AR024423A1 - PROCESO PARA LA PREPARACIoN DE TIAMETOXAM. - Google Patents

PROCESO PARA LA PREPARACIoN DE TIAMETOXAM.

Info

Publication number
AR024423A1
AR024423A1 ARP000103082A ARP000103082A AR024423A1 AR 024423 A1 AR024423 A1 AR 024423A1 AR P000103082 A ARP000103082 A AR P000103082A AR P000103082 A ARP000103082 A AR P000103082A AR 024423 A1 AR024423 A1 AR 024423A1
Authority
AR
Argentina
Prior art keywords
formula
hydrogen
alkyl
cycloalkyl
optionally substituted
Prior art date
Application number
ARP000103082A
Other languages
English (en)
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR024423A1 publication Critical patent/AR024423A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C257/00—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
    • C07C257/10—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
    • C07C257/22—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having nitrogen atoms of amidino groups further bound to nitrogen atoms, e.g. hydrazidines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C261/00—Derivatives of cyanic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C277/00—Preparation of guanidine or its derivatives, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C277/08—Preparation of guanidine or its derivatives, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups of substituted guanidines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D307/10—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/14—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyridine Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)

Abstract

Un método para producir compuestos de la formula 1 en donde: R1 es hidrogeno o alquilo C1-4; R2 es hidrogeno, alquilo C1-8, cicloalquilo C3-6, o unradical -N(R3)R4; o R2 y R6 son juntos -CH2-CH2-S-; R3 y R4, son hidrogeno, alquiloC1-4, cicloalquiloC 3-6, o un radical -CH2B; R6 es hidrogeno, alquilo C1-8,arilo o bencilo; o R3 y R6 son juntos -CH2-CH2-, -CH2-CH2-CH2-, -CH2-O-CH2, CH2-S-CH2- o -CH2-N(R5)-CH2-; X es CH-CN, CH-NO2 o N-NO2; A es un radicalheterocíclico, monocíclico o bíciclico,aromát ico o no aromático, opcionalmente sustituido; y B es fenilo, 3-piridilo, o tiazolilo opcionalmente sustituidoscaracterizados porque un compuesto de formula 2 en donde R2, R6 y X tienen el mismo significado que se da anteriormente en laformula 1, se hace reaccionar enla presencia de un catalizador de transferencia de fases y una base con un compuesto de la formula 3 en donde A y R1 tienen el mismo significado que se daanteriormente en la formula 1 y Q es un grupo saliente.
ARP000103082A 1999-06-23 2000-06-21 PROCESO PARA LA PREPARACIoN DE TIAMETOXAM. AR024423A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH117199 1999-06-23

Publications (1)

Publication Number Publication Date
AR024423A1 true AR024423A1 (es) 2002-10-02

Family

ID=4204160

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000103082A AR024423A1 (es) 1999-06-23 2000-06-21 PROCESO PARA LA PREPARACIoN DE TIAMETOXAM.

Country Status (24)

