AU2001252372A1 - Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by the NP Y5 receptor - Google Patents
Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by the NP Y5 receptorInfo
- Publication number
- AU2001252372A1 AU2001252372A1 AU2001252372A AU5237201A AU2001252372A1 AU 2001252372 A1 AU2001252372 A1 AU 2001252372A1 AU 2001252372 A AU2001252372 A AU 2001252372A AU 5237201 A AU5237201 A AU 5237201A AU 2001252372 A1 AU2001252372 A1 AU 2001252372A1
- Authority
- AU
- Australia
- Prior art keywords
- amino
- alkyl
- carbamoyl
- formula
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/76—Dibenzothiophenes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Emergency Medicine (AREA)
- Anesthesiology (AREA)
- Endocrinology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0010757 | 2000-05-05 | ||
| GBGB0010757.3A GB0010757D0 (en) | 2000-05-05 | 2000-05-05 | Chemical compounds |
| PCT/GB2001/001899 WO2001085714A1 (en) | 2000-05-05 | 2001-05-01 | Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by the np y5 receptor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001252372A1 true AU2001252372A1 (en) | 2001-11-20 |
Family
ID=9890945
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001252372A Abandoned AU2001252372A1 (en) | 2000-05-05 | 2001-05-01 | Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by the NP Y5 receptor |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US6967216B2 (ko) |
| EP (1) | EP1278739A1 (ko) |
| JP (1) | JP2003532723A (ko) |
| KR (1) | KR20020093975A (ko) |
| CN (1) | CN1440401A (ko) |
| AR (1) | AR028414A1 (ko) |
| AU (1) | AU2001252372A1 (ko) |
| BR (1) | BR0110548A (ko) |
| CA (1) | CA2406634A1 (ko) |
| GB (1) | GB0010757D0 (ko) |
| IL (1) | IL152230A0 (ko) |
| MX (1) | MXPA02010563A (ko) |
| NO (1) | NO20025286L (ko) |
| NZ (1) | NZ522188A (ko) |
| WO (1) | WO2001085714A1 (ko) |
| ZA (1) | ZA200208674B (ko) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN111825689A (zh) * | 2019-04-17 | 2020-10-27 | 中国医药研究开发中心有限公司 | 一种二氢吡唑啉酮类化合物的新晶型及其制备方法 |
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| EP1657240A4 (en) | 2003-08-18 | 2009-04-08 | Fujifilm Finechemicals Co Ltd | PYRIDYLTETRAHYDROPYRIDINE, PYRIDYLPIPERIDINE AND METHOD FOR THE PRODUCTION THEREOF |
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| TW200624427A (en) | 2004-09-20 | 2006-07-16 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
| WO2006034315A2 (en) * | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes |
| BRPI0515482A (pt) * | 2004-09-20 | 2008-07-22 | Xenon Pharmaceuticals Inc | derivados heterocìclicos e seus usos como agentes terapêuticos |
| WO2006034338A1 (en) * | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as mediators of stearoyl-coa desaturase |
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| BRPI0515488A (pt) * | 2004-09-20 | 2008-07-29 | Xenon Pharmaceuticals Inc | derivados de heterocìclicos e seu uso como agentes terapêuticos |
| EP2127676A3 (en) | 2004-11-01 | 2013-09-04 | Amylin Pharmaceuticals, LLC | Treatment of obesity and related disorders |
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| JPH1174077A (ja) | 1997-08-28 | 1999-03-16 | Junji Kido | ビニル系重合体を用いた積層型エレクトロルミネッセンス素子 |
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| AUPP285898A0 (en) | 1998-04-07 | 1998-04-30 | Fujisawa Pharmaceutical Co., Ltd. | Amido derivatives |
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| ATE329911T1 (de) | 1998-08-07 | 2006-07-15 | Applied Research Systems | Fsh mimetika zur behandlung von infertilität |
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| AU6190299A (en) | 1998-10-21 | 2000-05-08 | Dr. Reddy's Research Foundation | New compounds, their preparation and use |
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| GB0011013D0 (en) | 2000-05-09 | 2000-06-28 | Astrazeneca Ab | Chemical compounds |
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| NZ526623A (en) | 2000-12-22 | 2004-11-26 | Astrazeneca Ab | Carbazole derivatives and their use as neuropeptide Y5 receptor ligands |
| GB0121941D0 (en) | 2001-09-11 | 2001-10-31 | Astrazeneca Ab | Chemical compounds |
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2000
- 2000-05-05 GB GBGB0010757.3A patent/GB0010757D0/en not_active Ceased
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2001
- 2001-05-01 JP JP2001582315A patent/JP2003532723A/ja active Pending
- 2001-05-01 MX MXPA02010563A patent/MXPA02010563A/es unknown
- 2001-05-01 WO PCT/GB2001/001899 patent/WO2001085714A1/en active IP Right Grant
- 2001-05-01 BR BR0110548-5A patent/BR0110548A/pt not_active IP Right Cessation
- 2001-05-01 KR KR1020027014772A patent/KR20020093975A/ko not_active Application Discontinuation
- 2001-05-01 EP EP01925687A patent/EP1278739A1/en not_active Withdrawn
- 2001-05-01 AU AU2001252372A patent/AU2001252372A1/en not_active Abandoned
- 2001-05-01 CA CA002406634A patent/CA2406634A1/en not_active Abandoned
- 2001-05-01 US US10/275,529 patent/US6967216B2/en not_active Expired - Fee Related
- 2001-05-01 NZ NZ522188A patent/NZ522188A/en unknown
- 2001-05-01 IL IL15223001A patent/IL152230A0/xx unknown
- 2001-05-01 CN CN01812237A patent/CN1440401A/zh active Pending
- 2001-05-04 AR ARP010102135A patent/AR028414A1/es not_active Application Discontinuation
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2002
- 2002-10-25 ZA ZA200208674A patent/ZA200208674B/en unknown
- 2002-11-04 NO NO20025286A patent/NO20025286L/no not_active Application Discontinuation
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2005
- 2005-05-12 US US11/127,582 patent/US7332492B2/en not_active Expired - Lifetime
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN111825689A (zh) * | 2019-04-17 | 2020-10-27 | 中国医药研究开发中心有限公司 | 一种二氢吡唑啉酮类化合物的新晶型及其制备方法 |
| CN111825689B (zh) * | 2019-04-17 | 2023-05-05 | 中国医药研究开发中心有限公司 | 一种二氢吡唑啉酮类化合物的晶型及其制备方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1278739A1 (en) | 2003-01-29 |
| US20030225097A1 (en) | 2003-12-04 |
| IL152230A0 (en) | 2003-05-29 |
| MXPA02010563A (es) | 2003-03-10 |
| US6967216B2 (en) | 2005-11-22 |
| US7332492B2 (en) | 2008-02-19 |
| CN1440401A (zh) | 2003-09-03 |
| WO2001085714A1 (en) | 2001-11-15 |
| AR028414A1 (es) | 2003-05-07 |
| ZA200208674B (en) | 2004-02-10 |
| US20050209233A1 (en) | 2005-09-22 |
| NZ522188A (en) | 2004-04-30 |
| BR0110548A (pt) | 2003-04-01 |
| NO20025286D0 (no) | 2002-11-04 |
| KR20020093975A (ko) | 2002-12-16 |
| GB0010757D0 (en) | 2000-06-28 |
| NO20025286L (no) | 2002-11-04 |
| JP2003532723A (ja) | 2003-11-05 |
| CA2406634A1 (en) | 2001-11-15 |
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| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |