AU2006215785A1 - Novel processes for the preparation of a benzofuran - Google Patents

Novel processes for the preparation of a benzofuran Download PDF

Info

Publication number
AU2006215785A1
AU2006215785A1 AU2006215785A AU2006215785A AU2006215785A1 AU 2006215785 A1 AU2006215785 A1 AU 2006215785A1 AU 2006215785 A AU2006215785 A AU 2006215785A AU 2006215785 A AU2006215785 A AU 2006215785A AU 2006215785 A1 AU2006215785 A1 AU 2006215785A1
Authority
AU
Australia
Prior art keywords
formula
compound
pyrimidin
dimethyl
indole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2006215785A
Other languages
English (en)
Inventor
Martin Braun
Sorana Greiveldinger-Poenaru
Jurgen Jaeger
Laurent Schmitt
Peter Schneider
Chouaib Tahtaoui
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Arpida AG
Original Assignee
Arpida AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arpida AG filed Critical Arpida AG
Publication of AU2006215785A1 publication Critical patent/AU2006215785A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Indole Compounds (AREA)
AU2006215785A 2005-02-18 2006-02-10 Novel processes for the preparation of a benzofuran Abandoned AU2006215785A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EPEP/2005/001695 2005-02-18
EP2005001695 2005-02-18
PCT/EP2006/001179 WO2006087140A1 (en) 2005-02-18 2006-02-10 Novell processes for the preparation of a benzofuran

Publications (1)

Publication Number Publication Date
AU2006215785A1 true AU2006215785A1 (en) 2006-08-24

Family

ID=36283919

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2006215785A Abandoned AU2006215785A1 (en) 2005-02-18 2006-02-10 Novel processes for the preparation of a benzofuran
AU2006215788A Ceased AU2006215788B2 (en) 2005-02-18 2006-02-10 Novel processes for the preparation of a 2H-chromene

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU2006215788A Ceased AU2006215788B2 (en) 2005-02-18 2006-02-10 Novel processes for the preparation of a 2H-chromene

Country Status (22)

Country Link
US (2) US20080161561A1 (enExample)
EP (3) EP1856106A1 (enExample)
JP (2) JP2008530156A (enExample)
KR (2) KR20070106636A (enExample)
CN (4) CN101115746A (enExample)
AU (2) AU2006215785A1 (enExample)
BG (2) BG109937A (enExample)
BR (2) BRPI0607758A2 (enExample)
CA (2) CA2596668A1 (enExample)
CZ (2) CZ2007537A3 (enExample)
EE (2) EE200700051A (enExample)
HU (2) HUP0700604A3 (enExample)
IL (2) IL184404A0 (enExample)
MX (2) MX2007009282A (enExample)
NO (2) NO20073678L (enExample)
NZ (1) NZ556800A (enExample)
RO (2) RO122912B8 (enExample)
RU (2) RU2397980C2 (enExample)
TR (1) TR200705187T1 (enExample)
TW (2) TW200640912A (enExample)
WO (2) WO2006087143A1 (enExample)
ZA (2) ZA200706421B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101115746A (zh) * 2005-02-18 2008-01-30 阿皮德公开股份有限公司 用于制备苯并呋喃的新方法
US7947293B2 (en) 2008-04-08 2011-05-24 Arpida Ag Aqueous pharmaceutical formulation
MX2010011117A (es) * 2008-04-08 2011-02-24 Acino Pharma Ag Formulacion farmaceutica acuosa.
FR2949465B1 (fr) * 2009-09-01 2011-08-12 Pf Medicament Derives chromones, leur procede de preparation et leurs applications therapeutiques
CN110606831A (zh) * 2018-06-14 2019-12-24 上海度德医药科技有限公司 一种Iclaprim的新中间体及其制备方法和应用
CN110818693B (zh) * 2018-08-07 2023-06-02 上海度德医药科技有限公司 一种艾拉普林甲磺酸盐晶型b及其制备方法
CN109988156B (zh) * 2019-03-12 2021-12-28 广东中科药物研究有限公司 一种氨基嘧啶化合物
CN110372746A (zh) * 2019-07-11 2019-10-25 辽宁石油化工大学 一种合成β-胺基膦氧化合物的方法
CN110713483B (zh) * 2019-11-18 2023-04-07 上海医药工业研究院 艾拉普林中间体及艾拉普林的制备方法
CN110724135B (zh) * 2019-11-18 2023-04-28 上海医药工业研究院有限公司 一种艾拉普林中间体及其制备方法
CN110724108B (zh) * 2019-11-18 2023-04-28 上海医药工业研究院有限公司 一种艾拉普林中间体及其制备方法
CN110746361B (zh) * 2019-11-18 2023-04-21 上海医药工业研究院有限公司 一种艾拉普林中间体及其制备方法
CN110790753B (zh) * 2019-11-18 2023-04-07 上海医药工业研究院 艾拉普林对甲苯磺酸盐、其制备方法和应用
CN110818694B (zh) * 2019-11-18 2023-04-21 上海医药工业研究院有限公司 艾拉普林中间体及其应用
CN110642792B (zh) * 2019-11-18 2023-04-21 上海医药工业研究院有限公司 艾拉普林中间体的制备方法
CN113493461A (zh) * 2020-04-01 2021-10-12 上海医药工业研究院 一种七元杂环化合物或其盐、其制备方法及应用
CN117700410B (zh) * 2023-05-20 2025-07-04 山东康诺生物工程有限公司 一种3-(2-氯乙基)-2-甲基-9-羟基-4H-吡啶并[1,2-a]嘧啶-4-酮的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2709634A1 (de) * 1977-03-05 1978-09-07 Basf Ag Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4438267A (en) * 1980-11-11 1984-03-20 Daluge Susan M Monoheteroring compounds and their use
CA2238521C (en) * 1995-12-04 2005-08-16 F. Hoffmann-La Roche Ag Diaminopyrimidines, pharmaceutical compositions containing them and their use as antibacterial
WO2002010156A1 (en) * 2000-07-29 2002-02-07 Arpida Ag Benzofuran derivatives and their use as antibacterial agents
WO2003000657A1 (en) * 2001-06-20 2003-01-03 Daiichi Pharmaceutical Co., Ltd. Diamine derivatives
CN100443482C (zh) * 2003-07-11 2008-12-17 阿皮德公开股份有限公司 苯并呋喃衍生物及其在制备治疗由细菌引起的感染的药物中的用途
WO2005014586A1 (en) * 2003-08-08 2005-02-17 Arpida Ag Novel process for the preparation of 2h-chromenes
CN101115746A (zh) * 2005-02-18 2008-01-30 阿皮德公开股份有限公司 用于制备苯并呋喃的新方法

