ZA200903395B - Non-nucleoside reverse transcriptase inhibitors - Google Patents

Non-nucleoside reverse transcriptase inhibitors

Info

Publication number
ZA200903395B
ZA200903395B ZA200903395A ZA200903395A ZA200903395B ZA 200903395 B ZA200903395 B ZA 200903395B ZA 200903395 A ZA200903395 A ZA 200903395A ZA 200903395 A ZA200903395 A ZA 200903395A ZA 200903395 B ZA200903395 B ZA 200903395B
Authority
ZA
South Africa
Prior art keywords
reverse transcriptase
transcriptase inhibitors
nucleoside reverse
nucleoside
inhibitors
Prior art date
Application number
ZA200903395A
Other languages
English (en)
Inventor
Neville J Anthony
Robert Gomez
Samson M Jolly
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of ZA200903395B publication Critical patent/ZA200903395B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41921,2,3-Triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/16Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C07D249/18Benzotriazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ZA200903395A 2006-12-13 2009-05-18 Non-nucleoside reverse transcriptase inhibitors ZA200903395B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US87462906P 2006-12-13 2006-12-13

Publications (1)

Publication Number Publication Date
ZA200903395B true ZA200903395B (en) 2010-05-26

Family

ID=39277099

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200903395A ZA200903395B (en) 2006-12-13 2009-05-18 Non-nucleoside reverse transcriptase inhibitors

Country Status (29)

Country Link
US (2) US7781454B2 (fr)
EP (1) EP2121638B1 (fr)
JP (1) JP5123949B2 (fr)
KR (1) KR20090087481A (fr)
CN (1) CN101558050A (fr)
AR (1) AR064199A1 (fr)
AU (1) AU2007334598B2 (fr)
BR (1) BRPI0720196A2 (fr)
CA (1) CA2673093A1 (fr)
CL (1) CL2007003594A1 (fr)
CR (1) CR10843A (fr)
DO (1) DOP2009000138A (fr)
EA (1) EA200970572A1 (fr)
EC (1) ECSP099373A (fr)
GE (1) GEP20115320B (fr)
GT (1) GT200900158A (fr)
HN (1) HN2009001160A (fr)
IL (1) IL199103A0 (fr)
MA (1) MA31036B1 (fr)
MX (1) MX2009006285A (fr)
NI (1) NI200900103A (fr)
NO (1) NO20092636L (fr)
NZ (1) NZ577637A (fr)
PE (1) PE20081448A1 (fr)
SV (1) SV2009003294A (fr)
TN (1) TN2009000243A1 (fr)
TW (1) TW200831085A (fr)
WO (2) WO2008076223A1 (fr)
ZA (1) ZA200903395B (fr)

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JP5433582B2 (ja) 2007-11-14 2014-03-05 ジャンセン ファーマシューティカルズ, インコーポレイテッド. イミダゾ[1,2−a]ピリジン誘導体およびmGluR2受容体の正のアロステリック調節因子としてのその使用
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Also Published As

Publication number Publication date
BRPI0720196A2 (pt) 2013-12-31
EP2121638A2 (fr) 2009-11-25
NZ577637A (en) 2011-05-27
WO2008076223A1 (fr) 2008-06-26
US20100286192A1 (en) 2010-11-11
WO2008076225A3 (fr) 2008-08-07
GT200900158A (es) 2009-10-14
TW200831085A (en) 2008-08-01
IL199103A0 (en) 2010-03-28
CA2673093A1 (fr) 2008-06-26
NO20092636L (no) 2009-09-08
JP5123949B2 (ja) 2013-01-23
GEP20115320B (en) 2011-10-25
ECSP099373A (es) 2009-07-31
MX2009006285A (es) 2009-06-23
CR10843A (es) 2009-08-12
CN101558050A (zh) 2009-10-14
AU2007334598B2 (en) 2013-01-17
US20080275097A1 (en) 2008-11-06
AR064199A1 (es) 2009-03-18
PE20081448A1 (es) 2008-10-19
MA31036B1 (fr) 2009-12-01
DOP2009000138A (es) 2009-11-15
JP2010510989A (ja) 2010-04-08
US7781454B2 (en) 2010-08-24
WO2008076225A2 (fr) 2008-06-26
TN2009000243A1 (en) 2010-10-18
EA200970572A1 (ru) 2009-12-30
HN2009001160A (es) 2011-10-11
CL2007003594A1 (es) 2008-05-30
SV2009003294A (es) 2009-11-09
NI200900103A (es) 2010-01-26
KR20090087481A (ko) 2009-08-17
EP2121638B1 (fr) 2016-05-25
AU2007334598A1 (en) 2008-06-26

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