ZA201209237B - Furanyl compounds and the use thereof - Google Patents

Furanyl compounds and the use thereof

Info

Publication number
ZA201209237B
ZA201209237B ZA2012/09237A ZA201209237A ZA201209237B ZA 201209237 B ZA201209237 B ZA 201209237B ZA 2012/09237 A ZA2012/09237 A ZA 2012/09237A ZA 201209237 A ZA201209237 A ZA 201209237A ZA 201209237 B ZA201209237 B ZA 201209237B
Authority
ZA
South Africa
Prior art keywords
furanyl compounds
furanyl
compounds
Prior art date
Application number
ZA2012/09237A
Other languages
English (en)
Inventor
Leah M Fung
Kyle W H Chan
Cathy A Swindlehurst
Original Assignee
Novomedix Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novomedix Llc filed Critical Novomedix Llc
Publication of ZA201209237B publication Critical patent/ZA201209237B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
ZA2012/09237A 2010-06-07 2012-12-06 Furanyl compounds and the use thereof ZA201209237B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35230810P 2010-06-07 2010-06-07
PCT/US2011/039377 WO2011156321A1 (en) 2010-06-07 2011-06-07 Furanyl compounds and the use thereof

Publications (1)

Publication Number Publication Date
ZA201209237B true ZA201209237B (en) 2015-05-27

Family

ID=44210539

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2012/09237A ZA201209237B (en) 2010-06-07 2012-12-06 Furanyl compounds and the use thereof

Country Status (11)

Country Link
US (3) US8722731B2 (enExample)
EP (1) EP2576532B1 (enExample)
JP (1) JP5855095B2 (enExample)
CN (2) CN103108868B (enExample)
AU (1) AU2011265047B2 (enExample)
CA (1) CA2801778C (enExample)
MX (2) MX2012014273A (enExample)
NZ (1) NZ604018A (enExample)
SG (1) SG186229A1 (enExample)
WO (1) WO2011156321A1 (enExample)
ZA (1) ZA201209237B (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103108868B (zh) 2010-06-07 2015-11-25 诺沃梅迪科斯有限公司 呋喃基化合物及其用途
CN110818660B (zh) * 2012-09-21 2023-09-12 罗得岛医院 用于治疗癌症的β-羟化酶抑制剂
EP2925718B1 (en) 2012-11-30 2018-08-01 Novomedix, LLC Substituted biaryl sulfonamides and the use thereof
WO2015088977A1 (en) * 2013-12-10 2015-06-18 Emory University Targeted protease compositions and uses related thereto
CN106102775A (zh) 2014-02-07 2016-11-09 效应物治疗公司 治疗纤维变性疾病的方法
US10548908B2 (en) * 2016-09-15 2020-02-04 Nostopharma, LLC Compositions and methods for preventing and treating heterotopic ossification and pathologic calcification
CN115515685B (zh) * 2020-03-03 2025-04-08 皮克医疗公司 Eif4e抑制剂及其用途

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US9663483B2 (en) 2017-05-30
CN103108868A (zh) 2013-05-15
WO2011156321A1 (en) 2011-12-15
MX367469B (es) 2019-08-23
EP2576532A1 (en) 2013-04-10
JP2013528215A (ja) 2013-07-08
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CA2801778A1 (en) 2011-12-15
AU2011265047B2 (en) 2014-10-23
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NZ604018A (en) 2015-02-27
CN104860907A (zh) 2015-08-26
US20160024040A1 (en) 2016-01-28
AU2011265047A1 (en) 2013-01-10
US8722731B2 (en) 2014-05-13
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US9149527B2 (en) 2015-10-06
JP5855095B2 (ja) 2016-02-09

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