ATE502020T1 - Benzamid und heteroarylamid als p2x7- rezeptorantagonisten - Google Patents

Benzamid und heteroarylamid als p2x7- rezeptorantagonisten

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Publication number
ATE502020T1
ATE502020T1 AT02783358T AT02783358T ATE502020T1 AT E502020 T1 ATE502020 T1 AT E502020T1 AT 02783358 T AT02783358 T AT 02783358T AT 02783358 T AT02783358 T AT 02783358T AT E502020 T1 ATE502020 T1 AT E502020T1
Authority
AT
Austria
Prior art keywords
heteroarylamide
benzamide
receptor antagonists
antagonists
receptor
Prior art date
Application number
AT02783358T
Other languages
English (en)
Inventor
Allen DUPLANTIER
Chakrapani Subramanyam
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of ATE502020T1 publication Critical patent/ATE502020T1/de

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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D253/00—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/06—1,2,4-Triazines
    • C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/07—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D253/075—Two hetero atoms, in positions 3 and 5
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    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
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    • C07D263/18—Oxygen atoms
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AT02783358T 2001-11-12 2002-11-04 Benzamid und heteroarylamid als p2x7- rezeptorantagonisten ATE502020T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33678101P 2001-11-12 2001-11-12
PCT/IB2002/004613 WO2003042191A1 (en) 2001-11-12 2002-11-04 Benzamide and heteroarylamide as p2x7 receptor antagonists

Publications (1)

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ATE502020T1 true ATE502020T1 (de) 2011-04-15

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AT02783358T ATE502020T1 (de) 2001-11-12 2002-11-04 Benzamid und heteroarylamid als p2x7- rezeptorantagonisten

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EP (1) EP1448535B1 (de)
JP (1) JP4365218B2 (de)
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AP (1) AP2004003028A0 (de)
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AT (1) ATE502020T1 (de)
BR (1) BR0214044A (de)
CA (1) CA2466724C (de)
CY (1) CY1111405T1 (de)
DE (1) DE60239485D1 (de)
DK (1) DK1448535T3 (de)
EA (1) EA200400488A1 (de)
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