ZA200807756B - Novel 1,4-diaza-bicyclo[3.2.2] nonyl oxadiazolyl derivatives and their medical use - Google Patents
Novel 1,4-diaza-bicyclo[3.2.2] nonyl oxadiazolyl derivatives and their medical useInfo
- Publication number
- ZA200807756B ZA200807756B ZA200807756A ZA200807756A ZA200807756B ZA 200807756 B ZA200807756 B ZA 200807756B ZA 200807756 A ZA200807756 A ZA 200807756A ZA 200807756 A ZA200807756 A ZA 200807756A ZA 200807756 B ZA200807756 B ZA 200807756B
- Authority
- ZA
- South Africa
- Prior art keywords
- diseases
- disorders
- diaza
- bicyclo
- novel
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200600731 | 2006-05-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200807756B true ZA200807756B (en) | 2009-11-25 |
Family
ID=40616686
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200807756A ZA200807756B (en) | 2006-05-30 | 2007-05-29 | Novel 1,4-diaza-bicyclo[3.2.2] nonyl oxadiazolyl derivatives and their medical use |
Country Status (23)
| Country | Link |
|---|---|
| US (4) | US8158619B2 (fr) |
| EP (3) | EP2194056B1 (fr) |
| JP (2) | JP2009538866A (fr) |
| KR (1) | KR101458194B1 (fr) |
| CN (2) | CN101432286A (fr) |
| AT (3) | ATE518862T1 (fr) |
| AU (2) | AU2007267175A1 (fr) |
| BR (1) | BRPI0708843A2 (fr) |
| CA (2) | CA2653818A1 (fr) |
| DE (2) | DE602007006486D1 (fr) |
| DK (2) | DK2032574T3 (fr) |
| ES (1) | ES2342334T3 (fr) |
| IL (1) | IL193925A (fr) |
| MX (2) | MX2008014886A (fr) |
| MY (1) | MY147764A (fr) |
| NO (1) | NO20085398L (fr) |
| NZ (1) | NZ571288A (fr) |
| PL (1) | PL2032575T3 (fr) |
| PT (1) | PT2032575E (fr) |
| RU (1) | RU2427581C2 (fr) |
| UA (1) | UA95946C2 (fr) |
| WO (2) | WO2007138038A1 (fr) |
| ZA (1) | ZA200807756B (fr) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT2032575E (pt) | 2006-05-30 | 2010-07-09 | Neurosearch As | NOVO DERIVADO DE 1,4-DIAZA-BICICLO[3,2,2]NONIL-OXADIAZOLILO E A SUA APLICAÃO MéDICA |
| CA2667545A1 (fr) * | 2006-10-25 | 2008-05-02 | Neurosearch A/S | Composes de type oxadiazole et thiadiazole et leur utilisation comme modulateurs des recepteurs nicotiniques de l'acetylcholine |
| US7935695B2 (en) | 2007-08-17 | 2011-05-03 | Neurosearch A/S | 1,4-diaza-bicyclo[3.2.2]nonyl heteroaryl derivatives useful as nicotinic acetylcholine receptor ligands |
| JP2011513459A (ja) | 2008-03-11 | 2011-04-28 | ノイロサーチ アクティーゼルスカブ | ニコチン性アセチルコリン受容体のモジュレーターとして有用な、新規な１，４−ジアザ−ビシクロ［３．２．２］ノニルオキサジアゾリル誘導体 |
| US20110112078A1 (en) * | 2008-06-10 | 2011-05-12 | Neurosearch A/S | Novel oxadiazolyl-diazabicyclononane derivatives and their medical use |
| WO2010043539A1 (fr) * | 2008-10-13 | 2010-04-22 | Neurosearch A/S | Nouveaux dérivés d'oxadiazolyl-diazabicyclononane et leur utilisation médicale |
| WO2010063784A1 (fr) * | 2008-12-04 | 2010-06-10 | Neurosearch A/S | Nouveaux dérivés de diaza-bicyclononyl-phényle et leurs applications médicales |
| CA2750450A1 (fr) | 2009-01-26 | 2010-07-29 | Neurosearch A/S | Nouveaux derives d'indolyl-oxadiazolyl-diazabicyclononane et leur utilisation medicale et diagnostique |
| WO2010086280A1 (fr) | 2009-01-27 | 2010-08-05 | Neurosearch A/S | Nouveaux n-oxydes de dérivés de furanyl-oxadiazolyl-diazabicyclononane et leur utilisation médicale |
| WO2010086279A1 (fr) | 2009-01-27 | 2010-08-05 | Neurosearch A/S | Nouveaux dérivés de dibenzofuranyl-oxadiazolyl-diazabicyclononane, et utilisation médicale de ceux-ci |
| WO2010086278A1 (fr) | 2009-01-27 | 2010-08-05 | Neurosearch A/S | Nouveaux dérivés de benzodioxolyl-oxadiazolyl-diazabicyclononane et leur utilisation médicale |
| US20120071469A1 (en) * | 2009-05-14 | 2012-03-22 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.1]octane derivatives useful as nicotinic acetylcholine receptor modulators |
| JO3250B1 (ar) | 2009-09-22 | 2018-09-16 | Novartis Ag | إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 |
| EP2498826A1 (fr) | 2009-11-11 | 2012-09-19 | NeuroSearch AS | Dérivés de pyrrolyl-oxadiazolyl-diazabicyclononane marqués et leur utilisation dans des procédés de diagnostic |
