ZA200605587B - Novel phenylalanine derivative - Google Patents
Novel phenylalanine derivative Download PDFInfo
- Publication number
- ZA200605587B ZA200605587B ZA200605587A ZA200605587A ZA200605587B ZA 200605587 B ZA200605587 B ZA 200605587B ZA 200605587 A ZA200605587 A ZA 200605587A ZA 200605587 A ZA200605587 A ZA 200605587A ZA 200605587 B ZA200605587 B ZA 200605587B
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- ZA
- South Africa
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- pharmaceutically acceptable
- acceptable salts
- carbon atoms
- hydrogen atom
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Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Oncology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Transplantation (AREA)
- Endocrinology (AREA)
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- Emergency Medicine (AREA)
- Vascular Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2003425347 | 2003-12-22 | ||
| JP2004074943 | 2004-03-16 | ||
| JP2004159919 | 2004-05-28 | ||
| JP2004260319 | 2004-09-07 |
Publications (1)
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| ZA200605587B true ZA200605587B (en) | 2008-02-27 |
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| Application Number | Title | Priority Date | Filing Date |
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| ZA200605587A ZA200605587B (en) | 2003-12-22 | 2004-12-22 | Novel phenylalanine derivative |
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| Country | Link |
|---|---|
| US (2) | US7345049B2 (zh) |
| EP (3) | EP2615087A3 (zh) |
| JP (1) | JP4743659B2 (zh) |
| KR (2) | KR20110098980A (zh) |
| CN (2) | CN1917881B (zh) |
| AU (1) | AU2004303696B2 (zh) |
| BR (1) | BRPI0418026A (zh) |
| CA (1) | CA2550843C (zh) |
| ES (1) | ES2548853T3 (zh) |
| IL (1) | IL176469A (zh) |
| NO (1) | NO337628B1 (zh) |
| NZ (1) | NZ548420A (zh) |
| RU (1) | RU2390520C2 (zh) |
| WO (1) | WO2005061466A1 (zh) |
| ZA (1) | ZA200605587B (zh) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL223152B1 (pl) | 2000-08-18 | 2016-10-31 | Ajinomoto Kk | Pochodne fenyloalaniny, kompozycja farmaceutyczna oraz zastosowanie tych pochodnych |
| ATE345127T1 (de) * | 2000-09-29 | 2006-12-15 | Ajinomoto Kk | Neue phenylalanin-derivate |
| JP4470219B2 (ja) * | 2002-02-20 | 2010-06-02 | 味の素株式会社 | 新規フェニルアラニン誘導体 |
| CN100436429C (zh) * | 2003-02-20 | 2008-11-26 | 味之素株式会社 | 具有喹唑二酮骨架的苯丙氨酸衍生物的制造方法及制造中间体 |
| WO2005046697A1 (ja) * | 2003-11-14 | 2005-05-26 | Ajinomoto Co., Inc. | フェニルアラニン誘導体の徐放性経口投与製剤 |
| EP1683524B1 (en) * | 2003-11-14 | 2011-01-19 | Ajinomoto Co., Inc. | Solid dispersion or medicinal solid dispersion preparation of phenylalanine derivative |
| EP1688410B1 (en) * | 2003-11-27 | 2014-03-05 | Ajinomoto Co., Inc. | Crystal of phenylalanine derivative and process for producing the same |
| CN1917881B (zh) * | 2003-12-22 | 2014-11-26 | 味之素株式会社 | 新型苯基丙氨酸衍生物 |
| CN102503899B (zh) * | 2005-06-21 | 2014-09-24 | 味之素株式会社 | 苯基丙氨酸衍生物的结晶、其制备方法及其应用 |
| WO2007028789A1 (en) * | 2005-09-07 | 2007-03-15 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa | Quinazoline derivatives as antiviral agents |
| US20090111828A1 (en) * | 2005-11-23 | 2009-04-30 | Astrazeneca Ab | L-alanine derivatives |
| CA2635531C (en) * | 2005-12-29 | 2014-06-17 | Lexicon Pharmaceutical Inc. | Multicyclic amino acid derivatives and methods of their use |
| US7834050B2 (en) | 2006-03-29 | 2010-11-16 | Duke University | Small molecule insulin mimetics absent quinones |
| JP2009539815A (ja) * | 2006-06-09 | 2009-11-19 | アストラゼネカ アクチボラグ | 固形腫瘍の治療用のａ５ｂ１アンタゴニストとしてのＮ−（ベンゾイル）−Ｏ−［２−（ピリジン−２−イルアミノ）エチル］−Ｌ−チロシン誘導体と関連化合物 |
| EP2103601B1 (en) | 2006-11-22 | 2012-03-14 | Ajinomoto Co., Inc. | Process for production of phenylalanine derivatives having quinazolinedione skeletons and intermediates for the production |
| WO2008093065A1 (en) * | 2007-01-29 | 2008-08-07 | Astrazeneca Ab | L-ALANINE DERIVATIVES AS α5βL ANTAGONISTS |
| WO2008125811A1 (en) * | 2007-04-11 | 2008-10-23 | Astrazeneca Ab | N-[HETEROARYLCARBONYL]-S-THIENYL-L-ALANINE DERIVATIVES AS α5β1 ANTAGONISTS |
| EP2138482A4 (en) | 2007-04-19 | 2011-06-15 | Astellas Pharma Inc | BICYCLIC HETEROCYCLIC COMPOUND |
| WO2011094890A1 (en) | 2010-02-02 | 2011-08-11 | Argusina Inc. | Phenylalanine derivatives and their use as non-peptide glp-1 receptor modulators |
| WO2011122619A1 (ja) | 2010-03-29 | 2011-10-06 | 味の素株式会社 | フェニルアラニン誘導体の塩の結晶 |
| JP2013530963A (ja) | 2010-06-09 | 2013-08-01 | レセプトス インコーポレイテッド | 新規のｇｌｐ−１受容体安定化薬および調節薬 |
| DK2713722T3 (en) | 2011-05-31 | 2017-07-03 | Celgene Int Ii Sarl | Newly known GLP-1 receptor stabilizers and modulators |
| EP2791112B1 (en) | 2011-12-12 | 2020-09-23 | Celgene International II Sàrl | Carboxylic acid derivatives comprising four cycles acting as glp-1 receptor modulators for therapy of diseases such as diabetes |
| EP2842945B1 (en) | 2012-04-24 | 2016-10-26 | EA Pharma Co., Ltd. | Sulfonamide derivative and medicinal use thereof |
| CN102993105B (zh) * | 2012-12-19 | 2014-06-11 | 西南大学 | 1-甲基-2,4-喹唑啉二酮衍生物及其制备方法和应用 |
| KR102271179B1 (ko) * | 2013-06-11 | 2021-07-01 | 셀진 인터내셔널 Ii 에스에이알엘 | 신규의 glp-1 수용체 조절제 |
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- 2004-12-22 ZA ZA200605587A patent/ZA200605587B/en unknown
- 2004-12-22 KR KR1020117019338A patent/KR20110098980A/ko not_active Application Discontinuation
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- 2004-12-22 EP EP13152904.2A patent/EP2615087A3/en not_active Withdrawn
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- 2004-12-22 AU AU2004303696A patent/AU2004303696B2/en not_active Ceased
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- 2004-12-22 KR KR1020067014754A patent/KR101194176B1/ko active IP Right Grant
- 2004-12-22 EP EP14181015.0A patent/EP2803667A1/en not_active Withdrawn
- 2004-12-22 WO PCT/JP2004/019704 patent/WO2005061466A1/ja active Application Filing
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