AR077791A1 - Pesticidas mesoionicos - Google Patents

Pesticidas mesoionicos

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Publication number
AR077791A1
AR077791A1 ARP100102878A ARP100102878A AR077791A1 AR 077791 A1 AR077791 A1 AR 077791A1 AR P100102878 A ARP100102878 A AR P100102878A AR P100102878 A ARP100102878 A AR P100102878A AR 077791 A1 AR077791 A1 AR 077791A1
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AR
Argentina
Prior art keywords
independently selected
ring
cycloalkylalkyl
alkyl
halogen
Prior art date
Application number
ARP100102878A
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English (en)
Inventor
Ming Xu
My-Hanh Thi Tong
Kenneth Andrew Hughes
Wenming Zhang
Jr Caleb William Holyoke
George P Lahm
Jr Thomas Francis Pahutski
Original Assignee
Du Pont
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Publication of AR077791A1 publication Critical patent/AR077791A1/es

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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
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    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/22—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing ingredients stabilising the active ingredients
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    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/32—Ingredients for reducing the noxious effect of the active substances to organisms other than pests, e.g. toxicity reducing compositions, self-destructing compositions
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
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    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
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    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
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    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
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    • C07D513/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
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  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Toxicology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Catching Or Destruction (AREA)
  • Fodder In General (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

También se describen las composiciones que contienen los compuestos de la formula (1) y los métodos para controlar una plaga de invertebrados; el método comprende la etapa de poner la plaga de invertebrados o su ambiente en contacto con una cantidad biologicamente eficaz de un compuesto o una composicion de la presente solicitud. Reivindicacion 1: Un compuesto de la formula (1), un N-oxido, o sal de éste, caracterizado porque X es O o S; Y es O o S; A es O, S, NR3e o C(R3c)=C(R3d), siempre que la porcion C(R3c)=C(R3d) se oriente de manera que el átomo de carbono enlazado a R3d se conecte directamente al anillo de pirimidinio de la formula (1); Z es un enlace directo, O, S(O)n, NR6, C(R7)2O, OC(R7)2, C(=X1), C(=X1)E, EC(=X1), C(=NOR8) o C(=NN(R6)2); X1 es O, S o NR9; E es O, S o NR9a; R1 es H, halogeno, ciano, CHO, C(=O)OH, C(=O)NH2 o C(=S)NH2; o alquilo C1-8, alquenilo C2-8, alquinilo C2-8, cicloalquilo C3-10, alquilcicloalquilo C4-10, cicloalquilalquilo C4-10, cicloalquilcicloalquilo C6-14, alquilcicloalquilalquilo C5-10 o cicloalquenilo C3-6, cada uno insustituido o sustituido con al menos un sustituyente independientemente seleccionado del grupo consistente de halogeno, ciano, nitro, CHO, C(=O)OH, C(=O)NH2, C(=O)R10, C(=O)OR11, C(=O)NR12R13, C(=O)NR21NR22R23, OR11, S(O)nR10, SO2NR12R13, S(=O)(=NR21)R22, Si(R10)3 y Z1Qt; o un anillo de 3 a 10 miembros o un sistema anular de 7 a 11 miembros, cada anillo o sistema anular contiene miembros anulares seleccionados de átomos de carbono y hasta 4 heteroátomos independientemente seleccionados de hasta 2 O, hasta 2 S, y hasta 4 N, en donde hasta 3 miembros anulares del átomo de carbono son independientemente seleccionados de C(=O) y C(=S) y los miembros anulares del átomo de azufre son independientemente seleccionados de S(=O)u(=NR24)z, cada