AU2013292950C1 - Nitrogenous heterocyclic derivatives and their application in drugs - Google Patents

Nitrogenous heterocyclic derivatives and their application in drugs Download PDF

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AU2013292950C1
AU2013292950C1 AU2013292950A AU2013292950A AU2013292950C1 AU 2013292950 C1 AU2013292950 C1 AU 2013292950C1 AU 2013292950 A AU2013292950 A AU 2013292950A AU 2013292950 A AU2013292950 A AU 2013292950A AU 2013292950 C1 AU2013292950 C1 AU 2013292950C1
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alkyl
alkoxy
aryl
aliphatic
heteroaryl
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AU2013292950B2 (en
AU2013292950A1 (en
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Shengtian CAO
Jing Li
Runfeng LIN
Xiaojun Wang
Zhaohe Wang
Jiancun Zhang
Yingjun Zhang
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Sunshine Lake Pharma Co Ltd
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Assigned to SUNSHINE LAKE PHARMA CO., LTD. reassignment SUNSHINE LAKE PHARMA CO., LTD. Request for Assignment Assignors: NORTH & SOUTH BROTHER PHARMACY INVESTMENT COMPANY LIMITED
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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