0      0.0      4.0354       0.1250      9.0      9.0      9.0      9.0      9.0      6.0
      0.0620      7.0      9.0      2.0      9.0      2.0      6.0
      0.0320      4.0               1.0      6.0      0.0359       0.1250      6.0      9.0      0.0      9.0      0.0      4.0
      0.0620      6.0      7.0      0.0      7.0      0.0      3.0
      0.0320      2.0      4.0      0.0      7.0      0.0      2.0362       0.2500      9.0      4.0      9.0      9.0      8.0      6.0
      0.1250      7.0      8.0      9.0      9.0      4.0      3.0
      0.0620      2.0      7.0      9.0      9.0      0.0      3.0
      0.0320      0.0      4.0      0.0      9.0      0.0      3.0378       0.1250      9.0      9.0      9.0      9.0      9.0      9.0
      0.0620      9.0      9.0      9.0      9.0      9.0      8.0
      0.0320      9.0      9.0      9.0      9.0      9.0      8.0380       0.2500      9.0      9.0      8.0      9.0      8.0      7.0
      0.1250      9.0      9.0      2.0      9.0      2.0      7.0
      0.0620      8.0      9.0      2.0      9.0      0.0      7.0
      0.0320      7.0      9.0      0.0      9.0      0.0      3.0429       0.2500      9.0      9.0      0.0      7.0      0.0      2.0
      0.1250      6.0      7.0      0.0      7.0      0.0      2.0
      0.0620      6.0      6.0      0.0      4.0      0.0      1.0
      0.0320      4.0      4.0      0.0      2.0      0.0      1.0432       0.2500      9.0      9.0      9.0      9.0      4.0      7.0
      0.1250      9.0      9.0      7.0      9.0      2.0      7.0
      0.0620      9.0      8.0      4.0      9.0      0.0      4.0
      0.0320      9.0      8.0      0.0      9.0      0.0      4.0
                                      表IV(续)
                    E                                            O
                    C        C        C        M        S        R
                    H        Y        Y        O        A        Y
                    O        P        P        O        G        S化合物     施用率       R        I        S        V        P        A编号    (公斤/公顷)     C        R        E        A        Y        T431        0.2500      9.0      9.0      4.0      9.0      4.0      7.0
       0.1250      9.0      9.0      0.0      9.0      0.0      3.0
       0.0620      9.0      7.0      0.0      9.0      0.0      3.0
       0.0320      7.0      4.0      0.0      6.0      0.0      3.0445        0.2500      9.0      9.0      4.0      9.0      9.0      7.0
       0.1250      9.0      9.0      4.0      2.0      4.0      7.0
       0.0620      7.0      7.0      2.0      0.0      0.0      6.0
       0.0320      4.0      4.0      0.0      0.0      0.0      3.0448        0.2500      2.0      9.0      0.0      4.0      0.0      2.0
       0.1250      1.0      7.0      0.0      1.0      0.0      1.0
       0.0620      0.0               0.0      0.0      0.0      0.0517        0.2500      0.0      9.0      0.0      9.0      0.0      0.0
       0.1250      0.0      9.0      0.0      9.0      0.0      0.0
       0.0620      0.0      5.0      0.0      9.0      0.0      0.0
       0.0320      0.0      3.0      0.0      9.0      0.0      0.0528        0.2500      9.0      6.0      9.0      9.0      3.0      3.0
       0.1250      9.0      6.0      0.0      9.0      0.0      2.0
       0.0620      7.0      6.0      0.0      0.0      0.0      0.0
       0.0320      0.0      6.0      0.0      0.0      0.0      0.0
实施例189
对照除草性评估法
将本发明某些化合物的芽前及芽后除草性质与美国专利5,484,763及5,523,278所揭示的某些化合物比较。按照实施例185及186所述方法评估。结果如表V与VI所示。表V与VI中的数据用本发明实施例185的化合物编号或美国专利5,484,763及5,523,278所揭示化合物的对照化合物字母表示。
由表V与VI的数据可见，本发明化合物是比美国专利5,484,763及5,523,278所揭示的化合物更有效的除草剂。比较化合物字母                               YA                                        
Figure A9880989807262
B                                            CH3C                                            H
                                             表V
                                       芽前对比评估
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物     施用率     T      E      O      A     A       H      S      C      V      A      M      A      W      M编号    (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X4          0.5000    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    7.0    7.0    7.0
       0.2500    9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           7.0    7.0    7.0    7.0
       0.1250    9.0    9.0    6.0    9.0    6.0           7.0    9.0    9.0           9.0    7.0    7.0    7.0
       0.0625    9.0    7.0    7.0    9.0    9.0           4.0    9.0    9.0           9.0    7.0    5.0    7.0
       0.0313    9.0    7.0    7.0    9.0    9.0           2.0    9.0    9.0           3.0    7.0    2.0    3.0A          0.5000    7.0    5.0    2.0    9.0    9.0           2.0    0.0    3.0    0.0           3.0           0.0
       0.2500    6.0    6.0    2.0    7.0    9.0           0.0    0.0    2.0    0.0           3.0           0.0
       0.1250    5.0    3.5    1.5    5.0    7.0           0.0    0.0    2.5    0.0           0.5    0.0    0.0
       0.0625    0.0    2.0    0.0    2.5    4.5           0.0    0.0    0.0    0.0           0.5    0.0    0.0
       0.0320    0.0    0.0    0.0    5.5                  0.0    0.0    0.0           0.0    0.0    0.0    0.0
       0.0313    0.0    1.5    0.0    2.5    5.5           0.0    0.0    0.0    0.0           0.5    0.0    0.0
       0.0160    0.0    0.0    0.0    2.0                  0.0    0.0    0.0           0.0    0.0    0.0    0.0
                                        表V(续)
                                      芽前对比评估
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X6        0.5000     9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    9.0    9.0    9.0
     0.2500     9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    8.0    8.0    9.0
     0.1250     9.0    7.0    6.5    9.0    9.0    3.0    9.0    6.0    9.0    0.0    7.0    8.0    8.7    6.5
     0.0630     9.0    9.0    7.0    9.0    9.0    9.0           9.0    9.0    7.0           7.0    7.0    8.0
     0.0625     9.0    6.0    5.5    9.0    9.0    3.0    7.0    5.5    6.0    0.0    4.0    7.0    8.3    6.0
     0.0320     9.0    7.4    6.0    9.0    5.3    4.0    7.5    5.6    8.4    2.3    2.0    4.4    5.6    4.2
     0.0315     9.0    9.0    9.0    9.0    8.5    7.5           8.0    9.0    7.0           7.0    6.5    7.5
     0.0313     4.5    4.5    4.5    8.0    9.0    0.0    7.0    4.5    5.5    0.0    2.0    7.0    6.3    5.3
