BE2014C053I2 - - Google Patents

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Publication number
BE2014C053I2
BE2014C053I2 BE2014C053C BE2014C053C BE2014C053I2 BE 2014C053 I2 BE2014C053 I2 BE 2014C053I2 BE 2014C053 C BE2014C053 C BE 2014C053C BE 2014C053 C BE2014C053 C BE 2014C053C BE 2014C053 I2 BE2014C053 I2 BE 2014C053I2
Authority
BE
Belgium
Application number
BE2014C053C
Other languages
French (fr)
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of BE2014C053I2 publication Critical patent/BE2014C053I2/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
BE2014C053C 2002-10-11 2014-09-09 BE2014C053I2 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002298259 2002-10-11
PCT/JP2003/013070 WO2004033463A1 (ja) 2002-10-11 2003-10-10 2,3−ジヒドロ−6−ニトロイミダゾ[2,1−b]オキサゾール化合物

Publications (1)

Publication Number Publication Date
BE2014C053I2 true BE2014C053I2 (ko) 2022-08-30

Family

ID=32089299

Family Applications (1)

Application Number Title Priority Date Filing Date
BE2014C053C BE2014C053I2 (ko) 2002-10-11 2014-09-09

Country Status (27)

Country Link
US (1) US7262212B2 (ko)
EP (2) EP2570418A3 (ko)
JP (1) JP4186065B2 (ko)
KR (1) KR100723847B1 (ko)
CN (4) CN101172981A (ko)
AR (4) AR041198A1 (ko)
AU (1) AU2003272979B2 (ko)
BE (1) BE2014C053I2 (ko)
BR (1) BRPI0314344B8 (ko)
CA (1) CA2497569C (ko)
CY (2) CY1113578T1 (ko)
DK (1) DK1555267T3 (ko)
ES (1) ES2400179T3 (ko)
FR (1) FR14C0066I2 (ko)
HK (2) HK1085463A1 (ko)
HU (1) HUS1400046I1 (ko)
LU (1) LU92517I2 (ko)
MX (1) MXPA05003674A (ko)
MY (1) MY139244A (ko)
PL (3) PL404913A1 (ko)
PT (1) PT1555267E (ko)
RU (1) RU2326121C3 (ko)
SI (1) SI1555267T1 (ko)
TW (1) TWI347946B (ko)
UA (1) UA83200C2 (ko)
WO (1) WO2004033463A1 (ko)
ZA (1) ZA200501033B (ko)

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ES2314460T3 (es) * 2003-10-31 2009-03-16 Otsuka Pharmaceutical Co., Ltd. Compuestos de 2,3-dihidro-6-nitroimidazo (2,1-b)oxazol para el tratamiento de la tuberculosis.
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TW201434467A (zh) * 2005-10-05 2014-09-16 Otsuka Pharma Co Ltd 抗結核治療藥物及含彼之套組
JP5105818B2 (ja) * 2005-10-05 2012-12-26 大塚製薬株式会社 医薬組成物
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TW200800268A (en) * 2005-11-04 2008-01-01 Otsuka Pharma Co Ltd Medicinal composition showing improved drug absorbability
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AR070301A1 (es) 2007-05-08 2010-03-31 Otsuka Pharma Co Ltd Compuesto epoxi y metodo para producir el mismo
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EP2229368A1 (en) 2007-12-11 2010-09-22 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11beta-hydroxysteroid dehydrogenase 1
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US9643922B2 (en) 2008-08-18 2017-05-09 Yale University MIF modulators
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CN103524492A (zh) * 2013-10-23 2014-01-22 中国药科大学 侧链含硝基咪唑基团取代的喹诺酮类化合物、其制备及用途
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CN105732659B (zh) * 2014-12-12 2019-07-16 上海阳帆医药科技有限公司 硝基咪唑类化合物及其制备方法和在制药中的用途
BR112017015744A2 (pt) * 2015-01-29 2018-03-13 Medshine Discovery Inc composto apresentando uma estrutura de fórmula (i), um sal farmaceuticamente aceitável do mesmo ou um isômero ótico do mesmo, composição farmacêutica e uso do composto de fórmula (i) para o tratamento e prevenção de mycobacterium tuberculosis ou outras infecções microbianas
EP3275862B1 (en) * 2015-03-27 2020-08-12 Otsuka Pharmaceutical Co., Ltd. Method for producing 1-(4-hydroxyphenyl)-4-(4-trifluoromethoxyphenoxy)piperidine or salt thereof
CN106317072B (zh) * 2015-06-17 2020-03-17 盟科医药技术(上海)有限公司 用于分枝杆菌感染治疗的杂环化合物及其应用
EP3421454B9 (en) 2016-02-26 2023-08-09 Otsuka Pharmaceutical Co., Ltd. Piperidine derivative
CN105859628B (zh) * 2016-04-19 2018-08-07 清远职业技术学院 一种抗菌化合物对n咪唑苯甲醛缩邻甲苯胺希夫碱及其制备方法和应用
MX2019000858A (es) * 2016-07-22 2019-11-11 Medshine Discovery Inc Cristal y sal de nitroimidazol y metodo de fabricacion de los mismos.
JP7171726B2 (ja) 2017-08-16 2022-11-15 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッド 新規化合物
KR20210019056A (ko) 2018-06-11 2021-02-19 오츠카 세이야쿠 가부시키가이샤 델라마니드 함유 조성물
CN109705022A (zh) * 2018-12-28 2019-05-03 上海彩迩文生化科技有限公司 一种芳香胺中间体的制备方法
CN112300192B (zh) * 2019-08-02 2023-08-11 南京长澳医药科技有限公司 硝基咪唑类化合物及其制备方法和用途
CN110483549B (zh) * 2019-08-30 2021-03-05 沈阳药科大学 一种硝基咪唑吡喃类抗结核药物的制备方法
CN110615800A (zh) * 2019-10-16 2019-12-27 李丽丽 硝基咪唑类化合物及其制备方法和用途
CN112156088B (zh) * 2020-10-30 2021-08-31 健民药业集团股份有限公司 一种化合物在制备结核分枝杆菌抑制剂中的用途
CN113603706A (zh) * 2021-08-04 2021-11-05 深圳市泰力生物医药有限公司 德拉马尼的晶型、含有该晶型的活性药物和药物组合物
CN115368252B (zh) * 2022-09-19 2024-01-12 西北农林科技大学 一种4-胺基酚类衍生物及应用
CN116640106B (zh) * 2023-05-11 2024-03-08 郑州大学 一种苯基哌嗪类化合物及其制备方法、应用