| EP2513097A1 (fr) | 2009-12-18 | 2012-10-24 | NeuroSearch AS | Composés diazabicyclononyloxadiazole et leur utilisation en tant que modulateurs des récepteurs nicotiniques de l'acétylcholine |
| US8986654B2 (en) | 2011-04-15 | 2015-03-24 | Danpet Ab | Labelled and un-labelled methyl-pyrrolyl-oxadiazolyl-diazabicyclononane derivatives and their medical use |
| SG10202002990XA (en) | 2017-08-04 | 2020-05-28 | Skyhawk Therapeutics Inc | Methods and compositions for modulating splicing |
| BR112020021194A2 (pt) | 2018-04-18 | 2021-03-23 | Constallation Pharmaceuticals, Inc. | moduladores de enzimas modificadoras de metila, composições e usos dos mesmos |
| CN112262143A (zh) | 2018-05-21 | 2021-01-22 | 星座制药公司 | 甲基修饰酶的调节剂、其组合物和用途 |
| CN113660936A (zh) * | 2019-02-04 | 2021-11-16 | 斯基霍克疗法公司 | 用于调节剪接的方法和组合物 |
| CN114007613A (zh) | 2019-02-05 | 2022-02-01 | 斯基霍克疗法公司 | 用于调节剪接的方法和组合物 |
| EP3920928A4 (fr) | 2019-02-06 | 2022-09-28 | Skyhawk Therapeutics, Inc. | Procédés et compositions pour moduler l'épissage |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2809731B1 (fr) * | 2000-05-31 | 2002-07-19 | Sanofi Synthelabo | Derives de 1,4-diazabicyclo-[3.2.2] nonane-pheylisoxazole, leur preparation et leur application en therapeutique |
| FR2809732B1 (fr) * | 2000-05-31 | 2002-07-19 | Sanofi Synthelabo | DERIVES DE 4(-2-PHENYLTHIAZOL-5-yl)-1,4-DIAZABICYCLO-[3.2.2] NONANE, LEUR PREPARATION ET LEUR APPLICATION ENTHERAPEUTIQUE |
| FR2832713B1 (fr) * | 2001-11-23 | 2004-02-13 | Sanofi Synthelabo | Derives de 4-(1,3,4-thiadiazol-2-yl)-1,4-diazabicyclo[3.2.2] nonane, leur preparation et leur application en therapeutique |
| FR2832712B1 (fr) * | 2001-11-23 | 2004-02-13 | Sanofi Synthelabo | Derives de 4-(oxadiazol-3-yl)-1,4-diazabicyclo[3.2.2]nonane, leur preparation et leur application en therapeutique |
| PT1551835E (pt) * | 2002-09-30 | 2007-03-30 | Neurosearch As | Novos derivados de 1, 4-diazabicicloalcano, sua preparação e utilização |
| ES2280836T3 (es) | 2002-09-30 | 2007-09-16 | Neurosearch A/S | Nuevos derivados de 1,4-diazabicicloalcano, su preparacion y uso. |
| DE60309740T2 (de) * | 2002-11-11 | 2007-03-29 | Neurosearch A/S | 1,4-dizabicyclo(3,2,2)nonane derivative, verfahren zu ihrer herstellung und therapeutical verwendung |
| US6996399B2 (en) * | 2003-01-13 | 2006-02-07 | Micrel, Inc. | Wireless device and method using frequency hopping and sweep modes |
| ATE450263T1 (de) | 2004-02-04 | 2009-12-15 | Neurosearch As | Diazabicyclische aryl-derivate als cholinerge rezeptor-modulatoren |
| WO2006087306A2 (fr) | 2005-02-16 | 2006-08-24 | Neurosearch A/S | Nouveaux derives aryle diazabicycliques et leur utilisation medicale |
| PT2032575E (pt) | 2006-05-30 | 2010-07-09 | Neurosearch As | NOVO DERIVADO DE 1,4-DIAZA-BICICLO[3,2,2]NONIL-OXADIAZOLILO E A SUA APLICAÃO MéDICA |
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2007
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- 2007-05-29 MX MX2008014886A patent/MX2008014886A/es active IP Right Grant
- 2007-05-29 WO PCT/EP2007/055169 patent/WO2007138038A1/fr active Application Filing
- 2007-05-29 NZ NZ571288A patent/NZ571288A/en not_active IP Right Cessation
- 2007-05-29 DK DK07729590.5T patent/DK2032574T3/da active
- 2007-05-29 PL PL07729591T patent/PL2032575T3/pl unknown
- 2007-05-29 AU AU2007267175A patent/AU2007267175A1/en not_active Abandoned
- 2007-05-29 DE DE602007006486T patent/DE602007006486D1/de active Active
- 2007-05-29 EP EP10154049A patent/EP2194056B1/fr not_active Not-in-force
- 2007-05-29 RU RU2008139481/04A patent/RU2427581C2/ru not_active IP Right Cessation
- 2007-05-29 US US12/297,333 patent/US8158619B2/en active Active
- 2007-05-29 KR KR1020087031858A patent/KR101458194B1/ko not_active IP Right Cessation
- 2007-05-29 DK DK07729591.3T patent/DK2032575T3/da active
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