anillo o sistema anular opcionalmente sustituido con hasta 5 sustituyentes independientemente seleccionados de R14 siempre y cuando R1 sea halogeno, entonces Z es un enlace directo, S(=O), S(=O)2, OC(R7)2, C(=X1), EC(=X1), C(=NOR8) o C(=NN(R6)2); R2 es H, halogeno, ciano, hidroxi, amino, nitro, OCN, SCN, CHO, C(=O)OH, C(=O)NH2, C(=S)NH2, SO2NH2, C(=O)R18, C(=O)OR18, NHR18, NR18R19, C(=O)NR21R19, C(=S)NR21R19, SO2NR21R19, OC(=O)R21, OC(=O)OR18, OC(=O)NR21 R19, N(R21)C(=O)R21, N(R21)C(=O)OR19, N(R21)C(=O)NR21R22, OSO2R18, OSO2NR21R22, NR21SO2R18, NR21SO2NR21R22 o Si(R18R19R20); o alquilo C1-8, alquenilo C2-8, alquinilo C2-8, cicloalquilo C3-10, alquilcicloalquilo C4-10, cicloalquilalquilo C4-10, cicloalquilcicloalquilo C6-14, alquilcicloalquilalquilo C5-10, cicloalquenilo C3-8, alcoxi C1-8, cicloalcoxi C3-8, cicloalquilalcoxi C4-10, alqueniloxi C2-8, alquiniloxi C2-8, alquiltio C1-8, alquilsulfinilo C1-8, alquilsulfonilo C1-8, cicloalquiltio C3-8, cicloalquilsulfinilo C3-8, cicloalquilsulfonilo C3-8, cicloalquilalquiltio C4-10, cicloalquilalquilsulfinilo C4-10, cicloalquilalquilsulfonilo C4-10, alqueniltio C2-8, alquenilsulfinilo C2-8, alquenilsulfonilo C2-8, alquiniltio C2-8, alquinilsulfinilo C2-8 o alquinilsulfonilo C2-8, cada uno insustituido o sustituido con al menos un sustituyente independientemente seleccionado del grupo consistente de halogeno, ciano, nitro, CHO, C(=O)OH, C(=O)NH2, C(=O)R10, C(=O)OR11, C(=O)NR12R13, OR11, S(O)nR10, SO2NR12R13 y Si(R10)3; o un anillo de 3 a 10 miembros o un sistema anular de 7 a 11 miembros, cada anillo o sistema anular contiene miembros anulares seleccionados de átomos de carbono y hasta 4 heteroátomos independientemente seleccionados de hasta 2 O, hasta 2 S, y hasta 4 N, en donde hasta 3 miembros anulares del átomo de carbono son independientemente seleccionados de C(=O) y C(=S) y los miembros anulares del átomo de azufre son independientemente seleccionados de S(=O)u(=NR24)z, cada anillo o sistema anular opcionalmente sustituido con hasta 5 sustituyentes independientemente seleccionados de R15; R3a, R3b, R3c y R3d son independientemente H, halogeno, ciano, hidroxi, amino, nitro, SF5, OCN, SCN, CHO, C(=O)OH, C(=O)NH2, C(=S)NH2, SO2NH2, C(=O)R18, C(=O)OR18, NHR18, NR18R19, C(=O)NR21R19, C(=S)NR21R19, SO2NR21R19, OC(=O)R21, OC(=O)OR18, OC(=O)NR21R19, N(R21)C(=O)R21, N(R21)C(=O)OR19, N(R21)C(=O)NR21R22, OSO2R18, OSO2NR21R22, NR21 SO2R18, NR21SO2NR21R22, Si(R18R19R20) o Z1Qt; o alquilo C1-8, alquenilo C2-8, alquinilo C2-8, cicloalquilo C3-10, alquilcicloalquilo C4-10, cicloalquilalquilo C4-10, cicloalquilcicloalquilo C6-14, alquilcicloalquilalquilo C5-10, cicloalquenilo C3-8, alcoxi C1-8, cicloalcoxi C3-8, cicloalquilalcoxi C4-10, alqueniloxi C2-8, alquiniloxi C2-8, alquiltio C1-8, alquilsulfinilo C1-8, alquilsulfonilo C1-8, cicloalquiltio C3-8, cicloalquilsulfinilo C3-8, cicloalquilsulfonilo C3-8, cicloalquilalquiltio C4-10, cicloalquilalquilsulfinilo C4-10, cicloalquilalquilsulfonilo C4-10, alqueniltio C2-8, alquenilsulfinilo C2-8, alquenilsulfonilo C2-8, alquiniltio C2-8, alquinilsulfinilo C2-8 o alquinilsulfonilo C2-8, cada uno insustituido o sustituido con al menos un sustituyente independientemente seleccionado de R17; o R3a y R3b, o R3b y R3c, o R3c y R3d se toman juntos con los átomos de carbono adyacentes a los cuales están unidos para formar un anillo heterocíclico o carbocíclico de 5 a 7 miembros, cada anillo contiene miembros anulares seleccionados de átomos de carbono y hasta 3 heteroátomos independientemente seleccionados de hasta 2 O, hasta 2 S, y hasta 3 N, en donde hasta 2 miembros anulares del átomo de carbono son independientemente seleccionados de C(=O) y C(=S) y los miembros anulares del átomo de azufre son independientemente seleccionados de S(=O)n, cada anillo opcionalmente sustituido con hasta 3 sustituyentes independientemente seleccionados del grupo consistente de halogeno, ciano, hidroxi, amino, nitro, C(=O)OH, C(=O)NH2, SO2NH2, alquilo C1-4, haloalquilo C1-4, alquenilo C2-4, haloalquenilo C2-4, alquinilo C2-4, haloalquinilo C2-4, cicloalquilo C3-7, halocicloalquilo