NO20033398L - Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer - Google Patents
Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymerInfo
- Publication number
- NO20033398L NO20033398L NO20033398A NO20033398A NO20033398L NO 20033398 L NO20033398 L NO 20033398L NO 20033398 A NO20033398 A NO 20033398A NO 20033398 A NO20033398 A NO 20033398A NO 20033398 L NO20033398 L NO 20033398L
- Authority
- NO
- Norway
- Prior art keywords
- oxazolyl
- pyrrolyl
- thiazolyl
- inhibitors
- acid amide
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US26548601P | 2001-01-31 | 2001-01-31 | |
PCT/IB2001/002728 WO2002060898A1 (en) | 2001-01-31 | 2001-12-24 | Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20033398D0 NO20033398D0 (no) | 2003-07-30 |
NO20033398L true NO20033398L (no) | 2003-09-29 |
Family
ID=23010641
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20033398A NO20033398L (no) | 2001-01-31 | 2003-07-30 | Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer |
Country Status (24)
Country | Link |
---|---|
US (3) | US6559168B2 (no) |
EP (1) | EP1355907A1 (no) |
JP (1) | JP2004518691A (no) |
KR (1) | KR20030072614A (no) |
CN (1) | CN1489588A (no) |
BG (1) | BG108039A (no) |
BR (1) | BR0116850A (no) |
CA (1) | CA2436551A1 (no) |
CR (1) | CR7038A (no) |
CZ (1) | CZ20031903A3 (no) |
EA (1) | EA200300622A1 (no) |
EC (1) | ECSP034683A (no) |
EE (1) | EE200300362A (no) |
HU (1) | HUP0401305A2 (no) |
IL (1) | IL156412A0 (no) |
IS (1) | IS6844A (no) |
MA (1) | MA26985A1 (no) |
MX (1) | MXPA03006886A (no) |
NO (1) | NO20033398L (no) |
OA (1) | OA12542A (no) |
PL (1) | PL365443A1 (no) |
TN (1) | TNSN03050A1 (no) |
WO (1) | WO2002060898A1 (no) |
ZA (1) | ZA200305769B (no) |
Families Citing this family (75)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1371650A4 (en) * | 2001-03-23 | 2005-05-04 | Nippon Chemiphar Co | ACTIVATED RECEPTOR ACTIVATOR BY PEROXYSOME PROLIFIERS |
US20030055026A1 (en) | 2001-04-17 | 2003-03-20 | Dey L.P. | Formoterol/steroid bronchodilating compositions and methods of use thereof |
MXPA03010679A (es) * | 2001-05-23 | 2004-03-02 | Tanabe Seiyaku Co | Una composicion para acelerar la cicatrizacion de fractura osea. |
US20040180900A1 (en) * | 2001-05-23 | 2004-09-16 | Masaharu Takigawa | Therapeutic composition for repairing chondropathy |
EP1424078A4 (en) * | 2001-09-04 | 2009-03-25 | Ono Pharmaceutical Co | RESPIRATORY DISEASE MEDICINES COMPRISING A SPHINGOSINE-1-PHOSPHATE RECEPTOR REGULATING AGENT |
CZ2004747A3 (cs) * | 2001-12-21 | 2004-11-10 | Novo Nordisk A/S | Deriváty amidů jako GK aktivátory |
EP1465882B1 (en) * | 2001-12-21 | 2011-08-24 | X-Ceptor Therapeutics, Inc. | Hetrocyclic modulators of nuclear receptors |
GB0201677D0 (en) | 2002-01-25 | 2002-03-13 | Glaxo Group Ltd | Medicament dispenser |
WO2003063911A1 (fr) * | 2002-02-01 | 2003-08-07 | Anges Mg, Inc. | Compositions pharmaceutiques contenant un leurre et procede d'utilisation |
US20050158371A1 (en) * | 2002-02-12 | 2005-07-21 | Sumitomo Pharmaceuticals Co., Ltd. | Novel external agent |
KR101116627B1 (ko) * | 2002-06-27 | 2012-10-09 | 노보 노르디스크 에이/에스 | 치료제로서 아릴 카르보닐 유도체 |
GB0217196D0 (en) * | 2002-07-25 | 2002-09-04 | Glaxo Group Ltd | Medicament dispenser |
FI114917B (fi) * | 2002-08-29 | 2005-01-31 | Hormos Nutraceutical Oy Ltd | Lignaanikomplekseja |
WO2004047817A1 (en) * | 2002-11-27 | 2004-06-10 | Altana Pharma Ag | Pde4 and pde3/4 inhibitors for use in the treatment of cachexia |
