NO20033398L - Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer - Google Patents
Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymerInfo
- Publication number
- NO20033398L NO20033398L NO20033398A NO20033398A NO20033398L NO 20033398 L NO20033398 L NO 20033398L NO 20033398 A NO20033398 A NO 20033398A NO 20033398 A NO20033398 A NO 20033398A NO 20033398 L NO20033398 L NO 20033398L
- Authority
- NO
- Norway
- Prior art keywords
- oxazolyl
- pyrrolyl
- thiazolyl
- inhibitors
- acid amide
- Prior art date
Links
- 101100296720 Dictyostelium discoideum Pde4 gene Proteins 0.000 title 1
- 108010044467 Isoenzymes Proteins 0.000 title 1
- 101100082610 Plasmodium falciparum (isolate 3D7) PDEdelta gene Proteins 0.000 title 1
- -1 imidazolyl acid amide Chemical class 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 125000002971 oxazolyl group Chemical class 0.000 title 1
- 125000000168 pyrrolyl group Chemical class 0.000 title 1
- 125000000335 thiazolyl group Chemical group 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Virology (AREA)
- Neurology (AREA)
- Oncology (AREA)
- Biomedical Technology (AREA)
- Pulmonology (AREA)
- Neurosurgery (AREA)
- Communicable Diseases (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Molecular Biology (AREA)
- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Otolaryngology (AREA)
- Emergency Medicine (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26548601P | 2001-01-31 | 2001-01-31 | |
| PCT/IB2001/002728 WO2002060898A1 (en) | 2001-01-31 | 2001-12-24 | Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20033398D0 NO20033398D0 (no) | 2003-07-30 |
| NO20033398L true NO20033398L (no) | 2003-09-29 |
Family
ID=23010641
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20033398A NO20033398L (no) | 2001-01-31 | 2003-07-30 | Tiazolyl-, oksazolyl-, pyrrolyl-, og imidazolyl- syreamidderivater nyttige som inhibitorer av PDE4 isozymer |
Country Status (24)
| Country | Link |
|---|---|
| US (3) | US6559168B2 (es) |
| EP (1) | EP1355907A1 (es) |
| JP (1) | JP2004518691A (es) |
| KR (1) | KR20030072614A (es) |
| CN (1) | CN1489588A (es) |
| BG (1) | BG108039A (es) |
| BR (1) | BR0116850A (es) |
| CA (1) | CA2436551A1 (es) |
| CR (1) | CR7038A (es) |
| CZ (1) | CZ20031903A3 (es) |
| EA (1) | EA200300622A1 (es) |
| EC (1) | ECSP034683A (es) |
| EE (1) | EE200300362A (es) |
| HU (1) | HUP0401305A2 (es) |
| IL (1) | IL156412A0 (es) |
| IS (1) | IS6844A (es) |
| MA (1) | MA26985A1 (es) |
| MX (1) | MXPA03006886A (es) |
| NO (1) | NO20033398L (es) |
| OA (1) | OA12542A (es) |
| PL (1) | PL365443A1 (es) |
| TN (1) | TNSN03050A1 (es) |
| WO (1) | WO2002060898A1 (es) |
| ZA (1) | ZA200305769B (es) |
Families Citing this family (78)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002076957A1 (en) * | 2001-03-23 | 2002-10-03 | Nippon Chemiphar Co.,Ltd. | Activator for peroxisome proliferator-activated receptor |
| US20030055026A1 (en) | 2001-04-17 | 2003-03-20 | Dey L.P. | Formoterol/steroid bronchodilating compositions and methods of use thereof |
| EP1389467B1 (en) * | 2001-05-23 | 2013-07-03 | Mitsubishi Tanabe Pharma Corporation | Therapeutic composition for the regenerative treatment of cartilage diseases |
| JP4510384B2 (ja) | 2001-05-23 | 2010-07-21 | 田辺三菱製薬株式会社 | 骨折治癒促進用組成物 |
| EP1424078A4 (en) * | 2001-09-04 | 2009-03-25 | Ono Pharmaceutical Co | RESPIRATORY DISEASE MEDICINES COMPRISING A SPHINGOSINE-1-PHOSPHATE RECEPTOR REGULATING AGENT |
| EP1465882B1 (en) * | 2001-12-21 | 2011-08-24 | X-Ceptor Therapeutics, Inc. | Hetrocyclic modulators of nuclear receptors |
| RU2374236C2 (ru) * | 2001-12-21 | 2009-11-27 | Ново Нордиск А/С | Амидные производные в качестве активаторов gk |
| GB0201677D0 (en) | 2002-01-25 | 2002-03-13 | Glaxo Group Ltd | Medicament dispenser |
| EP1470826B1 (en) * | 2002-02-01 | 2009-01-28 | AnGes MG, Inc. | Decoy-containing pharmaceutical compositions for the treatment of aneurysms |
| US20050158371A1 (en) * | 2002-02-12 | 2005-07-21 | Sumitomo Pharmaceuticals Co., Ltd. | Novel external agent |
