NO20033398L - Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer - Google Patents
Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymerInfo
- Publication number
- NO20033398L NO20033398L NO20033398A NO20033398A NO20033398L NO 20033398 L NO20033398 L NO 20033398L NO 20033398 A NO20033398 A NO 20033398A NO 20033398 A NO20033398 A NO 20033398A NO 20033398 L NO20033398 L NO 20033398L
- Authority
- NO
- Norway
- Prior art keywords
- oxazolyl
- pyrrolyl
- thiazolyl
- inhibitors
- acid amide
- Prior art date
Links
- 101100296720 Dictyostelium discoideum Pde4 gene Proteins 0.000 title 1
- 108010044467 Isoenzymes Proteins 0.000 title 1
- 101100082610 Plasmodium falciparum (isolate 3D7) PDEdelta gene Proteins 0.000 title 1
- -1 imidazolyl acid amide Chemical class 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 125000002971 oxazolyl group Chemical class 0.000 title 1
- 125000000168 pyrrolyl group Chemical class 0.000 title 1
- 125000000335 thiazolyl group Chemical group 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Virology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Hematology (AREA)
- Molecular Biology (AREA)
- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Vascular Medicine (AREA)
- AIDS & HIV (AREA)
- Hospice & Palliative Care (AREA)
- Biotechnology (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26548601P | 2001-01-31 | 2001-01-31 | |
| PCT/IB2001/002728 WO2002060898A1 (en) | 2001-01-31 | 2001-12-24 | Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20033398D0 NO20033398D0 (no) | 2003-07-30 |
| NO20033398L true NO20033398L (no) | 2003-09-29 |
Family
ID=23010641
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20033398A NO20033398L (no) | 2001-01-31 | 2003-07-30 | Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer |
Country Status (24)
| Country | Link |
|---|---|
| US (3) | US6559168B2 (no) |
| EP (1) | EP1355907A1 (no) |
| JP (1) | JP2004518691A (no) |
| KR (1) | KR20030072614A (no) |
| CN (1) | CN1489588A (no) |
| BG (1) | BG108039A (no) |
| BR (1) | BR0116850A (no) |
| CA (1) | CA2436551A1 (no) |
| CR (1) | CR7038A (no) |
| CZ (1) | CZ20031903A3 (no) |
| EA (1) | EA200300622A1 (no) |
| EC (1) | ECSP034683A (no) |
| EE (1) | EE200300362A (no) |
| HU (1) | HUP0401305A2 (no) |
| IL (1) | IL156412A0 (no) |
| IS (1) | IS6844A (no) |
| MA (1) | MA26985A1 (no) |
| MX (1) | MXPA03006886A (no) |
| NO (1) | NO20033398L (no) |
| OA (1) | OA12542A (no) |
| PL (1) | PL365443A1 (no) |
| TN (1) | TNSN03050A1 (no) |
| WO (1) | WO2002060898A1 (no) |
| ZA (1) | ZA200305769B (no) |
Families Citing this family (78)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1371650A4 (en) * | 2001-03-23 | 2005-05-04 | Nippon Chemiphar Co | ACTIVATED RECEPTOR ACTIVATOR BY PEROXYSOME PROLIFIERS |
| US20030055026A1 (en) | 2001-04-17 | 2003-03-20 | Dey L.P. | Formoterol/steroid bronchodilating compositions and methods of use thereof |
| EP1389467B1 (en) * | 2001-05-23 | 2013-07-03 | Mitsubishi Tanabe Pharma Corporation | Therapeutic composition for the regenerative treatment of cartilage diseases |
| CA2447619A1 (en) * | 2001-05-23 | 2002-11-28 | Tanabe Seiyaku Co., Ltd. | A composition for accelerating bone fracture healing |
| US20040235794A1 (en) * | 2001-09-04 | 2004-11-25 | Shinji Nakade | Remedies for respiratory diseases comprising sphingosine-1-phosphate receptor controller |
| CN100506807C (zh) * | 2001-12-21 | 2009-07-01 | 诺沃挪第克公司 | 作为gk活化剂的酰胺衍生物 |
| US6696473B2 (en) * | 2001-12-21 | 2004-02-24 | X-Ceptor Therapeutics, Inc. | Heterocyclic modulators of nuclear receptors |
| GB0201677D0 (en) * | 2002-01-25 | 2002-03-13 | Glaxo Group Ltd | Medicament dispenser |
| US20040072726A1 (en) * | 2002-02-01 | 2004-04-15 | Ryuichi Morishita | Decoy-containing pharmaceutical compositions and method of using the same |
