NO20033398L - Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer - Google Patents

Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer

Info

Publication number
NO20033398L
NO20033398L NO20033398A NO20033398A NO20033398L NO 20033398 L NO20033398 L NO 20033398L NO 20033398 A NO20033398 A NO 20033398A NO 20033398 A NO20033398 A NO 20033398A NO 20033398 L NO20033398 L NO 20033398L
Authority
NO
Norway
Prior art keywords
oxazolyl
pyrrolyl
thiazolyl
inhibitors
acid amide
Prior art date
Application number
NO20033398A
Other languages
English (en)
Other versions
NO20033398D0 (no
Inventor
Anthony Marfat
Michael William Mckechney
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO20033398D0 publication Critical patent/NO20033398D0/no
Publication of NO20033398L publication Critical patent/NO20033398L/no

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    • C—CHEMISTRY; METALLURGY
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
NO20033398A 2001-01-31 2003-07-30 Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer NO20033398L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26548601P 2001-01-31 2001-01-31
PCT/IB2001/002728 WO2002060898A1 (en) 2001-01-31 2001-12-24 Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes

Publications (2)

Publication Number Publication Date
NO20033398D0 NO20033398D0 (no) 2003-07-30
NO20033398L true NO20033398L (no) 2003-09-29

Family

ID=23010641

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20033398A NO20033398L (no) 2001-01-31 2003-07-30 Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer

Country Status (24)

Country Link
US (3) US6559168B2 (no)
EP (1) EP1355907A1 (no)
JP (1) JP2004518691A (no)
KR (1) KR20030072614A (no)
CN (1) CN1489588A (no)
BG (1) BG108039A (no)
BR (1) BR0116850A (no)
CA (1) CA2436551A1 (no)
CR (1) CR7038A (no)
CZ (1) CZ20031903A3 (no)
EA (1) EA200300622A1 (no)
EC (1) ECSP034683A (no)
EE (1) EE200300362A (no)
HU (1) HUP0401305A2 (no)
IL (1) IL156412A0 (no)
IS (1) IS6844A (no)
MA (1) MA26985A1 (no)
MX (1) MXPA03006886A (no)
NO (1) NO20033398L (no)
OA (1) OA12542A (no)
PL (1) PL365443A1 (no)
TN (1) TNSN03050A1 (no)
WO (1) WO2002060898A1 (no)
ZA (1) ZA200305769B (no)

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EP1389467B1 (en) * 2001-05-23 2013-07-03 Mitsubishi Tanabe Pharma Corporation Therapeutic composition for the regenerative treatment of cartilage diseases
JP4510384B2 (ja) 2001-05-23 2010-07-21 田辺三菱製薬株式会社 骨折治癒促進用組成物
JPWO2003020313A1 (ja) * 2001-09-04 2004-12-16 小野薬品工業株式会社 スフィンゴシン−１−リン酸受容体調節剤からなる呼吸器疾患治療剤
EP1465882B1 (en) * 2001-12-21 2011-08-24 X-Ceptor Therapeutics, Inc. Hetrocyclic modulators of nuclear receptors
HUP0402309A3 (en) * 2001-12-21 2008-09-29 Novo Nordisk As Amide derivatives as glucokinase activators and pharmaceutical compositions containing them
GB0201677D0 (en) * 2002-01-25 2002-03-13 Glaxo Group Ltd Medicament dispenser
DE60231063D1 (de) * 2002-02-01 2009-03-19 Anges Mg Inc N zur behandlung von aneurysmen
US20050158371A1 (en) * 2002-02-12 2005-07-21 Sumitomo Pharmaceuticals Co., Ltd. Novel external agent
EP2471533A1 (en) * 2002-06-27 2012-07-04 Novo Nordisk A/S Aryl carbonyl derivatives as therapeutic agents
GB0217196D0 (en) * 2002-07-25 2002-09-04 Glaxo Group Ltd Medicament dispenser
FI114917B (fi) * 2002-08-29 2005-01-31 Hormos Nutraceutical Oy Ltd Lignaanikomplekseja
PL375631A1 (en) * 2002-11-27 2005-12-12 Altana Pharma Ag Pde4 and pde3/4 inhibitors for use in the treatment of cachexia
US7148248B2 (en) * 2002-11-29 2006-12-12 Masako Nozaki Method of treating or inhibiting the development of brain inflammation and sepsis
EP1424101A3 (en) * 2002-11-29 2004-08-18 NOZAKI, Masako Use of a leukotriene C4 and D4 receptor antagonist for the preparation of a medicament for treating or preventing brain inflammation and sepsis
DE60331367D1 (de) 2002-12-30 2010-04-01 Angiotech Int Ag Wirkstofffreisetzung von schnell gelierender polymerzusammensetzung
GB0302094D0 (en) 2003-01-29 2003-02-26 Pharmagene Lab Ltd EP4 receptor antagonists
US20050079548A1 (en) * 2003-07-07 2005-04-14 Plexxikon, Inc. Ligand development using PDE4B crystal structures
TWI359675B (en) 2003-07-10 2012-03-11 Dey L P Bronchodilating β-agonist compositions
GB0317516D0 (en) * 2003-07-25 2003-08-27 Pfizer Ltd Nicotinamide derivatives useful as PDE4 inhibitors
GB0317498D0 (en) * 2003-07-25 2003-08-27 Pfizer Ltd Compounds
US7153870B2 (en) 2003-07-25 2006-12-26 Pfizer Inc. Nicotinamide derivatives useful as PDE4 inhibitors
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US6894041B2 (en) 2005-05-17
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