C3-7, alquilcicloalquilo C4-8, haloalquilcicloalquilo C4-8, cicloalquilalquilo C4-8, halocicloalquilalquilo C4-8, alcoxi C1-6, haloalcoxi C1-6, alcoxicarbonilo C2-6, haloalcoxicarbonilo C2-6, alquilcarbonilo C2-6 y haloalquilcarbonilo C2-6; R3e es H, hidroxi, amino, CHO, C(=O)NH2, C(=S)NH2, SO2NH2, C(=O)R18, C(=O)OR18, NHR18, NR18R19, C(=O)NR21R19, C(=S)NR21R19, SO2NR21R19, OC(=O)R21, OC(=O)OR18, OC(=O)NR21R19, N(R21)C(=O)R21, N(R21)C(=O)OR19 , N(R21)C(=O)NR21R22, OSO2R18, OSO2NR21R22, NR21SO2R18, NR21SO2NR21R22, Si(R18R19R20) o Z1Qt; o alquilo C1-8, alquenilo C2-8, alquinilo C2-8, cicloalquilo C3-10, alquilcicloalquilo C4-10, cicloalquilalquilo C4-10, cicloalquilcicloalquilo C6-14, alquilcicloalquilalquilo C5-10, cicloalquenilo C3-8, alcoxi C1-8, cicloalcoxi C3-8, cicloalquilalcoxi C4-10, alqueniloxi C2-8, alquiniloxi C2-8, alquilsulfinilo C1-8, alquilsulfonilo C1-8, cicloalquilsulfinilo C3-8, cicloalquilsulfonilo C3-8, cicloalquilalquilsulfinilo C4-10, cicloalquilalquilsulfonilo C4-10, alquenilsulfinilo C2-8, alquenilsulfonilo C2-8, alquinilsulfinilo C2-8 o alquinilsulfonilo C2-8, cada uno insustituido o sustituido con al menos un sustituyente independientemente seleccionado de R17; o R3e y R3b, se toman juntos con los átomos de carbono adyacentes a los cuales están unidos para formar un anillo heterocíclico o carbocíclico de 5 a 7 miembros, cada anillo contiene miembros anulares seleccionados de átomos de carbono y hasta 3 heteroátomos independientemente seleccionados de hasta 2 O, hasta 2 S, y hasta 3 N, en donde hasta 2 miembros anulares del átomo de carbono son independientemente seleccionados de C(=O) y C(=S) y los miembros anulares del átomo de azufre son independientemente seleccionados de S(=O)n, cada anillo opcionalmente sustituido con hasta 3 sustituyentes independientemente seleccionados del grupo consistente de halogeno, ciano, hidroxi, amino, nitro, C(=O)OH, C(=O)NH2, SO2NH2, alquilo C1-4, haloalquilo C1-4, alquenilo C2-4, haloalquenilo C2-4, alquinilo C2-4, haloalquinilo C2-4, cicloalquilo C3-7, halocicloalquilo C3-7, alquilcicloalquilo C4-8, haloalquilcicloalquilo C4-8, cicloalquilalquilo C4-8, halocicloalquilalquilo C4-8, alcoxi C1-6, haloalcoxi C1-6, alcoxicarbonilo C2-6, haloalcoxicarbonilo C2-6, alquilcarbonilo C2-6 y haloalquilcarbonilo C2-6; cada R4 y R5 es independientemente H, halogeno, ciano, hidroxi, amino, nitro, OCN, SCN, CHO, C(=O)OH, C(=O)NH2, C(=S)NH2, o SO2NH2, o alquilo C1-6, alquenilo C2-6, alquinilo C2-6, cicloalquilo C3-8, alquilcicloalquilo C4-8, cicloalquilalquilo C4-8, cicloalquilcicloalquilo C6-12, alquilcicloalquilalquilo C5-8, cicloalquenilo C3-6, alcoxi C1-6, cicloalcoxi C3-6, cicloalquilalcoxi C4-8, alqueniloxi C2-6, alquiniloxi C2-6, cada uno insustituido o sustituido con al menos un sustituyente independientemente seleccionado del grupo consistente de halogeno, ciano, nitro, CHO, C(=O)OH, C(=O)NH2, C(=O)R10, C(=O)OR11; C(=O)NR12R13, OR11, S(O)nR10, SO2NR12R13 y Si(R10)3; o R4 y R5 se toman juntos con el átomo de carbono al cual están unidos para formar un anillo de 3 a 7 miembros que contiene miembros anulares seleccionados de átomos de carbono y hasta 2 heteroátomos independientemente seleccionados de un O, un S, y hasta 2 N, en donde hasta 2 miembros anulares del átomo de carbono son independientemente seleccionados de C(=O) y C(=S) y el miembro anular del átomo de azufre es seleccionado de S, S(O) o S(O)2, dicho anillo opcionalmente sustituido con hasta 4 sustituyentes independientemente seleccionados del grupo consistente de halogeno, ciano y alquilo C1-4; cada R6 es independientemente H; o alquilo C1-6, alquenilo C2-6, alquinilo C2-6, cicloalquilo C3-8, alquilcicloalquilo C4-8, cicloalquilalquilo C4-8, cicloalquilcicloalquilo C6-10, alquilcicloalquilalquilo C5-10, cicloalquenilo C3-6, alquilcarbonilo C2-6 o alcoxicarbonilo C2-6, cada uno insustituido o sustituido con al menos un sustituyente independientemente seleccionado del grupo consistente de halogeno, ciano, nitro, CHO, C(=O)OH, C(=O)NH2, C(=O)R10, C(=O)OR11, C(=O)NR12R13, OR11, S(O)nR10, SO2NR12
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