| US20050158371A1 (en) * | 2002-02-12 | 2005-07-21 | Sumitomo Pharmaceuticals Co., Ltd. | Novel external agent |
| AU2003243921B2 (en) * | 2002-06-27 | 2009-05-07 | Novo Nordisk A/S | Aryl carbonyl derivatives as therapeutic agents |
| GB0217196D0 (en) * | 2002-07-25 | 2002-09-04 | Glaxo Group Ltd | Medicament dispenser |
| FI114917B (fi) * | 2002-08-29 | 2005-01-31 | Hormos Nutraceutical Oy Ltd | Lignaanikomplekseja |
| JP2006508996A (ja) * | 2002-11-27 | 2006-03-16 | アルタナ ファルマ アクチエンゲゼルシャフト | 悪液質の治療における使用のための、pde4及びpde3/4インヒビター |
| EP1424101A3 (en) * | 2002-11-29 | 2004-08-18 | NOZAKI, Masako | Use of a leukotriene C4 and D4 receptor antagonist for the preparation of a medicament for treating or preventing brain inflammation and sepsis |
| US7148248B2 (en) * | 2002-11-29 | 2006-12-12 | Masako Nozaki | Method of treating or inhibiting the development of brain inflammation and sepsis |
| CA2511521C (en) | 2002-12-30 | 2012-02-07 | Angiotech International Ag | Drug delivery from rapid gelling polymer composition |
| GB0302094D0 (en) | 2003-01-29 | 2003-02-26 | Pharmagene Lab Ltd | EP4 receptor antagonists |
| US20050079548A1 (en) * | 2003-07-07 | 2005-04-14 | Plexxikon, Inc. | Ligand development using PDE4B crystal structures |
| TWI359675B (en) | 2003-07-10 | 2012-03-11 | Dey L P | Bronchodilating β-agonist compositions |
| US20050020587A1 (en) * | 2003-07-25 | 2005-01-27 | Pfizer Inc | Nicotinamide derivatives useful as PDE4 inhibitors |
| US7153870B2 (en) | 2003-07-25 | 2006-12-26 | Pfizer Inc. | Nicotinamide derivatives useful as PDE4 inhibitors |
| GB0317484D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Nicotinamide derivatives useful as pde4 inhibitors |
| US7132435B2 (en) | 2003-07-25 | 2006-11-07 | Pfizer Inc. | Compounds |
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- 2001-12-24 EP EP01273600A patent/EP1355907A1/en not_active Withdrawn
- 2001-12-24 WO PCT/IB2001/002728 patent/WO2002060898A1/en not_active Ceased
- 2001-12-24 EE EEP200300362A patent/EE200300362A/xx unknown
- 2001-12-24 PL PL01365443A patent/PL365443A1/xx not_active Application Discontinuation
- 2001-12-24 IL IL15641201A patent/IL156412A0/xx unknown
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- 2001-12-24 JP JP2002561466A patent/JP2004518691A/ja active Pending
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- 2003-07-25 ZA ZA200305769A patent/ZA200305769B/en unknown
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- 2003-07-29 CR CR7038A patent/CR7038A/es not_active Application Discontinuation
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Also Published As
| Publication number | Publication date |
|---|---|
| US20030186974A1 (en) | 2003-10-02 |
| CR7038A (es) | 2004-04-22 |
| MA26985A1 (fr) | 2004-12-20 |
| PL365443A1 (en) | 2005-01-10 |
| OA12542A (en) | 2006-06-05 |
| JP2004518691A (ja) | 2004-06-24 |
| US6559168B2 (en) | 2003-05-06 |
| HUP0401305A2 (hu) | 2004-10-28 |
| US20030130254A1 (en) | 2003-07-10 |
| BG108039A (en) | 2004-07-30 |
| ZA200305769B (en) | 2004-10-25 |
| CZ20031903A3 (cs) | 2004-07-14 |
| NO20033398D0 (no) | 2003-07-30 |
| CA2436551A1 (en) | 2002-08-08 |
| BR0116850A (pt) | 2004-02-25 |
| US6869945B2 (en) | 2005-03-22 |
| EA200300622A1 (ru) | 2003-12-25 |
| AU2002222429A2 (no) | 2002-08-12 |
| ECSP034683A (es) | 2003-08-29 |
| US6894041B2 (en) | 2005-05-17 |
| MXPA03006886A (es) | 2003-11-13 |
| WO2002060898A1 (en) | 2002-08-08 |
| US20020123520A1 (en) | 2002-09-05 |
| IS6844A (is) | 2003-06-16 |
| KR20030072614A (ko) | 2003-09-15 |
| IL156412A0 (en) | 2004-01-04 |
| EE200300362A (et) | 2003-12-15 |
| EP1355907A1 (en) | 2003-10-29 |
| CN1489588A (zh) | 2004-04-14 |
| TNSN03050A1 (fr) | 2005-12-23 |
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