AU2001286778B2 - Inhibitors of alpha4 mediated cell adhesion - Google Patents

Inhibitors of alpha4 mediated cell adhesion Download PDF

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Publication number
AU2001286778B2
AU2001286778B2 AU2001286778A AU2001286778A AU2001286778B2 AU 2001286778 B2 AU2001286778 B2 AU 2001286778B2 AU 2001286778 A AU2001286778 A AU 2001286778A AU 2001286778 A AU2001286778 A AU 2001286778A AU 2001286778 B2 AU2001286778 B2 AU 2001286778B2
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Australia
Prior art keywords
compound
group
dimethoxy
phenylalanine
formula
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Ceased
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AU2001286778A
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AU2001286778A1 (en
Inventor
Takayuki Kawaguchi
Toshiyuki Kume
Sumihiro Nomura
Ila Sircar
Mikiko Tsukimoto
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Mitsubishi Tanabe Pharma Corp
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Tanabe Seiyaku Co Ltd
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Publication of AU2001286778B2 publication Critical patent/AU2001286778B2/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
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  • Neurosurgery (AREA)
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  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Dermatology (AREA)
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  • Psychiatry (AREA)
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  • AIDS & HIV (AREA)
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  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
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AU2001286778A 2000-08-31 2001-08-27 Inhibitors of alpha4 mediated cell adhesion Ceased AU2001286778B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22912800P 2000-08-31 2000-08-31
US60/229,128 2000-08-31
PCT/US2001/026594 WO2002018320A2 (en) 2000-08-31 2001-08-27 INHIBITORS OF α4 MEDIATED CELL ADHESION

Publications (2)

Publication Number Publication Date
AU2001286778A1 AU2001286778A1 (en) 2002-06-06
AU2001286778B2 true AU2001286778B2 (en) 2005-02-10

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Application Number Title Priority Date Filing Date
AU2001286778A Ceased AU2001286778B2 (en) 2000-08-31 2001-08-27 Inhibitors of alpha4 mediated cell adhesion
AU8677801A Pending AU8677801A (en) 2000-08-31 2001-08-27 Inhibitors of alpha4 mediated cell adhesion

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU8677801A Pending AU8677801A (en) 2000-08-31 2001-08-27 Inhibitors of alpha4 mediated cell adhesion

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US (6) US7026501B2 (cg-RX-API-DMAC7.html)
EP (1) EP1315694B1 (cg-RX-API-DMAC7.html)
JP (1) JP3899022B2 (cg-RX-API-DMAC7.html)
KR (1) KR100528049B1 (cg-RX-API-DMAC7.html)
CN (1) CN1229334C (cg-RX-API-DMAC7.html)
AR (1) AR034556A1 (cg-RX-API-DMAC7.html)
AT (1) ATE292615T1 (cg-RX-API-DMAC7.html)
AU (2) AU2001286778B2 (cg-RX-API-DMAC7.html)
BR (1) BR0113629A (cg-RX-API-DMAC7.html)
CA (1) CA2418054C (cg-RX-API-DMAC7.html)
CZ (1) CZ303460B6 (cg-RX-API-DMAC7.html)
DE (1) DE60109943T2 (cg-RX-API-DMAC7.html)
DK (1) DK1315694T3 (cg-RX-API-DMAC7.html)
ES (1) ES2240509T3 (cg-RX-API-DMAC7.html)
HK (1) HK1052684B (cg-RX-API-DMAC7.html)
HU (1) HUP0302693A3 (cg-RX-API-DMAC7.html)
IL (2) IL154305A0 (cg-RX-API-DMAC7.html)
MX (1) MXPA03001837A (cg-RX-API-DMAC7.html)
MY (1) MY129000A (cg-RX-API-DMAC7.html)
NO (1) NO327861B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ524043A (cg-RX-API-DMAC7.html)
PL (1) PL206656B1 (cg-RX-API-DMAC7.html)
PT (1) PT1315694E (cg-RX-API-DMAC7.html)
RU (1) RU2250895C2 (cg-RX-API-DMAC7.html)
SI (1) SI1315694T1 (cg-RX-API-DMAC7.html)
TW (1) TWI224587B (cg-RX-API-DMAC7.html)
WO (1) WO2002018320A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA200301039B (cg-RX-API-DMAC7.html)

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