AR094932A1 - Formas sólidas de derivados heterocíclicos bicíclicos - Google Patents

Formas sólidas de derivados heterocíclicos bicíclicos

Info

Publication number
AR094932A1
AR094932A1 ARP140100645A ARP140100645A AR094932A1 AR 094932 A1 AR094932 A1 AR 094932A1 AR P140100645 A ARP140100645 A AR P140100645A AR P140100645 A ARP140100645 A AR P140100645A AR 094932 A1 AR094932 A1 AR 094932A1
Authority
AR
Argentina
Prior art keywords
methyl
pyridin
carboxamide
carbamoyl
dimethyl
Prior art date
Application number
ARP140100645A
Other languages
English (en)
Inventor
Furet Pascal
Chamoin Sylvie
Yeh Vince
Loren Jon
Molteni Valentina
Paul Collingwood Stephen
Bruce Ian
Shaw Duncan
Lewis Sarah
Michael Saunders Alex
Furminger Vikki
Turner Roy
Lv Lin
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of AR094932A1 publication Critical patent/AR094932A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Reivindicación 1: Un compuesto seleccionado a partir de: tartrato de N-(5-(2-(2,2-dimetil-pirrolidin-1-iI)-etil-carbamoil)-2-metil-piridin-3-il)-6-(1-metil-1H-pirazol-4-il)-pirazolo-[1,5-a]-piridin-3-carboxamida; complejo de N-(5-(2-(2,2-dimetil-pirrolidin-1-iI)-etil-carbamoil)-2-metil-piridin-3-il)-6-(1-metil-1H-pirazol-4-il)-pirazolo-[1,5-a]-piridin-3-carboxamida y Sacarina; maleato de N-(5-(2-(2,6-cis-dimetil-piperidin-1-il)-etil-carbamoil)-2-fluoro-fenil)-7-(1-metil-1H-pirazol-5-iI)-imidazo-[1,2-a]-piridin-3-carboxamida; y sacarinato de N-(5-(2-(2,6-cis-dimetil-piperidin-1-iI)-etil-carbamoil)-2-fluoro-fenil)-7-(1-metil-1H-pirazol-5-il)-imidazo-[1,2-a]-piridin-3-carboxamida. Reivindicación 4: Una forma cristalina de un compuesto seleccionado a partir de: L-tartrato de N-(5-(2-(2,2-dimetil-pirrolidin-1-iI)-etil-carbamoil)-2-metil-piridin-3-il)-6-(1-metil-1H-pirazol-4-il)-pirazolo-[1,5-a]-piridin-3-carboxamida; complejo de N-(5-(2-(2,2-dimetil-pirrolidin-1-il)-etil-carbamoil)-2-metil-piridin-3-il)-6-(1-metil-1H-pirazol-4-il)-pirazolo-[1,5-a]-piridin-3-carboxamida y Sacarina; maleato de N-(5-(2-(2,6-cis-dimetil-piperidin-1-iI)-etil-carbamoil)-2-fluoro-fenil)-7-(1-metil-1H-pirazol-5-il)-imidazo-[1,2-a]-piridin-3-carboxamida; y sacarinato de N-(5-(2-(2,6-cis-dimetil-piperidin-1-iI)-etil-carbamoil)-2-fluoro-fenil)-7-(1-metil-1H-pirazol-5-il)-imidazo-[1,2-a]-piridin-3-carboxamida.
ARP140100645A 2013-03-01 2014-02-28 Formas sólidas de derivados heterocíclicos bicíclicos AR094932A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN2013072060 2013-03-01

Publications (1)

Publication Number Publication Date
AR094932A1 true AR094932A1 (es) 2015-09-09

Family

ID=50288206

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140100645A AR094932A1 (es) 2013-03-01 2014-02-28 Formas sólidas de derivados heterocíclicos bicíclicos

Country Status (4)

Country Link
US (1) US9073921B2 (es)
AR (1) AR094932A1 (es)
TW (1) TW201443050A (es)
WO (1) WO2014132220A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11179376B2 (en) * 2017-12-20 2021-11-23 Sunshine Lake Pharma Co., Ltd. Salts of pyrazolo[1,5-a]pyridine derivative and use thereof

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