ZA200708086B - Treatment of Parkinson's disease, obstructive sleep apnea, dementia with Lewy bodies, vascular dementia with non-imidazole alkylamines histamine H3-receptor ligands - Google Patents

Treatment of Parkinson's disease, obstructive sleep apnea, dementia with Lewy bodies, vascular dementia with non-imidazole alkylamines histamine H3-receptor ligands

Info

Publication number
ZA200708086B
ZA200708086B ZA200708086A ZA200708086A ZA200708086B ZA 200708086 B ZA200708086 B ZA 200708086B ZA 200708086 A ZA200708086 A ZA 200708086A ZA 200708086 A ZA200708086 A ZA 200708086A ZA 200708086 B ZA200708086 B ZA 200708086B
Authority
ZA
South Africa
Prior art keywords
dementia
parkinson
disease
treatment
sleep apnea
Prior art date
Application number
ZA200708086A
Other languages
English (en)
Inventor
Schwartz Jean-Charles
Lecomte Jeanne-Marie
Original Assignee
Bioprojet Soc Civ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35169680&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200708086(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bioprojet Soc Civ filed Critical Bioprojet Soc Civ
Publication of ZA200708086B publication Critical patent/ZA200708086B/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4453Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ZA200708086A 2005-04-01 2007-09-20 Treatment of Parkinson's disease, obstructive sleep apnea, dementia with Lewy bodies, vascular dementia with non-imidazole alkylamines histamine H3-receptor ligands ZA200708086B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05290727A EP1707203A1 (en) 2005-04-01 2005-04-01 Treatment of parkinson's disease obstructive sleep apnea, dementia with lewy bodies, vascular dementia with non-imidazole alkylamines histamine H3- receptor ligands

Publications (1)

Publication Number Publication Date
ZA200708086B true ZA200708086B (en) 2008-10-29

Family

ID=35169680

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200708086A ZA200708086B (en) 2005-04-01 2007-09-20 Treatment of Parkinson's disease, obstructive sleep apnea, dementia with Lewy bodies, vascular dementia with non-imidazole alkylamines histamine H3-receptor ligands

Country Status (27)

Country Link
US (1) US8486947B2 (ru)
EP (2) EP1707203A1 (ru)
JP (3) JP5546761B2 (ru)
KR (1) KR101308527B1 (ru)
CN (1) CN101171009B (ru)
AU (1) AU2006228413C1 (ru)
BR (1) BRPI0612216B1 (ru)
CA (1) CA2603656C (ru)
CY (1) CY1114636T1 (ru)
DK (1) DK1863487T4 (ru)
EA (1) EA016007B1 (ru)
ES (1) ES2426008T5 (ru)
HR (1) HRP20130748T4 (ru)
MA (1) MA29353B1 (ru)
ME (1) ME01713B (ru)
MX (1) MX2007012162A (ru)
NO (1) NO343603B1 (ru)
NZ (1) NZ561940A (ru)
PL (1) PL1863487T5 (ru)
PT (1) PT1863487E (ru)
RS (1) RS52911B2 (ru)
SG (1) SG147415A1 (ru)
SI (1) SI1863487T2 (ru)
TN (1) TNSN07365A1 (ru)
UA (1) UA94902C2 (ru)
WO (1) WO2006103546A2 (ru)
ZA (1) ZA200708086B (ru)

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US9108948B2 (en) 2006-06-23 2015-08-18 Abbvie Inc. Cyclopropyl amine derivatives
NZ611323A (en) 2006-06-23 2014-10-31 Abbvie Bahamas Ltd Cyclopropyl amine derivatives as histamin h3 receptor modulators
FR2903904A1 (fr) * 2006-07-21 2008-01-25 Bioprojet Soc Civ Ile Association de modafinil et d'un antagoniste ou agoniste inverse du recepteur h3
CA2858816A1 (en) 2006-07-25 2008-01-31 Cephalon, Inc. Pyridizinone derivatives and uses thereof to treat diseases, disorders and/or conditions that may be mediated or modulated by inhibition of h3 receptors
US8153813B2 (en) 2007-12-20 2012-04-10 Abbott Laboratories Benzothiazole and benzooxazole derivatives and methods of use
MX2010008375A (es) 2008-01-30 2011-03-04 Cephalon Inc Star Derivados de piperidina espirocíclicos substituidos como ligandos de receptores de histamina-3 (h3).
FR2932479A1 (fr) * 2008-06-13 2009-12-18 Servier Lab Nouveaux derives azabicycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US9186353B2 (en) 2009-04-27 2015-11-17 Abbvie Inc. Treatment of osteoarthritis pain
US8853390B2 (en) 2010-09-16 2014-10-07 Abbvie Inc. Processes for preparing 1,2-substituted cyclopropyl derivatives
US9181275B2 (en) 2011-08-11 2015-11-10 Abbvie Inc. Mercaptoamidine derivatives and methods of use
WO2013151982A1 (en) 2012-04-03 2013-10-10 Arena Pharmaceuticals, Inc. Methods and compounds useful in treating pruritus, and methods for identifying such compounds
CN110292638A (zh) * 2012-10-05 2019-10-01 Vtv治疗有限责任公司 治疗轻度和中度阿尔茨海默病的方法
EP3391886A1 (en) 2017-04-19 2018-10-24 Novartis AG The use of a h3r inverse agonist for the treatment of shift work disorder
US11654283B2 (en) 2019-03-06 2023-05-23 Medtronic Xomed, Inc. Obstructive sleep apnea patient programmer for implantable devices
EP4248969A1 (en) 2022-03-23 2023-09-27 Bioprojet Use of pitolisant for treating severe fatigue

