ZA966666B - Derivatives of 5-0-desosaminyl 6-0-methyl erythronolide A, their preparation process and their use in the preparation of biologically active products. - Google Patents

Derivatives of 5-0-desosaminyl 6-0-methyl erythronolide A, their preparation process and their use in the preparation of biologically active products.

Info

Publication number
ZA966666B
ZA966666B ZA9606666A ZA966666A ZA966666B ZA 966666 B ZA966666 B ZA 966666B ZA 9606666 A ZA9606666 A ZA 9606666A ZA 966666 A ZA966666 A ZA 966666A ZA 966666 B ZA966666 B ZA 966666B
Authority
ZA
South Africa
Prior art keywords
preparation
desosaminyl
derivatives
biologically active
active products
Prior art date
Application number
ZA9606666A
Other languages
English (en)
Inventor
Alain Bonnet
Bernadette Chappert
Jacques Lagouardat
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of ZA966666B publication Critical patent/ZA966666B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
ZA9606666A 1995-10-09 1996-08-06 Derivatives of 5-0-desosaminyl 6-0-methyl erythronolide A, their preparation process and their use in the preparation of biologically active products. ZA966666B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9511861A FR2739620B1 (fr) 1995-10-09 1995-10-09 Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number Publication Date
ZA966666B true ZA966666B (en) 1997-08-06

Family

ID=9483377

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9606666A ZA966666B (en) 1995-10-09 1996-08-06 Derivatives of 5-0-desosaminyl 6-0-methyl erythronolide A, their preparation process and their use in the preparation of biologically active products.

Country Status (33)

Country Link
US (1) US6011142A (no)
EP (1) EP0854879B1 (no)
JP (1) JP4327248B2 (no)
KR (1) KR100451063B1 (no)
CN (1) CN1067401C (no)
AP (1) AP888A (no)
AR (1) AR004688A1 (no)
AT (1) ATE212034T1 (no)
AU (1) AU708351B2 (no)
BG (1) BG63752B1 (no)
BR (1) BR9610959A (no)
CA (1) CA2231562C (no)
CZ (1) CZ293430B6 (no)
DE (1) DE69618607T2 (no)
DK (1) DK0854879T3 (no)
EA (1) EA000765B1 (no)
EE (1) EE03878B1 (no)
ES (1) ES2171722T3 (no)
FR (1) FR2739620B1 (no)
GE (1) GEP20032899B (no)
HU (1) HUP9900136A3 (no)
IL (1) IL123613A0 (no)
MX (1) MX9802655A (no)
NO (1) NO312592B1 (no)
PL (1) PL183645B1 (no)
PT (1) PT854879E (no)
RO (1) RO118874B1 (no)
SI (1) SI0854879T1 (no)
SK (1) SK283619B6 (no)
TR (1) TR199800624T1 (no)
UA (1) UA52621C2 (no)
WO (1) WO1997013774A2 (no)
ZA (1) ZA966666B (no)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777282B1 (fr) * 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
KR20020007374A (ko) * 1999-04-16 2002-01-26 추후제출 매크롤라이드 항감염제
EP1171447A2 (en) 1999-04-16 2002-01-16 Ortho-McNeil Pharmaceutical, Inc. Ketolide antibacterials
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
GB0031312D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
ES2552682T3 (es) * 2003-03-10 2015-12-01 Merck Sharp & Dohme Corp. Agentes antibacterianos novedosos
WO2009055557A1 (en) * 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
WO2010048601A1 (en) 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Biodefenses using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
AU2010292010B2 (en) 2009-09-10 2016-01-07 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and MAC diseases
SI2550286T1 (sl) 2010-03-22 2016-04-29 Cempra Pharmaceuticals, Inc. Kristalne oblike makrolida in njihove uporabe
RU2608390C2 (ru) 2010-05-20 2017-01-18 Семпра Фармасьютикалз, Инк. Способы получения макролидов и кетолидов, и промежуточных соединений для их получения
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ，インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
RU2658050C2 (ru) 2012-03-27 2018-06-19 Семпра Фармасьютикалз, Инк. Парентеральные составы для введения макролидных антибиотиков
US9861616B2 (en) 2013-03-14 2018-01-09 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
CN105188712A (zh) 2013-03-15 2015-12-23 森普拉制药公司 用于制备大环内酯抗菌剂的收敛方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
DK90788A (da) * 1987-02-24 1988-08-25 Beecham Group Plc Erythromycinderivater
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
KR0166996B1 (ko) * 1992-04-22 1999-01-15 우에하라 아키라 5-o-데소사미닐에리쓰로노라이드a 유도체
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
EP0682038A4 (en) * 1993-01-26 1996-12-27 Taisho Pharmaceutical Co Ltd 5-O-DESOSAMINYLERYTHRONOLIDE DERIVATIVE.

Also Published As

Publication number Publication date
NO312592B1 (no) 2002-06-03
EP0854879B1 (fr) 2002-01-16
BG102350A (en) 1999-03-31
SK283619B6 (sk) 2003-10-07
FR2739620A1 (fr) 1997-04-11
EA000765B1 (ru) 2000-04-24
CN1067401C (zh) 2001-06-20
SK43198A3 (en) 1998-11-04
NO981630D0 (no) 1998-04-08
MX9802655A (es) 1998-11-30
JP4327248B2 (ja) 2009-09-09
DE69618607T2 (de) 2002-08-14
NO981630L (no) 1998-04-08
CZ293430B6 (cs) 2004-04-14
ES2171722T3 (es) 2002-09-16
BR9610959A (pt) 1999-03-02
PL183645B1 (pl) 2002-06-28
WO1997013774A2 (fr) 1997-04-17
EA199800280A1 (ru) 1998-10-29
DK0854879T3 (da) 2002-05-06
KR19990064100A (ko) 1999-07-26
UA52621C2 (uk) 2003-01-15
TR199800624T1 (xx) 1998-06-22
PT854879E (pt) 2002-07-31
EE9800109A (et) 1998-10-15
ATE212034T1 (de) 2002-02-15
US6011142A (en) 2000-01-04
PL326001A1 (en) 1998-08-17
IL123613A0 (en) 1998-10-30
GEP20032899B (en) 2003-02-25
AU7220896A (en) 1997-04-30
JPH11513401A (ja) 1999-11-16
DE69618607D1 (de) 2002-02-21
SI0854879T1 (en) 2002-08-31
HUP9900136A3 (en) 2000-04-28
AP888A (en) 2000-11-10
EP0854879A2 (fr) 1998-07-29
AR004688A1 (es) 1999-03-10
WO1997013774A3 (fr) 1997-05-29
CA2231562C (fr) 2006-11-28
KR100451063B1 (ko) 2004-12-17
EE03878B1 (et) 2002-10-15
HUP9900136A1 (hu) 1999-05-28
CZ105598A3 (cs) 1998-07-15
BG63752B1 (bg) 2002-11-29
FR2739620B1 (fr) 1997-12-19
RO118874B1 (ro) 2003-12-30
AU708351B2 (en) 1999-08-05
CA2231562A1 (fr) 1997-04-17
CN1199403A (zh) 1998-11-18

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