     0.0160     8.0    6.4    4.4    8.8    4.8    1.0    7.5    2.2    7.0    1.3    2.0    2.8    3.0    3.6
     0.0158     9.0    8.0    6.5    9.0    8.5    5.5           6.0    9.0    1.5           4.0    3.5    6.0
     0.0157     3.0    0.0    0.0    5.0           0.0           0.0    0.0    0.0                  3.5    2.3B        0.5000     5.0    8.0    0.0    9.0    7.0           5.0    5.0    4.0    1.0           4.0           1.0
     0.2500     2.0    3.0    0.0    9.0    9.0           2.0    5.0    6.0    1.0           2.0           0.0
     0.1250            2.0    0.0    9.0    5.0           0.0    3.0    2.0    0.0           2.0           0.0
     0.0625     3.0    0.0    0.0    6.0    0.0           0.0    0.0    0.0    0.0           0.0           0.0
     0.0313     0.0    0.0    0.0    9.0    0.0           0.0    0.0    0.0    0.0           0.0           0.0
                                        表V(续)
                                     芽前对比评估
                                                                                     G             O       T
                   A       A       C       C      G      I      I      E      S      L      G      R       R       Z
                   B       M       A       H      A      P      P      C      E      X      L      Y       Z       E
                   U       B       S       E      L      O      O      H      T      M      X      S       A       A化合物    施用率       T       E       O       A      A      H      S      C      V      A      M      A       W       M编号   (公斤/公顷)     H       L       B       L      P      E      S      G      I      W      A      T       R       X35        0.2500      9.0     9.0     9.0     9.0    9.0    9.0           9.0    9.0    9.0           6.0     8.0     8.0
      0.1250      9.0     9.0     9.0     9.0    9.0    9.0           9.0    9.0    9.0           8.0     9.0     8.0
      0.0625      9.0     9.0     9.0     9.0    8.0    7.0           9.0    9.0    7.0           7.0     7.0     8.0
      0.0313      9.0     9.0     7.0     9.0    7.0    6.0           7.0    9.0    5.0           6.0     6.0     7.0
      0.0156      9.0     8.0     6.0     9.0    7.0    4.0           6.0    7.0    1.0           3.0     3.0     5.0C         0.5000      9.0     6.0     5.5     7.0    7.5           2.0    6.0    5.0    0.0           4.0             0.0
      0.2500      9.0     2.0     0.0     3.0    6.0           0.0    4.0    4.0    0.0           4.0             0.0
      0.1250      4.0     2.0     0.0     5.0    2.0           0.0    2.0    2.0    0.0           2.0             0.0
      0.0625      2.0     3.0     0.0     4.0    2.0           0.0    0.0    0.0    0.0           2.0             0.0
      0.0313      0.0     3.0     1.0     3.0                  0.0    0.0    0.0    0.0           1.0             0.0
                                                        表VI
                                                     芽前对比评估
                                                                                  G             O      T
                   A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                   B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                   U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率       T      E      O      A      A      H      S      C      V      A      M      A      W      M编号    (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X4          0.5000     9.0    9.0    9.0    9.0    9.0           9.0    9.0    9.0           9.0    4.0    4.0    3.0
       0.2500     9.0    9.0    9.0    9.0    9.0           9.0    8.0    9.0           9.0    3.0    3.0    3.0
       0.1250     9.0    9.0    9.0    9.0    9.0           9.0    8.0    9.0           7.0    3.0    3.0    3.0
       0.0625     9.0    9.0    9.0    9.0    9.0           9.0    7.0    9.0           4.0    2.0    3.0    3.0
       0.0313     9.0    7.0    7.0    9.0    9.0           7.0    5.0    9.0           5.0    2.0    2.0    2.0
       0.0157     9.0    9.0    7.0    9.0    4.0                  2.0    8.0           6.0    2.0    2.0    2.0A          0.5000     9.0    9.0    9.0    9.0    9.0           9.0    2.0    2.0    4.5           4.5           4.0
       0.2500     9.0    9.0    9.0    9.0    8.3           9.0    2.7    2.7    4.6           3.6           3.8
       0.1250     9.0    7.0    8.9    7.9    6.4    7.5    8.4    1.8    3.0    4.6           2.9    4.3    4.2
       0.0625     8.6    6.9    7.9    7.1    5.4    6.0    7.5    1.0    2.1    4.6           2.6    4.0    3.7
       0.0320     9.0    9.0    0.0    9.0    8.5           9.0    1.0    1.0           4.3    2.3    3.8    4.0
       0.0313     7.8    5.6    6.9    6.3    4.2    5.7    6.8    0.6    1.6    4.0           2.1    3.8    3.4
       0.0160     3.0    7.0    0.0    9.0    5.5           5.5    1.0    1.0           3.5    2.0    2.8    3.8
       0.0157     7.0    6.0    7.6    5.8    3.8    5.0    5.0    0.5    1.2    4.0           2.0    3.5    3.1
                                       表VI(续)
                                     芽前对比评估
                                                                                G             O      T
                 A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                 B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                 U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率     T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)   H      L      B      L      P      E      S      G      I      W      A      T      R      X6         0.5000    9.0    9.0    7.0    9.0    9.0           9.0    7.0    9.0           7.0    5.0    6.0    3.0
      0.2500    9.0    9.0    8.0    9.0    9.0           9.0    6.0    9.0    7.0    6.0    5.0    5.0    3.5
      0.1250    9.0    9.0    7.0    9.0    9.0           9.0    7.0    9.0    7.0    6.0    4.5    2.5    3.5
      0.0640    9.0    9.0           9.0    9.0    9.0           3.0    7.0    6.0           1.0    3.0    5.0
      0.0630    9.0    6.5    2.5    7.0    5.0    5.0           1.5    2.0    4.8           1.8    1.5    4.5
      0.0625    9.0    9.0    4.0    9.0    9.0           9.0    2.0    9.0    7.0    4.0    1.5    2.0    3.5
      0.0320    9.0    9.0    2.3    6.5    3.0    9.0    9.0    1.0    6.0    5.5    5.0    1.5    2.5    3.8
      0.0315    9.0    6.0    1.5    5.0    3.0    4.0           1.0    2.5    3.8           1.0    0.8    4.3
      0.0313    9.0    8.0    0.0    9.0    9.0           8.0    2.0    7.0    7.0    4.0    1.5    1.5    3.5
