NO20033398D0 - Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer - Google Patents

Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer

Info

Publication number
NO20033398D0
NO20033398D0 NO20033398A NO20033398A NO20033398D0 NO 20033398 D0 NO20033398 D0 NO 20033398D0 NO 20033398 A NO20033398 A NO 20033398A NO 20033398 A NO20033398 A NO 20033398A NO 20033398 D0 NO20033398 D0 NO 20033398D0
Authority
NO
Norway
Prior art keywords
oxazolyl
pyrrolyl
thiazolyl
inhibitors
acid amide
Prior art date
Application number
NO20033398A
Other languages
English (en)
Other versions
NO20033398L (no
Inventor
Anthony Marfat
Michael William Mckechney
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO20033398D0 publication Critical patent/NO20033398D0/no
Publication of NO20033398L publication Critical patent/NO20033398L/no

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    • C—CHEMISTRY; METALLURGY
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
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  • Engineering & Computer Science (AREA)
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  • Virology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
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  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Molecular Biology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • AIDS & HIV (AREA)
  • Obesity (AREA)
NO20033398A 2001-01-31 2003-07-30 Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer NO20033398L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26548601P 2001-01-31 2001-01-31
PCT/IB2001/002728 WO2002060898A1 (en) 2001-01-31 2001-12-24 Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes

Publications (2)

Publication Number Publication Date
NO20033398D0 true NO20033398D0 (no) 2003-07-30
NO20033398L NO20033398L (no) 2003-09-29

Family

ID=23010641

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20033398A NO20033398L (no) 2001-01-31 2003-07-30 Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer

Country Status (24)

Country Link
US (3) US6559168B2 (no)
EP (1) EP1355907A1 (no)
JP (1) JP2004518691A (no)
KR (1) KR20030072614A (no)
CN (1) CN1489588A (no)
BG (1) BG108039A (no)
BR (1) BR0116850A (no)
CA (1) CA2436551A1 (no)
CR (1) CR7038A (no)
CZ (1) CZ20031903A3 (no)
EA (1) EA200300622A1 (no)
EC (1) ECSP034683A (no)
EE (1) EE200300362A (no)
HU (1) HUP0401305A2 (no)
IL (1) IL156412A0 (no)
IS (1) IS6844A (no)
MA (1) MA26985A1 (no)
MX (1) MXPA03006886A (no)
NO (1) NO20033398L (no)
OA (1) OA12542A (no)
PL (1) PL365443A1 (no)
TN (1) TNSN03050A1 (no)
WO (1) WO2002060898A1 (no)
ZA (1) ZA200305769B (no)

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US20030055026A1 (en) 2001-04-17 2003-03-20 Dey L.P. Formoterol/steroid bronchodilating compositions and methods of use thereof
JP4510383B2 (ja) * 2001-05-23 2010-07-21 田辺三菱製薬株式会社 軟骨疾患修復治療用組成物
KR20040007596A (ko) 2001-05-23 2004-01-24 다나베 세이야꾸 가부시키가이샤 골절 치료 촉진용 조성물
JPWO2003020313A1 (ja) * 2001-09-04 2004-12-16 小野薬品工業株式会社 スフィンゴシン−１−リン酸受容体調節剤からなる呼吸器疾患治療剤
JP2005518391A (ja) * 2001-12-21 2005-06-23 ノボ　ノルディスク　アクティーゼルスカブ Ｇｋ活性化剤としてのアミド誘導体
WO2003060078A2 (en) * 2001-12-21 2003-07-24 X-Ceptor Therapeutics, Inc. Heterocyclic modulators of nuclear receptors
GB0201677D0 (en) 2002-01-25 2002-03-13 Glaxo Group Ltd Medicament dispenser
US20040072726A1 (en) 2002-02-01 2004-04-15 Ryuichi Morishita Decoy-containing pharmaceutical compositions and method of using the same
US20050158371A1 (en) * 2002-02-12 2005-07-21 Sumitomo Pharmaceuticals Co., Ltd. Novel external agent
CA2744893A1 (en) * 2002-06-27 2004-01-08 Novo Nordisk A/S Aryl carbonyl derivatives as glucokinase activators
GB0217196D0 (en) * 2002-07-25 2002-09-04 Glaxo Group Ltd Medicament dispenser
FI114917B (fi) * 2002-08-29 2005-01-31 Hormos Nutraceutical Oy Ltd Lignaanikomplekseja
JP2006508996A (ja) * 2002-11-27 2006-03-16 アルタナ　ファルマ　アクチエンゲゼルシャフト 悪液質の治療における使用のための、ｐｄｅ４及びｐｄｅ３／４インヒビター
US7148248B2 (en) * 2002-11-29 2006-12-12 Masako Nozaki Method of treating or inhibiting the development of brain inflammation and sepsis
EP1424101A3 (en) * 2002-11-29 2004-08-18 NOZAKI, Masako Use of a leukotriene C4 and D4 receptor antagonist for the preparation of a medicament for treating or preventing brain inflammation and sepsis
WO2004060346A2 (en) 2002-12-30 2004-07-22 Angiotech International Ag Drug delivery from rapid gelling polymer composition
GB0302094D0 (en) 2003-01-29 2003-02-26 Pharmagene Lab Ltd EP4 receptor antagonists
US20050079548A1 (en) * 2003-07-07 2005-04-14 Plexxikon, Inc. Ligand development using PDE4B crystal structures
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