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Also Published As

Publication number Publication date
AR086485A2 (es) 2013-12-18
FR14C0066I2 (fr) 2015-05-22
EP1555267A4 (en) 2010-08-18
PL376157A1 (en) 2005-12-27
TW200420568A (en) 2004-10-16
PL217919B1 (pl) 2014-09-30
ES2400179T3 (es) 2013-04-08
CA2497569C (en) 2011-05-24
EP2570418A3 (en) 2013-07-03
RU2005114017A (ru) 2006-01-20
ZA200501033B (en) 2006-06-28
WO2004033463A1 (ja) 2004-04-22
PL409525A1 (pl) 2014-11-10
KR100723847B1 (ko) 2007-05-31
CN101255170A (zh) 2008-09-03
MY139244A (en) 2009-09-30
AR091771A2 (es) 2015-02-25
CN101172981A (zh) 2008-05-07
AU2003272979B2 (en) 2009-07-23
CY1113578T1 (el) 2016-06-22
EP1555267A1 (en) 2005-07-20
BRPI0314344B1 (pt) 2019-11-26
RU2326121C2 (ru) 2008-06-10
BR0314344A (pt) 2005-07-12
PL404913A1 (pl) 2013-09-30
US7262212B2 (en) 2007-08-28
MXPA05003674A (es) 2005-06-08
AR041198A1 (es) 2005-05-04
RU2326121C3 (ru) 2021-09-17
CN102532162B (zh) 2015-05-27
EP1555267B1 (en) 2013-01-16
DK1555267T3 (da) 2013-02-11
CA2497569A1 (en) 2004-04-22
UA83200C2 (en) 2008-06-25
KR20050061473A (ko) 2005-06-22
JP4186065B2 (ja) 2008-11-26
LU92517I2 (fr) 2014-10-13
AR089950A2 (es) 2014-10-01
US20060094767A1 (en) 2006-05-04
HK1171018A1 (en) 2013-03-15
CY2014041I1 (el) 2016-07-27
BRPI0314344B8 (pt) 2021-05-25
JP2004149527A (ja) 2004-05-27
CN102532162A (zh) 2012-07-04
SI1555267T1 (sl) 2013-05-31
CY2014041I2 (el) 2016-07-27
CN100366624C (zh) 2008-02-06
PT1555267E (pt) 2013-01-29
FR14C0066I1 (ko) 2014-10-17
AU2003272979A1 (en) 2004-05-04
TWI347946B (en) 2011-09-01
HK1085463A1 (en) 2006-08-25
HUS1400046I1 (hu) 2017-04-28
CN1705670A (zh) 2005-12-07
EP2570418A2 (en) 2013-03-20

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