AU2013214909A1 - Use of laquinimod for treating Crohn's disease patients who failed first-line anti-TNFa therapy - Google Patents
Use of laquinimod for treating Crohn's disease patients who failed first-line anti-TNFa therapy Download PDFInfo
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- AU2013214909A1 AU2013214909A1 AU2013214909A AU2013214909A AU2013214909A1 AU 2013214909 A1 AU2013214909 A1 AU 2013214909A1 AU 2013214909 A AU2013214909 A AU 2013214909A AU 2013214909 A AU2013214909 A AU 2013214909A AU 2013214909 A1 AU2013214909 A1 AU 2013214909A1
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4704—2-Quinolinones, e.g. carbostyril
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
Landscapes
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- Organic Chemistry (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (1)
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- 2013-02-01 JP JP2014555758A patent/JP2015505564A/ja not_active Withdrawn
- 2013-02-01 TW TW102104087A patent/TW201345527A/zh unknown
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| BR112014018485A2 (enExample) | 2017-06-20 |
| US20150359788A1 (en) | 2015-12-17 |
| WO2013116657A1 (en) | 2013-08-08 |
| AR089862A1 (es) | 2014-09-24 |
| AU2017200472A1 (en) | 2017-02-09 |
| JP2015505564A (ja) | 2015-02-23 |
| SG11201404214QA (en) | 2014-08-28 |
| CA2862865A1 (en) | 2013-08-08 |
| HK1202776A1 (en) | 2015-10-09 |
| EA201491460A1 (ru) | 2015-01-30 |
| EP2811832A4 (en) | 2015-09-23 |
| JP2017200926A (ja) | 2017-11-09 |
| US20170290822A1 (en) | 2017-10-12 |
| IL233557A0 (en) | 2014-08-31 |
| US20130203807A1 (en) | 2013-08-08 |
| KR20140138694A (ko) | 2014-12-04 |
| CN104093310A (zh) | 2014-10-08 |
| TW201345527A (zh) | 2013-11-16 |
| CN106063787A (zh) | 2016-11-02 |
| BR112014018485A8 (pt) | 2017-07-11 |
| US9161935B2 (en) | 2015-10-20 |
| EP2811832A1 (en) | 2014-12-17 |
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