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FR2579596B1 (fr) 1985-03-26 1987-11-20 Inst Nat Sante Rech Med (imidazolyl-4) piperidines, leur preparation et leur application en therapeutique
FR2671083B1 (fr) 1990-12-31 1994-12-23 Inst Nat Sante Rech Med Nouvelles 4-(4-imidazolyl) piperidines substituees en 1, leur preparation ainsi que leurs applications therapeutiques.
ES2108107T3 (es) 1991-02-27 1997-12-16 Seed Capital Investments Derivados de imidazol que tienen actividad antagonista en el receptor h3 de histamina.
EP0619818B1 (en) 1991-12-18 1996-07-10 Schering Corporation Imidazoylalkyl substituted with a six membered nitrogen containing heterocyclic ring
IL104125A (en) 1991-12-18 2000-08-31 Schering Corp Imidazolyl or imidazoylalkyl substituted with a four or five membered nitrogen containing heterocyclic ring and pharmaceutical compositions comprising them
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JP3522790B2 (ja) 1993-06-08 2004-04-26 花王株式会社 H3−レセプター刺激薬
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Also Published As

Publication number Publication date
SG147415A1 (en) 2008-11-28
UA94902C2 (ru) 2011-06-25
CA2603656A1 (en) 2006-10-05
JP2016106142A (ja) 2016-06-16
ES2426008T5 (es) 2020-03-20
RS52911B2 (sr) 2019-11-29
AU2006228413C1 (en) 2012-02-02
EA200702135A1 (ru) 2008-04-28
BRPI0612216A2 (pt) 2010-10-26
MX2007012162A (es) 2007-11-22
SI1863487T1 (sl) 2013-09-30
DK1863487T4 (da) 2019-10-14
CA2603656C (en) 2015-06-16
US20090318433A1 (en) 2009-12-24
ME01713B (me) 2014-09-20
HRP20130748T4 (hr) 2019-11-15
PL1863487T5 (pl) 2021-08-09
CY1114636T1 (el) 2016-10-05
JP5546761B2 (ja) 2014-07-09
JP2008534572A (ja) 2008-08-28
RS52911B (en) 2014-02-28
US8486947B2 (en) 2013-07-16
NO343603B1 (no) 2019-04-08
EP1707203A1 (en) 2006-10-04
MA29353B1 (fr) 2008-03-03
JP5955872B2 (ja) 2016-07-20
WO2006103546A3 (en) 2007-03-01
KR20080002904A (ko) 2008-01-04
TNSN07365A1 (fr) 2008-12-31
CN101171009A (zh) 2008-04-30
SI1863487T2 (sl) 2019-11-29
ES2426008T3 (es) 2013-10-18
EA016007B1 (ru) 2012-01-30
EP1863487B1 (en) 2013-05-29
CN101171009B (zh) 2012-11-07
PL1863487T3 (pl) 2014-10-31
EP1863487A2 (en) 2007-12-12
WO2006103546A2 (en) 2006-10-05
KR101308527B1 (ko) 2013-09-17
DK1863487T3 (da) 2013-08-12
HRP20130748T1 (en) 2013-10-11
AU2006228413B2 (en) 2011-09-15
PT1863487E (pt) 2013-08-29
EP1863487B2 (en) 2019-07-17
AU2006228413A1 (en) 2006-10-05
NZ561940A (en) 2010-06-25
NO20075086L (no) 2007-12-27
JP2014062126A (ja) 2014-04-10
BRPI0612216B1 (pt) 2022-04-19

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