Also Published As

Publication number Publication date
IL184405A0 (en) 2007-10-31
CN102140094B (zh) 2012-06-06
RO122912B1 (ro) 2010-04-30
AU2006215788B2 (en) 2011-10-20
RO122853B1 (ro) 2010-03-30
MX2007009283A (es) 2008-02-19
NO20073701L (no) 2007-09-03
NZ556800A (en) 2011-01-28
WO2006087140A1 (en) 2006-08-24
HUP0700605A3 (en) 2008-02-28
EE200700051A (et) 2007-12-17
CN102140094A (zh) 2011-08-03
HUP0700605A2 (en) 2008-01-28
BRPI0607758A2 (pt) 2010-03-23
RU2007134583A (ru) 2009-03-27
CA2596668A1 (en) 2006-08-24
RO122912B8 (ro) 2010-09-30
RU2397980C2 (ru) 2010-08-27
CZ2007537A3 (cs) 2008-02-20
WO2006087143A8 (en) 2008-11-27
JP2008530156A (ja) 2008-08-07
ZA200706422B (en) 2008-09-25
TR200705187T1 (tr) 2007-11-21
KR20070106635A (ko) 2007-11-02
CN101115743A (zh) 2008-01-30
NO20073678L (no) 2007-09-03
MX2007009282A (es) 2008-02-19
BG109937A (bg) 2008-05-30
JP2009505943A (ja) 2009-02-12
US20080161561A1 (en) 2008-07-03
CN101115746A (zh) 2008-01-30
RU2007134584A (ru) 2009-03-27
HUP0700604A2 (en) 2008-01-28
EP1856109A1 (en) 2007-11-21
EP1856106A1 (en) 2007-11-21
IL184404A0 (en) 2007-10-31
ZA200706421B (en) 2008-11-26
EE200700050A (et) 2007-12-17
US20080221324A1 (en) 2008-09-11
KR20070106636A (ko) 2007-11-02
TW200640912A (en) 2006-12-01
CZ2007536A3 (cs) 2008-02-20
BG109938A (bg) 2008-05-30
CN102079727A (zh) 2011-06-01
CN101115743B (zh) 2011-04-13
EP2270003A1 (en) 2011-01-05
HUP0700604A3 (en) 2008-02-28
TW200640914A (en) 2006-12-01
CA2596669A1 (en) 2006-08-24
WO2006087143A1 (en) 2006-08-24
AU2006215788A1 (en) 2006-08-24
BRPI0607797A2 (pt) 2010-10-19

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Legal Events

Date Code Title Description
DA3 Amendments made section 104

Free format text: THE NATURE OF THE AMENDMENT IS: AMEND THE INVENTION TITLE TO READ NOVEL PROCESSES FOR THE PREPARATION OF A BENZOFURAN

MK4 Application lapsed section 142(2)(d) - no continuation fee paid for the application