      0.0160    5.7    7.7    0.0    3.0    2.7    6.0    7.5    0.7    3.7    5.5    2.5    1.5    2.0    3.5
      0.0158    5.0    3.0    0.0    0.0    0.0    2.5           0.0    0.0    3.0           0.5    0.0    4.0
      0.0157    8.0    7.0    0.0    9.0    4.0           7.0    2.0    7.0           4.0    2.0    2.0    2.0B         0.5000    9.0    9.0    9.0    9.0    8.0           9.0    6.0    5.0    7.5           6.0           5.5
      0.2500    9.0    9.0    9.0    8.0    8.0           8.0    5.0    5.0    7.0           5.5           6.0
      0.1250    9.0    8.0    8.0    9.0    7.0           8.0    4.0    4.0    6.0           4.5           5.5
      0.0625    9.0    8.0    8.0    7.0    7.0           8.0    2.0    2.0    5.5           4.5           5.0
      0.0313    8.0    6.0    7.0    7.0    7.0           7.0    2.0    0.0    5.5           4.0           5.5
      0.0157    8.0    2.0    6.0    3.0    5.0           6.0    0.0    0.0    5.5           3.5           5.0
                                             表VI(续)
                                           芽前对比评估
                                                                                 G             O      T
                  A      A      C      C      G      I      I      E      S      L      G      R      R      Z
                  B      M      A      H      A      P      P      C      E      X      L      Y      Z      E
                  U      B      S      E      L      O      O      H      T      M      X      S      A      A化合物    施用率      T      E      O      A      A      H      S      C      V      A      M      A      W      M编号   (公斤/公顷)    H      L      B      L      P      E      S      G      I      W      A      T      R      X35        0.0315     9.0    9.0    5.0    9.0           4.0           2.0    2.0    4.0           1.0    1.5    5.0
      0.0158     9.0    5.0    2.0    9.0    2.0    3.0           1.0    2.0    3.5           0.5    1.0    4.5C         0.5000     9.0    9.0    9.0    5.0    9.0           7.0    0.0    2.0    4.5           4.5           3.0
      0.2500     9.0    7.0    7.0    4.0    6.0           6.0    0.0    0.0    2.5           3.0           2.5
      0.1250     9.0    8.0    7.0    3.0    6.0           7.0    0.0    0.0    2.0           2.5           1.5
      0.0625     9.0    7.0    7.0    3.0    5.0           5.0    0.0    0.0    3.0           2.5           1.5
      0.0313     9.0    6.0    8.0    3.0    3.0           6.0    0.0    0.0    1.5           2.0           2.0
      0.0157     8.0    6.0    3.0    0.0    2.0           2.0    0.0    0.0    1.0           2.0           1.5

Claims (33)

1.一种化合物，它具有如下结构：
Figure A9880989800021
其中
R为C1-C6烷基、C1-C6卤代烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR4或NR5R6；
R1与R2分别为氢、卤素、C1-C6烷基、C3-C7环烷基、C1-C6卤代烷基、C3-C6烯基、C3-C6卤代烯基、C3-C6炔基、OR7、S(O)nR8或NR9R10，当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它任选地穿插氧、硫或氮，且任选地被一至三个甲基或一个或多个卤原子取代；
R3为卤素或A2R11；
X为氢、卤素或C1-C4烷基；
X1为氢、卤素、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素、氰基、R12、X2R12、X3R12、X2X3R12或X3X2R12；
X2为O、S(O)p或NR13；
X3为-C(＝A3)-、-C(＝NOR14)-或-C(＝N-NR13R50)；
R4、R5、R6、R7、R8、R9、R10、R11与R14分别为氢、C1-C6烷基、C3-C7环烷基、C2-C8烷氧基烷基、C2-C6烯基、C2-C6炔基或苄基；
R12为氢，
C1-C8烷基、C3-C7环烷基、C2-C8烯基、C5-C6环烯基或C2-C8炔基，其中各基团任选地被下列任何组合取代：1至6个卤原子、1至3个C1-C20烷氧基，它任选地被一个C1-C6烷氧基、苄氧基或C1-C6烷硫基取代、1或2个C1-C10卤代烷氧基、1或2个NR15R16基团、1至3个S(O)qR17基团、1或2个氰基、1或2个C3-C7环烷基、1个硫氰基、1个O(SO2)R17基团、1个O(NO2)基团、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)SR19基团、1或2个C(O)NR20R21基团、1至3个X4R22基团、1或2个P(O)(OR23)2基团、1或2个Si(R24)3基团、
1个4至10元单环或稠合双环杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1或2个苯基，其中各苯基分别任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C3-C7环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，或
茚满基，它任选地被下列任何组合取代：1或2个卤原子、1或2个C1-C4烷基、1个C1-C4烷氧基、1个或C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基、或X4R22基团；
R13为氢、C1-C8烷氧基烷基、C1-C6烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基、SO2R51或1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基，且当R13及R12及其所连接的氮原子结合在一起时，形成了5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢、Si(R31)3、C(O)NR35R36、C(O)R33、SO2R47、
C1-C20烷基，它被下列基团取代：一个羟基、苄氧基、硝基、OC(O)R33、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、P(O)(OH)NH2、P(O)(OH)(OR23)、C(O)NR35OR23、氰基或2-二氧戊环基，
1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、或C1-C4卤代烷磺酰基，
C3-C20烯基，它任选地被下列基团取代：1至3个卤原子、1个羟基、1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它任选地被下列基团取代：一个羟基、C1-C6烷氧基、C1-C4烷基、C2-C4烯基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个羟基、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，
苄基，其苯环上任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团，或
4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢、
C1-C6烷基、C3-C7环烷基、C2-C6烯基或C2-C6炔基，其中各基团任选地被一个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个CO2R26基团，
C(O)R43，或
CO2R42；
R16与R21分别为氢、C1-C6烷基、C1-C4烷氧基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17、R18、R25、R30、R33、R45及R51分别为NR46R48、-N＝CR46R48、任选地被一个C1-C6烷氧基、噻吩或呋喃基取代的C1-C8烷基、C1-C6卤代烷基、C3-C8环烷基、CO2R23、任选地被苯基取代的C2-C6烯基，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团，或
5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R19与R26分别为氢、C1-C20烷基、C1-C8卤代烷基、C3-C7环烷基、C3-C7卤代环烷基、C3-C20烯基、C3-C8卤代烯基、C5-C8环烯基、C5-C8卤代环烯基、C3-C8炔基、C3-C8卤代炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、C1-C6硫烷基、C2-C20烷氧烷氧基、苯基、OSi(R47)3、OC(O)R33、C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
2-、3或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基、C3-C8环烷基、二噁烷或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R34、R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢、氰基、C1-C6烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
m、n、p与q分别为0、1或2的整数；
R29为氢、C1-C4烷基或C1-C4卤代烷基；
R24、R31、R41及R47分别为C1-C4烷基、
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；
R23、R39、R40、R42、R43、R44、R46及R48分别为氢、C2-C6烯基、C3-C8环烷基、
C1-C8烷基，它任选地被一或二个C1-C4烷氧基取代；
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，且
当R46与R48及其所连接的原子结合在一起时，为5至12元单环或稠合双环杂环或环烷基环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；及
A、A1、A2、A3、A4、X4及X5分别为O或S；
及其光学异构体、非对映异构体和/或互变异构体。
2.根据权利要求1所述的化合物，其中
R为C1-C6烷基、C1-C6卤代烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR4或NR5R6；
R1与R2分别为氢、卤素、C1-C6烷基、C3-C7环烷基、C1-C6卤代烷基、C3-C6烯基、C3-C6卤代烯基、C3-C6炔基、OR7、S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它任选地穿插氧、硫或氮，且任选地被一至三个甲基或一个或多个卤原子取代；
R3为卤素或A2R11；
X为氢、卤素或C1-C4烷基；
X1为氢、卤素、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素、氰基、R12、X2R12、X3R12、X2X3R12或X3X2R12；
X2为O、S(O)p或NR13；
X3为-C(＝A3)-或-C(＝NOR14)-；