| AU2003243921B2 (en) * | 2002-06-27 | 2009-05-07 | Novo Nordisk A/S | Aryl carbonyl derivatives as therapeutic agents |
| GB0217196D0 (en) * | 2002-07-25 | 2002-09-04 | Glaxo Group Ltd | Medicament dispenser |
| FI114917B (fi) * | 2002-08-29 | 2005-01-31 | Hormos Nutraceutical Oy Ltd | Lignaanikomplekseja |
| US20060079540A1 (en) * | 2002-11-27 | 2006-04-13 | Altana Pharma Ag | Pde4 and pde3/4 inhibitors for use in the treatment of cachexia |
| US7148248B2 (en) * | 2002-11-29 | 2006-12-12 | Masako Nozaki | Method of treating or inhibiting the development of brain inflammation and sepsis |
| EP1424101A3 (en) * | 2002-11-29 | 2004-08-18 | NOZAKI, Masako | Use of a leukotriene C4 and D4 receptor antagonist for the preparation of a medicament for treating or preventing brain inflammation and sepsis |
| ATE457716T1 (de) | 2002-12-30 | 2010-03-15 | Angiotech Int Ag | Wirkstofffreisetzung von schnell gelierender polymerzusammensetzung |
| GB0302094D0 (en) | 2003-01-29 | 2003-02-26 | Pharmagene Lab Ltd | EP4 receptor antagonists |
| US20050079548A1 (en) * | 2003-07-07 | 2005-04-14 | Plexxikon, Inc. | Ligand development using PDE4B crystal structures |
| TWI359675B (en) | 2003-07-10 | 2012-03-11 | Dey L P | Bronchodilating β-agonist compositions |
| US7132435B2 (en) | 2003-07-25 | 2006-11-07 | Pfizer Inc. | Compounds |
| GB0317498D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Compounds |
| US20050020587A1 (en) * | 2003-07-25 | 2005-01-27 | Pfizer Inc | Nicotinamide derivatives useful as PDE4 inhibitors |
| GB0317484D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Nicotinamide derivatives useful as pde4 inhibitors |
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- 2001-12-24 OA OA1200300177A patent/OA12542A/en unknown
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- 2001-12-24 IL IL15641201A patent/IL156412A0/xx unknown
- 2001-12-24 CZ CZ20031903A patent/CZ20031903A3/cs unknown
- 2001-12-24 PL PL01365443A patent/PL365443A1/xx not_active Application Discontinuation
- 2001-12-24 EA EA200300622A patent/EA200300622A1/ru unknown
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- 2001-12-24 JP JP2002561466A patent/JP2004518691A/ja active Pending
- 2001-12-24 EP EP01273600A patent/EP1355907A1/en not_active Withdrawn
- 2001-12-24 CN CNA018224431A patent/CN1489588A/zh active Pending
- 2001-12-24 KR KR10-2003-7010071A patent/KR20030072614A/ko not_active Ceased
- 2001-12-24 CA CA002436551A patent/CA2436551A1/en not_active Abandoned
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2002
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- 2002-11-20 US US10/300,950 patent/US6869945B2/en not_active Expired - Fee Related
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- 2003-07-25 ZA ZA200305769A patent/ZA200305769B/en unknown
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- 2003-07-29 CR CR7038A patent/CR7038A/es not_active Application Discontinuation
- 2003-07-30 NO NO20033398A patent/NO20033398L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US6559168B2 (en) | 2003-05-06 |
| HUP0401305A2 (hu) | 2004-10-28 |
| EE200300362A (et) | 2003-12-15 |
| EA200300622A1 (ru) | 2003-12-25 |
| US6894041B2 (en) | 2005-05-17 |
| ZA200305769B (en) | 2004-10-25 |
| US20030186974A1 (en) | 2003-10-02 |
| OA12542A (en) | 2006-06-05 |
| PL365443A1 (en) | 2005-01-10 |
| IL156412A0 (en) | 2004-01-04 |
| AU2002222429A2 (es) | 2002-08-12 |
| WO2002060898A1 (en) | 2002-08-08 |
| CR7038A (es) | 2004-04-22 |
| US20020123520A1 (en) | 2002-09-05 |
| IS6844A (is) | 2003-06-16 |
| US6869945B2 (en) | 2005-03-22 |
| MXPA03006886A (es) | 2003-11-13 |
| CA2436551A1 (en) | 2002-08-08 |
| MA26985A1 (fr) | 2004-12-20 |
| US20030130254A1 (en) | 2003-07-10 |
| ECSP034683A (es) | 2003-08-29 |
| EP1355907A1 (en) | 2003-10-29 |
| KR20030072614A (ko) | 2003-09-15 |
| BG108039A (en) | 2004-07-30 |
| BR0116850A (pt) | 2004-02-25 |
| TNSN03050A1 (fr) | 2005-12-23 |
| JP2004518691A (ja) | 2004-06-24 |
| CN1489588A (zh) | 2004-04-14 |
| CZ20031903A3 (cs) | 2004-07-14 |
| NO20033398D0 (no) | 2003-07-30 |
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