ATE378336T1 - Imidazopyridine als hemmstoffe cyclin abhängiger kinasen - Google Patents

Imidazopyridine als hemmstoffe cyclin abhängiger kinasen

Info

Publication number
ATE378336T1
ATE378336T1 AT03786514T AT03786514T ATE378336T1 AT E378336 T1 ATE378336 T1 AT E378336T1 AT 03786514 T AT03786514 T AT 03786514T AT 03786514 T AT03786514 T AT 03786514T AT E378336 T1 ATE378336 T1 AT E378336T1
Authority
AT
Austria
Prior art keywords
imidazopyridines
inhibitors
cyclin dependent
dependent kinases
kinases
Prior art date
Application number
AT03786514T
Other languages
English (en)
Inventor
Michael Dwyer
Timothy Guzi
Kamil Paruch
Ronald Doll
Kartik Keertikar
Viyyoor Girijavallabhan
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of ATE378336T1 publication Critical patent/ATE378336T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT03786514T 2002-09-19 2003-09-17 Imidazopyridine als hemmstoffe cyclin abhängiger kinasen ATE378336T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41206302P 2002-09-19 2002-09-19

Publications (1)

Publication Number Publication Date
ATE378336T1 true ATE378336T1 (de) 2007-11-15

Family

ID=32030794

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03786514T ATE378336T1 (de) 2002-09-19 2003-09-17 Imidazopyridine als hemmstoffe cyclin abhängiger kinasen

Country Status (18)

Country Link
US (2) US6992080B2 (de)
EP (1) EP1539756B1 (de)
JP (1) JP4845379B2 (de)
KR (1) KR20050052500A (de)
CN (1) CN100549011C (de)
AR (1) AR041291A1 (de)
AT (1) ATE378336T1 (de)
AU (1) AU2003295332B2 (de)
CA (1) CA2499639C (de)
DE (1) DE60317529T2 (de)
ES (1) ES2293068T3 (de)
IL (1) IL167433A (de)
MX (1) MXPA05003058A (de)
MY (1) MY133311A (de)
NZ (1) NZ538566A (de)
TW (1) TWI351405B (de)
WO (1) WO2004026867A2 (de)
ZA (1) ZA200502278B (de)

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CN102015693B (zh) 2008-02-21 2014-10-29 默沙东公司 作为erk抑制剂的化合物
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GB0906472D0 (en) 2009-04-15 2009-05-20 Astex Therapeutics Ltd New compounds
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PH12012500778A1 (en) 2009-10-30 2012-11-26 Janssen Pharmaceutica Nv IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS
AR080754A1 (es) 2010-03-09 2012-05-09 Janssen Pharmaceutica Nv Derivados de imidazo (1,2-a) pirazina y su uso como inhibidores de pde10
JP5938352B2 (ja) 2010-03-11 2016-06-22 ギリアード コネチカット， インコーポレイテッド イミダゾピリジンｓｙｋ阻害剤
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CN106687139A (zh) 2014-07-14 2017-05-17 吉利德科学公司 用于治疗癌症的组合
CN108700594B (zh) 2015-11-18 2021-06-29 建新公司 多囊性肾病的生物标志物及其用途
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Also Published As

Publication number Publication date
CA2499639C (en) 2011-11-08
HK1071757A1 (en) 2005-07-29
WO2004026867A2 (en) 2004-04-01
AU2003295332A1 (en) 2004-04-08
AU2003295332B2 (en) 2007-01-18
TW200407322A (en) 2004-05-16
MY133311A (en) 2007-11-30
AR041291A1 (es) 2005-05-11
JP4845379B2 (ja) 2011-12-28
WO2004026867A3 (en) 2004-08-05
DE60317529D1 (de) 2007-12-27
IL167433A (en) 2011-03-31
JP2006507254A (ja) 2006-03-02
KR20050052500A (ko) 2005-06-02
US7452902B2 (en) 2008-11-18
ZA200502278B (en) 2006-05-31
US20060030555A1 (en) 2006-02-09
TWI351405B (en) 2011-11-01
ES2293068T3 (es) 2008-03-16
US6992080B2 (en) 2006-01-31
EP1539756A2 (de) 2005-06-15
CA2499639A1 (en) 2004-04-01
US20040097517A1 (en) 2004-05-20
DE60317529T2 (de) 2008-09-25
CN100549011C (zh) 2009-10-14
MXPA05003058A (es) 2005-05-27
CN1703414A (zh) 2005-11-30
EP1539756B1 (de) 2007-11-14
NZ538566A (en) 2008-02-29

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