R4、R5、R6、R7、R8、R9、R10、R11与R14分别为氢、C1-C6烷基、C3-C7环烷基、C2-C6烯基、C2-C6炔基或苄基；
R12为氢，
C1-C6烷基、C3-C7环烷基、C2-C6烯基、C5-C6环烯基或C2-C6炔基，其中各基团任选地被下列任何组合取代：1至6个卤原子、1至3个C1-C20烷氧基、1或2个C1-C10卤代烷氧基、1或2个NR15R16基团、1至3个S(O)qR17基团、1或2个氰基、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)NR20R21基团、1至3个X4R22基团、1或2个P(O)(OR23)2基团、1或2个Si(R24)3基团、
1个4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C3-C7环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
当R12与R13及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基、或X4R22基团；
R13为氢、C1-C6烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基或SO2R51，且当R13及R12与所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢、Si(R31)3、
C1-C20烷基，它被下列基团取代：一个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、P(O)(OH)NH2、P(O)(OH)(OR23)、C(O)NHOR23、氰基或2-二氧戊环基，
1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、或C1-C4卤代烷磺酰基，
C3-C20烯基，它任选地被下列基团取代：1至3个卤原子、1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NHOR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它任选地被下列基团取代：一个C1-C6烷氧基、C1-C4烷基、C2-C4烯基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NHOR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NHOR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基、它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，
苄基、其苯环上任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团，或
4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢、
C1-C6烷基、C3-C7环烷基、C2-C6烯基或C2-C6炔基，其中各基团任选地被一个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
C(O)R43；
R16与R21分别为氢、C1-C6烷基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17、R18、R25、R30、R33、R45及R51分别为C1-C4烷基、C1-C4卤代烷基、CO2R23、C2-C6烯基，它任选地被苯基取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团，或
5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R19与R26分别为氢、C1-C20烷基、C1-C8卤代烷基、C3-C7环烷基、C3-C7卤代环烷基、C3-C20烯基、C3-C8卤代烯基、C5-C8环烯基、C5-C8卤代环烯基、C3-C8炔基、C3-C8卤代炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
2-、3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R34、R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢、氰基、C1-C6烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
m、n、p与q分别为0、1或2的整数；
R29为氢、C1-C4烷基或C1-C4卤代烷基；
R24、R31、R41及R47分别为C1-C4烷基、
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；
R23、R39、R40、R42、R43、R44、R46及R48分别为氢、C1-C4烷基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，且
A、A1、A2、A3、A4、X4及X5分别为O或S；
及其光学异构体、非对映异构体和/或互变异构体。
3.根据权利要求1所述的化合物，它具有下式结构：
Figure A9880989800131
4.根据权利要求3所述的化合物，其中
R为C1-C4烷基、C1-C4卤代烷基、C3-C4烯基、C3-C4炔基或苄基；
R1为卤素或C1-C4卤代烷基；
R2为氢、卤素或C1-C4卤代烷基；
X与X1分别为氢或卤素；
Z为O或S；
Y为氰基、R12、X2R12或X3X2R12；
X2为O、S或NR13；
R12为氢，
C1-C6烷基、C3-C7环烷基、C2-C6烯基、C5-C6环烯基或C2-C6炔基，其中各基团任选地被下列任何组合取代：1至3个卤原子、1或2个C1-C20烷氧基、1或2个C1-C10卤代烷基、1个NR15R16基团、1个S(O)qR17基团、1或2个氰基、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)SR19基团、1或2个C(O)NR20R21基团、1或2个X4R22基团、1个P(O)(OR23)2基团、1个Si(R24)3基团、
1个4至10元单环或稠合双环杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它任选地被下列任何组合取代：1至3个卤原子、1个C1-C6烷基、1个C1-C6烷氧基、1个C3-C7环烷基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，
苯基，它任选地被下列任何组合取代：1或2个卤原子、1至3个C1-C4烷基、1或2个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团；
R13为氢、C2-C6烷氧基烷基、C1-C4烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基或SO2R51；
R14为氢、C1-C6烷基、C3-C7环烷基、C2-C8烷氧基烷基、C2-C6烯基、C2-C6炔基或苄基；
R16与R21分别为氢、C1-C6烷基、C1-C4烷氧基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；且
R32为氢、
Si(R47)3，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、C1-C6硫烷基、C2-C20烷氧烷氧基、苯基、OSi(R47)3、OC(O)R33、C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基、C3-C8环烷基、二噁烷或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子。
5.根据权利要求4所述的化合物，其中
R为C1-C4烷基；
R1为C1-C4卤代烷基；
R2为氢；
Y为R12、OR12、C(O)NR13R12、C(O)R12、CO2R12、C(O)SR12或C(＝NOR14)；
R12为氢、
C1-C6烷基或C2-C6烯基，其中各基团任选地被下列任何组合取代：1至3个卤原子、1或2个C1-C6烷氧基、1个C1-C10卤代烷氧基、1个NR15R16基团、1个S(O)qR17基团、1或2个氰基、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)NR20R21基团、1个X4R22基团、1个P(O)(OR23)2基团、1个OC(O)R33基团、
1个咪唑环，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
1个邻苯二甲酰亚胺环，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
1个四元有机铵基团，或
1个苯基，它任选地被下列任何组合取代：1至3个卤原子、1个C1-C4烷基、1个C1-C4烷氧基或1个X5R27基团，或
苯基，它任选地被下列任何组合取代：1或2个卤原子、1至3个C1-C4烷基、1个C1-C4烷氧基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团或1个N(R29)SO2R30基团；
R13为氢、C1-C6烷氧基烷基、C1-C4烷基、OR23、氰基或SO2R51；
R22与R27分别为氢、C(O)R33、SO2R47、
C1-C4烷基，它被下列基团取代：一个C1-C6烷氧基、CO2R32、C(O)R33、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NHOR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C6烯基，它任选地被1个C1-C6烷氧基、CO2R32、C(O)R33或C(OR34)2基团取代，
C3-C6炔基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1或2个C1-C4烷基、1或2个C1-C4烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，或
苄基、其苯环上任选地被下列任何组合取代：1至3个卤原子、1或2个C1-C4烷基、1或2个C1-C4烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团；
R15为氢、
C1-C4烷基，它任选地被1个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
C(O)R43；
R16为氢、C1-C4烷基、P(O)(OR44)2、SO2R45、C(O)R46、或
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R17、R18、R25、R30、R33、R45及R51分别为NR46R48、C1-C4烷基、C1-C4卤代烷基、
C2-C6烯基，它任选地被苯基取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团；
R19与R26分别为氢、C1-C4烷基、C3-C6烯基、C3-C6炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
C1-C4烷基，它任选地被一个CO2R48、OC(O)R33或C1-C4烷氧基取代，
C1-C4卤代烷基，
C3-C8环烷基，
C3-C8卤代环烷基，
C3-C6烯基，它任选地被一个苯基取代，
C3-C6卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C6炔基，它任选地被一个苯基取代，
C3-C6卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基、或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R35与R49分别为氢或C1-C4烷基，且R36与R50分别为氢、氰基、C1-C4烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
R23为氢或C1-C4烷基；且
A为O。
6.根据权利要求5所述的化合物，其中：
R为甲基；
R1为三氟甲基；
X1为氢；
X为氢或氟；
Y为R12、CO2R12、C(O)R12或C(O)NR13R12；
R12为氢、
C1-C6烷基，它任选地被下列任何组合取代：1至3个卤原子、1个羟基、1或2个C1-C4烷氧基、1个C1-C4卤代烷氧基、1个SO2R17基团、1或2个氰基、1个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)NR20R21基团、1个P(O)(OR23)2基团或1个OC(O)R33基团，
C2-C6烯基，它任选地被下列任何组合取代：1个C(O)R18基团或1个CO2R19基团，
Figure A9880989800181
R13为氢、C1-C4烷基或SO2R51；
R14为氢、C1-C4烷基或苄基；
R18、R23、R56及R57分别为氢或C1-C3烷基；
R52、R53、R54及R55分别为氢、C1-C3烷基、C2-C3烯基、C1-C3烷氧基或卤素，但其限制条件为R52、R53、R54及R55中至少一者为氢；
R19为氢、C1-C4烷基、C3-C6烯基、C3-C6炔基、苄基、吡啶基或碱金属、碱土金属、铵或有机铵阳离子；
R22为氢、C(O)R33、SO2R47；
C1-C4烷基，它任选地被一个氰基取代，
C3-C6烯基，或
C3-C6炔基；
R32为氢、
C1-C4烷基，它任选地被一个CO2R48或C1-C4烷氧基取代，
C1-C4卤代烷基、
C3-C6烯基，它任选地被1个苯基取代，
C3-C6炔基，它任选地被1个苯基取代，
C1-C4烷基，它被1个吡啶基、呋喃基、噻吩基、四氢呋喃基或NR49R50基团取代，或
碱金属、碱土金属、铵或有机铵阳离子；
R35及R49分别为氢或C1-C4烷基；
R36为SO2R51或C1-C3烷氧基；
R17、R33及R51分别为C1-C4烷基、C1-C4卤代烷基、NR46R48、C3-C6环烷基或异噁唑环；
R46与R48分别为氢、C1-C4烷基或苄基；
R47为C1-C4烷基；
R50为C1-C4烷基或
苯基，它任选地分别经1个或多个分别选自下列之基团取代：卤素、氰基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；及
A1为O。
7.根据权利要求6所述的化合物，其中：
Y为C1-C3烷基、CO2R32、卤甲基、氰甲基、C(CH3)2CO2R32、C1-C3烷氧乙基、C1-C3烷氧甲基、羟甲基、CHO、C(O)CH3、CH(CH3)(C1-C4烷氧基)、C(CH3)2CN、CH[O(C1-C3烷基)]2、CH2SO2R17、C(O)NHSO2R51、
