ZA959675B - 6-Aryl pyrido (2,3-d) pyrimidines and naphthydridines for inhibiting protein tyrosine kinase mediated cellular proliferation - Google Patents

6-Aryl pyrido (2,3-d) pyrimidines and naphthydridines for inhibiting protein tyrosine kinase mediated cellular proliferation

Info

Publication number
ZA959675B
ZA959675B ZA959675A ZA959675A ZA959675B ZA 959675 B ZA959675 B ZA 959675B ZA 959675 A ZA959675 A ZA 959675A ZA 959675 A ZA959675 A ZA 959675A ZA 959675 B ZA959675 B ZA 959675B
Authority
ZA
South Africa
Prior art keywords
naphthydridines
pyrimidines
tyrosine kinase
protein tyrosine
cellular proliferation
Prior art date
Application number
ZA959675A
Other languages
English (en)
Inventor
Clifton John Blankley
Annette Marian Doherty
James Marino Hamby
Robert Lee Panek
Mel Conrad Schroeder
Howard Daniel Hollis Showalter
Cleo Connolly
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of ZA959675B publication Critical patent/ZA959675B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA959675A 1994-11-14 1995-11-14 6-Aryl pyrido (2,3-d) pyrimidines and naphthydridines for inhibiting protein tyrosine kinase mediated cellular proliferation ZA959675B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US33905194A 1994-11-14 1994-11-14

Publications (1)

Publication Number Publication Date
ZA959675B true ZA959675B (en) 1996-05-29

Family

ID=23327276

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA959675A ZA959675B (en) 1994-11-14 1995-11-14 6-Aryl pyrido (2,3-d) pyrimidines and naphthydridines for inhibiting protein tyrosine kinase mediated cellular proliferation

Country Status (7)

Country Link
US (1) US5733913A (ko)
JP (1) JP4221530B2 (ko)
KR (1) KR100385520B1 (ko)
IL (1) IL115256A0 (ko)
SI (1) SI0790997T1 (ko)
UA (1) UA61047C2 (ko)
ZA (1) ZA959675B (ko)

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Also Published As

Publication number Publication date
SI0790997T1 (en) 2000-06-30
UA61047C2 (en) 2003-11-17
JPH10509452A (ja) 1998-09-14
JP4221530B2 (ja) 2009-02-12
US5733913A (en) 1998-03-31
KR100385520B1 (ko) 2003-10-10
IL115256A0 (en) 1995-12-31

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