Country Link
EP (1) EP1187833B1 (es)
JP (1) JP4588951B2 (es)
KR (1) KR100644739B1 (es)
CN (1) CN1247572C (es)
AR (1) AR024423A1 (es)
AT (1) ATE364042T1 (es)
AU (1) AU773966B2 (es)
BR (1) BR0011839B1 (es)
CA (1) CA2369404C (es)
CY (1) CY1106743T1 (es)
CZ (1) CZ300093B6 (es)
DE (1) DE60035109T2 (es)
DK (1) DK1187833T3 (es)
ES (1) ES2284506T3 (es)
HU (1) HU228645B1 (es)
IL (1) IL146580A0 (es)
MX (1) MXPA01012639A (es)
PL (1) PL202732B1 (es)
PT (1) PT1187833E (es)
RU (1) RU2258704C2 (es)
TW (1) TWI254713B (es)
UA (1) UA73306C2 (es)
WO (1) WO2001000623A1 (es)
ZA (1) ZA200110388B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006073973A2 (en) 2004-12-31 2006-07-13 Reddy Us Therapeutics, Inc. Novel benzylamine derivatives as cetp inhibitors
US8604055B2 (en) 2004-12-31 2013-12-10 Dr. Reddy's Laboratories Ltd. Substituted benzylamino quinolines as cholesterol ester-transfer protein inhibitors
DE102008052795B4 (de) 2008-10-22 2012-01-26 Balchem Corp. Verfahren zur Herstellung von Fettsäureestern ein- oder mehrwertiger Alkohole unter Verwendung spezieller hydroxyfunktioneller quartärer Ammoniumverbindungen als Katalysatoren
US9199967B2 (en) 2011-08-18 2015-12-01 Dr. Reddy's Laboratories Ltd. Substituted heterocyclic amine compounds as cholestryl ester-transfer protein (CETP) inhibitors
CA2850022C (en) 2011-09-27 2018-05-01 Dr. Reddy's Laboratories, Ltd. 5 - benzylaminomethyl - 6 - aminopyrazolo [3,4-b] pyridine derivatives as cholesteryl ester-transfer protein (cetp) inhibitors useful for the treatment of atherosclerosis
CN102372702A (zh) * 2011-11-17 2012-03-14 安徽省化工研究院 噻虫嗪的制备方法
CN103787922B (zh) * 2014-03-04 2016-06-01 新昌县鸿吉电子科技有限公司 一种合成硝基取代化合物的工业催化方法
CN103880832B (zh) * 2014-04-04 2016-06-15 连云港市金囤农化有限公司 一种噻虫嗪的制备方法
GB2514927B (en) * 2014-05-28 2019-04-17 Rotam Agrochem Int Co Ltd Thiamethoxam and uses thereof
GB2511010B (en) * 2014-05-28 2017-05-03 Rotam Agrochem Int Co Ltd Method of producing thiamethoxam
GB2564284A (en) * 2014-05-28 2019-01-09 Rotam Agrochem Int Co Ltd Thiamethoxam and uses thereof
CN107400123A (zh) * 2017-08-28 2017-11-28 江苏绿叶农化有限公司 一种噻虫嗪的生产方法
EP3480196A1 (en) 2017-11-02 2019-05-08 Jiangsu Rotam Chemistry Co., Ltd Process for the preparation of thiamethoxam
AR124935A1 (es) 2021-03-01 2023-05-24 Syngenta Crop Protection Ag Formulaciones plaguicidas

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2822050B2 (ja) * 1989-02-04 1998-11-05 日本バイエルアグロケム株式会社 ２―ニトロイミノイミダゾリジン類の製法
JP3159859B2 (ja) * 1994-02-09 2001-04-23 日本バイエルアグロケム株式会社 殺虫性ニトロ化合物
DE19904310A1 (de) * 1999-01-28 2000-08-03 Bayer Ag Verfahren zur Herstellung heterocyclischer Verbindungen

Also Published As

Publication number Publication date
RU2258704C2 (ru) 2005-08-20
BR0011839B1 (pt) 2010-11-03
ATE364042T1 (de) 2007-06-15
ZA200110388B (en) 2002-06-20
JP4588951B2 (ja) 2010-12-01
KR100644739B1 (ko) 2006-11-13
PL202732B1 (pl) 2009-07-31
CN1247572C (zh) 2006-03-29
WO2001000623A1 (en) 2001-01-04
AU773966B2 (en) 2004-06-10
PL352401A1 (en) 2003-08-25
CA2369404C (en) 2010-06-08
TWI254713B (en) 2006-05-11
CY1106743T1 (el) 2012-05-23
JP2003503409A (ja) 2003-01-28
CZ300093B6 (cs) 2009-01-28
AU5684700A (en) 2001-01-31
MXPA01012639A (es) 2002-06-21
DK1187833T3 (da) 2007-10-08
BR0011839A (pt) 2002-03-05
CA2369404A1 (en) 2001-01-04
HU228645B1 (en) 2013-04-29
UA73306C2 (en) 2005-07-15
CN1356998A (zh) 2002-07-03
EP1187833B1 (en) 2007-06-06
CZ20014524A3 (cs) 2002-03-13
DE60035109D1 (de) 2007-07-19
ES2284506T3 (es) 2007-11-16
DE60035109T2 (de) 2008-02-07
PT1187833E (pt) 2007-09-05
EP1187833A1 (en) 2002-03-20
IL146580A0 (en) 2002-07-25
KR20020022712A (ko) 2002-03-27
HUP0202050A3 (en) 2004-09-28
HUP0202050A2 (en) 2002-09-28

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Legal Events

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FG Grant, registration
FD Application declared void or lapsed, e.g., due to non-payment of fee