Figure A9880989800191
R53、R54、R55及R56分别为氢或甲基，但其限制条件为R53、R54及R55中至少一者为氢；
R22为氰甲基、甲基、乙基、烯丙基、或炔丙基；
R32为氢，
C1-C4烷基，它任选地被1个CO2R48基团取代，
C1-C4卤代烷基，
C3-C6烯基或
C3-C6炔基；且
R35为氢。
8.根据权利要求1所述的化合物，它选自：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-(二甲氨基)乙酯；
2-{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-(对-乙苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}丙酸甲酯；
{{6-{5-[3，6-二氢3-甲基-4(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}乙酸甲酯；
3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-(6-氟-3-甲基-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸乙酯；
1-甲基-3-{3-(6-(2-丙炔氧基)间-甲苯基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-{3-{6-[(1-苯并咪唑羰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-{3-{6-{[(间-氰苯基)氨基甲酰基]甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸烯丙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸3-苯基-2-丙炔酯；
{{2-{5-[3，6-二氢-3-甲基-2，6二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基)-对-甲苯基}氧基}乙酸1-甲基-2-丙炔酯；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸2-氯乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2，2，2-三氟乙酯；
3-[3-(2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)2，4(1H，3H)-嘧啶二酮；
2-[3-(6-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，4-二甲苯基}氧基}乙酸甲酯；
3-{3-{6-{[(间-氰苯基)氨基甲酰基]甲氧基}-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
1-甲基-3-{3-[(甲磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(邻-甲氧苯基)-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酰基}甲磺酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}丙酸2-丙炔酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈；
3-[3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}丙酸；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲氧乙酰胺；
2-{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-4-甲氧苯氧基}丙酸甲酯；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-(甲磺酰基)乙酰胺；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-(甲磺酰基)丙酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲基-N-(甲磺酰基)乙酰胺；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-甲基-N-(甲磺酰基)乙酰胺；
2-{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}-N-(乙磺酰基)乙酰胺；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-噻吩羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，苯甲酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲氧乙酸酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二乙基-1，2-苯并异噻唑-3-乙腈；
3-[6-氟-3-(甲氧甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，5-异噁唑羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，环丙烷羧酸酯；
3-(乙酰基-1，2-苯并异噻唑-5-基)-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
3-[3-(1-甲氧乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸苄酯；
N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-[(对-甲苄基)磺酰基]-1，2-苯并异噻唑-3-甲酰胺；
N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲酰胺；
3-[3-(1-羟乙基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲醛，3-(二甲基缩醛)；
3-(6-氟-3-甲基-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲醛，3-(二甲基缩醛)；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-羧酸；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-甲基-1，2-苯并异噻唑-3-乙腈；
N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙氧甲基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸甲酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-呋喃甲酸酯；
N-[(间-氯苄基)磺酰基]-5[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；及
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲基氨基甲酸酯。
9.一种防治不需要的植物品种的方法，包括对所述植物的叶部或含其种子或其他繁殖器官的土壤或水施用除草有效量的如权利要求1所述的化合物。
10.根据权利要求9所述的方法，其中该化合物为如权利要求2所述的化合物。
11.根据权利要求9所述的方法，其中该化合物具有下式结构：
Figure A9880989800261
12.根据权利要求11所述的方法，其中该化合物为如权利要求4所述的化合物。
13.根据权利要求9所述的方法，其中该化合物为如权利要求8所述的化合物。
14.根据权利要求9所述的方法，其中该化合物系在作物植株、作物种子或其他作物繁殖器官存在下施用到不需要的植物品种的叶部或含其种子或其他繁殖器官的土壤或水中。
15.根据权利要求14所述的方法，其中该作物为谷类作物。
16.根据权利要求15所述的方法，其中该谷类作物系选自玉米、小麦及稻。
17.根据权利要求16所述的方法，其中该谷类作物为玉米，化合物选自下列：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-(二甲氨基)乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(对-乙苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}乙酸甲酯；
3-[3-(二溴甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸1-甲基-2-丙炔酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
1-甲基-3-{3-[(甲磺酰基)甲基]-1，2-苯并异噻唑-5-基}-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(邻-甲氧苯基)-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
N-{{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酰基}甲磺酰胺；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-乙腈；
3-[3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲基-N-(甲磺酰基)乙酰胺；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲基氨基甲酸酯；
N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-羧酸；与
N-(苄磺酰基)-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-甲酰胺。
18.根据权利要求16所述的方法，其中该谷类作物为小麦，该化合物选自：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-(二甲氨基)乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}丙酸甲酯；
3-(6-氟-3-甲基-1，2-苯并异噁唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-{3-{6-[(1-苯并咪唑基羰基)甲氧基]-间-甲苯基}-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸烯丙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸3-苯基-2-丙炔酯；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸2-氯乙酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸2，2，2-三氟乙酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-2，4-二甲苯基}氧基}乙酸甲酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲氧乙酰胺；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}-N-甲基-N-(甲磺酰基)乙酰胺；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯；
3-(3-乙酰基-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
N-[(间-氯苄基)磺酰基]-5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；与
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺。
19.根据权利要求16所述的方法，其中该谷类作物为稻，化合物选自下列：
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸异丙酯；
{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
3-[3-(6-甲氧基-间-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}乙酸乙酯；
1-甲基-3-[3-(6-(2-丙炔氧基)间-甲苯基]-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-{6-{[(间-氰苯基)氨基甲酰基]甲氧基}间-甲苯基}-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4-(1H，3H)-嘧啶二酮；
3-[3-(2-甲氧基-对-甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-[3-(6-甲氧基-3，4-二甲苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
3-[3-{6-{[(间-氰苯基)氨基甲酰基]甲氧基}间-甲苯基}-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
{邻-[5-(3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