EP1424101A3 (en) * | 2002-11-29 | 2004-08-18 | NOZAKI, Masako | Use of a leukotriene C4 and D4 receptor antagonist for the preparation of a medicament for treating or preventing brain inflammation and sepsis |
US7148248B2 (en) * | 2002-11-29 | 2006-12-12 | Masako Nozaki | Method of treating or inhibiting the development of brain inflammation and sepsis |
JP2006516548A (ja) | 2002-12-30 | 2006-07-06 | アンジオテック インターナショナル アクツィエン ゲゼルシャフト | 迅速ゲル化ポリマー組成物からの薬物送達法 |
GB0302094D0 (en) | 2003-01-29 | 2003-02-26 | Pharmagene Lab Ltd | EP4 receptor antagonists |
US20050079548A1 (en) * | 2003-07-07 | 2005-04-14 | Plexxikon, Inc. | Ligand development using PDE4B crystal structures |
GB0317482D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Nicotinamide derivatives useful as pde4 inhibitors |
GB0317516D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Nicotinamide derivatives useful as PDE4 inhibitors |
GB0317498D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Compounds |
GB0317484D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Nicotinamide derivatives useful as pde4 inhibitors |
US7132435B2 (en) | 2003-07-25 | 2006-11-07 | Pfizer Inc. | Compounds |
US7153870B2 (en) | 2003-07-25 | 2006-12-26 | Pfizer Inc. | Nicotinamide derivatives useful as PDE4 inhibitors |
US20050020587A1 (en) * | 2003-07-25 | 2005-01-27 | Pfizer Inc | Nicotinamide derivatives useful as PDE4 inhibitors |
US20050187278A1 (en) * | 2003-08-28 | 2005-08-25 | Pharmacia Corporation | Treatment or prevention of vascular disorders with Cox-2 inhibitors in combination with cyclic AMP-specific phosphodiesterase inhibitors |
MXPA06002521A (es) * | 2003-09-05 | 2006-06-20 | Altana Pharma Ag | Uso de inhibidores de pde4 para el tratamiento de diabetes mellitus. |
US7534894B2 (en) * | 2003-09-25 | 2009-05-19 | Wyeth | Biphenyloxy-acids |
GB0324269D0 (en) | 2003-10-16 | 2003-11-19 | Pharmagene Lab Ltd | EP4 receptor antagonists |
AU2005203930C1 (en) | 2004-01-06 | 2012-02-23 | Vtv Therapeutics Llc | Heteroaryl-ureas and their use as glucokinase activators |
US20090042951A1 (en) * | 2004-02-20 | 2009-02-12 | Robert Danziger | Blood Pressure Reduction in Salt-Sensitive Hypertension |
WO2005102388A1 (ja) * | 2004-04-26 | 2005-11-03 | Ono Pharmaceutical Co., Ltd. | 新規なblt2介在性疾患、blt2結合剤および化合物 |
CN101031293A (zh) * | 2004-05-06 | 2007-09-05 | 普莱希科公司 | Pde4b抑制剂及其应用 |
US7655680B2 (en) * | 2004-05-17 | 2010-02-02 | Otsuka Pharmaceutical Co., Ltd. | Thiazole compound and use thereof |
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BG108039A (en) | 2004-07-30 |
CN1489588A (zh) | 2004-04-14 |
US20030186974A1 (en) | 2003-10-02 |
US6559168B2 (en) | 2003-05-06 |
BR0116850A (pt) | 2004-02-25 |
AU2002222429A2 (no) | 2002-08-12 |
US6894041B2 (en) | 2005-05-17 |
EE200300362A (et) | 2003-12-15 |
IL156412A0 (en) | 2004-01-04 |
ZA200305769B (en) | 2004-10-25 |
EA200300622A1 (ru) | 2003-12-25 |
TNSN03050A1 (fr) | 2005-12-23 |
OA12542A (en) | 2006-06-05 |
US20030130254A1 (en) | 2003-07-10 |
EP1355907A1 (en) | 2003-10-29 |
NO20033398D0 (no) | 2003-07-30 |
US6869945B2 (en) | 2005-03-22 |
CR7038A (es) | 2004-04-22 |
JP2004518691A (ja) | 2004-06-24 |
CZ20031903A3 (cs) | 2004-07-14 |
CA2436551A1 (en) | 2002-08-08 |
PL365443A1 (en) | 2005-01-10 |
MXPA03006886A (es) | 2003-11-13 |
MA26985A1 (fr) | 2004-12-20 |
IS6844A (is) | 2003-06-16 |
ECSP034683A (es) | 2003-08-29 |
HUP0401305A2 (hu) | 2004-10-28 |
US20020123520A1 (en) | 2002-09-05 |
WO2002060898A1 (en) | 2002-08-08 |
KR20030072614A (ko) | 2003-09-15 |
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