3-[3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α-乙基-1，2-苯并异噻唑-3-乙腈；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二乙基-1，2-苯并异噻唑-3-乙腈；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，5-异噁唑羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，环丙烷羧酸酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-羧酸甲酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-α，α-二甲基-1，2-苯并异噻唑-3-乙酸苄酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；与
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺。
20.根据权利要求14所述的方法，其中作物为大豆。
21.根据权利要求20所述的方法，其中化合物系选自下列：
2-{{2-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-对-甲苯基}氧基}丙酸甲酯；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
1-甲基-3-(3-甲基-1，2-苯并异噻唑-5-基]-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-{{6-{5-[3，6-二氢-3-甲基-4-(三氟甲基)-2，6-二氧-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-3，4-二甲苯基}氧基}丙酸甲酯；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
3-[3-(邻-甲氧苯基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
2-{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸2-丙炔酯；
{邻-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-1，2-苯并异噻唑-3-基}-苯氧基}乙酸2-丙炔酯；
3-{3-[(烯丙氧基)甲基]-1，2-苯并异噻唑-5-基}-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
{{2-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噁唑-3-基}-对-甲苯基}氧基}乙酸甲酯；
{{6-{5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-6-氟-1，2-苯并异噻唑-3-基}-间-甲苯基}氧基}乙酸甲酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，苯甲酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-噻吩羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，甲氧乙酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，环丙烷羧酸酯；
3-[3-(羟甲基)-1，2-苯并异噻唑-5-基]-1-甲基-6-(三氟甲基)-2，4(1H，3H)-嘧啶二酮，2-呋喃甲酸酯；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(甲丙基磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(乙磺酰基)-1，2-苯并异噻唑-3-甲酰胺；
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(异丙基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺；与
5-[3，6-二氢-3-甲基-2，6-二氧-4-(三氟甲基)-1(2H)-嘧啶基]-N-(二甲基氨磺酰基)-1，2-苯并异噻唑-3-甲酰胺。
22.根据权利要求9所述的方法，其中该化合物以约0.001公斤/公顷至1公斤/公顷的施用率施加到不需要的植物品种的叶部或含其种子或其他繁殖器官的土壤或水中。
23.一种除草组合物，它包含惰性固体或液体载体及除草有效量的如权利要求1所述的化合物。
24.根据权利要求23所述的组合物，其中该化合物为如权利要求2所述的化合物。
25.根据权利要求23所述的组合物，其中该化合物有下式结构：
26.根据权利要求25所述的组合物，其中该化合物为权利要求4所述的化合物。
27.根据权利要求23所述的组合物，其中该化合物为如权利要求8所述的化合物。
28.一种中间化合物，它具有下式结构：
Figure A9880989800332
其中
R1与R2分别为氢、卤素、C1-C6烷基、C3-C7环烷基、C1-C6卤代烷基、C3-C6烯基、C3-C6卤代烯基、C3-C6炔基、OR7、S(O)nR8或NR9R10，当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它任选地穿插氧、硫或氮，且任选地被一至三个甲基或一个或多个卤原子取代；
X为氢、卤素或C1-C4烷基；
X1为氢、卤素、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素、氰基、R12、X2R12、X3R12、X2X3R12或X3X2R12；
X2为O、S(O)p或NR13；
X3为-C(＝A3)-、-C(＝NOR14)-或-C(＝N-NR13R50)；
R4、R5、R6、R7、R8、R9、R10与R14分别为氢、C1-C6烷基、C3-C7环烷基、C2-C8烷氧基烷基、C2-C6烯基、C2-C6炔基或苄基；
R12为氢，
C1-C8烷基、C3-C7环烷基、C2-C8烯基、C5-C6环烯基或C2-C8炔基，其中各基团任选地被下列任何组合取代：1至6个卤原子、1至3个C1-C20烷氧基，它任选地被一个C1-C6烷氧基、苄氧基或C1-C6烷硫基取代，1或2个C1-C10卤代烷氧基、1或2个NR15R16基团、1至3个S(O)qR17基团、1或2个氰基、1或2个C3-C7环烷基、1个硫氰基、1个O(SO2)R17基团、1个O(NO2)基团、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)SR19基团、1或2个C(O)NR20R21基团、1至3个X4R22基团、1或2个P(O)(OR23)2基团、1或2个Si(R24)3基团、
1个4至10元单环或稠合双环杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1或2个苯基，其中各苯基分别任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C3-C7环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，或
茚满基，它任选地被下列任何组合取代：1或2个卤原子、1或2个C1-C4烷基、1个C1-C4烷氧基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基、或X4R22基团；
R13为氢、C1-C8烷氧基烷基、C1-C6烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基、SO2R51或1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基，且当R13及R12及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢、Si(R31)3、C(O)NR35R36、C(O)R33、SO2R47、
C1-C20烷基，它被下列基团取代：一个羟基、苄氧基、硝基、OC(O)R33、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、P(O)(OH)NH2、P(O)(OH)(OR23)、C(O)NR35OR23、氰基或2-二氧戊环基，
1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、或C1-C4卤代烷磺酰基，
C3-C20烯基，它任选地被下列基团取代：1至3个卤原子、1个羟基、1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它任选地被下列基团取代：一个羟基、C1-C6烷氧基、C1-C4烷基、C2-C4烯基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个羟基、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1至3个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，
苄基、它任选地于苯环上经下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团，或
4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢、
C1-C6烷基、C3-C7环烷基、C2-C6烯基或C2-C6炔基，其中各基团任选地被一个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个CO2R26基团，
C(O)R43，或
CO2R42；
R16与R21分别为氢、C1-C6烷基、C1-C4烷氧基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17、R18、R25、R30、R33、R45及R51分别为NR46R48、
-N＝CR46R48、C1-C8烷基，它任选地被一个C1-C6烷氧基、噻吩或呋喃基取代，C1-C6卤代烷基、C3-C8环烷基、CO2R23、C2-C6烯基，它任选地被苯基取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团，或
5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R19与R26分别为氢、C1-C20烷基、C1-C8卤代烷基、C3-C7环烷基、C3-C7卤代环烷基、C3-C20烯基、C3-C8卤代烯基、C5-C8环烯基、C5-C8卤代环烯基、C3-C8炔基、C3-C8卤代炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、C1-C6硫烷基、C2-C20烷氧烷氧基、苯基、OSi(R47)3、OC(O)R33、C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
2-、3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基、C3-C8环烷基、二噁烷或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R34、R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢、氰基、C1-C6烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
m、n、p与q分别为0、1或2的整数；
R29为氢、C1-C4烷基或C1-C4卤代烷基；
R24、R31、R41及R47分别为C1-C4烷基、
苄基，它任选地被一个或多个分别选自下列的基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；
R23、R39、R40、R42、R43、R44、R46及R48分别为氢、C2-C6烯基、C3-C8环烷基、
C1-C8烷基，它任选地被一或二个C1-C4烷氧基取代；
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，且
当R46与R48及其所连接的原子结合在一起时，为5至12元单环或稠合双环杂环或环烷基环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；及
A、A1、A3、A4、X4及X5分别为O或S；
及其光学异构体、非对映异构体和/或互变异构体。
29.根据权利要求28所述的化合物，其中：
R1与R2分别为氢、卤素、C1-C6烷基、C3-C7环烷基、C1-C6卤代烷基、C3-C6烯基、C3-C6卤代烯基、C3-C6炔基、OR7、S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它任选地穿插氧、硫或氮，且任选地被一至三个甲基或一个或多个卤原子取代；
X为氢、卤素或C1-C4烷基；
X1为氢、卤素、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素、氰基、R12、X2R12、X3R12、X2X3R12或X3X2R12；
X2为O、S(O)p或NR13；
X3为-C(＝A3)-或-C(＝NOR14)-；
R4、R5、R6、R7、R8、R9、R10与R14分别为氢、C1-C6烷基、C3-C7环烷基、C2-C6烯基、C2-C6炔基或苄基；
R12为氢，
C1-C6烷基、C3-C7环烷基、C2-C6烯基、C5-C6环烯基或C2-C6炔基，其中各基团任选地被下列任何组合取代：1至6个卤原子、1至3个C1-C20烷氧基、1或2个C1-C10卤代烷氧基、1或2个NR15R16基团、1至3个S(O)qR17基团、1或2个氰基、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)NR20R21基团、1至3个X4R22基团、1或2个P(O)(OR23)2基团、1或2个Si(R24)3基团、
1个4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C3-C7环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基、或X4R22基团；
R13为氢、C1-C6烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基或SO2R51，且当R13及R12及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢、Si(R31)3、
C1-C20烷基，它被下列基团取代：一个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、P(O)(OH)NH2、P(O)(OH)(OR23)、C(O)NR35OR23、氰基或2-二氧戊环基，
1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、或C1-C4卤代烷磺酰基，
C3-C20烯基，它任选地被下列基团取代：1至3个卤原子、1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NHOR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它任选地被下列基团取代：一个C1-C6烷氧基、C1-C4烷基、C2-C4烯基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NHOR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NHOR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基、它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，
苄基、它任选地于苯环上经下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团，或
4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢、
C1-C6烷基、C3-C7环烷基、C2-C6烯基或C2-C6炔基，其中各基团任选地被一个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
C(O)R43，
R16与R21分别为氢、C1-C6烷基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17、R18、R25、R30、R33、R45及R51分别为C1-C4烷基，C1-C4卤代烷基、CO2R23、
C2-C6烯基，它任选地被苯基取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团，或
5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R19及R26分别为氢、C1-C20烷基、C1-C8卤代烷基、C3-C7环烷基、C3-C7卤代环烷基、C3-C20烯基、C3-C8卤代烯基、C5-C8环烯基、C5-C8卤代环烯基、C3-C8炔基、C3-C8卤代炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
2-、3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R34、R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢、氰基、C1-C6烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
m、n、p与q分别为0、1或2的整数；
R29为氢、C1-C4烷基或C1-C4卤代烷基；
R24、R31、R41及R47分别为C1-C4烷基、
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；
R23、R39、R40、R42、R43、R44、R46及R48分别为氢、C1-C4烷基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，且
A、A1、A3、A4、X4及X5分别为O或S；
及其光学异构体、非对映异构体和/或互变异构体。
30.根据权利要求28所述的化合物，其中
R1与R2分别为氢、卤素、C1-C6烷基、C3-C7环烷基、C1-C6卤代烷基、C3-C6烯基、C3-C6卤代烯基、C3-C6炔基、OR7、S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它任选地穿插氧、硫或氮，且任选地被一至三个甲基或一个或多个卤原子取代；
X为氢、卤素或C1-C4烷基；
X1为氢、卤素、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素、氰基、R12、X2R12、X3R12、X2X3R12或X3X2R12；
X2为O、S(O)p或NR13；
X3为-C(＝A3)-、-C(＝NOR14)-或-C(＝N-NR13R50)；
R4、R5、R6、R7、R8、R9、R10与R14分别为氢、C1-C6烷基、C3-C7环烷基、C2-C8烷氧基烷基、C2-C6烯基、C2-C6炔基或苄基；
R12为氢，
C1-C8烷基、C3-C7环烷基、C2-C8烯基、C5-C6环烯基或C2-C8炔基，其中各基团任选地被下列任何组合取代：1至6个卤原子、1至3个C1-C20烷氧基，它任选地被一个C1-C6烷氧基、苄氧基或C1-C6烷硫基取代，1或2个C1-C10卤代烷氧基、1或2个NR15R16基基团、1至3个S(O)qR17基团、1或2个氰基、1或2个C3-C7环烷基、1个硫氰基、1个O(SO2)R17基团、1个O(NO2)基团、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)SR19基团、1或2个C(O)NR20R21基团、1至3个X4R22基团、1或2个P(O)(OR23)2基团、1或2个Si(R24)3基团、
1个4至10元单环或稠合双环杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1或2个苯基，其中各苯基分别任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C3-C7环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，或
茚满基，它任选地被下列任何组合取代：1或2个卤原子、1或2个C1-C4烷基、1个C1-C4烷氧基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基、或X4R22基团；
R13为氢、C1-C8烷氧基烷基、C1-C6烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基、SO2R51或1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基，且当R13及R12及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢、Si(R31)3、C(O)NR35R36、C(O)R33、SO2R47、
C1-C20烷基，它被下列基团取代：一个羟基、苄氧基、硝基、OC(O)R33、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、P(O)(OH)NH2、P(O)(OH)(OR23)、C(O)NR35OR23、氰基或2-二氧戊环基，
1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、或C1-C4卤代烷磺酰基，
C3-C20烯基，它任选地被下列基团取代：1至3个卤原子、1个羟基、1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它任选地被下列基团取代：一个羟基、一个C1-C6烷氧基、C1-C4烷基、C2-C4烯基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个羟基、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，
苄基，它任选地于苯环上经下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团，或
4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢、
C1-C6烷基、C3-C7环烷基、C2-C6烯基或C2-C6炔基，其中各基团任选地被一个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个CO2R26基团，
C(O)R43，或
CO2R42；
R16与R21分别为氢、C1-C6烷基、C1-C4烷氧基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17、R18、R25、R30、R33、R45及R51分别为NR46R48、
-N＝CR46R48、C1-C8烷基，它任选地被一个C1-C6烷氧基、噻吩或呋喃基取代，C1-C6卤代烷基、C3-C8环烷基、CO2R23、C2-C6烯基，它任选地被苯基取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团，或
5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R19与R26分别为氢、C1-C20烷基、C1-C8卤代烷基、C3-C7环烷基、C3-C7卤代环烷基、C3-C20烯基、C3-C8卤代烯基、C5-C8环烯基、C5-C8卤代环烯基、C3-C8炔基、C3-C8卤代炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、C1-C6硫烷基、C2-C20烷氧烷氧基、苯基、OSi(R47)3、OC(O)R33、C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
2-、3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基、C3-C8环烷基、二噁烷或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R34、R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢、氰基、C1-C6烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
m、n、p与q分别为0、1或2的整数；
R29为氢、C1-C4烷基或C1-C4卤代烷基；
R24、R31、R41及R47分别为C1-C4烷基、
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；
R23、R39、R40、R42、R43、R44、R46及R48分别为氢、C2-C6烯基、C3-C8环烷基、
C1-C8烷基，它任选地被一或二个C1-C4烷氧基取代；
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，且
当R46与R48及其所连接的原子结合在一起时，为5至12元单环或稠合双环杂环或环烷基环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；及
A、A1、A3、A4、X4及X5分别为O或S；
及其光学异构体、非对映异构体和/或互变异构体。
31.根据权利要求30所述的化合物，其中
R1为卤素或C1-C4卤代烷基，
R2为氢、卤素或C1-C4卤代烷基；
X与X1分别为氢或卤素；
Z为O或S；
Y为氰基、R12、X2R12或X3X2R12；
X2为O、S或NR13；
X3为-C(＝A3)-、-C(＝NOR14)-或-C(＝N-NR13R50)；
R12为氢，
C1-C6烷基、C3-C7环烷基、C2-C6烯基、C5-C6环烯基或C2-C6炔基，其中各基团任选地被下列任何组合取代：1至3个卤原子、1或2个C1-C20烷氧基、1或2个C1-C10卤代烷氧基、1个NR15R16基团、1个S(O)qR17基团、1或2个氰基、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)SR19基团、1或2个C(O)NR20R21基团、1或2个X4R22基团、1个P(O)(OR23)2基团、1个Si(R24)3基团、
1个4至10元单环或稠合双环杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1个苯基，它任选地被下列任何组合取代：1至3个卤原子、1个C1-C6烷基、1个C1-C6烷氧基、1个C3-C7环烷基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，或
苯基，它任选地被下列任何组合取代：1或2个卤原子、1至3个C1-C4烷基、1或2个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
R13为氢、C2-C6烷氧基烷基、C1-C4烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基或SO2R51；
R28为卤素；
R22与R27分别为氢、Si(R31)3、C(O)NR35R36、C(O)R33、SO2R47、
C1-C20烷基，它被下列基团取代：一个羟基、苄氧基、硝基、OC(O)R33、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、P(O)(OH)NH2、P(O)(OH)(OR23)、C(O)NR35OR23、氰基或2-二氧戊环基，
1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、或C1-C4卤代烷磺酰基，
C3-C20烯基，它任选地被下列基团取代：1至3个卤原子、1个羟基、1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它任选地被下列基团取代：一个羟基、C1-C6烷氧基、C1-C4烷基、C2-C4烯基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个羟基、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，
苄基，其苯环上任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团，或
4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢、
C1-C6烷基、C3-C7环烷基、C2-C6烯基或C2-C6炔基，其中各基团任选地被一个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个CO2R26基团，
C(O)R43，或
CO2R42；
R14为氢、C1-C6烷基、C3-C7环烷基、C2-C8烷氧基烷基、C2-C6烯基，C2-C6炔基或苄基；
R16与R21分别为氢、C1-C6烷基、C1-C4烷氧基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R17、R18、R25、R30、R33、R45及R51分别为NR46R48、
-N＝CR46R48、C1-C8烷基，它任选地被一个C1-C6烷氧基、噻吩或呋喃基取代，C1-C6卤代烷基、C3-C8环烷基、CO2R23、C2-C6烯基，它任选地被苯基取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团，或
5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R19与R26分别为氢、C1-C20烷基、C1-C8卤代烷基、C3-C7环烷基、C3-C7卤代环烷基、C3-C20烯基、C3-C8卤代烯基、C5-C8环烯基、C5-C8卤代环烯基、C3-C8炔基、C3-C8卤代炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、C1-C6硫烷基、C2-C20烷氧烷氧基、苯基、OSi(R47)3、OC(O)R33、C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基、C3-C8环烷基、二噁烷或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R34、R37及R38分别为C1-C6烷基；
R35与R49分别氢或C1-C6烷基，且R36与R50分别为氢、氰基、C1-C6烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
q为0、1或2的整数；
R29为氢、C1-C4烷基或C1-C4卤代烷基；
R24、R31、R41及R47分别为C1-C4烷基、
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；
R23、R39、R40、R42、R43、R44、R46及R48分别为氢、C2-C6烯基、C3-C8环烷基、
C1-C8烷基，它任选地被一或二个C1-C4烷氧基取代；
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，且
A、A1、A3、A4、X4及X5分别为O或S；
及其光学异构体、非对映异构体和/或互变异构体。
32.一种制备有下式结构的化合物的方法
Figure A9880989800531
其中
R为C1-C6烷基、C1-C6卤代烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR4或NR5R6；
R1与R2分别为氢、卤素、C1-C6烷基、C3-C7环烷基、C1-C6卤代烷基、C3-C6烯基、C3-C6卤代烯基、C3-C6炔基、OR7、S(O)nR8或NR9R10，且当R1与R2及其所连接的原子结合在一起时，代表4至7元饱和或不饱和环，它任选地穿插氧、硫或氮，且任选地被一至三个甲基或一个或多个卤原子所取代；
X为氢、卤素或C1-C4烷基；
X1为氢、卤素、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；
Y为卤素、氰基、R12、X2R12、X3R12、X2X3R12或X3X2R12；
X2为O、S(O)p或NR13；
X3为-C(＝A3)-、-C(＝NOR14)-或-C(＝N-NR13R50)；
R4、R5、R6、R7、R8、R9、R10与R14分别为氢、C1-C6烷基、C3-C7环烷基、C2-C8烷氧基烷基、C2-C6烯基、C2-C6炔基或苄基；
R12为氢，
C1-C8烷基、C3-C7环烷基、C2-C8烯基、C5-C6环烯基或C2-C8炔基，其中各基团任选地被下列任何组合取代：1至6个卤原子、1至3个C1-C20烷氧基，它任选地被一个C1-C6烷氧基、苄氧基或C1-C6烷硫基取代，1或2个C1-C10卤代烷基、1或2个NR15R16基团、1至3个S(O)qR17基团、1或2个氰基、1或2个C3-C7环烷基、1个硫氰基、1个O(SO2)R17基团、1个O(NO2)基团、1或2个C(O)R18基团、1或2个CO2R19基团、1或2个C(O)SR19基团、1或2个C(O)NR20R21基团、1至3个X4R22基团、1或2个P(O)(OR23)2基团、1或2个Si(R24)3基团、
1个4至10元单环或稠合双环杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1或2个X4R22基团；
1个四元有机铵基团，或
1或2个苯基，其中各苯基分别任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C3-C7环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团或1个X5R27基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基、1个C3-C6环烷基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，或
茚满基，它任选地被下列任何组合取代：1或2个卤原子、1或2个C1-C4烷基、1个C1-C4烷氧基、1个C1-C4卤代烷基、1个C1-C4烷硫基、1个氰基、1个硝基、1个C(O)R25基团、1个CO2R26基团、1个X4R22基团、1个CH＝CHR22基团、1个CH2CH(R28)R22基团，或1个N(R29)SO2R30基团，
且当R12与R13及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基、或X4R22基团；
R13为氢、C1-C8烷氧基烷基、C1-C6烷基、C3-C7环烷基、C3-C6烯基、C3-C6炔基、苄基、OR23、氰基、SO2R51或1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基，且当R13及R12及其所连接的氮原子结合在一起时，为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R28为卤素；
R22与R27分别为氢、Si(R31)3、C(O)NR35R36、C(O)R33、SO2R47、
C1-C20烷基，它被下列基团取代：一个羟基、苄氧基、硝基、OC(O)R33、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、P(O)(OH)NH2、P(O)(OH)(OR23)、C(O)NR35OR23、氰基或2-二氧戊环基，
1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基、或
1个5至12元单环或稠合双环杂环，它任选地被1个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、或C1-C4卤代烷磺酰基，
C3-C20烯基，它任选地被下列基团取代：1至3个卤原子、1个羟基、1个C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或1个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C5-C8环烯基，它任选地被下列基团取代：一个羟基、C1-C6烷氧基、C1-C4烷基、C2-C4烯基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
C3-C10炔基，它任选地被下列基团取代：1个羟基、C1-C6烷氧基、CO2R32、C(O)R33、C(A4R34)2、C(O)NR35R36、C(O)ON＝CR37R38、C(O)NR35OR23、氰基或2-二氧戊环基，或一个苯基、二氢呋喃酮或呋喃酮环，其中各环任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基、它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团或1个C(O)R33基团，
苄基、它任选地于苯环上经下列任何组合取代：1至3个卤原子、1至3个C1-C6烷基、1至3个C1-C6烷氧基、1个C1-C4卤代烷基、1个C1-C4卤代烷氧基、1个氰基、1个硝基、1个NR39R40基团、或1个C(O)R33基团，或
4至10元杂环，它任选地被下列任何组合取代：1或2个氧代基、1或2个硫代基、1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基；
R15与R20分别为氢、
C1-C6烷基、C3-C7环烷基、C2-C6烯基或C2-C6炔基，其中各基团任选地被一个CO2R42基团取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基或1至3个C1-C4卤代烷氧基，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个CO2R26基团，
C(O)R43，或
CO2R42；
R16与R21分别为氢、C1-C6烷基、C1-C4烷氧基、C3-C7环烷基、C2-C6烯基，C3-C7环烯基、C2-C6炔基、P(O)(OR44)2、SO2R45、C(O)R46、
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团，或
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基或1个X4R22基团；
R17、R18、R25、R30、R33、R45及R51分别为NR46R48、-N＝CR46R48、C1-C8烷基，它任选地被一个C1-C6烷氧基、噻吩或呋喃基取代，C1-C6卤代烷基、C3-C8环烷基、CO2R23、C2-C6烯基，它任选地被苯基取代，
苄基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基或1个X4R22基团，
苯基，它任选地被下列任何组合取代：1至3个卤原子、1至3个C1-C4烷基、1至3个C1-C4卤代烷基、1至3个C1-C4烷氧基、1至3个C1-C4卤代烷氧基、1个硝基、1个氰基、或1个X4R22基团，或
5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基、C1-C4卤代烷磺酰基或X4R22基团；
R19与R26分别为氢、C1-C20烷基、C1-C8卤代烷基、C3-C7环烷基、C3-C7卤代环烷基、C3-C20烯基、C3-C8卤代烯基、C5-C8环烯基、C5-C8卤代环烯基、C3-C8炔基、C3-C8卤代炔基、Si(R41)3、苄基、苯基、糠基、吡啶基、噻吩基、羟亚氨基、或碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R32为氢、
Si(R47)3，
二(C1-C4烷基)亚氨基，
C1-C20烷基，它任选地被一个CO2R48、C1-C6烷氧基、C1-C6硫烷基、C2-C20烷氧烷氧基、苯基、OSi(R47)3、OC(O)R33、C3-C7环烷基或二(C1-C4烷基)亚氨基取代，
C1-C15卤代烷基，
C3-C8环烷基，它任选地被一个CO2R48基团取代，
C3-C8卤代环烷基，
C3-C20烯基，它任选地被一个苯基取代，
C3-C15卤代烯基，
C5-C8环烯基，
C5-C8卤代环烯基，
C3-C20炔基，它任选地被一个苯基取代，
C3-C20卤代炔基，
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，
2-、3-或4-吡啶基，
2-或3-呋喃基，
2-或3-噻吩基，
2-四氢呋喃基，
C1-C4烷基，它被一个吡啶基、呋喃基、噻吩基、四氢呋喃基、C3-C8环烷基、二噁烷或NR49R50基团取代，或
碱金属、碱土金属、锰、铜、锌、钴、银、镍、铵或有机铵阳离子；
R34、R37及R38分别为C1-C6烷基；
R35与R49分别为氢或C1-C6烷基，且R36与R50分别为氢、氰基、C1-C6烷基、SO2R51或苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、及C1-C4卤代烷氧基，或当R35与R36或R49与R50及其所连接的氮原子结合在一起时，可为5至12元单环或稠合双环杂环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；
m、n、p与q分别为0、1或2的整数；
R29为氢、C1-C4烷基或C1-C4卤代烷基；
R24、R31、R41及R47分别为C1-C4烷基、
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基；
R23、R39、R40、R42、R43、R44、R46及R48分别为氢、C2-C6烯基、C3-C8环烷基、
C1-C8烷基，它任选地被一或二个C1-C4烷氧基取代；
苄基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，或
苯基，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基及C1-C4卤代烷氧基，且
当R46与R48及其所连接的原子结合在一起时，为5至12元单环或稠合双环杂环或环烷基环，它任选地被一个或多个分别选自下列之基团取代：卤素、氰基、硝基、氨基、羟基、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基、C1-C4卤代烷氧基或C1-C4卤代烷磺酰基；及
A、A1、A3、A4、X4及X5分别为O或S；该方法包括使下式胺：
Figure A9880989800591
其中X、X1、Y与Z的定义同上，与下式2-二烷氨基-6H-1，3-噁嗪-6-酮其中R1与R2如上述说明，在有机酸存在下反应，形成下式的中间化合物
Figure A9880989800593
其中R1、R2、X、X1、Y与Z的定义同上，使该中间化合物与下式亲电子物Z1R其中R的定义同上，Z1为氯，溴或碘，在碱存在下反应。
33.一种制备下式化合物的方法
Figure A9880989800601
其中
X为氢、卤素或C1-C4烷基；
X1为氢、卤素、C1-C4烷基、C1-C4卤代烷基、C1-C4烷氧基或C1-C4卤代烷氧基；
Z为O或S(O)m；且
m为0、1或2的整数，
该方法包括使下式化合物其中X、X1与Z的定义同上，与氯或溴在酸之存在下反应。
CN98809898A 1997-09-17 1998-09-15 作为除草剂的取代的3－(1,2－苯并异噻唑或异噁唑－5－基)－取代的嘧啶 Pending CN1273585A (zh)

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CN114276287A (zh) * 2021-12-27 2022-04-05 浙江工业大学 N-(取代苄氧基)酰胺类化合物及其制备方法和应用
CN116354953A (zh) * 2022-12-31 2023-06-30 西北农林科技大学 含苯并噻唑类化合物的除草组合物

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